Search results for " activity"

showing 10 items of 4540 documents

Simple dialkyl pyrazole-3,5-dicarboxylates show in vitro and in vivo activity against disease-causing trypanosomatids.

2017

SUMMARYThe synthesis and antiprotozoal activity of some simple dialkyl pyrazole-3,5-dicarboxylates (compounds 2–6) and their sodium salts (pyrazolates) (compounds 7–9) against Trypanosoma cruzi, Leishmania infantum and Leishmania braziliensis are reported. In most cases the studied compounds showed, especially against the clinically significant amastigote forms, in vitro activities higher than those of the reference drugs (benznidazole for T. cruzi and glucantime for Leishmania spp.); furthermore, the low non-specific cytotoxicities against Vero cells and macrophages shown by these compounds led to good selectivity indexes, which are 8–72 times higher for T. cruzi amastigotes and 15–113 tim…

0301 basic medicineTrypanosomamedicine.drug_classTrypanosoma cruziParasitemiaLeishmania braziliensisMicrobiology03 medical and health sciencesMiceIn vivoChlorocebus aethiopsparasitic diseasesmedicineAnimalsChagas DiseaseDicarboxylic AcidsLeishmania infantumAmastigoteTrypanosoma cruziVero CellsLeishmaniaMice Inbred BALB CbiologyMacrophagesbiology.organism_classificationLeishmaniaLeishmania braziliensisTrypanocidal Agentsantichagasic activitypyrazole030104 developmental biologyInfectious DiseasesBenznidazoleleishmanicidal activityAntiprotozoalcytotoxicityPyrazolesAnimal Science and ZoologyParasitologyFemaleLeishmania infantummedicine.drug
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Effects of innovative and conventional sanitizing treatments on the reduction of Saccharomycopsis fibuligera defects on industrial durum wheat bread

2016

Wickerhamomyces anomalus, Hyphopichia burtonii and Saccharomycopsis fibuligera are spoilage yeasts causing chalk mold defects on sliced bread packaged under modified atmosphere. The first objective of this study, carried out in a bread-making company for two consecutive years, was to genetically identify yeasts isolated from spoiled sliced bread in Modified Atmosphere Packaging (MAP) and to determine the dominant species among identified strains. The second objective was to evaluate the effects of hydrogen peroxide and silver solution 12% (HPS) treatment in the leavening cells and cooling chambers, in comparison with the conventional Ortho-Phenylphenol (OPP) fumigating treatment, on the inc…

0301 basic medicineWater activityBaked goodsWickerhamomyces anomalus030106 microbiologyFood spoilageSaccharomycopsismedicine.disease_causeMicrobiology03 medical and health sciences0404 agricultural biotechnologyYeastsMoldmedicineBaked goodFood scienceChalk mold defects; Baked goods; 26S sequencing; MAP packaging; Water activity; Environmental biodecontaminationTriticumLeavening agent26S sequencingChalk mold defectChemistryEnvironmental biodecontaminationTemperatureMAP packagingWaterBreadHydrogen Peroxide04 agricultural and veterinary sciencesGeneral MedicineSettore AGR/15 - Scienze E Tecnologie AlimentariContamination040401 food scienceYeastRNA RibosomalModified atmosphereChalk mold defectsFood ScienceWater activity
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Employ of Citrus By-product as Fat Replacer Ingredient for Bakery Confectionery Products

2020

Citrus fruits processing is one of the foremost industrial activities in Sicily and the main residual by-product consists in peels and seeds (known as "pastazzo"). Traditionally this by-product has been used for different purposes, and only most recently, it has been described as source of a wide range of healthy bioactive compounds and dietary fibers. In the present work, a debittered food grade orange fiber (DOF), extracted from orange juice by-product, was experimentally obtained and tested as fat-replacer at different percentages (30, 50, and 70%) in bakery confectionery products (brioches). The DOF showed high total fiber content, low water activity and a high water binding capacity. T…

0301 basic medicineWater activityEndocrinology Diabetes and Metabolism030209 endocrinology & metabolismlcsh:TX341-641Orange (colour)fat replacementfunctional food03 medical and health sciencesIngredient0302 clinical medicineorange juice wasteBy-productFood scienceWater contentfunctional foodsNutritionOriginal ResearchOrange juice030109 nutrition & dieteticsNutrition and DieteticsChemistrybakery confectionery productsdietary fiberbakery confectionery productDietary fiberWater bindinglcsh:Nutrition. Foods and food supplyFood Science
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Complete Genome Sequence of Lactobacillus rhamnosus Strain BPL5 (CECT 8800), a Probiotic for Treatment of Bacterial Vaginosis

2016

ABSTRACT Lactobacillus rhamnosus BPL5 (CECT 8800), is a probiotic strain suitable for the treatment of bacterial vaginosis. Here, we report its complete genome sequence deciphered by PacBio single-molecule real-time (SMRT) technology. Analysis of the sequence may provide insight into its functional activity.

0301 basic medicineWhole genome sequencingStrain (chemistry)030106 microbiologyfood and beveragesBiologymedicine.diseasebiology.organism_classificationMicrobiologylaw.invention03 medical and health sciencesProbiotic030104 developmental biologyLactobacillus rhamnosuslawGeneticsmedicineFunctional activityProkaryotesBacterial vaginosisMolecular BiologyGenome Announcements
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Barrel cortex: What is it good for?

2017

The rodent whisker system, with barrel cortex as its most prominent structure, has evolved into a powerful model system to study sensory processing. However, despite the vast amount of data collected on barrel cortex neural activity patterns, as well as its circuitry and plasticity, the precise behavioral and cognitive operations for which this structure is needed are still elusive. Proposed functions of barrel cortex include detection, discrimination, coordination of whisker movements during exploratory locomotion or active touch, and associative learning. Departing from a definition of what exactly constitutes a function and how the involvement of a brain area in a specific task can be es…

0301 basic medicineanimal structuresSensory processingmedicine.medical_treatmentBarrel (horology)Somatosensory system03 medical and health sciencesNeural activityMice0302 clinical medicineCognitionmedicineAnimalsBehavior AnimalGeneral NeuroscienceCognitionSomatosensory CortexBarrel cortexAssociative learningRats030104 developmental biologyVibrissaePsychologyNeuroscience030217 neurology & neurosurgeryCognitive loadNeuroscience
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Identification and control of moulds responsible for black spot spoilage in dry-cured ham.

2016

The aims of this work were to identify moulds responsible for black spot spoilage in the drying and cellar stages of dry-cured ham processing and evaluate the effectiveness of preventive actions for controlling this alteration. Four mould strains isolated from spoiled hams were identified by morphological characteristics and the ITS and β-tubulin sequencing. Two of them were Cladosporium oxysporum, one was C. cladosporioides and the remaining one was C. herbarum. These spoiling strains reproduced the black spots on dry-cured ham-based media and ham slices. Additionally, the effect of water activity (aw) conditions reached throughout dry-cured ham ripening and the activity of the protective …

0301 basic medicinebiologyWater activityFood spoilageSus scrofaFood preservationfood and beveragesRipeningPenicillium chrysogenumbiology.organism_classificationPenicillium chrysogenumMeat Products03 medical and health sciences030104 developmental biologyFood PreservationFood MicrobiologyFood microbiologyAnimalsMicrobial InteractionsFood scienceDesiccationCladosporiumFood ScienceBlack spotCladosporiumMeat science
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Physical Activity and Brain Health.

2019

Physical activity (PA) has been central in the life of our species for most of its history, and thus shaped our physiology during evolution. However, only recently the health consequences of a sedentary lifestyle, and of highly energetic diets, are becoming clear. It has been also acknowledged that lifestyle and diet can induce epigenetic modifications which modify chromatin structure and gene expression, thus causing even heritable metabolic outcomes. Many studies have shown that PA can reverse at least some of the unwanted effects of sedentary lifestyle, and can also contribute in delaying brain aging and degenerative pathologies such as Alzheimer’s Disease, diabetes, and multiple s…

0301 basic medicinebrain healthIrisinlcsh:QH426-470Dopaminemyokinesphysical activityDiseaseReviewmyokineexercise and neurodegenerationexercise and aging03 medical and health sciences0302 clinical medicineSettore BIO/10 - BiochimicaMyokineGeneticsMedicineHumansEpigeneticsSettore BIO/06 - Anatomia Comparata E CitologiaExerciseGenetics (clinical)Sedentary lifestylelactatebusiness.industryMultiple sclerosisBrain-Derived Neurotrophic FactorBrainCognitionNeurodegenerative Diseasesmedicine.diseaselcsh:Genetics030104 developmental biologyBDNFAntidepressantbusinessNeuroscience030217 neurology & neurosurgeryHormoneEndocannabinoidsGenes
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Mesoglea Extracellular Matrix Reorganization during Regenerative Process in Anemonia viridis (Forskål, 1775)

2021

Given the anatomical simplicity and the extraordinary ability to regenerate missing parts of the body, Cnidaria represent an excellent model for the study of the mechanisms regulating regenerative processes. They possess the mesoglea, an amorphous and practically acellular extracellular matrix (ECM) located between the epidermis and the gastrodermis of the body and tentacles and consists of the same molecules present in the ECM of vertebrates, such as collagen, laminin, fibronectin and proteoglycans. This feature makes cnidarians anthozoans valid models for understanding the ECM role during regenerative processes. Indeed, it is now clear that its role in animal tissues is not just tissue su…

0301 basic medicinecollagenAnemonia viridis Collagen Enzymatic activity Histology Morphology Regeneration Animals Collagen Type I Extracellular Matrix Sea Anemones Regeneration Wound HealingTentacleQH301-705.5enzymatic activityContext (language use)Anemonia viridisMesogleaArticleCollagen Type ICatalysisInorganic ChemistryExtracellular matrixhistology03 medical and health sciences0302 clinical medicinemorphologyAnimalsPhysical and Theoretical ChemistryBiology (General)Molecular BiologyQD1-999SpectroscopyWound HealingbiologyRegeneration (biology)Organic ChemistryGeneral MedicineRegenerative processExtracellular MatrixComputer Science ApplicationsCell biologyFibronectinChemistrySea Anemones030104 developmental biologyregenerationbiology.proteinAnemonia viridis; collagen; enzymatic activity; histology; morphology; regenerationWound healing<i>Anemonia viridis</i>030217 neurology & neurosurgeryInternational Journal of Molecular Sciences
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Polyphosphate Reverses the Toxicity of the Quasi-Enzyme Bleomycin on Alveolar Endothelial Lung Cells In Vitro

2021

Simple Summary Bleomycin (BLM) is a medication introduced used to treat various types of cancer, including testicular cancer, ovarian cancer, and Hodgkin’s disease. Its most serious side effect is pulmonary fibrosis and impaired lung function. Using A549 human lung cells it is shown that, in parallel to an increased cell toxicity and DNA damage, BLM causes a marked enlargement of the cell nucleus. This effect is abolished by inorganic polyphosphate (polyP), if this physiological polymer is administered together with BLM. The detoxification of BLM is–most likely–caused by the upregulation of the gene encoding the BLM hydrolase which inactivates BLM in vitro and in vivo. This study contribute…

0301 basic medicinecongenital hereditary and neonatal diseases and abnormalitiesCancer ResearchDNA damageBleomycinlcsh:RC254-282Article03 medical and health scienceschemistry.chemical_compound0302 clinical medicineanti-SARS-CoV-2 activityDownregulation and upregulationprevention of fibrosischemistry.chemical_classificationbleomycinpulmonary fibrosisurogenital systemChemistryCell growthCOVID-19nutritional and metabolic diseasespolyphosphatelcsh:Neoplasms. Tumors. Oncology. Including cancer and carcinogensMolecular biologyIn vitroChromatin030104 developmental biologyEnzymeOncology030220 oncology & carcinogenesisToxicityCancers
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Photocatalytic Activity of Polymer Nanoparticles Modulates Intracellular Calcium Dynamics and Reactive Oxygen Species in HEK-293 Cells

2018

Optical modulation of living cells activity by light-absorbing exogenous materials is gaining increasing interest, due to the possibility both to achieve high spatial and temporal resolution with a minimally invasive and reversible technique and to avoid the need of viral transfection with light-sensitive proteins. In this context, conjugated polymers represent ideal candidates for photo-transduction, due to their excellent optoelectronic and biocompatibility properties. In this work, we demonstrate that organic polymer nanoparticles, based on poly(3-hexylthiophene) conjugated polymer, establish a functional interaction with an in vitro cell model (Human Embryonic Kidney cells, HEK-293). Th…

0301 basic medicineconjugated polymerHistologylcsh:BiotechnologyCellBiomedical EngineeringBioengineeringContext (language use)02 engineering and technologyCalcium in biology03 medical and health sciencesCa2+ imaginglcsh:TP248.13-248.65medicineViability assaybio-organic electronicsOriginal Researchreactive oxygen specieschemistry.chemical_classificationReactive oxygen speciesorganic semiconductorHEK 293 cellsBioengineering and BiotechnologyPhotocatalytic ActivityTransfection021001 nanoscience & nanotechnologyConjugated Polymer NanoparticlesCytosol030104 developmental biologymedicine.anatomical_structurechemistryBiophysicsIntracellular Calcium Dynamicsphotomodulationlight0210 nano-technologycell optical stimulationBiotechnologyFrontiers in Bioengineering and Biotechnology
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