Search results for "relationship"

showing 10 items of 3616 documents

Cytotoxic activity of some natural and synthetic guaianolides

2005

Several natural guaianolides and synthetic derivatives of repin (1) were tested and found to be active against tumor cell replication. Repin (1) and both mono- and di-halohydrin analogues (2, 7-9, 11, 12) showed significant antitumor potency. A more effective compound (17) was obtained by esterificating repin with the paclitaxel side chain.

PaclitaxelStereochemistryPharmaceutical ScienceEpoxideSesquiterpeneAnalytical Chemistrychemistry.chemical_compoundStructure-Activity RelationshipDrug DiscoveryTumor Cells CulturedPotencyHumansCytotoxicityPharmacologychemistry.chemical_classificationMolecular StructureChemistryOrganic ChemistrySettore CHIM/06 - Chimica OrganicaAntineoplastic Agents PhytogenicIn vitroTerpenoidCentaurea Asteraceae sesquiterpene lactonesComplementary and alternative medicinePaclitaxelMolecular MedicineDrug Screening Assays AntitumorSesquiterpenesLactone
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Capsaicin differentially modulates voltage-activated calcium channel currents in dorsal root ganglion neurones of rats

2005

It is discussed whether capsaicin, an agonist of the pain mediating TRPV1 receptor, decreases or increases voltage-activated calcium channel (VACC) currents (ICa(V)). ICa(V) were isolated in cultured dorsal root ganglion (DRG) neurones of rats using the whole cell patch clamp method and Ba 2+ as charge carrier. In large diameter neurones (>35Am), a concentration of 50AM was needed to reduce ICa(V) (activated by depolarizations to 0 mV) by 80%, while in small diameter neurones (30Am), the IC50 was 0.36 AM. This effect was concentration dependent with a threshold below 0.025 AM and maximal blockade (>80%) at 5AM. The current–voltage relation was shifted to the hyperpolarized direction with an…

Pain ThresholdPatch-Clamp TechniquesTRPV1TRPV Cation ChannelsN-type calcium channelSecond Messenger SystemsMembrane PotentialsGanglia SpinalAnimalsL-type calcium channelPatch clampRats WistarMolecular BiologyCell SizeNeuronsDose-Response Relationship DrugVoltage-dependent calcium channelChemistryGeneral NeuroscienceCalcium channelT-type calcium channelCalciseptineAnatomyRatsRats Inbred LewBiophysicsCalcium ChannelsNeurology (clinical)CapsaicinSignal TransductionDevelopmental BiologyBrain Research
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The beatles: tradition, avant-garde... and expressiveness

2019

Resumen: La música de The Beatles, tras su enorme éxito a través del tiempo, esconde diversos secretos que hunden sus raíces no solo en las tendencias coetáneas más evidentes -Pop Art, hippismo, cómic-, sino también en otras mucho más alejadas y sorprendentes que se refieren al manejo de las emociones, desde diversas herramientas armónicas procedentes de la música académica con la manifiesta influencia de las artes visuales, la pintura, la fotografía o la iconología sobre los álbumes del grupo. La continua búsqueda expresiva en The Beatles convirtió la música de la banda de Liverpool en una síntesis perfecta entre vanguardia y tradición a causa de la convergencia entre texto y sonido y, sob…

Paintingbusiness.industryMovement (music)TradiciónHippiemedia_common.quotation_subjectPhotographyArt historyPopular MusicGeneral MedicineArtComicsMúsica PopularIconologyArteConvergence (relationship)businessHumanitiesArtMusicMúsicaTraditionmedia_commonRevista humanidades
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Erratum for “Simple Relationships for the Optimal Design of Paired Drip Laterals on Uniform Slopes”

2017

In the original paper, errors in exponents of Eq. (11b) were detected. The corrected Eq. (11b) is reported.

Paired lateralSettore AGR/08 - Idraulica Agraria E Sistemazioni Idraulico-ForestaliOptimal length.MicroirrigationDesign relationship
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Intravenous morphine for management of cancer pain.

2010

Summary In recent years, a growing interest in palliative care and in routes of administration other than oral have prompted more aggressive measures to improve the efficacy of analgesic interventions in patients with difficult pain conditions. This review provides an overview of the use of intravenous morphine to control pain in patients with cancer. Intravenous morphine has been increasingly used in different clinical situations—including breakthrough pain, poor pain control with escalating doses of oral opioids, retitrating patients with acute pain, treating patients with long-standing poor pain control and unpredictable needs, and optimising opioid therapy to prevent incident pain assoc…

Palliative careDose-Response Relationship DrugMorphinebusiness.industryAnalgesicPsychological interventionCancerPainmedicine.diseasePain ladderAnalgesics OpioidOncologyOpioidAnesthesiaNeoplasmsChronic DiseaseInjections IntravenousMorphineMedicineHumansbusinessCancer painmedicine.drugPain MeasurementThe Lancet. Oncology
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THE IMPACT OF THE PANDEMIC ON QUALITY OF LIFE

2021

This paper aims to highlight how the situation related to the spread of Covid-19 infection has disrupted the lives of all citizens, changing their lifestyles. A year ago, the World Health Organisation declared the spread of the virus, which established the start of the pandemic. This situation has had major repercussions on people’s lives, affecting not only their mental and physical wellbeing but also brought about various effects of social isolation. Social distancing has forced people to change their habits and experiment with new ways of working, going to school and relating to each other. New technologies have proved very useful in this respect, as they have been able to make people fe…

Pandemic didactics technology relationship well-being
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Which factors influence orthodontists in their decision to extract? A questionnaire survey

2019

Background To evaluate the relative influence of different criteria in the choice between extraction and nonextraction treatment in current orthodontics, and to assess how the percentage of extractions has evolved over time. Material and methods Pre-treatment records (panoramic radiograph, lateral cephalogram, study casts and photographs) of fourteen cases in permanent dentition (adult or adolescent) with class I molar relationship and moderate anterior crowding were evaluated by 28 orthodontists. For each case, each orthodontist filled out a questionnaire reporting his treatment plan proposal (extraction or nonextraction) and the importance of specific parameters in his decision-making pro…

Panoramic radiographMolar relationshipAnterior crowdingOrthodontics02 engineering and technology03 medical and health sciences0302 clinical medicineTreatment planMedicineSurveyRadiation treatment planningGeneral DentistryExtractions; Orthodontics; Survey; Treatment planningOrthodonticsProfessional careerbusiness.industryResearchQuestionnaire030206 dentistry021001 nanoscience & nanotechnology:CIENCIAS MÉDICAS [UNESCO]CrowdingExtractionsUNESCO::CIENCIAS MÉDICAS0210 nano-technologybusinessTreatment planning
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Neuropharmacology of vision in goldfish: A review

2009

AbstractThe goldfish is one of the few animals exceptionally well analyzed in behavioral experiments and also in electrophysiological and neuroanatomical investigations of the retina. To get insight into the functional organization of the retina we studied color vision, motion detection and temporal resolution before and after intra-ocular injection of neuropharmaca with known effects on retinal neurons. Bicuculline, strychnine, curare, atropine, and dopamine D1- and D2-receptor antagonists were used. The results reviewed here indicate separate and parallel processing of L-cone contribution to different visual functions, and the influence of several neurotransmitters (dopamine, acetylcholin…

Parallel processing (psychology)genetic structuresColor visionDopamineMotion PerceptionGlycineColorRetinachemistry.chemical_compoundMotionGABADopamineGoldfishmedicineElectroretinographyParallel processingAnimalsNeurotransmitterNeuropharmacologyVision Oculargamma-Aminobutyric AcidRetinaNeurotransmitter AgentsColor VisionDose-Response Relationship DrugFlickerStrychnineBicucullineSensory Systemseye diseasesAcetylcholineOphthalmologymedicine.anatomical_structurechemistryTime Perceptionsense organsPsychologyNeurosciencemedicine.drugVision Research
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Growth in a time of external imbalances

2019

Abstract Globalization and financial integration have increased in the last three decades giving rise to cumulated large external imbalances. The question we address in this paper is whether economic growth can be affected by these external imbalances. We estimate an augmented growth equation with the external stock position of the countries measured by the net foreign asset position. Unlike previous literature, we use non-parametric methods that capture non-linearities and heterogeneity, and apply them to a sample that includes 106 developed and developing countries for the period 1983-2011. Contrary to the neoclassical theory, we find that improvements in the external position foster grow…

Parameter heterogeneityEconomics and Econometrics050208 finance05 social sciencesNet foreign assetsFinancial integrationDeveloping countryMonetary economicsLucas paradoxGlobalizationNegative relationship0502 economics and businessOpenness to experienceEconomicsNet foreign assets050207 economicsStock (geology)Economic growth
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Neuroglobin and cytoglobin overexpression protects human SH-SY5Y neuroblastoma cells against oxidative stress-induced cell death

2006

Although reactive oxygen species (ROS) at physiological concentrations are required for normal cell function, excessive production of ROS is detrimental to cells. Neuroglobin and cytoglobin are two globins, whose functions are still a matter of debate. A potential role in the detoxification of ROS is suggested. The influence of neuroglobin and cytoglobin on cell death after oxidative stress in human neuroblastoma SH-SY5Y cells was evaluated. Exposure of SH-SY5Y cells to paraquat or H(2)O(2) resulted in a concentration- and time-dependent induction of apoptotic and necrotic cell death. H(2)O(2) was 16 times more potent to induce cell death as compared to paraquat. SH-SY5Y cells transfected w…

ParaquatProgrammed cell deathTime FactorsBlotting WesternGene ExpressionNeuroglobinNerve Tissue ProteinsBiologymedicine.disease_causeNeuroblastomaCell Line TumormedicineHumansGlobinCell DeathDose-Response Relationship DrugHerbicidesGeneral NeuroscienceCytoglobinCytoglobinHydrogen PeroxideTransfectionFlow CytometryOxidantsMolecular biologyGlobinsOxidative StressApoptosisCell cultureNeuroglobinOxidative stressNeuroscience letters
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