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showing 10 items of 8115 documents

High chemoselectivity of CS dipolarophile in 1,3-dipolar cycloaddition of nitrilimines and 1,2,4-triazepin-5-one derivatives: experimental, theoreti…

2005

Substituted 2,7-dimethyl-3-thioxo-3,4,5,6-tetrahydro-2H-[1,2,4]triazepin-5-one reacts as a dipolarophile with several N-aryl-C-ethoxycarbonylnitrilimines, in equimolar quantities, to give, in all cases, two types of products: diethyl 3-(p-aryl)-2-[N′-(p-aryl)-N′-(2′,7′-dimethyl-5′-oxo-5′,6′-dihydro-2H-[1,2,4]triazepin-3′-yl)-hydrazino]-2,3-dihydro[1,3,4]thiadiazole-2,5-dicarboxylate (3a–3c in 20–25% yield) and ethyl 4-(p-aryl)-5-imino-1,4-dihydro[1,3,4]thiadiazole carboxylate (4a–4c in 45–50% yield). When 1:2 stoichiometry was used, the formation of product 3 (50%) was favoured. The reaction is entirely chemo- and regioselective. The structures of the compounds obtained, where aryl stands f…

ArylOrganic ChemistryRegioselectivityMedicinal chemistrychemistry.chemical_compoundchemistryNucleophileYield (chemistry)Electrophile13-Dipolar cycloadditionOrganic chemistryCarboxylatePhysical and Theoretical ChemistryChemoselectivityJournal of Physical Organic Chemistry
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Trienediolates of hexadienoic acids in synthesis. Addition to unsaturated ketones. A convergent approach to the synthesis of retinoic acids

1995

Abstract The regioselectivity of the addition of the lithium trienediolates generated from hexa-2,4dienoic acids 1 and 2 or the dihydropyran-2ones 4 and 5 to unsaturated ketones 6 is studied. Equilibration conditions favour reaction of the trienediolates through their ω carbon, and the ketones according to 1,2- and 1,4-additions. β-Ionone 6a and the aryl-butenone 6b lead to the 1,2-ω-adducts 8 , which undergo a facile acid catalyzed dehydration to retmoic acids 11 . On reaction with the unsaturated ketone 6b or with the aryl ketones 21 , the trimethyldihydropyran-2one S leads to γ-adducts derived from deprotonation of the chain methyl mbstituent along with the 1,4-ω-adducts.

ArylOrganic Chemistrychemistry.chemical_elementRegioselectivitymedicine.diseaseBiochemistrychemistry.chemical_compoundDeprotonationchemistryAcid catalyzedUnsaturated ketoneDrug DiscoverymedicineOrganic chemistryLithiumDehydrationCarbonTetrahedron
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ChemInform Abstract: Trienediolates of Hexadienoic Acids in Synthesis. Addition to Unsaturated Ketones. A Convergent Approach to the Synthesis of Ret…

2010

Abstract The regioselectivity of the addition of the lithium trienediolates generated from hexa-2,4dienoic acids 1 and 2 or the dihydropyran-2ones 4 and 5 to unsaturated ketones 6 is studied. Equilibration conditions favour reaction of the trienediolates through their ω carbon, and the ketones according to 1,2- and 1,4-additions. β-Ionone 6a and the aryl-butenone 6b lead to the 1,2-ω-adducts 8 , which undergo a facile acid catalyzed dehydration to retmoic acids 11 . On reaction with the unsaturated ketone 6b or with the aryl ketones 21 , the trimethyldihydropyran-2one S leads to γ-adducts derived from deprotonation of the chain methyl mbstituent along with the 1,4-ω-adducts.

Arylchemistry.chemical_elementRegioselectivityGeneral Medicinemedicine.diseaseTerpenechemistry.chemical_compoundDeprotonationchemistryAcid catalyzedmedicineOrganic chemistryLithiumDehydrationCarbonChemInform
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Redécouverte d'une faune pléistocène dans les remplissages karstiques de Tam Hang au Laos : premiers résultats.

2008

12 pages; The discovery of a Pleistocene fauna in karstic fills at TamHang in Laos: preliminary results. TamHang, located in northeastern Laos, in the Hua Pan province, is a reference site not only for its numerous archaeological and human remains, but also for its two faunal assemblages, whose composition suggests different dating in the Pleistocene. Discovered in 1934 by Jacques Fromaget, a new excavation of the site has been undertaken in 2003. During this campaign, at Tam Hang south, 575 isolated teeth of mammals were extracted from a deep layer of calcareous breccia. This assemblage corresponds to that one described by Arambourg and Fromaget [C. Arambourg, J. Fromaget, Le gisement quat…

Asie du Sud-Est continentale010506 paleontologyPleistocene[SHS.ARCHEO]Humanities and Social Sciences/Archaeology and PrehistoryBiostratigraphy010502 geochemistry & geophysicsSouth-East Asia mainland01 natural sciencesTam HangSoutheast asiaPhanerozoicMilieu karstiqueKarstic system0105 earth and related environmental sciences[ SDU.STU.PG ] Sciences of the Universe [physics]/Earth Sciences/PaleontologyGeneral Engineering15. Life on landArchaeologyPleistoceneLaos[ SHS.ARCHEO ] Humanities and Social Sciences/Archaeology and PrehistoryClastic rockQuaternary[SDU.STU.PG]Sciences of the Universe [physics]/Earth Sciences/PaleontologyCenozoicGeology
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El día a día del trabajo social en Salud: funciones y disfunciones

2010

Este artículo aporta información sobre la Asociación Española de Trabajo Social y Salud, su Delegación en la Comunidad Valenciana y la jornada que celebró en noviembre 2009, cuyo lema era: 'El día a día del Trabajo Social en Salud: funciones y disfunciones' y su objetivo propiciar un espacio de intercambio, análisis, reflexión y proposición sobre la práctica diaria en el campo de la salud por parte de los trabajadores sociales, para una mejor praxis profesional, una mayor atención integral, una mayor eficiencia asistencial, una mayor satisfacción de los ciudadanos y una mayor rentabilidad social de la intervención social en el ámbito sanitario. This article describes the Spanish Association…

Asociación Española de Trabajo Social y Salud Trabajo Social en Salud intervención social en el ámbito sanitario práctica de los trabajadores sociales sanitarios. Spanish Association of Social Work and Health Social Work in Health Healthy social worker's Trainee. Artículo:SOCIOLOGÍA::Cambio y desarrollo social [UNESCO]UNESCO::SOCIOLOGÍA::Cambio y desarrollo social
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Mafie straniere e 'ndrangheta al nord. Una sfida alla tenuta dell'art. 416 bis?

2014

L'autore analizza i percorsi giurisprudenziali riguardanti l'applicazione del delitto di associazione mafiosa al fenomeno delle mafie straniere e delle mafie "storiche" in aree non tradizionali (coma la 'ndrangheta al Nord), con l'obbiettivo di verificare la conformità o meno di tali percorsi alle interpretazioni consolidate. Secondo l'autore, soltanto con riferimento ad alcuni recenti approdi giurisprudenziali concernenti l'espansione della 'ndrangheta in Piemonte e in Liguria si registra un mutamento degli orientamenti consolidati in materia, sul versante in particolare dei requisiti oggettivi del metodo mafioso di cui al 3° comma dell'art. 416 bis c.p.

Associazione di tipo mafioso mafie straniere 'ndrangheta metodo mafiosoSettore IUS/17 - Diritto Penale
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Sulla requisitoria del P.G. nel processo Dell’Utri: un vero e proprio atto di fede nel concorso esterno

2012

L'Autore commenta a caldo il "caso Dell'Utri" in ordine al concorso esterno in associazione mafiosa, puntando l'attenzione sugli ambigui rapporti tra impresa e associazioni criminali

Associazione mafiosaConcorso esternoSettore IUS/17 - Diritto Penale
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A Roma una mafia c'è e si vede

2015

All''analisi critica della giurisprudenza in tema di esportabilità dell' inquadramento entro la cornice del delitto di associazione mafiosa dei fatti contestati agli indagati in un noto processo romano si accompagnano alcune proposte de iure condendo.

Associazione mafiosa- organizzazione territoriale esportabilità del modelloSettore IUS/17 - Diritto Penale
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Tethyan magnetostratigraphy from Pizzo Mondello (Sicily) and correlation to the Late Triassic Newark astrochronological polarity time scale

2004

We present the magnetostratigraphy and stable isotope stratigraphy from an expanded (~430-m-thick) Upper Triassic marine limestone section at Pizzo Mondello, Sicily, and review published biostratigraphic information that can be used to defi ne the location of the conodont Carnian-Norian and Norian- Rhaetian boundaries in this section. Pizzo Mondello offers good potential for magnetostratigraphic correlation of marine biostratigraphic and chemostratigraphic data with the continental Newark astrochronological polarity time scale (APTS) for development of an integrated Late Triassic time scale. The relatively stable average values of 18O centered on 0‰ are a strong indication that the Cherty …

AstrochronologybiologyPaleontologyGeologyastrochronological polarity time scaleBiostratigraphyOverprintingbiology.organism_classificationPaleontologyGeophysicsStratigraphyTethyStratigraphic sectionRadiometric datingmagnetostratigraphybiostratigraphyNewarkConodontSicilyLate TriassicGeologyMagnetostratigraphyGeological Society of America Bulletin
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Pharmacological blockade of the fatty acid amide hydrolase (FAAH) alters neural proliferation, apoptosis and gliosis in the rat hippocampus, hypothal…

2015

Endocannabinoids participate in the control of neurogenesis, neural cell death and gliosis. The pharmacological effect of the fatty acid amide hydrolase (FAAH) inhibitor URB597, which limits the endocannabinoid degradation, was investigated in the present study. Cell proliferation (phospho-H3(+) or BrdU(+) cells) of the main adult neurogenic zones as well as apoptosis (cleaved caspase-3(+)), astroglia (GFAP(+)), and microglia (Iba1(+) cells) were analyzed in the hippocampus, hypothalamus and striatum of rats intraperitoneally treated with URB597 (0.3 mg/kg/day) at one dose/4-days resting or 5 doses (1 dose/day). Repeated URB597 treatment increased the plasma levels of the N-acylethanolamine…

AstrocitosNeurobiologia del desenvolupamentAmidohidrolasasCannabinoid receptorCarbamatos:Chemicals and Drugs::Amino Acids Peptides and Proteins::Proteins::Intracellular Signaling Peptides and Proteins::Apoptosis Regulatory Proteins::Caspases [Medical Subject Headings]:Phenomena and Processes::Cell Physiological Phenomena::Cell Physiological Processes::Cell Differentiation::Neurogenesis [Medical Subject Headings]medicine.medical_treatment:Chemicals and Drugs::Carbohydrates::Monosaccharides::Hexoses::Glucose [Medical Subject Headings]Apoptosis:Phenomena and Processes::Physiological Phenomena::Body Constitution::Body Weights and Measures::Body Size::Body Weight [Medical Subject Headings]chemistry.chemical_compound:Chemicals and Drugs::Amino Acids Peptides and Proteins::Proteins::Membrane Proteins::Receptors Cell Surface::Receptors G-Protein-Coupled::Receptors Cannabinoid::Receptor Cannabinoid CB1 [Medical Subject Headings]0302 clinical medicine:Chemicals and Drugs::Organic Chemicals::Carboxylic Acids::Acids Acyclic::Carbamates [Medical Subject Headings]Fatty acid amide hydrolaseReceptor cannabinoide CB1:Organisms::Eukaryota::Animals [Medical Subject Headings]FAAHGliosishealth care economics and organizations:Chemicals and Drugs::Nucleic Acids Nucleotides and Nucleosides::Nucleosides::Deoxyribonucleosides::Deoxyuridine::Bromodeoxyuridine [Medical Subject Headings]:Chemicals and Drugs::Lipids::Glycerides::Triglycerides [Medical Subject Headings]Original Research0303 health sciencesNeurogenesisBenzamidas:Chemicals and Drugs::Polycyclic Compounds::Steroids::Cholestanes::Cholestenes::Cholesterol [Medical Subject Headings]Endocannabinoid systemEtanolaminas3. Good healthEndocannabinoides:Chemicals and Drugs::Lipids::Fatty Acids::Fatty Acids Unsaturated::Fatty Acids Monounsaturated::Oleic Acids [Medical Subject Headings]CannabinoidesMicroglíalipids (amino acids peptides and proteins)medicine.symptomColesterol:Chemicals and Drugs::Organic Chemicals::Hydrocarbons::Terpenes::Cannabinoids [Medical Subject Headings]:Chemicals and Drugs::Lipids::Fatty Acids::Palmitic Acids [Medical Subject Headings]psychological phenomena and processesProliferación celularmedicine.medical_specialtyCerebroNeurogenesiseducationBiologyBromodesoxiuridina:Anatomy::Nervous System::Neuroglia::Microglia [Medical Subject Headings]Triglicéridoslcsh:RC321-571Ácidos oléicosRatas03 medical and health sciencesCellular and Molecular NeuroscienceInternal medicineHipocampomedicineCaspasa 3:Anatomy::Nervous System::Central Nervous System::Brain::Limbic System::Hippocampus [Medical Subject Headings]:Phenomena and Processes::Cell Physiological Phenomena::Cell Physiological Processes::Cell Growth Processes::Cell Proliferation [Medical Subject Headings]lcsh:Neurosciences. Biological psychiatry. Neuropsychiatry030304 developmental biologyPalmitoylethanolamide:Chemicals and Drugs::Chemical Actions and Uses::Pharmacologic Actions::Molecular Mechanisms of Pharmacological Action::Neurotransmitter Agents::Endocannabinoids [Medical Subject Headings]:Chemicals and Drugs::Enzymes and Coenzymes::Enzymes::Hydrolases::Amidohydrolases [Medical Subject Headings]Cannabinoids:Anatomy::Cells::Neuroglia::Astrocytes [Medical Subject Headings]Peso corporalEnergy metabolism:Anatomy::Nervous System::Central Nervous System::Brain [Medical Subject Headings]:Anatomy::Nervous System::Central Nervous System::Brain::Limbic System::Hypothalamus [Medical Subject Headings]URB597:Phenomena and Processes::Cell Physiological Phenomena::Cell Physiological Processes::Cell Death [Medical Subject Headings]:Diseases::Pathological Conditions Signs and Symptoms::Pathologic Processes::Gliosis [Medical Subject Headings]:Chemicals and Drugs::Organic Chemicals::Amines::Amino Alcohols::Ethanolamines [Medical Subject Headings]Muerte celular:Phenomena and Processes::Cell Physiological Phenomena::Cell Physiological Processes::Cell Death::Apoptosis [Medical Subject Headings]:Organisms::Eukaryota::Animals::Chordata::Vertebrates::Mammals::Rodentia::Muridae::Murinae::Rats [Medical Subject Headings]EndocrinologyURB597chemistryGliosisnervous systemGlucosaCannabinoidEnergy Metabolism:Chemicals and Drugs::Organic Chemicals::Amides::Benzamides [Medical Subject Headings]HipotálamoÁcidos palmíticos030217 neurology & neurosurgeryNeuroscienceFrontiers in Cellular Neuroscience
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