6533b827fe1ef96bd1285a3c

RESEARCH PRODUCT

Triazolopyridines. Part 26: The preparation of novel [1,2,3]triazolo[1,5-a]pyridine sulfoxides

Belén AbarcaFrédéric R. LerouxRafael Ballesteros-garridoRafael Ballesteros-garridoRafael BallesterosFrançoise Colobert

subject

chemistry.chemical_compoundchemistryStereochemistryOrganic ChemistryDrug DiscoveryPyridineSubstituentHalideRegioselectivityTriazolopyridineRing (chemistry)BiochemistryMedicinal chemistry

description

Abstract The regioselective synthesis of new triazolopyridine halides and sulfoxides with the substituent in all different ring positions of [1,2,3]triazolo[1,5- a ]pyridines is presented. The triazolo ring opening reaction of some representative sulfoxides to obtain disubstituted pyridines is also studied.

yearjournalcountryeditionlanguage
2008-04-01Tetrahedron
https://doi.org/10.1016/j.tet.2008.02.011