Search results for "radical"

showing 10 items of 1401 documents

Intermolecular oxidative dehydrogenative 3,3′-coupling of benzo[b]furans and benzo[b]thiophenes promoted by DDQ/H+: total synthesis of shandougenine B

2016

With an excess of a strong acid, 2,3-dichloro-5,6-dicyano-1,4-quinone (DDQ) is shown to promote metal-free intermolecular oxidative dehydrogenative (ODH) 3,3'-coupling of 2-aryl-benzo[b]furans and 2-aryl-benzo[b]thiophenes up to 92% yield as demonstrated with 9 substrates. Based on the analysis of oxidation potentials and molecular orbitals combined with EPR, NMR and UV-Vis observations, the studied reaction is initiated by a DDQ-substrate charge transfer complex and presumably proceeds via oxidation of the substrate into an electrophilic radical cation that further reacts with another molecule of a neutral substrate. The coupling reactivity can easily be predicted from the oxidation potent…

116 Chemical sciencesEFFICIENTfree radicalscoupling reactionsvapaat radikaalit010402 general chemistryPhotochemistry01 natural sciencesMedicinal chemistryCoupling reactionoxidative dehydrogenationC BOND FORMATIONSCHOLL REACTIONELECTRON-TRANSFERMolecular orbitalReactivity (chemistry)luonnonaineiden synteesiDIPHOSPHINE LIGANDSta116BASIS-SETSCATALYZED STEREOSELECTIVE REACTIONS010405 organic chemistryChemistryOrganic ChemistrykytkentäreaktiotSubstrate (chemistry)Total synthesishapettava dehydroganaatiolaskennallinen kemiaCharge-transfer complex0104 chemical sciencesRadical ionsynthesis of natural productsACIDElectrophileCATION-RADICALSHETEROCYCLESOrganic Chemistry Frontiers
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Synthesis, Stability and Relaxivity of TEEPO-Met: An Organic Radical as a Potential Tumour Targeting Contrast Agent for Magnetic Resonance Imaging

2018

Cancer is a widespread and life-threatening disease and its early-stage diagnosis is vital. One of the most effective, non-invasive tools in medical diagnostics is magnetic resonance imaging (MRI) with the aid of contrast agents. Contrast agents that are currently in clinical use contain metals, causing some restrictions in their use. Also, these contrast agents are mainly non-specific without any tissue targeting capabilities. Subsequently, the interest has notably increased in the research of organic, metal-free contrast agents. This study presents a new, stable organic radical, TEEPO-Met, where a radical moiety 2,2,6,6-tetraethylpiperidinoxide (TEEPO) is attached to an amino acid, methio…

116 Chemical sciencesPharmaceutical ScienceContrast Media01 natural sciencesAnalytical Chemistrylaw.inventionGLUCOSENuclear magnetic resonancePiperidineslawHeterocyclic CompoundsNeoplasmsDrug DiscoveryMoietymagneettitutkimusSpin labelElectron paramagnetic resonanceta116orgaaniset yhdisteetmedicine.diagnostic_testMolecular StructureChemistryPhantoms ImagingRelaxation (NMR)radicalsMagnetic Resonance Imaging3. Good healthChemistry (miscellaneous)Molecular MedicineMRIRadical010402 general chemistryvapaat radikaalitImaging phantomArticleCyclic N-OxidesvarjoainetutkimusnitroxidesmedicineAnimalsHumanscontrast agentstyppiyhdisteetPhysical and Theoretical Chemistrymethionine010405 organic chemistryOrganic ChemistryElectron Spin Resonance SpectroscopyMagnetic resonance imagingIN-VITRO3126 Surgery anesthesiology intensive care radiologynitroxides; radicals; methionine; contrast agents; MRI; NMR; EPRIn vitroNMRTRANSPORT0104 chemical sciencesREDUCTIONSPIN-LABEL1182 Biochemistry cell and molecular biologyEPRMolecules; Volume 23; Issue 5; Pages: 1034
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Radical sex role ideology and the Finnish gender role movement in the late 1960s

2022

An active discussion of gender roles and the need to renegotiate them took place in the late 1960s in Finland. While previous studies have associated this ‘sex role debate’ with the independent civic organisation Association 9, this article focuses on the wider gender role movement. The article analyses the interplay and differences among the Finnish Women’s Democratic League, the Committee for Women’s Status, and Association 9’s grassroots activism between 1965 and 1970. It demonstrates that similar ideas about sex roles were presented simultaneously in two public spheres: the dominant public, where the ideas were promoted by Association 9, and the people’s democratic counterpublic, which …

1960-lukunaisetHistoryradikalismigender role movementnaishistoriajärjestötnaisen asemasukupuoliGender Studiestasa-arvofeminismi1960sradical sex role ideologypublic spheresukupuoliroolitradikaalifeminisminaisasiajärjestötnaisasialiikkeetFinlandWomen's History Review
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CCDC 2097024: Experimental Crystal Structure Determination

2021

Related Article: Anni I. Taponen, Awatef Ayadi, Manu K. Lahtinen, Itziar Oyarzabal, Sébastien Bonhommeau, Mathieu Rouzières, Corine Mathonière, Heikki M. Tuononen, Rodolphe Clérac, Aaron Mailman|2021|J.Am.Chem.Soc.|143|15912|doi:10.1021/jacs.1c07468

3-methylpyridinium-1235-dithiadiazolyl radical cation 77'88'-tetracyanoquinodimethane radical anion propanenitrile solvateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 2097023: Experimental Crystal Structure Determination

2021

Related Article: Anni I. Taponen, Awatef Ayadi, Manu K. Lahtinen, Itziar Oyarzabal, Sébastien Bonhommeau, Mathieu Rouzières, Corine Mathonière, Heikki M. Tuononen, Rodolphe Clérac, Aaron Mailman|2021|J.Am.Chem.Soc.|143|15912|doi:10.1021/jacs.1c07468

3-methylpyridinium-1235-dithiadiazolyl radical cation 77'88'-tetracyanoquinodimethane radical anionSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Nanoparticles of a polyaspartamide-based brush copolymer for modified release of sorafenib: In vitro and in vivo evaluation.

2017

Abstract In this paper, we describe the preparation of polymeric nanoparticles (NPs) loaded with sorafenib for the treatment of hepatocellular carcinoma (HCC). A synthetic brush copolymer, named PHEA-BIB-ButMA (PBB), was synthesized by Atom Trasnfer Radical Polymerization (ATRP) starting from the α-poly( N -2-hydroxyethyl)- d , l -aspartamide (PHEA) and poly butyl methacrylate (ButMA). Empty and sorafenib loaded PBB NPs were, then, produced by using a dialysis method and showed spherical morphology, colloidal size, negative ζ potential and the ability to allow a sustained sorafenib release in physiological environment. Sorafenib loaded PBB NPs were tested in vitro on HCC cells in order to e…

3003MaleHepatocellular carcinomamedicine.medical_treatmentPharmaceutical Science02 engineering and technologyATRPPharmacology01 natural sciencesDrug Delivery SystemsCopolymerChemistryATRP; Hepatocellular carcinoma; Sorafenib; Tumor targeting; α-Poly(N-2-hydroxyethyl)-DL-aspartamide; 3003Liver NeoplasmsSorafenib021001 nanoscience & nanotechnologyDrug delivery0210 nano-technologymedicine.drugSorafenibNiacinamideCarcinoma HepatocellularCell SurvivalRadical polymerizationIntraperitoneal injectionL-aspartamideMice NudeAntineoplastic AgentsEnhanced permeability and retention effect010402 general chemistryPolymethacrylic AcidsIn vivoCell Line TumormedicineAnimalsHumansneoplasmsProtein Kinase InhibitorsPhenylurea Compoundstechnology industry and agriculturedigestive system diseasesIn vitro0104 chemical sciencesDrug LiberationTumor targetingDelayed-Action PreparationsBiophysicsα-Poly(N-2-hydroxyethyl)-DNanoparticlesα-Poly(N-2-hydroxyethyl)-DL-aspartamidePeptidesJournal of controlled release : official journal of the Controlled Release Society
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The Two Dimensions of Narcissistic Personality and Support for the Radical Right: The Role of Right–Wing Authoritarianism, Social Dominance Orientati…

2020

This paper offers an explanation of the link between grandiose narcissism and support for radical right parties. Drawing on representative data of the GESIS Panel ( N = 2827), focusing on support for the German radical right populist party Alternative for Germany in 2016 and treating grandiose narcissism as a two–dimensional concept, it is shown that the effects of grandiose narcissism are indirect rather than direct. The paper also reveals that it is mainly narcissistic rivalry that accounts for radical right party support, whereas narcissistic admiration has a protecting relationship. Finally, our results indicate that the indirect effects of narcissistic rivalry on radical right party s…

3207 Social PsychologySocial psychology (sociology)Social Psychology300 Social sciences sociology & anthropologymedia_common.quotation_subject05 social sciencesImmigrationRight-wing authoritarianism050109 social psychology050105 experimental psychologyRadical rightPsychologieNarcissistic personalityNarcissismmedicine0501 psychology and cognitive sciencesmedicine.symptomPsychologySocial psychologySocial dominance orientation10095 Institute of Sociologymedia_commonEuropean Journal of Personality
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CCDC 1834563: Experimental Crystal Structure Determination

2018

Related Article: Serhii Krykun, Vincent Croué, Magali Allain, Zoia Voitenko, Juan Aragó, Enrique Ortí, Sébastien Goeb, Marc Sallé|2018|J.Mater.Chem.C|6|13190|doi:10.1039/C8TC04730H

48-bis[45-bis(methylsulfanyl)-2H-13-dithiol-2-ylidene]-48-dihydrobenzo[12-b:45-b']bisthiophene radical cation hexafluorophosphate tetrahydrofuran solvateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 2182459: Experimental Crystal Structure Determination

2022

Related Article: Anni I. Taponen, Awatef Ayadi, Noora Svahn, Manu K. Lahtinen, Mathieu Rouzières, Rodolphe Clérac, Heikki M. Tuononen, Aaron Mailman|2022|Cryst.Growth Des.|22|7110|doi:10.1021/acs.cgd.2c00795

4-(1-n-butylpyridinium-3-yl)-1235-dithiadiazolyl radical trifluoromethanesulfonateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 1863394: Experimental Crystal Structure Determination

2018

Related Article: Anni I. Taponen, Joanne W. L. Wong, Kristina Lekin, Abdeljalil Assoud, Craig M. Robertson, Manu Lahtinen, Rodolphe Clérac, Heikki M. Tuononen, Aaron Mailman, Richard T. Oakley|2018|Inorg.Chem.|57|13901|doi:10.1021/acs.inorgchem.8b02416

4-(3H-1235-diselenadiazol-4-yl)pyridine radicalSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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