Search results for "l-5"

showing 10 items of 373 documents

CCDC 1534754: Experimental Crystal Structure Determination

2017

Related Article: Xiang-Yu Chen, Qiang Liu, Pankaj Chauhan, Sun Li, Anssi Peuronen, Kari Rissanen, Ehsan Jafari, Dieter Enders|2017|Angew.Chem.,Int.Ed.|56|6241|doi:10.1002/anie.201702881

4-(3-methyl-4-nitro-12-oxazol-5-yl)-5-(thiophen-2-yl)-56-dihydro[11'-biphenyl]-3(4H)-oneSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 872438: Experimental Crystal Structure Determination

2012

Related Article: B.Abu Thaher, P.Koch, D.Schollmeyer, S.Laufer|2012|Acta Crystallogr.,Sect.E:Struct.Rep.Online|68|o632|doi:10.1107/S1600536812004096

4-(4-Fluorophenyl)-1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-5-amineSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 2009112: Experimental Crystal Structure Determination

2020

Related Article: Jonathan Bould, Kamil Lang, Kaplan Kirakci, Luis Cerdán, Daniel Roca-Sanjuán, Antonio Francés-Monerris, William Clegg, Paul G. Waddell, Marcel Fuciman, Tomáš Polívka, Michael G. S. Londesborough|2020|Inorg.Chem.|59|17058|doi:10.1021/acs.inorgchem.0c02277

5'6':67-conjuncto-(22'-dichloro-11'33'44'-hexamethyl-6'7':8'9':9'10'-tri-muH-nido-decaborane)-(77'88'10'-pentamethyl-56:89:910-tri-muH-nido-decaborane) 5'6':67-conjuncto-(22'-dichloro-11'33'44'-hexamethyl-6'7':8'9':9'10'-tri-muH-nido-decaborane)-(77'88'1010'-hexamethyl-56:89:910-tri-muH-nido-decaborane)Space GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 2169529: Experimental Crystal Structure Determination

2023

Related Article: Renè Hommelsheim, Sandra Bausch, Arjuna Selvakumar, Mostafa Amer, Khai-Nghi Truong, Kari Rissanen, Carsten Bolm|2023|Chem.-Eur.J.|29|e202203729|doi:10.1002/chem.202203729

5-methyl-3-phenyl-5a67899a-hexahydro-[123]triazolo[51-c][124]benzothiadiazin-5-one unknown solvateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 1571124: Experimental Crystal Structure Determination

2017

Related Article: Toms Rekis, Agris Be¯rzinš, Inese Sarcevica, Artis Kons, Ma¯rtinš Balodis, Lia¯na Orola, Heike Lorenz, Andris Actinš|2018|Cryst.Growth Des.|18|264|doi:10.1021/acs.cgd.7b01203

6-(2-(4-methoxyphenyl)-1H-benzimidazol-5-yl)-5-methyl-45-dihydropyridazin-3(2H)-oneSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Contaminación atmosférica en la Península Ibérica medida con Sentinel-5P

2021

Este estudio está basado en el análisis de la contaminación atmosférica sobre la Península Ibérica mediante el uso de técnicas de teledetección. La metodología utilizada ha sido el procesamiento de imágenes tomadas por el satélite Sentinel-5P, sensor TROPOMI, mediante código en Python. En el trabajo hemos generado la cartografía del monóxido de carbono y de dióxido de nitrógeno para el mes de marzo de los años 2019 y 2020. Durante el mes de marzo de 2020, la contaminación atmosférica se vio reducida debido a las duras restricciones que vivió la población debido al COVID-19, por lo que vemos la importancia de realizar este tipo de estudios para conocer el comportamiento de la atmósfera y el …

:GEOGRAFÍA [UNESCO]contaminación atmosféricaTROPOMIsentinel-5PNO2península IbéricaUNESCO::GEOGRAFÍA
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Application of tRNS to improve multiple sclerosis fatigue: a pilot, single-blind, sham-controlled study

2019

We evaluated the effects of transcranial random noise stimulation (tRNS) on fatigue in 17 subjects with relapsing–remitting multiple sclerosis with low physical disability. Two different patient groups underwent real or sham stimulation for 10 days, targeting the primary motor cortex of the dominant side or contralateral to the most compromised limb. In the ‘real group’, beneficial effects were observed using the Modified Fatigue Impact Scale (p = 0.04; physical subscale: p = 0.03), the subscales ‘change in health’ (p = 0.006) and ‘role limitations due to physical problems’ (p = 0.001) of the Multiple Sclerosis Quality of Life-54, and by assessing the patient impression of perceived fatigue…

AdultMale0301 basic medicinemedicine.medical_specialtyPhysical disabilityNeurologyFatigue treatmentStimulationTranscranial Direct Current StimulationSeverity of Illness IndexPlacebosYoung Adult03 medical and health sciencesMultiple Sclerosis Relapsing-Remitting0302 clinical medicinePhysical medicine and rehabilitationOutcome Assessment Health CaremedicineHumansMultiple sclerosiSingle-Blind MethodBeneficial effectsFatigueBiological Psychiatrybusiness.industryMSQoL-54Multiple sclerosisMotor CortextRNSmedicine.diseaseFatigue impact scalePsychiatry and Mental health030104 developmental biologyPrimary motor areaNeurologyQuality of LifeFemaleMFISNeurology (clinical)Single blindPrimary motor cortexbusiness030217 neurology & neurosurgeryJournal of Neural Transmission
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Synthesis and antifungal activity of new N-(1-phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides

2002

N-(1-Phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides 6, with a Benodanil-like structure, were synthesized by refluxing in acetic acid the corresponding benzotriazinones 5 with potassium iodide for 1 h in order to study the role on the antifungal activity of the N-substitution with an aromatic heterocyclic system on benzamide moiety. Among the tested iododerivatives, compounds 6d,f,g,h possess interesting activities toward some phytopathogenic fungal strains.

AntifungalAntifungal AgentsIndazolesMagnetic Resonance SpectroscopySpectrophotometry Infraredmedicine.drug_classStereochemistryColony Count MicrobialPharmaceutical Sciencechemistry.chemical_elementCarboxamideMicrobial Sensitivity TestsIodineChemical synthesisAcetic acidchemistry.chemical_compoundN-(1-phenyl-4-carbetoxypyrazol-5-yl)-2-iodobenzamides N-(indazol-3-yl)-2-iodobenzamides N-(indazol-3-yl)-2-iodobenzamides antifungal activityDrug DiscoverymedicineMoietyBenzamideChemistryFungiSettore CHIM/08 - Chimica FarmaceuticaBenzamidesPyrazolesIl Farmaco
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Mode and mechanism of neurotensin action in rat proximal colon

1997

Abstract This study examined the mechanism of action of neurotensin on intraluminal pressure in rat proximal colon. The direct and indirect contractile response to neurotensin (100 nM) was abolished in Ca 2+ -free solution, and was antagonized by nifedipine (1–5–10 nM) and potentiated by Bay K 8644 (methyl 1,4-dihydro-2,6-dimethyl-3-nitro-4-(2-trifluoromethylphenyl)-pyridine-5-carboxylate) (10–100–1000 nM). Neurotensin, in the presence of nifedipine (10 nM) and atropine (1 μM), induced a tetrodotoxin-insensitive inhibitory effect, which was antagonized by SR 48692 (2[(1-(7-chloro-4-quinolinyl)-5-(2,6-dimethoxy-phenyl)pyrazol-3-yl) carbonyl amino]tricyclo (3.3.1.1. 3.7 ) decan-2-carboxylic a…

Atropinemedicine.medical_specialtyNifedipineColonchemistry.chemical_elementCholinergic AgonistsIn Vitro TechniquesCalciumInhibitory postsynaptic potentialApaminCholinergic Antagonistschemistry.chemical_compoundNifedipineInternal medicinemedicineAnimalsReceptors NeurotensinRats WistarNeurotensinPharmacologyChemistryMuscle Smooth3-Pyridinecarboxylic acid 14-dihydro-26-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)- Methyl esterBethanecholCalcium Channel BlockersRatsCalcium Channel AgonistsEndocrinologyApaminMechanism of actionQuinolinesExcitatory postsynaptic potentialBiophysicsPyrazolesCalciummedicine.symptomMuscle Contractionmedicine.drugMuscle contractionNeurotensinEuropean Journal of Pharmacology
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Lures for red palm weevil trapping systems: aggregation pheromone and synthetic kairomone

2015

[EN] BACKGROUNDThe optimisation of the lure is essential for the implementation of trapping systems to control insect pests. In this work, the response of the red palm weevil (RPW), Rhynchophorus ferrugineus Olivier, to increasing emission rates of its aggregation pheromone (ferrugineol) and the efficacy of a convenient synthetic kairomone based on fermentation odours (ethyl acetate and ethanol) have been evaluated in different years and locations along the Mediterranean basin. RESULTSIn general, although capture data and emission had noticeable variability among locations, significantly fewer RPW were captured in pyramidal Picusan (R) traps with the lowest ferrugineol emission rates tested…

Behavior AnimalEthanolMass trappingmonitoringEthyl acetateRhynchophorus ferrugineuRhynchophorus ferrugineusPheromonesmass trappingmonitoringSettore AGR/11 - Entomologia Generale E ApplicataQUIMICA ORGANICAInsect HormonesInsect ScienceAnimalsWeevilsPest Control BiologicalAgronomy and Crop Science4-methyl-5-nonanol
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