Search results for "stil"

showing 10 items of 1452 documents

Microleakage comparison of glass-ionomer and white mineral trioxide aggregate used as a coronal barrier in nonvital bleaching

2011

Objectives: There is some evidence that the pH at the root surface is reduced by intracoronal placement of bleaching pastes, which is known to enhance osteoclastic activity. Therefore, it is recommended that a protective barrier be used over the canal filling to prevent leakage of bleaching agents. Glass-ionomer (GI) is commonly used as a coronal barrier before nonvital bleaching. Because mineral trioxide aggregate (MTA) creates high alkalinity after mixing with water, using MTA as a protective barrier over the canal filling may not only prevent leakage of bleaching agents and microorganisms, but may prevent cervical resorption. The aim of this study was to evaluate sealing ability of white…

Mineral trioxide aggregategenetic structuresGlass ionomer cementDentistryIn Vitro Techniqueschemistry.chemical_compoundTooth BleachingHumansHydrogen peroxideAluminum CompoundsGeneral DentistryDental LeakageChemistrybusiness.industrySilicatesOxidesCalcium Compounds:CIENCIAS MÉDICAS [UNESCO]ResorptionCementoenamel junctionDrug CombinationsOtorhinolaryngologyDistilled waterGlass Ionomer CementsCoronal planeUNESCO::CIENCIAS MÉDICASSurgerysense organsSodium perboratebusiness
researchProduct

Radioprotective activity and cytogenetic effect of resveratrol in human lymphocytes: An in vitro evaluation

2012

Trans-resveratrol is a natural occurring polyphenol, obtained from grapes and other berries. This compound has shown antioxidant, anti-inflammatory, immunostimulant or anti-carcinogenic properties. Our aim was to evaluate the radioprotective efficacy, in vitro, of trans-resveratrol against radiation-induced chromosomal damage and to study the genotoxicity and cytotoxicity of this polyphenol in cell cultures without irradiation. The study was carried out by the pre-treatment of human lymphocytes at concentrations from 0 to 219μM of trans-resveratrol. The results showed that all concentrations tested reduced radiation-induced chromosomal damage compared with cells with any treatment. Maximum …

Mitotic indexProliferation indexmedicine.drug_classRadiation-Protective AgentsSister chromatid exchangePharmacologyBiologyResveratrolToxicologymedicine.disease_causeImmunostimulantchemistry.chemical_compoundStilbenesMitotic IndexmedicineHumansLymphocytesCytotoxicityCells CulturedCell ProliferationChromosome AberrationsGeneticsDose-Response Relationship DrugMutagenicity TestsCell growthfood and beveragesGeneral MedicinechemistryGamma RaysResveratrolSister Chromatid ExchangeGenotoxicityFood ScienceFood and Chemical Toxicology
researchProduct

Preventing root caries development under oral biofilm challenge in an artificial mouth

2013

Objectives: To study the preventive effects of chlorhexidine against root caries under oral biofilm in an artificial mouth. Study Design: Sixteen human tooth-root disks were inoculated with a salivary sample that was produced by mixing the unstimulated saliva of three adults who had no untreated caries. The disks were incubated in an artificial mouth fed with a 5% sucrose solution three times daily for one week. Eight disks received a twice daily rinse of 0.12% chlorhexidine (test group). The other eight disks were rinsed in distilled water (control). The biofilm was then studied with three techniques: colony forming unit (CFU) counting, scanning electron microscopy (SEM) and confocal laser…

Models AnatomicSalivaOdontologíaBacterial growthMicrobiologymedicineHumansGeneral DentistryRoot cariesColony-forming unitMouthOral Medicine and PathologyChemistryChlorhexidineChlorhexidineBiofilm:CIENCIAS MÉDICAS [UNESCO]Ciencias de la saludDemineralizationOtorhinolaryngologyDistilled waterRoot CariesBiofilmsUNESCO::CIENCIAS MÉDICASAnti-Infective Agents LocalSurgeryResearch-Articlemedicine.drug
researchProduct

Heterocyclic and Phenyl Double-Bond-Locked Combretastatin Analogues Possessing Potent Apoptosis-inducing activity in HL60 and in MDR Cell lines

2005

Two new series of combretastatin (CA-4) analogues have been prepared. The alkenyl motif of CA-4 was replaced either by a five-membered heterocyclic (isoxazoline or isoxazole) or by a six-membered ring (pyridine or benzene). The new compounds have been evaluated for their effects on tubulin assembly and for cytotoxic and apoptotic activities. Five compounds (18b, 20a, 21a, 34b, and 35b) demonstrated an attractive profile of cytotoxicity (IC501 microM) and apoptosis-inducing activity but poor antitubulin activity. The isoxazoline derivatives 18b, 20a, and 21a, demonstrated potent apoptotic activity different from that of natural CA-4. Their ability to block most cells in the G2 phase suggests…

Models MolecularA-4 ANALOGSDouble bondHL60StereochemistryPyridinesTUBULINApoptosisANTINEOPLASTIC AGENTSchemistry.chemical_compoundStructure-Activity RelationshipCell Line TumorDrug DiscoveryStilbenesBenzene DerivativesHumansIsoxazoleBIOLOGICAL EVALUATIONCytotoxicitychemistry.chemical_classificationCombretastatinbiologyCOLCHICINEDEATHIsoxazolesDrug Resistance MultipleTubulinANTIMITOTIC ANTITUMOR AGENTSMULTIDRUGchemistryApoptosisCell cultureDrug Resistance NeoplasmDISCOVERYbiology.proteinMolecular MedicineDrug Screening Assays AntitumorSOLID TUMOR-THERAPY
researchProduct

Revised structure of trans-resveratrol: Implications for its proposed antioxidant mechanism

2015

The crystal structure of trans-resveratrol has been redetermined by X-ray diffraction. The newly refined structure demonstrates that the previously reported, dynamically disordered hydrogen-bonding network is rather the superposition of two crystallographically independent molecules of trans-resveratrol. This latter arrangement possesses a well-defined hydrogen-bonding network in a unit cell of double the previously reported volume. While not meant as a criticism of the proposed antioxidant mechanism itself, the present studies clearly show that the X-ray diffraction data should no longer be used for its additional support.

Models MolecularDiffractionStereochemistryClinical BiochemistryStructure (category theory)Pharmaceutical ScienceCrystal structureCrystallography X-Ray010402 general chemistry01 natural sciencesBiochemistryAntioxidantsStructure-Activity RelationshipStilbenesDrug DiscoveryMoleculeMolecular BiologyMolecular StructureTrans-resveratrol010405 organic chemistryHydrogen bondChemistryOrganic ChemistryHydrogen Bondingdisorder0104 chemical sciencesCrystallographyResveratrolMechanism (philosophy)Molecular MedicineX-ray structuresuperstructureSuperstructure (condensed matter)Bioorganic & Medicinal Chemistry Letters
researchProduct

Structural determinants of resveratrol for cell proliferation inhibition potency: experimental and docking studies of new analogs.

2010

International audience; Resveratrol is the subject of intense research because of the abundance of this compound in the human diet and as one of the most valuable natural chemopreventive agents. Further advances require new resveratrol analogs be used to identify the structural determinants of resveratrol for the inhibition potency of cell proliferation by comparing experimental and docking studies. Therefore, we synthesized new trans/(E)- and cis/(Z)-resveratrol - analogs not reported to date - by modifying the hydroxylation pattern of resveratrol and a double bond geometry. We included them in a larger panel of 14 molecules, including (Z)-3,5,4'-trimethoxystilbene, the most powerful molec…

Models MolecularMESH : HydroxidesMESH : DNAMESH: Cell CycleMESH: TubulinResveratrolHydroxylationchemistry.chemical_compound0302 clinical medicineTubulinMESH: StilbenesDrug DiscoveryStilbenesHydroxidesMESH : Cell ProliferationDocking studiesMESH : Colchicine0303 health sciencesCell CycleMESH: DNAStereoisomerismGeneral MedicineMESH : TubulinMESH: Hydroxides3. Good healthColon cancerBiochemistryMESH : Stereoisomerism030220 oncology & carcinogenesisMESH: Models MolecularMESH: Cell Line TumorStereochemistryMESH : Models MolecularStereoisomerismMESH : Stilbenes03 medical and health sciencesCell Line TumorMESH: Cell ProliferationMESH : Cell Cycle[SDV.BBM] Life Sciences [q-bio]/Biochemistry Molecular BiologyHumans[SDV.BBM]Life Sciences [q-bio]/Biochemistry Molecular BiologyBinding site[ SDV.BBM ] Life Sciences [q-bio]/Biochemistry Molecular BiologyTubulin polymerization030304 developmental biologyCell ProliferationPharmacologyCombretastatinBinding SitesMESH: HumansCell growthMESH : Cell Line TumorOrganic ChemistryMESH : HumansDNAMESH: StereoisomerismMESH: ColchicinechemistryPolymethoxy-stilbenesMESH: Binding SitesDocking (molecular)Cell cultureResveratrolResveratrol; Polymethoxy-stilbenes; Tubulin polymerization; Colon cancer; Docking studiesColchicineMESH : Binding Sites
researchProduct

Topology and accessibility of the transmembrane helices and the sensory site in the bifunctional transporter DcuB of Escherichia coli.

2011

C(4)-Dicarboxylate uptake transporter B (DcuB) of Escherichia coli is a bifunctional transporter that catalyzes fumarate/succinate antiport and serves as a cosensor of the sensor kinase DcuS. Sites and domains of DcuB were analyzed for their topology relative to the cytoplasmic or periplasmic side of the membrane and their accessibility to the water space. For the topology studies, DcuB was fused at 33 sites to the reporter enzymes PhoA and LacZ that are only active when located in the periplasm or the cytoplasm, respectively. The ratios of the PhoA and LacZ activities suggested the presence of 10 or 11 hydrophilic loops, and 11 or 12 α-helical transmembrane domains (TMDs). The central part…

Models MolecularRecombinant Fusion ProteinsMolecular Sequence Datalac operonTopologyBiochemistryProtein Structure SecondaryPolyethylene GlycolsProtein structureBacterial ProteinsCatalytic DomainStilbenesAmino Acid SequenceCysteineBinding sitePeptide sequenceDicarboxylic Acid TransportersEscherichia coli K12ChemistryEscherichia coli ProteinsCell MembranePeriplasmic spaceAlkaline PhosphataseTransmembrane domainMembrane proteinBiochemistryLac OperonEthylmaleimideSulfonic AcidsHydrophobic and Hydrophilic InteractionsCysteineBiochemistry
researchProduct

An in vitro evaluation of the efficacy of a novel iontophoresis fluoride tray on remineralization

2013

Objectives: The aim of this study is to determine the effects on remineralization of a novel iontophoresis device called "Fluorinex", conventional (acidulated phosphat fluoride) APF gel treatment, and conventional ionthophoresis device comparatively by laser fluorescence measurements. Study Design: Artificial incipient carious lesions were created on immature, 60 intact premolar and molar teeth with no defects. The specimens were randomly allocated to four groups. In the first group 1.23% APF gel was applied to specimens by conventional method for 4 minutes and in the second group 2% (sodium fluoride) NaF solution applied by conventional iontophoresis device for 4 minutes. In Fluorinex grou…

MolarRemineralisationChromatographyIontophoresisbusiness.industryResearchDentistryLaser fluorescenceOdontología:CIENCIAS MÉDICAS [UNESCO]Ciencias de la saludCommunity and Preventive Dentistrychemistry.chemical_compoundmedicine.anatomical_structurechemistryDistilled waterSodium fluorideUNESCO::CIENCIAS MÉDICASPremolarMedicinebusinessGeneral DentistryFluoride
researchProduct

Bond strength and elemental analysis of oxidized dentin bonded to resin modified glass ionomer based restorative material

2019

Background This study aimed to investigate the influence of hesperidin application on the bonding of resin-modified glass ionomer-based restorative material to dentin treated with oxygen-induced endodontic irrigants. Material and Methods One hundred human permanent molars were categorized into five groups (n= 20/group), treated with various irrigants as follows: Group C; distilled water (control group), Group SH; 5.25% NaOCl, Group SH+H; 5.25% NaOCl + 5 % hesperidin, Group HP; 10% H2O2, Group HP+H; 10% H2O2 + 5 % hesperidin. Specimens were bonded with RMGI based restorative material. For each group, half of the specimens were evaluated for µSBS by a universal testing machine and the other h…

MolarUniversal testing machineChemistryBond strengthResearch0206 medical engineeringGlass ionomer cement030206 dentistry02 engineering and technology:CIENCIAS MÉDICAS [UNESCO]020601 biomedical engineeringOperative Dentistry and Endodontics03 medical and health sciencesHesperidinchemistry.chemical_compound0302 clinical medicinemedicine.anatomical_structureDistilled waterstomatognathic systemElemental analysisUNESCO::CIENCIAS MÉDICASDentinmedicineGeneral DentistryNuclear chemistry
researchProduct

The effect of bacterial cellulose nanocrystals on the shear bond strength of resin modified glass ionomer cement to dentin

2020

Background The present study aimed to investigate the effect of bacterial cellulose nanocrystals (BCNC) on the shear bond strength (SBS) of resin modified glass ionomer cement (RMGIC) to dentin. Material and Methods A total of 48 freshly extracted intact third molars were randomly divided into four main groups with three different concentrations (0.3%, 0.5% and 1% wt) of BCNC with RMGIC and control group without BCNC. These specimens were kept in distilled water at 37° C for 24h. Shear bond strength was examined, using the universal testing machine. Kruskal-Wallis test and Dunn`s post-hoc test were applied for analysis of data. P<0.05 was considered as the level of significance. Results The…

MolarUniversal testing machineMaterials scienceResearchGlass ionomer cementShear bondchemistry.chemical_compoundmedicine.anatomical_structureDistilled waterNanocrystalchemistryBacterial celluloseBiomaterials and Bioengineering in DentistryDentinmedicineComposite materialGeneral DentistryUNESCO:CIENCIAS MÉDICAS
researchProduct