ChemInform Abstract: Microwave-Assisted Tandem Organocatalytic Peptide-Coupling Intramolecular aza-Michael Reaction: α,β-Unsaturated N-Acyl Pyrazoles as Michael Acceptors.

6533b7dafe1ef96bd126ea7a

RESEARCH PRODUCT

ChemInform Abstract: Microwave-Assisted Tandem Organocatalytic Peptide-Coupling Intramolecular aza-Michael Reaction: α,β-Unsaturated N-Acyl Pyrazoles as Michael Acceptors.

María Sánchez-roselló Cristina Mulet Marta Guerola Carlos Del Pozo Santos Fustero

subject

chemistry.chemical_classification Tandem education Enantioselective synthesis Peptide General Medicine Conjugated system behavioral disciplines and activities Combinatorial chemistry humanities Coupling (electronics)chemistry Organocatalysis Intramolecular force Michael reaction lipids (amino acids peptides and proteins)

description

Conjugated N-acyl pyrazoles are successfully employed in the organocatalytic enantioselective intramolecular aza-Michael reaction as ester surrogates.

year	journal	country	edition	language
2015-04-16	ChemInform

https://doi.org/10.1002/chin.201518046

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