Search results for "wistar"

showing 10 items of 1094 documents

Comparison of segmental-dependent permeability in human and in situ perfusion model in rat.

2017

Abstract Nowadays, alternative methods have been developed to predict intestinal permeability values in human as in vitro, in situ or ex vivo methods. They were developed by the necessity to avoid the problems of the human permeability experiments. However, determination of human permeability is needed to properly validate the alternative methods. For this reason, recently, Dahlgren et al. published an indirect method based on a deconvolution technique to estimate the human permeability in different gastrointestinal segments (jejunum, ileum and colon). Therefore, the objective of this research was to demonstrate that Doluisio technique is a useful method to predict the human permeability in…

Malemedicine.medical_specialtyColonIn situ perfusionPharmaceutical Science02 engineering and technology030226 pharmacology & pharmacyPermeability03 medical and health sciences0302 clinical medicineIleummedicineAnimalsHumansRats WistarAlternative methodsIntestinal permeabilityChemistry021001 nanoscience & nanotechnologymedicine.diseaseSurgeryPerfusionPermeability (earth sciences)JejunumAtenololIntestinal AbsorptionKetoprofenDeconvolution0210 nano-technologyBiomedical engineeringMetoprololEuropean journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
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Modulation by nitric oxide of spontaneous mechanical activity in rat proximal colon.

1999

Summary 1 In order to examine the role of nitric oxide (NO) in the tonic neural inhibition in rat proximal colon, the effects of Nω-nitro- l-arginine methyl ester (L-NAME) were studied on the spontaneous contractions of circular muscle (monitored as intraluminal pressure changes) and of longitudinal muscle (detected as isometric tension changes). 2 L-NAME (3 × 10−−6–3 × 10−−4 m) caused a concentration-dependent increase in the amplitude of circular contractions, without affecting those of longitudinal muscle. This effect was prevented by l-arginine (1–5 × 10−−3 m), but not d-arginine. 3 In the presence of tetrodotoxin (10−−6 m), which per se induced increase of the pressure waves, L-NAME (1…

Malemedicine.medical_specialtyColonIsometric exerciseNeurotransmissionIn Vitro TechniquesInhibitory postsynaptic potentialNitric OxideNitric oxideTonic (physiology)chemistry.chemical_compoundInternal medicineIsometric ContractionmedicineAnimalsDrug InteractionsEnzyme InhibitorsRats WistarGuanethidinePharmacologyDose-Response Relationship DrugGeneral NeuroscienceMuscle SmoothRatsEndocrinologyNG-Nitroarginine Methyl EsterchemistryTetrodotoxinHexamethoniummedicine.drugMuscle ContractionJournal of autonomic pharmacology
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Modulatory role of magnesium on the contractile response of rat aorta to several agonists in normal and calcium-free medium.

1993

Abstract Acute withdrawal of external Mg2+ increased basal tone of rat isolated aorta incubated in the presence of Ca2+. Above normal levels of Mg2+ (1–4 Mm) inhibited basal tone while much higher levels of the divalent cation (64–256 Mm) evoked contractile responses regardless of the presence of Ca2+. Contractile responses to noradrenaline (1μm) and KCl (80 Mm) were inhibited by addition of cumulative concentrations of Mg2+. Acetylcholine-induced contractions in the presence of physiological concentrations of Mg2+ (1 Mm) decreased gradually to the basal tone, but a sustained contraction was observed in the absence of this ion. In Ca2+-free medium, acetylcholine-induced phasic responses ind…

Malemedicine.medical_specialtyContraction (grammar)Muscle RelaxationPharmaceutical Sciencechemistry.chemical_elementAorta ThoracicCalciumIn Vitro TechniquesMuscle Smooth VascularDivalentPotassium ChlorideNorepinephrineInternal medicinemedicineExtracellularAnimalsMagnesiumRats WistarPharmacologychemistry.chemical_classificationAcetylcholineCulture MediaRatsKineticsMuscle relaxationEndocrinologychemistryCalciummedicine.symptomIsotonic SolutionsExtracellular SpaceMagnesium DeficiencyVasoconstrictionAcetylcholinemedicine.drugMuscle contractionMuscle ContractionThe Journal of pharmacy and pharmacology
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Regulation of argininosuccinate synthetase level by corticosteroid and pancreatic hormones during perinatal period.

1995

The urea cycle takes place in the hepatocyte of ureothelic animals. The conversion of ammonia into urea involves five reactions. The first 2 take place in the matrix of the mitochondria, the last 2 occur in the cytosol. Argininosuccinate synthetase (AS) is the third reaction of the urea cycle. It catalyses the condensation of citrulline and aspartate into arginonosuccinate. We have previously reported that rat AS activity was present in the cytosol and the outer membrane of the mitochondria. We have shown that, at the activity level, the colocation of AS was changing during fetal and neonatal development and was under the control of corticosteroid and pancreatic hormones. However, an unreso…

Malemedicine.medical_specialtyCytoplasmHydrocortisoneClinical BiochemistryArgininosuccinate synthaseMitochondria LiverMitochondrionArgininosuccinate SynthaseDexamethasoneDiabetes Mellitus Experimentalchemistry.chemical_compoundAdrenal Cortex HormonesPregnancyInternal medicinemedicineCitrullineAnimalsRats WistarMolecular BiologyPancreatic hormoneCells CulturedHypophysectomybiologyAdrenalectomyCell BiologyGeneral MedicineGlucagonPancreatic HormonesRatsCytosolmedicine.anatomical_structureEndocrinologychemistryAnimals NewbornLiverHepatocyteUrea cyclebiology.proteinFemaleHormoneMolecular and cellular biochemistry
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Improved Bone Biomechanical Properties in Rats after Oral Xylitol Administration

1999

The effects of 5, 10, and 20% dietary xylitol supplementations on the biomechanical properties, histological architecture, and the contents of collagen, pyridinoline, and deoxypyridinoline in long bones of rats were studied. Tibiae were used for the three-point bending test, and femurs were used for the torsion and loading test of the femoral neck. The 10 and 20% oral xylitol administrations caused a significant increase of tibial stress, femoral shear stress, and stress of the femoral neck as compared with the controls. Parallel, but not significant, effects were also seen in the 5% xylitol supplementation group. No significant differences in strain or Young's modulus of the tibiae were de…

Malemedicine.medical_specialtyDeoxypyridinolineEndocrinology Diabetes and MetabolismAdministration OralDentistryXylitolBone and Boneschemistry.chemical_compoundEndocrinologyInternal medicinemedicineAnimalsOrthopedics and Sports MedicineFemurFemurTibiaAmino AcidsRats WistarXylitolFemoral neckPyridinolineTibiabusiness.industrymusculoskeletal systemBiomechanical PhenomenaRatscarbohydrates (lipids)Trabecular bonemedicine.anatomical_structureEndocrinologychemistryCollagenbusinessBone volumeCalcified Tissue International
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Effects of Intraaccumbens Microinjections of Quinpirole on Head Turning and Circling Movement in the Rat

1998

This study was designed to evaluate whether nucleus accumbens dopamine D2 receptors are involved in the initiation of the movement, as distinguished from its execution. For this purpose, the effects of the quinpirole-induced increase of nucleus accumbens dopamine D2 receptor activity were observed on specific parameters of the circling behavior and of its first stage, the head-turning (HT) movement. The experiments were performed on rats with unilateral 6-hydroxydopamine (6-OHDA) lesion of the pars compacta of the substantia nigra and d-amphetamine i.p. (3 mg/kg). Bilateral intraaccumbens microinjections of quinpirole (1, 5, and 10 microg/0.5 microl), an agonist of the D2 receptor family, w…

Malemedicine.medical_specialtyDextroamphetamineQuinpiroleMicroinjectionsClinical BiochemistrySubstantia nigraNucleus accumbensToxicologyBiochemistryNucleus AccumbensBehavioral NeuroscienceQuinpiroleDopamine Uptake InhibitorsDopamine receptor D2Internal medicineBasal gangliamedicineAnimalsRats WistarOxidopamineBiological PsychiatryPharmacologyDose-Response Relationship DrugPars compactaChemistrySympathectomy ChemicalDextroamphetamineBody movementRatsEndocrinologyDopamine AgonistsSympatholyticsStereotyped BehaviorNeurosciencemedicine.drugPharmacology Biochemistry and Behavior
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Anti-inflammatory effects of cerebrocrast in a model of rat paw edema and on mononuclear THP-1 cells.

2002

Cerebrocrast (IOS 1.1212; 4-[2-(difluoromethoxy)phenyl]-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylic acid di(2-propoxyethyl) diester) is a novel derivative of 1,4-dihydropyridine, which does not antagonize Ca(2+) influx in neuronal tissues. Since several classical dihydropyridines possess anti-inflammatory properties, we first studied the effects of cerebrocrast in a model of rat paw edema induced by carrageenan. Cerebrocrast had a preventative effect in this model of inflammation, with maximal activity (32-45% inhibition) in the 0.1-0.25 mg kg(-1) range. It was ineffective when added after the injection of carrageenan. Subsequent in vitro experiments showed that cerebrocrast in the mi…

Malemedicine.medical_specialtyDihydropyridinesmedicine.drug_classmedicine.medical_treatmentAnti-Inflammatory AgentsInflammationNeuroprotectionAnti-inflammatoryMonocyteschemistry.chemical_compoundInternal medicineForelimbmedicineTumor Cells CulturedAnimalsEdemaHumansTHP1 cell lineRats WistarPharmacologyDose-Response Relationship Drugbusiness.industryBiological activityCarrageenanRatsDisease Models AnimalEndocrinologyCytokinechemistryTumor necrosis factor alphamedicine.symptombusinessEuropean journal of pharmacology
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Effect of low levels of dietary fish oil on fatty acid desaturation and tissue fatty acids in obese and lean rats

1995

The effect of very low levels of dietary long-chain n-3 fatty acids on delta 6 desaturation of linoleic acid (18:2n-6) and alpha-linolenic acid (18:3n-3), and on delta 5 desaturation of dihomo-gamma-linolenic acid (20:3n-6), in liver microsomes and its influence on tissue fatty acids were examined in obese and lean Zucker rats and in Wistar rats. Animals fed for 12 wk a balanced diet containing ca. 200 mg of long-chain polyunsaturated n-3 fatty acids per 100 g of diet were compared to those fed the same amount of alpha-linolenic acid. Low amounts of long-chain n-3 fatty acids greatly inhibited delta 6 desaturation of 18:2n-6 and delta 5 desaturation of 20:3n-6, while delta 6 desaturation of…

Malemedicine.medical_specialtyDocosahexaenoic Acids030309 nutrition & dieteticsLinoleic acidPhospholipidBlood lipidsKidneyBiochemistryLinoleic Acid03 medical and health scienceschemistry.chemical_compoundFish OilsSpecies SpecificityInternal medicinemedicineAnimalsRats WistarComputingMilieux_MISCELLANEOUS030304 developmental biologychemistry.chemical_classification0303 health sciencesChemistryMyocardiumOrganic ChemistryBody WeightFatty AcidsFatty acidCell BiologyOrgan SizeFish oilDietary FatsRatsRats Zucker[SDV.BBM.BC]Life Sciences [q-bio]/Biochemistry Molecular Biology/Biomolecules [q-bio.BM]EndocrinologyHuman nutritionBiochemistryLinoleic AcidsLiverDocosahexaenoic acidMicrosomes LiverRATArachidonic acid
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Effects of dietary treatment of rats with eicosapentaenoic acid or docosahexaenoic acid on hepatic lipid metabolism

1998

(1) Effects of dietary treatment of male albino rats with eicosapentaenoic acid (EPA) or docosahexaenoic acid on hepatic mitochondrial lipid metabolism have been investigated. (2) Mitochondria isolated from rats given these treatments were shown to have increased ability to respire on acyl-CoA esters in the presence of malonate. This effect was expressed with most of the long-chain acyl-CoA esters used as substrates. When malonate in the incubations was replaced with malate, mitochondria from treated animals were found to exhibit diminished rates of respiration on polyunsaturated acyl-CoA esters, in particular linolenoyl-, eicosapentaenoyl- and docosahexaenoyl-CoA. This phenomenon could not…

Malemedicine.medical_specialtyDocosahexaenoic AcidsMitochondria LiverBiochemistryLipid peroxidationchemistry.chemical_compoundFish OilsInternal medicinemedicineAnimalsRats WistarMolecular Biologychemistry.chemical_classificationFatty acidLipid metabolismCell BiologyMetabolismLipid MetabolismEicosapentaenoic acidDietRatsEndocrinologyEicosapentaenoic AcidLiverchemistryBiochemistryDocosahexaenoic acidCarnitine biosynthesislipids (amino acids peptides and proteins)Lipid PeroxidationCarnitine palmitoyltransferase IResearch ArticleBiochemical Journal
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The effects of different basal levels of anxiety on the behavioral shift analyzed in the central platform of the elevated plus maze.

2015

The aim of the present research was to study the effects of different basal levels of anxiety on the behavioral shift studied in the central platform of the elevated plus maze. To this purpose, quantitative and multivariate analyses, the latter based on transition matrix elaboration, were carried out on Wistar and on DA/Han rats the latter belonging to a strain characterized by different reactivity to anxiogenic stimuli. Wistar rats spent 74.11 ± 5.11 s in the central platform, whereas DA/Han significantly more: 127.08 ± 9.87. Per cent distributions evidenced a clear-cut difference in walking activities (46.25% in Wistar, 28.4% in DA/Han rats) and in the sniffing activities (45.82% in Wista…

Malemedicine.medical_specialtyElevated plus mazeMaze learningWistar ratAnxietyMotor ActivitySettore BIO/09 - FisiologiaBehavioral NeuroscienceBasal (phylogenetics)SniffingInternal medicinemedicineAnimalsMotor activityRats WistarMaze LearningBehavioral shiftBehavior AnimalMultivariate analysiRats Inbred StrainsDA/Han ratRatsEndocrinologyAnxiogenicMultivariate AnalysisExploratory BehaviorAnxietyTransition matricesmedicine.symptomElevated plus mazePsychologyDecision makingNeuroscienceBehavioural brain research
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