0000000001313269

AUTHOR

Arturo Tortosa

showing 3 related works from this author

Organocatalytic enantioselective functionalization of indoles in the carbocyclic ring with cyclic imines

2019

[EN] An organocatalytic enantioselective functionalization in the carbocyclic ring of indoles with benzoxathiazine 2,2-dioxides is described using a quinine-derived bifunctional organocatalyst. This aza-Friedel-Crafts reaction provides 4-indolyl, 5-indolyl and 7-indolyl sulfamidate derivatives in good yields (up to 99%) and with moderate to high enantioselectivities (up to 86% ee).

Alkylation02 engineering and technologyAlkylation010402 general chemistryRing (chemistry)01 natural sciencesHydroxyindolesCatalysisKetiminesReaccions químiqueschemistry.chemical_compoundMaterials ChemistryFriedel-Crafts reactionBifunctionalFriedel–Crafts reactionConstructionAsymmetric-SynthesisChemistryInhibitorsEnantioselective synthesisGeneral Chemistry021001 nanoscience & nanotechnologyCombinatorial chemistry0104 chemical sciencesFISICA APLICADASurface modification0210 nano-technologyQuímica orgànicaDerivatives
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CCDC 1846586: Experimental Crystal Structure Determination

2018

Related Article: Carlos Vila, Arturo Tortosa, Gonzalo Blay, M. Carmen Muñoz, José R. Pedro|2019|New J.Chem.|43|130|doi:10.1039/C8NJ05577G

Space GroupCrystallographyCrystal System4-(5-hydroxy-1H-indol-4-yl)-34-dihydro-2H-12lambda63-benzoxathiazine-22-dioneCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 1875758: Experimental Crystal Structure Determination

2018

Related Article: Carlos Vila, Arturo Tortosa, Gonzalo Blay, M. Carmen Muñoz, José R. Pedro|2019|New J.Chem.|43|130|doi:10.1039/C8NJ05577G

Space GroupCrystallographyCrystal SystemCrystal StructureCell Parameters68-dichloro-4-(4-hydroxy-1H-indol-5-yl)-34-dihydro-2lambda613-benzothiadiazine-22(1H)-dione monohydrateExperimental 3D Coordinates
researchProduct