Search results for "tuli"

showing 10 items of 223 documents

Cytotoxicity of Artesunic Acid Homo- and Heterodimer Molecules toward Sensitive and Multidrug-Resistant CCRF-CEM Leukemia Cells

2010

A novel approach to circumvent multidrug resistance is hybridization of natural products in dimers. We analyzed homodimers of two artesunic acid molecules and heterohybrids of artesunic acid and betulin in human CCRF-CEM and multidrug-resistant P-glycoprotein-overexpressing CEM/ADR5000 leukemia cells. Multidrug-resistant cells were not cross-resistant to the novel compounds. Collateral sensitivity was observed for artesunic acid homodimer. Artesunic acid and artesunic acid homodimer induced G0/G1 cell cycle arrest, apoptosis, and formation of reactive oxygen species.

Spectrometry Mass Electrospray IonizationMagnetic Resonance SpectroscopyCell SurvivalApoptosischemistry.chemical_compoundCell Line TumorDrug DiscoverymedicineHumansCytotoxicitychemistry.chemical_classificationReactive oxygen speciesFormazansLeukemiaBetulinCell CycleSuccinatesCell cycleFlow Cytometrymedicine.diseaseArtemisininsTriterpenesMultiple drug resistanceLeukemiachemistryBiochemistryDrug Resistance NeoplasmCell cultureApoptosisMolecular MedicineReactive Oxygen SpeciesJournal of Medicinal Chemistry
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INTRA- AND INTERSPECIFIC VARIATION IN INTERNAL STRUCTURES OF THE GENUSSTENOSARINA(BRACHIOPODA, TEREBRATULIDA) USING LANDMARKS

2001

Abstract Although a number of brachiopod genera have been defined mainly from their internal structures, the fixity of those structures has rarely been investigated. Variability of the rather simple loops of two New Caledonian species of the Recent genus Stenosarina (Terebratulida), one species having a variant with endemic morphology, provides insight into the relationship between the two species. Procrustes methods based on landmarks are used. Intra-population variability is found to be of the same order of magnitude as inter-population variability. Moreover, the morphological distance between the endemic variant and the other specimens is greater than the distance between the two species…

StenosarinaPaleontologyVariation (linguistics)GenusPaleontologyZoologyMorphology (biology)Interspecific competitionBiologybiology.organism_classificationTerebratulidaJournal of Paleontology
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Activity of lupane triterpenoids from Maytenus species as inhibitors of nitric oxide and prostaglandin E2

2005

In the present study, we report that three new lupane triterpenes (1-3), in addition to 16 known ones (4-19), were isolated from the root bark of Maytenus cuzcoina and the leaves of Maytenus chiapensis. Their structures were elucidated by spectral analysis, including homonuclear and heteronuclear correlation NMR experiments (COSY, ROESY, HSQC, and HMBC). The natural compounds and derivatives 6a, 6b, 9a, and 9b have been tested for potential anti-inflammatory activity, and several compounds including 3-epicalenduladiol (2), 11alpha-hydroxy-glochidone (3), rigidenol (6), acetoxy-rigidenol (6a), 11alpha-acetoxy-30-chloro-3-oxo-lup-20(29)-ene (6b), betulin (9), 28-acetoxy-betulin (9a), epibetul…

StereochemistryClinical BiochemistryPharmaceutical SciencePharmacognosyNitric OxideBiochemistryDinoprostoneTerpeneCelastraceaeMiceStructure-Activity Relationshipchemistry.chemical_compoundTriterpeneDrug DiscoveryAnimalsMolecular Biologychemistry.chemical_classificationBetulinbiologyMaytenusMacrophagesSpectrum AnalysisOrganic ChemistryBiological activityBacterial InfectionsMaytenusbiology.organism_classificationAntineoplastic Agents PhytogenicTriterpenesTerpenoidEndotoxinsPlant LeaveschemistryMolecular MedicineBioorganic & Medicinal Chemistry
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Jekaterinai Ripai veltīto apsveikumu kolekcija

2018

Raksts par vēsturnieci, bijušo Latvijas Valsts Universitātes Vēstures un filoloģijas fakultātes dekāni (1961-1963) un Studentu zinātniskās biedrības sekcijas zinātnisko vadītāju docenti Jekaterinu Ripu (1902-1993) un viņai veltīto vēstuļu un apsveikumu kolekciju, kas glabājas Latvijas Universitātes Muzeja Vēstures kolekcijā.

Studentu zinātniskā biedrībaStudent scientific societygreetings:HUMANITIES and RELIGION::History and philosophy subjects::History subjects::History [Research Subject Categories]Faculty of History and PhilologyVēstures un filoloģijas fakultāteapsveikumiJekaterina RipaIlgvars Butulis
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Pluralismo político y rol del moderador en tertulias televisivas: Al Rojo Vivo y Las Mañanas de Cuatro

2019

Las tertulias televisivas poseen gran relevancia en el nuevo ciclo político abierto en España en 2014. Con vistas a analizar el grado de pluralismo político y el rol del moderador que se despliega en ellas, se ha tomado una muestra de 50 programas (25 de “Al Rojo Vivo” y 25 de “Las Mañanas de Cuatro”). La perspectiva es cualitativa respecto al alcance del marco permitido y cuantitativa en cuanto al tratamiento que reciben los partidos políticos. Las variables registradas están relacionadas con quién, cuánto y cómo interviene en el programa. Se ha obtenido el número de intervenciones que realiza un partido por cada contraargumento que recibe de los periodistas. Del análisis se extraen conclu…

Tertulias políticasDebateTelevisiónPeriodismoComunicaciónPluralismo:3 - Ciencias sociales:316 - Comunicación [CDU]:0 - Generalidades.::070 - Periódicos. Prensa. Periodismo. Ciencias de la información [CDU]MIGUEL HERNÁNDEZ COMMUNICATION JOURNAL
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La mascota del magistrado

2010

Es bien conocida la importancia de las tertulias en el siglo XVIII. Sin llegar a la trascendencia de las francesas, también las hubo en España, especialmente en el reinado de Carlos III. Pero en el caso analizado, la tertulia semanal en casa del abogado José Bermúdez tiene un carácter político (presencia de embajadores), cultural (origen de la primera biografía de Cervantes) y de entretenimiento. El presente artículo centra su atención en este último aspecto. (A)

TertuliasMagistradosUNESCO::HISTORIA::Historia por épocas::Historia antiguaNovatoresSociabilidad:HISTORIA::Historia por épocas::Historia antigua [UNESCO]
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Cytotoxic phytochemicals from the crude extract of Tetrapleura tetraptera fruits towards multi-factorial drug resistant cancer cells.

2020

Abstract Ethnopharmacological relevance Tetrapleura tetraptera is an African medicinal spice used in traditional medicine to treat several ailments including cancer. Aim of the study The present study was designed to evaluate the cytotoxicity of the dichloromethane-methanol (1:1) extract of the fruits of Tetrapleura tetraptera (TTF) and its constituents: (3R, 4S)-3,4-dimethyloxetan-2-one (1), luteolin (2), stigmasterol (4), 3-O-[6′-O-undecanoyl-β-D-glucopyranosyl]stigmasterol (6), olean-12-en-3-β-O-D-glucopyranoside (7), 3-O-β-D-glucopyranosyl-(1 → 6)-β-D-glucopyranosylurs-12-en-28-oic acid (8), 3-O-β-D-glucopyranosyl-(1 → 3)-β-D-glucopyranosyl-27-hydroxyolean-12-ene-28-oic acid (9), methyl…

Tetrapleura tetrapteraPhytochemicalsApoptosis03 medical and health scienceschemistry.chemical_compoundInhibitory Concentration 500302 clinical medicineBetulinic acidNeoplasmsDrug DiscoveryCytotoxic T cellHumansTetrapleuraCytotoxicity030304 developmental biologyPharmacologychemistry.chemical_classificationMembrane Potential Mitochondrial0303 health sciencesReactive oxygen speciesbiologyDose-Response Relationship DrugPlant ExtractsHep G2 Cellsbiology.organism_classificationHCT116 CellsMolecular biologyAntineoplastic Agents PhytogenicDrug Resistance MultipleMatrix MetalloproteinasesOxidative StresschemistryApoptosisDrug Resistance Neoplasm030220 oncology & carcinogenesisCaspasesFruitCancer cellReactive Oxygen SpeciesLuteolinSignal TransductionJournal of ethnopharmacology
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Botulinum toxin injections into the detrusor

2011

Text miningbusiness.industryUrologyMedicinePharmacologybusinessBotulinum toxinmedicine.drugBJU International
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Does low concentration mycotoxin exposure induce toxicity in HepG2 cells through oxidative stress?

2020

The purpose of this study was to determine whether exposure to low concentrations of deoxynivalenol (DON), T-2 toxin (T-2) and patulin (PAT) in a human hepatocellular carcinoma cell line (HepG2) exerts toxic effects through mechanisms related to oxidative stress, and how cells deal with such exposure. Cell viability was determined by the MTT and protein content (PC) assays over 24, 48 and 72 h. The IC

Time FactorsCell SurvivalHealth Toxicology and MutagenesisMitochondria LiverHepatic carcinoma010501 environmental sciencesToxicologymedicine.disease_cause01 natural sciencesPatulinInhibitory Concentration 5003 medical and health scienceschemistry.chemical_compoundmedicineHumansMycotoxinVolume concentration0105 earth and related environmental sciencesMembrane Potential Mitochondrial0303 health sciencesDose-Response Relationship DrugToxinChemistry030302 biochemistry & molecular biologyfood and beveragesHep G2 CellsMycotoxinsMolecular biologydigestive system diseasesOxidative StressT-2 ToxinPatulinHepg2 cellsToxicityHepatocytesLipid PeroxidationReactive Oxygen SpeciesTrichothecenesOxidative stressToxicology Mechanisms and Methods
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Modeling the effect of ethanol vapor on the germination time of Penicillium chrysogenum.

2005

The influence of ethanol vapor on germination of Penicillium chrysogenum was determined on yeast nitrogen base plus glucose agar medium at 25 degrees C. Ethanol vapors were generated by 0 to 6% (wt/wt) ethanol solutions at the bottom of hermetically closed petri dishes. The logistic equation was used to describe the data as the percentage of germination versus time and to estimate the germination time. The effect of ethanol concentration on germination time was described by a new reparameterized equation, resulting in an estimated limiting ethanol concentration of 4.3%. Up to 3% ethanol, all spores germinated, and the germination time increased with increasing ethanol concentration. At 3.5 …

Time FactorsWater activityconidial germinationphbreadGerm tubePenicillium chrysogenumshelf-life extensionMicrobiologyModels BiologicalLevensmiddelenmicrobiologieAgar platechemistry.chemical_compoundFood Preservationwater activityBotanyFood scienceVLAGEthanolbiologyDose-Response Relationship DrugEthanolspoilagetemperatureSpores FungalPenicillium chrysogenumbiology.organism_classificationYeastSporeKineticsLogistic Modelschemistryclostridium-botulinumGerminationFood Microbiologygrowth-rateFood ScienceJournal of food protection
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