Efficient palladium catalyzed synthesis of heteroaromatic sulfoxides

6533b7d0fe1ef96bd125ac3b

RESEARCH PRODUCT

Efficient palladium catalyzed synthesis of heteroaromatic sulfoxides

Françoise Colobert Frédéric R. Leroux Rafael Ballesteros-garrido Rafael Ballesteros Belén Abarca

subject

chemistry.chemical_compound Chemistry Yield (chemistry)Organic Chemistry Drug Discovery Pyridine Thiophene chemistry.chemical_element Triazolopyridine Biochemistry Combinatorial chemistry Catalysis Palladium

description

Abstract The present Letter describes the efficient synthesis of novel heteroaromatic sulfoxides by means of a palladium catalyzed heteroarylation of sulfenate anions. Triazolopyridine, pyridine and thiophene sulfoxides can be obtained under mild conditions and in high yield from the corresponding heteroaryl bromides.

year	journal	country	edition	language
2007-09-01	Tetrahedron Letters

https://doi.org/10.1016/j.tetlet.2007.07.165

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