Search results for "inflammation"

showing 10 items of 2662 documents

Mast cell-derived mediators promote murine neutrophil effector functions

2013

Mast cells are able to trigger life-saving immune responses in murine models for acute inflammation. In such settings, several lines of evidence indicate that the rapid and protective recruitment of neutrophils initiated by the release of mast cell-derived pro-inflammatory mediators is a key element of innate immunity. Herein, we investigate the impact of mast cells on critical parameters of neutrophil effector function. In the presence of activated murine bone marrow-derived mast cells, neutrophils freshly isolated from bone marrow rapidly lose expression of CD62L and up-regulate CD11b, the latter being partly driven by mast cell-derived TNF and GM-CSF. Mast cells also strongly enhance neu…

PhagocytosisImmunologyApoptosisInflammation610 Medicine & healthmast cellsBiology142-005 142-005Neutrophil ActivationlungMiceImmune systemPhagocytosisneutrophilsmedicineAnimalsImmunology and AllergyCells CulturedMice Knockout2403 ImmunologyInnate immune systemTumor Necrosis Factor-alpharodentGranulocyte-Macrophage Colony-Stimulating FactorPneumoniaGeneral MedicineFlow CytometryMast cellMice Mutant StrainsCell biologycell activationMice Inbred C57BLInterleukin 33medicine.anatomical_structureinflammationImmunology2723 Immunology and AllergyTumor necrosis factor alphamedicine.symptomCell activation
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Natural Products and Inflammation

2017

Inflammation (or inflammatory reaction) is the response to body aggression by a pathogen agent, an allergen, a toxic compound, a tissue lesion, etc.[...]

Pharmaceutical ScienceInflammation010402 general chemistrymedicine.disease_cause01 natural sciencesAnalytical ChemistryLesionlcsh:QD241-441Allergenlcsh:Organic chemistryDrug DiscoveryHumansMedicinePhysical and Theoretical ChemistryPathogenInflammationBiological Products010405 organic chemistrybusiness.industryAggressionOrganic Chemistry0104 chemical sciencesEditorialn/aChemistry (miscellaneous)ImmunologyMolecular Medicinemedicine.symptombusinessMolecules
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Pentoxifylline and Oxypurinol: Potential Drugs to Prevent the “Cytokine Release (Storm) Syndrome” Caused by SARS-CoV-2?

2020

Background: COVID-19, caused by SARS-CoV-2, is a potentially lethal, rapidly-expanding pandemic and many efforts are being carried out worldwide to understand and control the disease. COVID-19 patients may display a cytokine release syndrome, which causes severe lung inflammation, leading, in many instances, to death. Objective: This paper is intended to explore the possibilities of controlling the COVID-19-associated hyperinflammation by using licensed drugs with anti-inflammatory effects. Hypothesis: We have previously described that pentoxifylline alone, or in combination with oxypurinol, reduces the systemic inflammation caused by experimentally-induced pancreatitis in rats. Pentoxifyl…

Pharmacology0303 health sciencesbusiness.industryInflammationmedicine.diseaseSystemic inflammationPentoxifyllineProinflammatory cytokine03 medical and health scienceschemistry.chemical_compoundCytokine release syndrome0302 clinical medicinechemistry030220 oncology & carcinogenesisDrug DiscoveryImmunologyMedicineAcute pancreatitisPancreatitismedicine.symptomXanthine oxidasebusiness030304 developmental biologymedicine.drugCurrent Pharmaceutical Design
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SAR150640, a selective β3-adrenoceptor agonist, prevents human myometrial remodelling and activation of matrix metalloproteinase in an in vitro model…

2010

Background and purpose:  The uterine pathophysiology underlying inflammatory conditions such as chorioamnionitis remains largely unclear. As we have shown that β3-adrenoceptors act as regulators of myometrial inflammation, we wanted to investigate the potential role of β3-adrenoceptors in preventing uterine remodelling induced by inflammation. Experimental approach:  The consequences of human chorioamnionitis on myometrial remodelling were characterized by Sirius Red staining and metalloproteinase (MMP) expression, and compared with the effects of incubating human myometrial samples with Escherichia coli lipopolysaccharide (LPS) in vitro. We also assessed the effect of SAR150640, a selectiv…

PharmacologyAgonistmedicine.medical_specialtyMetalloproteinasemedicine.drug_classMyometriumInflammationMatrix metalloproteinaseMMP9BiologyChorioamnionitismedicine.diseasechemistry.chemical_compoundEndocrinologychemistryInternal medicinemedicinemedicine.symptomSirius RedBritish Journal of Pharmacology
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Nitric oxide, derived from inducible nitric oxide synthase, decreases hypoxia inducible factor-1α in macrophages during aspirin-induced mesenteric in…

2010

Background and purpose:  Nitric oxide (NO) modulates expression of hypoxia inducible factor-1 (HIF-1), a transcription factor regulating function of myeloid cells. Here, we have assessed the role played by NO, formed by inducible NOS (iNOS), in the inflammation induced by aspirin in the gut, by modulating HIF-1 activity. Experimental approach:  The role of iNOS-derived NO on leucocyte–endothelial interactions induced by aspirin was evaluated by intravital microscopy in mesenteric venules of rats pretreated with selective iNOS inhibitors, 1400W or l-N6-(1-iminoethyl)-lysine. NO was localized by fluorescence microscopy, using DAF-FM. iNOS, HIF-1α and CD36 were localized by immunohistochemistr…

PharmacologyAspirinmedicine.medical_specialtybiologyChemistryCD36InflammationNitric oxideNitric oxide synthasechemistry.chemical_compoundEndocrinologyHypoxia-inducible factorsInternal medicinemedicinebiology.proteinmedicine.symptomImmunostainingIntravital microscopymedicine.drugBritish Journal of Pharmacology
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GABA and GABA receptors in the gastrointestinal tract: from motility to inflammation

2015

Although an extensive body of literature confirmed γ-aminobutyric acid (GABA) as mediator within the enteric nervous system (ENS) controlling gastrointestinal (GI) function, the true significance of GABAergic signalling in the gut is still a matter of debate. GABAergic cells in the bowel include neuronal and endocrine-like cells, suggesting GABA as modulator of both motor and secretory GI activity. GABA effects in the GI tract depend on the activation of ionotropic GABAA and GABAC receptors and metabotropic GABAB receptors, resulting in a potential noteworthy regulation of both the excitatory and inhibitory signalling in the ENS. However, the preservation of GABAergic signalling in the gut …

PharmacologyChemistryGABAA receptorGABAB receptorPharmacologyInflammatory Bowel DiseasesInhibitory postsynaptic potentialSettore BIO/09 - FisiologiaGastrointestinal TractMetabotropic receptorReceptors GABAGABA receptorAnimalsHumansGABAergicEnteric nervous systemGastrointestinal MotilityGABA • GABAA receptors • GABAB receptors • Gastrointestinal motility • Inflammationgamma-Aminobutyric Acid5-HT receptorPharmacological Research
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Differential effects of leflunomide on leukocytes: Inhibition of ratin vivo adhesion and humanin vitro oxidative burst without affecting surface mark…

1994

Leflunomide has been shown to combat effectively autoimmune diseases in a number of animal models, as well as chronic polyarthritis of humans. Here we report on the effects of this novel drug on the adherence of leukocytes to endothelium, an essential event in establishment and maintenance of inflammation. The entry of cells into tissues is dependent on interactions of adhesion molecules. The process of diapedesis, which these molecules control, involves three phases: tethering, triggering of receptors on endothelial cells and firm attachment of leukocytes to these cells. The interaction of LECAM-1 (constitutively expressed on circulating leukocytes) and P- and E-selectins on the vessel wll…

PharmacologyEndotheliumCell adhesion moleculeImmunologyInflammationBiologyToxicologyIn vitroCell biologyRespiratory burstmedicine.anatomical_structureIntegrin alpha MImmunologymedicinebiology.proteinPharmacology (medical)medicine.symptomLeflunomidemedicine.drugHumaninAgents and Actions
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The nitric oxide related therapeutic phenomenon: a challenging task.

2002

Nitric oxide (NO), produced from L-arginine by the activity of constitutive and inducible NO synthases, has been implicated in a wide range of physiological and pathophysiological processes. Low concentrations of this mediator play homeostatic roles, whereas NO is up-regulated in a number of pathological states and can have damaging effects. Pharmacological modulation of NO levels or NO biosynthesis may be a therapeutic strategy for a number of conditions, although the reported results can be some times controversial. Inhibitors of NO synthases exhibit different selectivity for the neuronal, endothelial or inducible isoforms, which contributes to their beneficial and detrimental effects. Re…

PharmacologyGene isoformbiologyInflammationNitric OxideNitric oxideNitric oxide synthasePathogenesischemistry.chemical_compoundMediatorchemistryMechanism of actionDrug DiscoveryImmunologymedicinebiology.proteinAnimalsHumansmedicine.symptomNeuroscienceHomeostasisCurrent pharmaceutical design
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Recent progress in revealing the biological and medical significance of the non-neuronal cholinergic system.

2015

This special issue of International Immunopharmacology is the proceedings of the Fourth International Symposium on Non-neuronal Acetylcholine that was held on August 28-30, 2014 at the Justus Liebig University of Giessen in Germany. It contains original contributions of meeting participants covering the significant progress in understanding of the biological and medical significance of the non-neuronal cholinergic system extending from exciting insights into molecular mechanisms regulating this system via miRNAs over the discovery of novel cholinergic cellular signaling circuitries to clinical implications in cancer, wound healing, immunity and inflammation, cardiovascular, respiratory and …

PharmacologyInflammationWound HealingStem CellseducationImmunologyRespiratory Tract DiseasesBiologyImmunopharmacologyAcetylcholineMicroRNAsGene Expression RegulationCardiovascular DiseasesNeoplasmsImmunologyCholinergic systemImmunology and AllergyCholinergicAnimalsNeuroscienceSignal TransductionInternational immunopharmacology
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Effects of triterpenes on the immune system.

2010

Ethnopharmacological relevance: Triterpenes, which comprise a broad chemical group of active principles, are implicated in the mechanisms of action and pharmacological effects of many medicinal plants used in folk medicine against diseases in which the immune system is implicated. They have been described as anti-inflammatory, antiviral, antimicrobial, and antitumoral agents, as well as being immunomodulator compounds. Several of them are implicated in the resolution of immune diseases, although their effects have not always been clearly correlated. Aim of the review: The aim of this review is to compile relevant data on the mechanisms of action of triterpenes isolated from active ethnomedi…

PharmacologyMechanism (biology)Anti-HIV AgentsInflammationNF-κBComputational biologyBiologyAntimicrobialMajor histocompatibility complexTriterpeneschemistry.chemical_compoundImmune systemCucurbitacinschemistryAdjuvants ImmunologicImmune SystemDrug DiscoveryImmunologymedicinebiology.proteinAnimalsHumansmedicine.symptomMedicinal plantsTranscription FactorsJournal of ethnopharmacology
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