Search results for " ACTIVATION"

showing 10 items of 1535 documents

Implication of eNOS Uncoupling in Cardiovascular Disease

2017

Under physiological conditions, nitric oxide (NO) is produced in the vasculature mainly by the endothelial nitric oxide synthase (eNOS). Endothelial NO relaxes blood vessels, inhibits platelet activity, and protects against atherosclerosis. Under pathological conditions such as hypertension, diabetes, and hypercholesterolemia, eNOS may become uncoupled. Uncoupled eNOS generates superoxide at the expense of NO and contributes substantially to oxidative stress and endothelial dysfunction. Major mechanisms of eNOS uncoupling include deficiency of the eNOS cofactor tetrahydrobiopterin, deficiency of the eNOS substrate L-arginine, and eNOS S-glutathionylation. Reversal of eNOS uncoupling may rep…

chemistry.chemical_classificationmedicine.medical_specialtyReactive oxygen speciesbiologybusiness.industrySuperoxideTetrahydrobiopterinbiology.organism_classificationmedicine.disease_causemedicine.diseaseNitric oxidechemistry.chemical_compoundEndocrinologychemistryEnosInternal medicinemedicinePlatelet activationEndothelial dysfunctionbusinessOxidative stressmedicine.drugReactive Oxygen Species
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Trace element determination in sediments: a comparative study between neutron activation analysis (NAA) and inductively coupled plasma-mass spectrome…

2000

An inductively coupled plasma-mass spectrometry (ICP-MS) method has been employed for trace element determination in five real sediment samples and a standard reference material. These samples were mineralized by dry ashing at 550°C and fused at 1100°C for 30 min with lithium metaborate. Dissolved samples were measured by a semiquantitative methodology with external calibration and with Rh as an internal standard. More than 50 elements have been measured. As a reference technique, a direct analysis of the solid samples was carried out by neutron activation analysis. Results obtained by ICP-MS have been compared with those obtained by neutron activation analysis (NAA) by applying the paired …

chemistry.chemical_compoundAshingChemistryAnalytical chemistryTrace elementSample preparationNeutron activation analysisMass spectrometryInductively coupled plasma mass spectrometrySpectroscopyAnalytical ChemistryNeutron activationLithium metaborateMicrochemical Journal
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A Versatile Palladium/Triphosphane System for Direct Arylation of Heteroarenes with Chloroarenes at Low Catalyst Loading

2010

International audience; Put a ring on it: The use of an air-stable, robust palladium/tridentate phosphane catalyst in direct C[BOND]H and C[BOND]Cl activation reactions is reported (see scheme; DMAc=N,N-dimethylacetamide, TBAB=tetra-n-butylammonium bromide). Electron-rich, electron-poor, and polysubstituted furans (X=O), thiophenes (X=S), pyrroles (X=NR5), and thiazoles were arylated with chloroarenes in the presence of the catalyst.

chemistry.chemical_elementRing (chemistry)010402 general chemistry01 natural sciencesCatalysisCatalysischemistry.chemical_compound[ CHIM.CATA ] Chemical Sciences/CatalysisBromidePolymer chemistryOrganic chemistryheterocyclesbiologyChemistry010405 organic chemistrydirect arylationGeneral Chemistry[CHIM.CATA]Chemical Sciences/CatalysisGeneral Medicinebiology.organism_classificationpalladium0104 chemical sciencesC[BOND]H activationTriphosphanesynthetic methodsTetraPalladiumAngewandte Chemie
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The hedgehog receptor patched is involved in cholesterol transport.

2011

International audience; BACKGROUND: Sonic hedgehog (Shh) signaling plays a crucial role in growth and patterning during embryonic development, and also in stem cell maintenance and tissue regeneration in adults. Aberrant Shh pathway activation is involved in the development of many tumors, and one of the most affected Shh signaling steps found in these tumors is the regulation of the signaling receptor Smoothened by the Shh receptor Patched. In the present work, we investigated Patched activity and the mechanism by which Patched inhibits Smoothened. METHODOLOGY/PRINCIPAL FINDINGS: Using the well-known Shh-responding cell line of mouse fibroblasts NIH 3T3, we first observed that enhancement …

ciliumlcsh:MedicineyeastBiochemistryReceptors G-Protein-CoupledTransmembrane Transport ProteinsMicechemistry.chemical_compound0302 clinical medicineMolecular Cell Biology[SDV.IDA]Life Sciences [q-bio]/Food engineeringMembrane Receptor SignalingBiomacromolecule-Ligand InteractionsSonic hedgehoglcsh:ScienceComputingMilieux_MISCELLANEOUS0303 health sciencesMultidisciplinaryMechanisms of Signal TransductionVeratrum Alkaloids[SDV.IDA] Life Sciences [q-bio]/Food engineeringdrosophilaSmoothened ReceptorLipidsHedgehog signaling pathwayCell biologySterolsSmoothened ReceptorAlimentation et Nutritionembryonic structurescilMembranes and Sorting[SDV.NEU]Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]Signal transductionvesicular traffickingSignal TransductionResearch Articleprimary ciliumPatched ReceptorsPatchedsignal-transductionanimal structuresCyclopamine[SPI.GPROC] Engineering Sciences [physics]/Chemical and Process EngineeringBiophysicsReceptors Cell Surfacepathway activationSaccharomyces cerevisiaetransduction du signalBiology03 medical and health sciencessonic hedgehoglipidAnimalsHumansFood and NutritionHedgehog Proteins[SPI.GPROC]Engineering Sciences [physics]/Chemical and Process EngineeringBiology030304 developmental biologyPatched Receptorsprotein signalsCell Membranelcsh:RProteinscholesterolBiological TransportTransmembrane Proteinssterol-sensing domainchemistry[ SDV.NEU ] Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]NIH 3T3 Cellscholesterol;lipid;cell trafficking; yeast;drosophila;cells ; pathway activation; vesicular trafficking; signal-transduction; sonic hedgehog;sterol-sensing domain; primary cilium;protein signalsbiology.proteincellslcsh:Qcell traffickingSmoothened030217 neurology & neurosurgery
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Integrin α2β1 Mediates Isoform-Specific Activation of p38 and Upregulation of Collagen Gene Transcription by a Mechanism Involving the α2 Cytoplasmic…

1999

Two collagen receptors, integrins alpha1beta1 and alpha2beta1, can regulate distinct functions in cells. Ligation of alpha1beta1, unlike alpha2beta1, has been shown to result in recruitment of Shc and activation of the Ras/ERK pathway. To identify the downstream signaling molecules activated by alpha2beta1 integrin, we have overexpressed wild-type alpha2, or chimeric alpha2 subunit with alpha1 integrin cytoplasmic domain in human osteosarcoma cells (Saos-2) lacking endogenous alpha2beta1. The chimeric alpha2/alpha1 chain formed a functional heterodimer with beta1. In contrast to alpha2/alpha1 chimera, forced expression of alpha2 integrin resulted in upregulation of alpha1 (I) collagen gene …

collagenIntegrinsReceptors CollagenTranscription GeneticintegrinIntegrincytoplasmic domainCDC42Biologyp38 MAPKTransfectionCD49cp38 Mitogen-Activated Protein KinasesCollagen receptorTumor Cells CulturedHumansProtein IsoformsCell BiologyMolecular biologyCell biologyUp-RegulationEnzyme ActivationIntegrin alpha Mbiology.proteinIntegrin beta 6Original ArticleSignal transductionMitogen-Activated Protein KinasesITGA6Signal TransductionThe Journal of Cell Biology
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Neuromuscular adaptations to single-session combined strength and endurance training in untrained men : an examination of the order effect

2013

Understanding the adaptations to single-session combined strength (S) and endurance (E) training has received increased attention in scientific literature through the expand-ing use of combined training programs for practical purposes. However, the intra-session exercise order when performing both E and S in the same training session may limit potential strength development, as the neuromuscular adaptations to either training mode alone are very different. Research on the effect of the intra-session exercise order of combined training on various training-induced adaptations, i.e. the order effect, is currently limited, especially with regard to the neuromuscular adaptations. Therefore, the …

combined trainingneural activationhermo-lihastoimintakestävyysharjoitteluorder effectinterference effectsuper-imposed twitch techniquevoimaharjoittelustrength
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Activity and kinetics of DNA dependent DNA and RNA polymerases n xeroderma pigmentosum and in normal human skin.

1971

1. DNA dependent DNA polymerase (E.C.2.7.7.7) was prepared from human normal and from Xeroderma pigmentosum skin. 2. DNA polymerase from normal skin has the same Michaelis constant with native and denatured DNA as templateKm= 120 ± 11 µg DNA/ml, with differing maximum reaction velocities. 3. The enzyme from Xeroderma pigmentosum has the same Michaelis constant for denatured DNA as the enzyme from normal skin, but with native DNA as template, theKmvalue is lower (97.2 ± 9.8). The maximum reaction velocities of the Xeroderma pigmentosum enzyme with native resp. denatured DNA as template are the same. 4. DNA dependent RNA polymerases (E.C.2.7.7.6) from normal and Xeroderma pigmentosum skin wer…

congenital hereditary and neonatal diseases and abnormalitiesXeroderma pigmentosumDNA polymeraseDNA polymerase IIDermatologyTritiumEndonucleasechemistry.chemical_compoundmedicineHumansskin and connective tissue diseasesPolymeraseSkinCarbon IsotopesXeroderma PigmentosumDNA clampintegumentary systembiologynutritional and metabolic diseasesRNA NucleotidyltransferasesGeneral MedicineDNAClinical Enzyme Testsmedicine.diseaseMolecular biologyEnzyme ActivationchemistryDNA Nucleotidyltransferasesbiology.proteinPrimer (molecular biology)DNAArchiv fur dermatologische Forschung
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Enhanced Lipid Peroxidation and Platelet Activation in the Early Phase of Type 1 Diabetes Mellitus

2003

Background— To investigate early events possibly related to the development of diabetic angiopathy, we examined whether 8-iso-prostaglandin F 2α (8-iso-PGF 2α ) formation, a marker of in vivo oxidant stress, is altered in different stages of type 1 diabetes (T1DM) and whether it correlates with the rate of thromboxane (TX) A 2 biosynthesis, a marker of in vivo platelet activation. We also investigated the relationship between inflammatory markers and F 2 -isoprostane formation in this setting. Methods and Results— A cross-sectional study was performed in 23 insulin-treated patients aged <18 years with new-onset T1DM (≤6 weeks, group A), matched for age and gender with 23 patients with s…

diabetes mellitus; inflammation; plateletsMalemedicine.medical_specialtyAdolescentThromboxaneInflammationDiabetic angiopathyDinoprostTimeThromboxane A2Reference ValuesPhysiology (medical)Internal medicineDiabetes mellitusHumansInsulinMedicinePlatelet activationChildInterleukin 6InflammationF2-IsoprostanesType 1 diabetesbiologyInterleukin-6Tumor Necrosis Factor-alphabusiness.industryPlatelet Activationmedicine.diseaseThromboxane B2Oxidative StressC-Reactive ProteinCross-Sectional StudiesDiabetes Mellitus Type 1Endocrinologydiabetes mellitusplateletsDisease Progressionbiology.proteinFemaleTumor necrosis factor alphaLipid Peroxidationmedicine.symptomCardiology and Cardiovascular MedicinebusinessBiomarkersFollow-Up StudiesCirculation
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Optimal inter-stimulus interval for interpolated twitch technique when using double pulse stimulation

2013

Interpolated twitch technique is a method frequently used to assess voluntary activa- tion. This method uses electrically evoked twitch superimposed on the voluntary activi- ty and its comparison with the twitch in rested muscle i.e. control twitch, to evaluate completeness of muscle activation. The purpose of this study was to investigate the ef- fect of interval in paired stimulation on control twitch in young and elderly individuals with bent and flexed knee positions. Supramaximal electrical stimulation consisted of one single stimulus and eight paired stimulation with intervals from 5 to 40ms, with increments of 5ms. In evoked twitches normalized peak torque amplitude (NPT), time to pe…

doubletittpaired stimulivoluntary activationlihaksetbiomekaniikkainterpolated twitch techniqueärsykkeet
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Acute incremental endurance performance and explosive strength training period : muscle activity, acid-base balance and hormonal responses

2015

Johdanto. Akuutin kestävyys- ja voimaharjoituksen fysiologiset vasteet ilmenevät luurankolihaksissa, hengitys- ja verenkiertoelimistössä, sekä endokriinisessa että immuunijärjestelmässä. Nämä vasteet voivat heikentää suorituskykyä, ja esimerkiksi happo-emästasapaino on tarkoin säädelty negatiivisten seurausten varalta. Lihasten toimintaa voidaan tutkia elektromyografialla (EMG), ja nykyään on myös mahdollista käyttää tekstiilielektrodeja, jotka mahdollistavat lihasryhmien sähköisen aktiivisuuden tallentamisen normaalin liikkumisen aikana. Tämän tutkimuksen tarkoituksena oli tutkia yhteyksiä etu- ja takareisien lihasaktiivisuuksien ja happo-emästasapainon välillä, vertailla lihasaktiivisuuks…

elektromyografiaEMG shortskestävyysharjoitteluacid-base balancehappo-emästasapainolihaksetincremental exercise testmuscle activation
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