Search results for "tmax"

showing 9 items of 9 documents

Polyoxypregnanes as safe, potent, and specific ABCB1-inhibitory pro-drugs to overcome multidrug resistance in cancer chemotherapy in vitro and in vivo

2021

Multidrug resistance (MDR) mediated by ATP binding cassette subfamily B member 1 (ABCB1) is significantly hindering effective cancer chemotherapy. However, currently, no ABCB1-inhibitory drugs have been approved to treat MDR cancer clinically, mainly due to the inhibitor specificity, toxicity, and drug interactions. Here, we reported that three polyoxypregnanes (POPs) as the most abundant constituents of Marsdenia tenacissima (M. tenacissima) were novel ABCB1-modulatory pro-drugs, which underwent intestinal microbiota-mediated biotransformation in vivo to generate active metabolites. The metabolites at non-toxic concentrations restored chemosensitivity in ABCB1-overexpressing cancer cells v…

ABCC1 ATP binding cassette subfamily C member 1IC50 half maximal inhibitory concentrationMultidrug resistancePharmacologyNADPH reduced nicotinamide adenine dinucleotide phosphateF bioavailabilitychemistry.chemical_compoundPCR polymerase chain reaction0302 clinical medicineMDR multidrug resistanceECL electrochemiluminescencet1/2 elimination half-lifeLC–MS liquid chromatography coupled with mass spectrometryN.D. not detectedGeneral Pharmacology Toxicology and PharmaceuticsBBB blood–brain barriermedia_commonATF3 activating transcription factor 30303 health sciencesChemistryABC ATP-binding cassetteNMPA National Medical Products AdministrationPXR pregnane X receptorSDS-PAGE sodium dodecyl sulfate-polyacrylamide gel electrophoresisHBSS Hankʹs balanced salt solutionABCB1Combination chemotherapyProdrugMarsdenia tenacissimaCmax peak concentrationPaclitaxelGAPDH glyceraldehyde-3-phosphate dehydrogenase030220 oncology & carcinogenesisBHI brain heart infusionOriginal ArticleAUC0–∞ area under plasma concentration vs. time curveMRT mean residence timeDrugmedia_common.quotation_subjectRM1-950Vd volume of distributionABCB1 ATP binding cassette subfamily B member 1UIC-2 mouse monoclonal ABCB1 antibodyABCG2 ATP binding cassette subfamily G member 2Combination chemotherapyCYP cytochrome P450 isozymePI propidium iodideTEER transepithelial electrical resistance03 medical and health sciencesPBS phosphate buffer salineFBS fetal bovine serumDox doxorubicinIn vivoPOP polyoxypregnanemedicine030304 developmental biologyEVOM epithelial tissue voltohmmeterTmax time for peak concentrationCancerLBE lowest binding energyPE phycoerythrinmedicine.diseaseMultiple drug resistancePolyoxypregnanePapp apparent permeabilityN.A. not applicableCancer cellH&E hematoxylin and eosinMDR1a multidrug resistance protein 1aTherapeutics. PharmacologyqPCR quantitative PCRM. tenacissima Marsdenia tenacissimaCL clearanceSD standard derivationActa Pharmaceutica Sinica B
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Multi-layer intrusion detection system with ExtraTrees feature selection, extreme learning machine ensemble, and softmax aggregation

2019

Abstract Recent advances in intrusion detection systems based on machine learning have indeed outperformed other techniques, but struggle with detecting multiple classes of attacks with high accuracy. We propose a method that works in three stages. First, the ExtraTrees classifier is used to select relevant features for each type of attack individually for each (ELM). Then, an ensemble of ELMs is used to detect each type of attack separately. Finally, the results of all ELMs are combined using a softmax layer to refine the results and increase the accuracy further. The intuition behind our system is that multi-class classification is quite difficult compared to binary classification. So, we…

Artificial intelligencelcsh:Computer engineering. Computer hardwareExtreme learning machineEnsemble methodsComputer scienceBinary numberlcsh:TK7885-7895Feature selection02 engineering and technologyIntrusion detection systemlcsh:QA75.5-76.95Machine learning0202 electrical engineering electronic engineering information engineeringVDP::Teknologi: 500::Informasjons- og kommunikasjonsteknologi: 550Multi layerExtreme learning machinebusiness.industryIntrusion detection system020206 networking & telecommunicationsPattern recognitionComputer Science ApplicationsBinary classificationFeature selectionSignal ProcessingSoftmax function020201 artificial intelligence & image processinglcsh:Electronic computers. Computer scienceArtificial intelligencebusinessClassifier (UML)EURASIP Journal on Information Security
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Deep CNN-ELM Hybrid Models for Fire Detection in Images

2018

In this paper, we propose a hybrid model consisting of a Deep Convolutional feature extractor followed by a fast and accurate classifier, the Extreme Learning Machine, for the purpose of fire detection in images. The reason behind using such a model is that Deep CNNs used for image classification take a very long time to train. Even with pre-trained models, the fully connected layers need to be trained with backpropagation, which can be very slow. In contrast, we propose to employ the Extreme Learning Machine (ELM) as the final classifier trained on pre-trained Deep CNN feature extractor. We apply this hybrid model on the problem of fire detection in images. We use state of the art Deep CNN…

Contextual image classificationArtificial neural networkComputer sciencebusiness.industryPattern recognition02 engineering and technologyConvolutional neural networkBackpropagationSupport vector machine03 medical and health sciences0302 clinical medicineSoftmax function0202 electrical engineering electronic engineering information engineering020201 artificial intelligence & image processingArtificial intelligencebusinessClassifier (UML)030217 neurology & neurosurgeryExtreme learning machine
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Fast Neural Machine Translation Implementation

2018

This paper describes the submissions to the efficiency track for GPUs at the Workshop for Neural Machine Translation and Generation by members of the University of Edinburgh, Adam Mickiewicz University, Tilde and University of Alicante. We focus on efficient implementation of the recurrent deep-learning model as implemented in Amun, the fast inference engine for neural machine translation. We improve the performance with an efficient mini-batching algorithm, and by fusing the softmax operation with the k-best extraction algorithm. Submissions using Amun were first, second and third fastest in the GPU efficiency track.

FOS: Computer and information sciencesFocus (computing)Computer Science - Computation and LanguageMachine translationComputer sciencebusiness.industrycomputer.software_genreTrack (rail transport)Softmax functionArtificial intelligenceInference enginebusinesscomputerComputation and Language (cs.CL)
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2021

This paper proposes a new method for blind mesh visual quality assessment (MVQA) based on a graph convolutional network. For that, we address the node classification problem to predict the perceived visual quality. First, two matrices representing the 3D mesh are considered: a graph adjacency matrix and a feature matrix. Both matrices are used as input to a shallow graph convolutional network. The network consists of two convolutional layers followed by a max-pooling layer to provide the final feature representation. With this structure, the Softmax classifier predicts the quality score category without the reference mesh’s availability. Experiments are conducted on four publicly available …

General Computer Sciencebusiness.industryComputer scienceNode (networking)Feature extractionGeneral EngineeringPattern recognitionFeature (computer vision)Softmax functionGraph (abstract data type)General Materials SciencePolygon meshArtificial intelligenceAdjacency matrixbusinessRepresentation (mathematics)IEEE Access
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Multimodal biometric recognition systems using deep learning based on the finger vein and finger knuckle print fusion

2020

Recognition systems using multimodal biometrics attracts attention because they improve recognition efficiency and high-security level compared to the unimodal biometrics system. In this study, the authors present a secure multimodal biometrics recognition system based on the deep learning method that uses convolutional neural networks (CNNs). The authors propose two multimodal architectures using the finger knuckle print (FKP) and the finger vein (FV) biometrics with different levels of fusion: the features level fusion and scores level fusion. The features extraction for FKP and FV are performed using transfer learning CNN architectures: AlexNet, VGG16, and ResNet50. The key step aims to …

Image fusionBiometricsbusiness.industryComputer scienceDeep learningFeature extractionComputingMethodologies_IMAGEPROCESSINGANDCOMPUTERVISIONWord error rate020206 networking & telecommunicationsPattern recognition02 engineering and technologyConvolutional neural networkSupport vector machineSignal ProcessingSoftmax function0202 electrical engineering electronic engineering information engineering020201 artificial intelligence & image processingComputer Vision and Pattern RecognitionArtificial intelligenceElectrical and Electronic EngineeringbusinessSoftwareIET Image Processing
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In vitro evaluation of poloxamer in situ forming gels for bedaquiline fumarate salt and pharmacokinetics following intramuscular injection in rats

2019

Graphical abstract

In situPO Propylene oxideIV IntravenousP338 Poloxamer 338lcsh:RS1-441Pharmaceutical Sciencechemistry.chemical_compoundn Sample sizeSD Standard deviationIM Intramuscularchemistry.chemical_classificationC0 Analyte plasma concentration at time zeroDoE Design of experimentsUV UltravioletPharmacology. TherapyK2.EDTA Potassium ethylenediaminetetraacetic acidLC–MS/MS Liquid chromatography-tandem mass spectrometryH&E Hematoxylin and eosintmax Sampling time to reach the maximum observed analyte plasma concentrationIn situ forming gelsCMC Critical micellar concentrationCmax Maximum observed analyte plasma concentrationIntramuscular injectionDN Dose normalizedGPT Gel point temperaturePLGA Poly-(DL-lactic-co-glycolic acid)TFA Trifluoroacetic acidCAN AcetonitrileATP Adenosine 5′ triphosphateSalt (chemistry)Polyethylene glycolPoloxamerArticlelcsh:Pharmacy and materia medicaPharmacokineticsIn vivoUHPLC Ultra-high performance liquid chromatographyPharmacokineticsAUClast Area under the analyte concentration versus time curve from time zero to the time of the last measurable (non-below quantification level) concentrationEO Ethylene oxideNMP N-methyl-2-pyrrolidoneComputingMethodologies_COMPUTERGRAPHICSAUC∞ Area under the analyte concentration vs time curve from time zero to infinite timeP407 Poloxamer 407In vitro releasePoloxamerCMT Critical micellar temperatureGel erosionIn vitrot1/2 Apparent terminal elimination half-lifechemistryMDR-TB Multi-drug resistant tuberculosisAUC80h Area under the analyte concentration versus time curve from time zero to 80 htlast Sampling time until the last measurable (non-below quantification level) analyte plasma concentrationMRM Multiple reaction monitoringNuclear chemistrySustained releaseInternational Journal of Pharmaceutics: X
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A Comparative Analysis of Multiple Biasing Techniques for $Q_{biased}$ Softmax Regression Algorithm

2021

Over the past many years the popularity of robotic workers has seen a tremendous surge. Several tasks which were previously considered insurmountable are able to be performed by robots efficiently, with much ease. This is mainly due to the advances made in the field of control systems and artificial intelligence in recent years. Lately, we have seen Reinforcement Learning (RL) capture the spotlight, in the field of robotics. Instead of explicitly specifying the solution of a particular task, RL enables the robot (agent) to explore its environment and through trial and error choose the appropriate response. In this paper, a comparative analysis of biasing techniques for the Q-biased softmax …

business.industryComputer scienceObstacle avoidanceSoftmax functionQ-learningRobotReinforcement learningMobile robotArtificial intelligencebusinessTrial and errorAction selection2021 International Conference on Artificial Intelligence and Mechatronics Systems (AIMS)
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Maksimaalisen rasvan hapettumispisteen (Fatmax-pisteen) päivittäinen vaihtelu ja sen määrittäminen sykevälivaihtelun avulla

2007

sykefatmax-pisterasvahapettuminenvaihtelu
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