Oligopeptide der β-Carbolin-3-carbonsäure - Synthese und Affinität zu Benzodiazepinrezeptoren

6533b82dfe1ef96bd1291b9f

RESEARCH PRODUCT

Oligopeptide der β-Carbolin-3-carbonsäure - Synthese und Affinität zu Benzodiazepinrezeptoren

Walter E. Müller Klaus-peter Lippke Walter Schunack

subject

chemistry.chemical_compound Oligopeptide Dipeptide Membrane chemistry Stereochemistry Drug Discovery Pharmaceutical Science Biological activity Tripeptide Receptor

description

Es wurden Oligopeptide der β-Carbolin-3-carbonsaure dargestellt und deren Affinitat zum Benzodiazepinrezeptor in Mausehirn-Membranen bestimmt. Uber Struktur-Affinitatsbeziehungen wird berichtet. Oligopeptides of β-Carboline-3-carboxylic Acid - Synthesis and Benzodiazepine Receptor Affinity Oligopeptides of β-carboline-3-carboxylic acid were prepared and tested with respect to their affinity for the benzodiazepine receptor in mouse brain membranes. Structure-affinity relationships are reported.

year	journal	country	edition	language
1987-01-01	Archiv der Pharmazie

https://doi.org/10.1002/ardp.19873200210

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