Search results for "rito"

showing 10 items of 2948 documents

The CO-releasing molecule CORM-3 protects against articular degradation in the K/BxN serum transfer arthritis model.

2010

Contains fulltext : 89015.pdf (Publisher’s version ) (Closed access) Carbon monoxide-releasing molecules can counteract inflammatory responses. The aim of this study was to investigate whether tricarbonylchloro(glycinate)ruthenium (II) (CORM-3) is able to control the effector phase of experimental arthritis. Arthritis was induced in C57Black-6 mice by an intraperitoneal injection of serum from arthritic K/BxN mice. CORM-3 was administered intraperitoneally at 10 mg/kg/day (5 mg/kg twice a day) from days 0 to 10 and animals were sacrificed on day 11. Serum levels of osteocalcin and prostanoids were measured by enzyme-linked immunosorbent assay and radioimmunoassay. Gene expression was determ…

Cartilage ArticularMaleSerummedicine.medical_specialtymedicine.medical_treatmentIntraperitoneal injectionArthritisMice TransgenicHMGB1Auto-immunity transplantation and immunotherapy [N4i 4]RutheniumMicechemistry.chemical_compoundMice Inbred NODInternal medicineOrganometallic CompoundsmedicineAnimalsPharmacologyCarbon MonoxidebiologyChemistryProstaglandin D2 synthaseRadioimmunoassaymedicine.diseaseArthritis ExperimentalMice Inbred C57BLDisease Models AnimalEndocrinologyRANKLbiology.proteinOsteocalcinProstaglandin D2Infection and autoimmunity [NCMLS 1]European Journal of Pharmacology
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Architettura estone: case nuove e vecchi problemi

2005

Le riviste internazionali: Estonia. «Maja» e «Ehituskunst» sono le voci della giovane generazione di architetti

Casa Estonia RivisteSettore SPS/10 - Sociologia Dell'Ambiente E Del Territorio
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Bile acid-derived mono- and diketals—synthesis, structural characterization and self-assembling properties

2010

Three oxo-derivatives of bile acid methyl esters have been used as starting compounds in the preparation of novel bile acid monoketals with 1,2-benzenediol (catechol) and 2,3-naphthalenediol, as well as mono- and diketals with pentaerythritol. Monoketals of pentaerythritol showed a tendency to form thermoreversible gels in many aromatic solvents and the methyl lithocholate derivative proved to be a supergelator able to form a gel with t-butylbenzene at a concentration as low as 0.5% w/v. Whereas the naphthalenediol ketals formed film-type materials in the studied solvents, the catechol ketals underwent rapid crystallization into X-ray quality single crystals. Single crystal X-ray structures…

CatecholBile acidmedicine.drug_classOrganic ChemistryDiastereomerCrystal structureBiochemistryPentaerythritollaw.inventionchemistry.chemical_compoundchemistrylawSelf assemblingmedicineOrganic chemistryPhysical and Theoretical ChemistryCrystallizationSingle crystalOrganic & Biomolecular Chemistry
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Synthesis and antiproliferative activity of substituted 3[2-(1H-indol-3-yl)-1,3-thiazol-4-yl]-1H-pyrrolo[3,2-b]pyridines, marine alkaloid nortopsenti…

2014

A large number of indolyl-4-azaindolyl thiazoles, nortopsentin analogues, were conveniently synthesized. The antiproliferative activity of the new derivatives was examined against four human tumor cell lines with different histologic origin. Seven derivatives consistently reduced the growth of the experimental models independently of TP53 gene status and exhibited the highest activity against the malignant peritoneal mesothelioma (STO) cell line. The most active compound of this series acts as a CDK1 inhibitor, and was found to cause cell cycle arrest at G 2 /M phase, to induce apoptosis by preventing the phosphorylation of survivin in Thr 34 and to increase the cytotoxic activity of paclit…

Cell cycle checkpointCDK1 InhibitorsAntiproliferative Activity CDK1 Inhibitors Diffuse Malignant Peritoneal Mesothelioma Nortopsentin Analogues SurvivinPyridinesStereochemistrySurvivinDiffuse Malignant Peritoneal MesotheliomaAntineoplastic AgentsApoptosisAntiproliferative Activity; CDK1 Inhibitors; Diffuse Malignant Peritoneal Mesothelioma; Nortopsentin Analogues; SurvivinBiochemistryCell LineAntiproliferative ActivityStructure-Activity Relationshipchemistry.chemical_compoundDrug DiscoverySurvivinHumansCytotoxic T cellProtein Kinase InhibitorsCell ProliferationPharmacologyCyclin-dependent kinase 1AlkaloidOrganic ChemistrySettore CHIM/08 - Chimica FarmaceuticaPaclitaxelchemistryCell cultureApoptosisNortopsentin AnaloguesMolecular Medicine
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Sustainable viticulure in Brazil's context : a proposition

2015

The thesis involves the proposition of a framework for the sustainability of viticulture in Brazil using a territorial approach built from two exploratory studies in Brazilian wine regions of Campanha Gaúcha and Vale do São Francisco based on preliminary studies. Those studies involved technical visits in three countries (France, Italy and Spain) and frameworks’ observations in another five (South Africa, Australia, New Zealand, USA and Chile). The framework proposed is called BaccuS. It is structured on a matrix basis, with an axis corresponding to dimensions and other to guidelines, both in ascending order of complexity and development. There are eighteen topics that represent areas to ac…

CertificationVigne et vin[SHS.GEO] Humanities and Social Sciences/Geography[SDV.SA.STA] Life Sciences [q-bio]/Agricultural sciences/Sciences and technics of agricultureWineBrésil[SDE.BE] Environmental Sciences/Biodiversity and EcologySustainabilityCahier des chargesDéveloppement durableStandard développement durableTerritoireSustainable viticultureTerritoryVale do São FranciscoCampanha GaúchaViticulture durableBrazil
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HIPEC for gynaecological malignancies: A last update (Review)

2023

Advanced-stage gynaecological cancer represents a clinical entity with challenging surgical treatment in an effort to optimize prognosis. Hyperthermic intraperitoneal chemotherapy (HIPEC) following cytoreductive surgery (CRS) has been reported as a method potentially eligible to improve prognosis. However, no definitive conclusions have yet been made on which types of cancer and which context HIPEC may actually have a beneficial impact. The present review discusses the efficacy and safety of HIPEC as a treatment option for patients with primary/recurrent ovarian, endometrial and cervix cancer, as well as peritoneal sarcomatosis. A literature search was conducted using MeSH terms for each top…

Cervix cancerEndometrium cancerOvarian cancerGynaecological malignanciePeritoneal sarcomatosiCytoreductive surgeryHyperthermic Intraperitoneal ChemotherapyUpdate.Settore MED/40 - Ginecologia E Ostetricia
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Hydrologie, Changement Climatique, Adaptation, Ressource en Eau en Bourgogne : rapport final du projet HYCCARE Bourgogne

2016

HYCCARE Bourgogne est un projet de recherche-action dont l’objectif est de mettre à disposition des décideurs locaux des outils qui leur permettront de mieux prendre en compte le risque lié aux impacts du changement climatique sur la ressource en eau.

Changement climatiqueterritoireMots-clés : changement climatiquegouvernancecollectifsgestion de l’eauadaptationhydrologiebassin versant[SDU.STU.CL] Sciences of the Universe [physics]/Earth Sciences/Climatology[SDU.STU.CL]Sciences of the Universe [physics]/Earth Sciences/Climatologyressource en eauBourgognegestion de l'eauRessources en eaupolitiques « climat »modélisation
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Theory for polaritonic quantum tunneling

2022

I investigate the tunneling decay rate of a polaritonic system formed by a strong coupling between a vacuum cavity mode and $N$ metastable systems. Using a simple model potential, I find the instanton solutions controlling the low-temperature tunneling rate. The resulting rate modification due to the cavity is proportional to the mean of the second power of the light-matter coupling. No collective effect that would enhance the rates by a factor of $\sqrt{N}$ is present, which is in line with the results in the thermal activation regime.

Chemical Physics (physics.chem-ph)Quantum PhysicsPhysics - Chemical PhysicsFOS: Physical scienceskvanttimekaniikkaQuantum Physics (quant-ph)kvanttifysiikkapolaritonit
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Prediction of acute toxicity of organophosphorus pesticides using topological indices

2007

Topological indices were used in the prediction of the acute toxicity (intraperitoneal and oral LD(50)) of organophosphorus pesticides on rats. Models with six variables for the prediction of LD(50)-i.p. (r = 0.849, Q(2) = 0.613) and eight variables for LD(50)-oral (r = 0.906, Q(2) = 0.701) were selected. External group and cross-validation by use of leave-n-out tests were also performed in order to assess the stability and the prediction performance of the selected topological models.

ChemistryAdministration OralQuantitative Structure-Activity RelationshipBioengineeringGeneral MedicineTopologyAcute toxicityRatsLethal Dose 50Organophosphorus CompoundsDrug DiscoveryAnimalsRegression AnalysisMolecular MedicineComputer SimulationPesticidesOrganophosphorus pesticidesInjections IntraperitonealSAR and QSAR in Environmental Research
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Thy-1 (CD90) regulates the extravasation of leukocytes during inflammation.

2010

Human Thy-1 (CD90) has been shown to mediate adhesion of inflammatory cells to activated microvascular endothelial cells via interaction with Mac-1 (CD11b/CD18) in vitro. Since there are no data showing the physiological relevance of Thy-1 for the recruitment of inflammatory cells in vivo, different inflammation models were investigated in Thy-1-deficient mice and littermate controls. In thioglycollate-induced peritonitis, the number of neutrophils and monocytes was significantly diminished in Thy-1-deficient mice. During acute lung inflammation, the extravasation of eosinophils and monocytes into the lung was significantly reduced in Thy-1-deficient mice. Moreover, during chronic lung infl…

ChemokineMice 129 StrainNeutrophilsmedicine.medical_treatmentT-LymphocytesImmunologyInflammationCD18In Vitro TechniquesPeritonitisMonocytesMiceCell MovementCell AdhesionLeukocytesImmunology and AllergyMedicineAnimalsHumansCD90Thy-1InflammationMice KnockoutTransplantation Chimerabiologybusiness.industryInterleukinsEndothelial CellsPneumoniaExtravasationTransplantationEosinophilsMice Inbred C57BLCytokineIntegrin alpha MImmunologybiology.proteinThy-1 Antigensmedicine.symptomChemokinesbusinessextravasationPeptide HydrolasesEuropean journal of immunology
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