Search results for " Staphylococcus aureus"

showing 7 items of 67 documents

Pyrrolomycins as antimicrobial agents. Microwave-assisted organic synthesis and insights into their antimicrobial mechanism of action

2019

Abstract New compounds able to counteract staphylococcal biofilm formation are needed. In this study we investigate the mechanism of action of pyrrolomycins, whose potential as antimicrobial agents has been demonstrated. We performed a new efficient and easy method to use microwave organic synthesis suitable for obtaining pyrrolomycins in good yields and in suitable amount for their in vitro in-depth investigation. We evaluate the inhibitory activity towards Sortase A (SrtA), a transpeptidase responsible for covalent anchoring in Gram-positive peptidoglycan of many surface proteins involved in adhesion and in biofilm formation. All compounds show a good inhibitory activity toward SrtA, havi…

Staphylococcus aureusClinical BiochemistryPharmaceutical ScienceMicrobial Sensitivity Testsmedicine.disease_causeSettore BIO/19 - Microbiologia Generale01 natural sciencesBiochemistrychemistry.chemical_compoundBacterial ProteinsDrug DiscoverymedicinePyrrolesEnzyme InhibitorsMicrowavesMolecular BiologyEnzyme Assays010405 organic chemistryChemistryOrganic ChemistryBiofilmN-Acetylmuramoyl-L-alanine AmidaseAntimicrobialAminoacyltransferasesAntimicrobial resistance Pyrrolomycins Sortase A Staphylococcus aureus In-silico docking studies MAOS Pharmacokinetics studies Murein hydrolase activitySettore CHIM/08 - Chimica Farmaceutica0104 chemical sciencesAnti-Bacterial AgentsMolecular Docking Simulation010404 medicinal & biomolecular chemistryCysteine EndopeptidasesBiochemistryMechanism of actionDocking (molecular)Staphylococcus aureusSettore CHIM/03 - Chimica Generale E InorganicaSortase ABiofilmsPseudomonas aeruginosaMolecular MedicineOrganic synthesisPeptidoglycanmedicine.symptom
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Rapid differentiation between livestock-associated and livestock-independent Staphylococcus aureus CC398 clades.

2013

Staphylococcus aureus clonal complex 398 (CC398) isolates cluster into two distinct phylogenetic clades based on single-nucleotide polymorphisms (SNPs) revealing a basal human clade and a more derived livestock clade. The scn and tet(M) genes are strongly associated with the human and the livestock clade, respectively, due to loss and acquisition of mobile genetic elements. We present canonical single-nucleotide polymorphism (canSNP) assays that differentiate the two major host-associated S. aureus CC398 clades and a duplex PCR assay for detection of scn and tet (M). The canSNP assays correctly placed 88 S. aureus CC398 isolates from a reference collection into the human and livestock clade…

Staphylococcus aureusLivestockPsychologie appliquéelcsh:MedicineBiologySettore MED/42 - Igiene Generale E Applicatamedicine.disease_causeStaphylococcal infectionsPolymorphism Single NucleotideAnimal DiseasesMicrobiologylaw.invention03 medical and health sciencesPhylogeneticslawmedicineAnimalsHumansMRSA ST398 clades differentiationCladelcsh:SciencePhylogenyPolymerase chain reaction030304 developmental biology0303 health sciencesMultidisciplinaryPhylogenetic tree030306 microbiologylcsh:RStaphylococcal InfectionsSciences bio-médicales et agricolesmedicine.diseaseMethicillin-resistant Staphylococcus aureus3. Good healthGenes BacterialStaphylococcus aureuslcsh:QMobile genetic elementsBiologieResearch ArticlePLoS ONE
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Effect of temperature on the release of carvacrol and cinnamaldehyde incorporated into polymeric systems to control growth and biofilms ofEscherichia…

2015

This study assessed the effect of temperature on the release of essential oil components incorporated by melt compounding into polymeric films. Specifically, polyethylene-co-vinylacetate (EVA) films containing carvacrol (CAR) and cinnamaldehyde (ALD), alone and in combination, were prepared and their surface and mechanical properties and antibacterial and anti-biofilm activity against Escherichia coli and Staphylococcus aureus were evaluated. The addition of ALD and CAR did not provoke variation in the surface morphology of EVA and allowed their delivery. At 37°C, films containing CAR, ALD or their combination (25+75%) were found to have the strongest bactericidal effect, whereas at lower t…

Staphylococcus aureusMorphology (linguistics)Aquatic Sciencemedicine.disease_causeApplied Microbiology and BiotechnologybiofilmCinnamaldehydelaw.inventionchemistry.chemical_compoundlawOils VolatileEscherichia colimedicineOrganic chemistryCarvacrolAcroleinEscherichia coliEssential oilWater Science and TechnologyAcroleinBiofilmtemperatureAnti-Bacterial Agentsantibacterial polymerchemistryStaphylococcus aureusBiofilmsMonoterpenesStaphylococcus aureuCymenesPolyvinylsPolyethylenestemperature; antibacterial polymers; biofilm; essential oil components; Escherichia coli; Staphylococcus aureusessential oil componentNuclear chemistryBiofouling
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The chemical composition of the aerial parts of Stachys spreitzenhoferi (Lamiaceae) growing in Kythira Island (Greece), and their antioxidant, antimi…

2022

The Stachys L. genus has been used in traditional medicine to treat skin inflammations, stomach disorders, and stress. The aim of this study was to investigate the chemical profile and biological activity of the methanolic extract of Stachys spreitzenhoferi Heldr. (Lamiaceae) aerial parts, collected on the island of Kythira, South Greece. The analysis by liquid chromatography coupled with electrospray ionization and high-resolution mass spectrometry [LC-(-)ESI/HRMSn] of the methanol extract revealed the occurrence of thirty-six compounds - flavonoids, phenylethanoid glycosides, iridoids, quinic acid derivatives, aliphatic alcohol glycosides, and oligosaccharides - highlighting the substanti…

Staphylococcus aureusQuinic AcidPlant ScienceAntiproliferative activityHorticultureAntimicrobial activityBiochemistryAntioxidantsAntimicrobial activity; Antioxidant effects; Antiproliferative activity; LC-(−)ESI/HRMS(n); Lamiaceae; Stachys spreitzenhoferi Heldr.; Anti-Bacterial Agents; Antioxidants; Flavonoids; Glycosides; Greece; Humans; Iridoids; Methanol; Plant Components Aerial; Plant Extracts; Quinic Acid; Reactive Oxygen Species; Staphylococcus aureus; Superoxide Dismutase; U937 Cells; Anti-Infective Agents; Lamiaceae; StachysAnti-Infective AgentsHumansIridoidsStachys spreitzenhoferi HeldrGlycosidesMolecular BiologyFlavonoidsLamiaceaeGreecePlant ExtractsSuperoxide DismutaseMethanolStachys spreitzenhoferi Heldr.LC-(−)ESI/HRMS(n)AerialGeneral MedicineU937 CellsAntioxidant effectPlant Components AerialAnti-Bacterial AgentsAntioxidant effectsStachysPlant ComponentsReactive Oxygen Species
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Control of biofilm formation by poly-ethylene-co-vinyl acetate films incorporating nisin.

2010

The aim of this study was to evaluate the effect of poly-ethylene-co-vinyl acetate (EVA) films incorporating different concentrations (0.1%, 0.5% and 1%) of nisin on the biofilm-forming ability of Listeria monocytogenes ATCC 7644, Staphylococcus aureus 815 and Staphylococ-cus epidermidis ATCC 35984. Nisin was incorporated into two grades of EVA (EVA14 and EVA28) in the melt during a common film-blowing operation. The efficacy of EVA/nisin films was evaluated by biofilm biomass measurements and Live/Dead staining in combination with fluorescence microscopy. In order to evaluate whether the nisin incorporation could modify the film surface properties, contact angle measurements and scanning e…

Staphylococcusmedicine.disease_causeApplied Microbiology and BiotechnologyBacterial AdhesionNisin polymeric film biofilmMicrobiologyContact anglechemistry.chemical_compoundListeria monocytogenesStaphylococcus epidermidisStaphylococcus epidermidispolycyclic compoundsFluorescence microscopemedicineVinyl acetateNisinNisinListeria monocytogeneNisin; Polymeric film; Biofilm; Listeria monocytogenes; Staphylococcus aureus; Staphylococcus epidermidisbiologyBiofilmBiofilmFood PackagingGeneral Medicinebiochemical phenomena metabolism and nutritionbiology.organism_classificationListeria monocytogenesAnti-Bacterial AgentsSettore ING-IND/22 - Scienza E Tecnologia Dei MaterialiPolymeric filmchemistryStaphylococcus aureusBiofilmsStaphylococcus aureuPolyvinylsBiotechnologyNuclear chemistryApplied microbiology and biotechnology
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Antibacterial Activity of Flavonoids Against Methicillin-resistant Staphylococcus aureus strains

2000

An experimental and theoretical study was performed on the anti-staphylococcal activity of 18 natural and synthetic flavonoids against methicillin-resistant Staphylococcus aureus strains. The analysed flavonoids belong to three well-differentiated structural patterns: chalcones, flavanones and flavones. The quantitative analysis of the anti-staphylococcal activity of the compounds was carried out by determining their percent inhibition degree. The hierarchical cluster analysis method was used to analyse the anti-MRSA activity of the compounds. With this methodology, the flavonoids were classified into four groups according to their anti-staphylococcal activity (high, sufficient, intermediat…

Statistics and ProbabilityStaphylococcus aureusChalconeStereochemistryFlavonoidMicrobial Sensitivity Testsmedicine.disease_causeFlavonesGeneral Biochemistry Genetics and Molecular BiologyStructure-Activity Relationshipchemistry.chemical_compoundChalconemedicineAnimalsCluster AnalysisHumansStructure–activity relationshipFlavonoidschemistry.chemical_classificationGeneral Immunology and MicrobiologyApplied MathematicsGeneral MedicineStaphylococcal InfectionsMethicillin-resistant Staphylococcus aureusAnti-Bacterial AgentschemistryBiochemistryStaphylococcus aureusModeling and SimulationMethicillin ResistanceGeneral Agricultural and Biological SciencesAntibacterial activityQuantitative analysis (chemistry)Journal of Theoretical Biology
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MRSA ST22-IVa (EMRSA-15 clone) in Palermo, Italy

2010

Summary: Epidemic spread of methicillin-resistant Staphylococcus aureus (MRSA) strains carrying the Staphylococcal Chromosomal Cassettes (SCC) mec type IV is being increasingly reported in many geographical areas. A survey to determine the prevalence and characteristics of MRSA SCCmec IV isolates identified in four general hospitals in Palermo, Italy, was carried out. During the period February–June 2009, SCCmec type IVa has been found in 12 out of 94 isolates. Nine isolates from all hospitals and all strains from a NICU outbreak occurring in the same period were attributed with the ST22-IVa (EMRSA-15) clone. In our setting, due to the changing MRSA epidemiology, detection of SCCmec IV coul…

clone (Java method)Methicillin-Resistant Staphylococcus aureusMeticillinEpidemiologyDrug resistanceMRSAMolecular typingmedicine.disease_causeHospitals GeneralMicrobiologylcsh:Infectious and parasitic diseasesDisease OutbreaksMolecular typingEpidemic spreadPrevalenceMedicineHumanslcsh:RC109-216EMRSA-15business.industrylcsh:Public aspects of medicinePublic Health Environmental and Occupational HealthOutbreaklcsh:RA1-1270General MedicineStaphylococcal Infectionsbiochemical phenomena metabolism and nutritionbacterial infections and mycosesVirologyInfectious DiseasesCross-Sectional StudiesItalyStaphylococcus aureusST22-IVAsense organsbusinessmedicine.drugBeta lactam antibioticsJournal of Infection and Public Health
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