6533b860fe1ef96bd12c3880

RESEARCH PRODUCT

ChemInform Abstract: A New Method for the Regioselective Synthesis of β-Enamino Acid Derivatives.

Santos FusteroMa Dolores DíazRaquel Pérez Carlón

subject

chemistry.chemical_compoundchemistryRegioselectivityImidazolechemistry.chemical_elementGeneral MedicineBoronCombinatorial chemistryCatalysis

description

Abstract A mild, simple and efficient route to β-enamino imidazole carbonilic derivatives 3 by reaction of ketimines with N,N′ -carbonyl diimidazole in the presence of boron triflouride as catalyst has been developed. The conversion of 3 to esters has also been explored.

https://doi.org/10.1002/chin.199332231