Search results for " surface"

showing 10 items of 2838 documents

Folate-mediated targeting of polymeric conjugates of gemcitabine.

2005

The synthesis of two new macromolecular prodrugs for active tumor targeting was set up. Gemcitabine (2'-deoxy-2',2'-difluorocytidine) was conjugated to alpha,beta-poly(N-2-hydroxyethyl)-DL-aspartamide (PHEA) through succinyl or diglycolyl hydrolysable spacers. The targeting agent folic acid was attached to the macromolecular backbone through the aminocaproic spacer. The two conjugates [PHEA-(5'-succinylgemcitabine)-1'-carboxypentyl-folamide and PHEA-(5'-diglycolyl-gemcitabine)-1'-carboxypentyl-folamide], were purified and extensively characterised by spectroscopic (UV, IR and NMR) and chromatographic analyses to determine the correct chemical structure, the purity degree and the reaction yi…

Antimetabolites AntineoplasticTime FactorsStereochemistryCell SurvivalpolyaspartamideChemical structurePharmaceutical ScienceReceptors Cell SurfaceConjugated systemDeoxycytidineDrug Delivery SystemsFolic AcidCell Line Tumorfolate-mediated targetingExtracellularHumansProdrugsIncubationPolyhydroxyethyl MethacrylateDrug CarriersDose-Response Relationship DrugChemistrypolymeric conjugateFolate Receptors GPI-AnchoredSuccinatesHydrogen-Ion ConcentrationGemcitabineIn vitroBiochemistryCell cultureCarrier ProteinsMacromoleculeConjugateInternational journal of pharmaceutics
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Role of the virulence plasmid pR99 and the metalloprotease Vvp in resistance of Vibrio vulnificus serovar E to eel innate immunity

2007

Vibrio vulnificus biotype 2 serovar E (VSE) is a bacterial pathogen that produces a haemorrhagic septicaemia called vibriosis in eels. Its ability to grow in blood is conferred by a recently described virulence plasmid [Lee CT, Amaro C, Wu KM, Valiente E, Chang YF, Tsai SF, et al. A common virulence plasmid in biotype 2 Vibrio vulnificus and its dissemination aided by a conjugal plasmid. Journal of Bacteriology, submitted for publication.]. In this study, we analyzed the role of this plasmid together with the role played by the metalloprotease (Vvp) in the interaction between bacteria and eel innate immunity. To this end, we compared and statistically analyzed the differences in resistance …

Antimicrobial peptidesVirulenceMicrobial Sensitivity TestsVibrio vulnificusAquatic ScienceMicrobiologyPlasmidAnti-Infective AgentsBacterial ProteinsPhagocytosisBacteriologyAnimalsEnvironmental ChemistryImmunity MucosalVibrio vulnificusPathogenAntigens BacterialPhagocytesInnate immune systembiologyComplement Fixation TestsTransferrinMetalloendopeptidasesGeneral MedicineAnguillabiology.organism_classificationAntibodies BacterialVirologyImmunity InnateAntigens SurfaceMutationAlternative complement pathwayMuramidaseAntimicrobial Cationic PeptidesPlasmidsFish & Shellfish Immunology
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Negative-pressure cavitation extraction of cajaninstilbene acid and pinostrobin from pigeon pea [Cajanus cajan (L.) Millsp.] leaves and evaluation of…

2011

Abstract In this study, an efficient negative-pressure cavitation extraction (NPCE) technique was developed to extract cajaninstilbene acid (CSA) and pinostrobin (PI) from pigeon pea [Cajanus cajan (L.) Millsp.] leaves. The operating parameters were optimised using single-factor experiment and central composite design combined with response surface methodology. Well-fitting models for the extraction of CSA and PI were successfully established. From the economic perspective, the selected operating parameters were: extraction pressure −0.075 MPa, extraction temperature 45 °C, material size 40 mesh, ethanol concentration 80%, extraction time 30 min, liquid/solid ratio 30:1 and 4 extraction cyc…

AntioxidantChromatographyABTSCentral composite designbiologyChemistryDPPHmedicine.medical_treatmentExtraction (chemistry)General Medicinebiology.organism_classificationAnalytical ChemistryCajanuschemistry.chemical_compoundBotanymedicineResponse surface methodologyLegumeFood ScienceFood Chemistry
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Ionic liquid gels and antioxidant carbon nanotubes: Hybrid soft materials with improved radical scavenging activity

2019

Hypothesis: Performances of materials are frequently affected by the action of radicals that can induce their degradation. To overcome the above issue, natural antioxidants (AOs) can be added during manufacturing. Considering the high instability of AOs, they have been adsorbed on carbon nanomaterials surface. However, the inclusion of functionalized carbon nanomaterials into gel matrix could enhance the antioxidant efficiency and represent an easy way to disperse and handle the active species.Experiments: Carboxypropyl functionalized carbon nanotubes (f-CNT), pure or with physically adsorbed alpha-tocopherol (f-CNT-VE) and quercetin (f-CNT-Q), were incorporated in some ionic liquid gels (I…

AntioxidantRadicalmedicine.medical_treatmentNatural antioxidants02 engineering and technologyCarbon nanotubeIonic liquid010402 general chemistry01 natural sciencesCarbon nanotubelaw.inventionNatural antioxidantBiomaterialschemistry.chemical_compoundColloid and Surface ChemistryAdsorptionRheologylawmedicineThin filmChemistrySettore CHIM/06 - Chimica Organica021001 nanoscience & nanotechnology0104 chemical sciencesSurfaces Coatings and FilmsElectronic Optical and Magnetic MaterialsCoating materialChemical engineeringIonic liquidHybrid ionic liquid gelDegradation (geology)0210 nano-technologyJournal of Colloid and Interface Science
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Stevia rebaudiana Bertoni as a natural antioxidant/antimicrobial for high pressure processed fruit extract: Processing parameter optimization

2013

Response surface methodology was used to evaluate the optimal high pressure processing treatment (300-500 MPa, 5-15 min) combined with Stevia rebaudiana (Stevia) addition (0-2.5% (w/v)) to guarantee food safety while maintaining maximum retention of nutritional properties. A fruit extract matrix was selected and Listeria monocytogenes inactivation was followed from the food safety point of view while polyphenoloxidase (PPO) and peroxidase (POD) activities, total phenolic content (TPC) and antioxidant capacity (TEAC and ORAC) were studied from the food quality point of view. A combination of treatments achieved higher levels of inactivation of L. monocytogenes and of the oxidative enzymes, s…

Antioxidantmedicine.medical_treatmentAntioxidantsAnalytical ChemistryPascalizationFood PreservationOxidative enzymeBotanymedicineSteviaFood scienceResponse surface methodologyPeroxidasePlant ProteinsMangiferabiologyCaricaPlant ExtractsChemistryGeneral Medicinebiology.organism_classificationListeria monocytogenesSteviaAnti-Bacterial AgentsStevia rebaudianaPoint of deliveryFruitFood PreservativesFood qualityCatechol OxidaseCitrus sinensisFood ScienceFood Chemistry
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Solvent-free microwave-assisted extraction of polyphenols from olive tree leaves: Antioxidant and antimicrobial properties

2017

International audience; Response surface methodology (RSM) and artificial neural networks (ANN) were evaluated and compared in order to decide which method was the most appropriate to predict and optimize total phenolic content (TPC) and oleuropein yields in olive tree leaf (Olea europaea) extracts, obtained after solvent-free microwave- assisted extraction (SFMAE). The SFMAE processing conditions were: microwave irradiation power 250-350 W, extraction time 2-3 min, and the amount of sample 5-10 g. Furthermore, the antioxidant and antimicrobial activities of the olive leaf extracts, obtained under optimal extraction conditions, were assessed by several in vitro assays. ANN had better predic…

Antioxidantmedicine.medical_treatment[SDV]Life Sciences [q-bio]Pharmaceutical ScienceAntioxidantsAnalytical Chemistrychemistry.chemical_compoundDrug Discovery[SDV.IDA]Life Sciences [q-bio]/Food engineeringAntimicrobial; Antioxidant; Oleuropein; Olive leaves; Optimization; Solvent-free microwave extraction; Organic ChemistryOlive leavesMicrowaves04 agricultural and veterinary sciences040401 food scienceAnti-Bacterial AgentsChemistry (miscellaneous)Molecular MedicineAntioxidantAntibacterial activityOptimizationStaphylococcus aureusMicrobial Sensitivity TestsArticlelcsh:QD241-4410404 agricultural biotechnologyOlive leaflcsh:Organic chemistryOleuropeinOleaStaphylococcus epidermidismedicine[SPI.GPROC]Engineering Sciences [physics]/Chemical and Process EngineeringResponse surface methodologyPhysical and Theoretical ChemistryOleuropeinolive leaves; solvent-free microwave extraction; oleuropein; antioxidant; antimicrobial; optimizationChromatographyPlant ExtractsExtraction (chemistry)Organic ChemistryPolyphenolsolive leaves;solvent-free microwave extraction;oleuropein;antioxidant;antimicrobial;optimizationPlant LeaveschemistryPolyphenolYield (chemistry)Solvent-free microwave extractionSolventsAntimicrobialNeural Networks Computer
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Functional Role of Lipoprotein Receptors in Alzheimers Disease

2008

The LDL receptor gene family constitutes a class of structurally closely related cell surface receptors fulfilling diverse functions in different organs, tissues, and cell types. The LDL receptor is the prototype of this family, which also includes the VLDLR, ApoER2/LRP8, LRP1 and LRP1B, as well as Megalin/GP330, SorLA/LR11, LRP5, LRP6 and MEGF7. Recently several lines of evidence have positioned the LDL receptor gene family as one of the key players in Alzheimer's disease (AD) research. Initially this receptor family was of high interest due to its key function in cholesterol/apolipoprotein E (ApoE) uptake, with the epsilon4 allele of ApoE as the strongest genetic risk factor for late-onse…

Apolipoprotein EAmyloid beta-PeptidesbiologyChemistryEndosomeLRP1BLRP1Cell biologyAmyloid beta-Protein PrecursorApolipoproteins ECholesterolReceptors LDLNeurologyAlzheimer DiseaseCell surface receptormental disordersLDL receptorAmyloid precursor proteinbiology.proteinAnimalsHumansNeurology (clinical)ReceptorCurrent Alzheimer Research
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Hölder stability for Serrin’s overdetermined problem

2015

In a bounded domain \(\varOmega \), we consider a positive solution of the problem \(\Delta u+f(u)=0\) in \(\varOmega \), \(u=0\) on \(\partial \varOmega \), where \(f:\mathbb {R}\rightarrow \mathbb {R}\) is a locally Lipschitz continuous function. Under sufficient conditions on \(\varOmega \) (for instance, if \(\varOmega \) is convex), we show that \(\partial \varOmega \) is contained in a spherical annulus of radii \(r_i 0\) and \(\tau \in (0,1]\). Here, \([u_\nu ]_{\partial \varOmega }\) is the Lipschitz seminorm on \(\partial \varOmega \) of the normal derivative of u. This result improves to Holder stability the logarithmic estimate obtained in Aftalion et al. (Adv Differ Equ 4:907–93…

Applied Mathematics010102 general mathematicsMathematical analysisRegular polygonSerrin’s problemFunction (mathematics)Directional derivativeLipschitz continuity01 natural sciencesDomain (mathematical analysis)010101 applied mathematicsOverdetermined systemCombinatoricsBounded functionOverdetermined problemHarnack’s inequalityStationary surface0101 mathematicsStabilityMethod of moving planeHarnack's inequalityMathematicsAnnali di Matematica Pura ed Applicata (1923 -)
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Separation of halloysite/kaolinite mixtures in water controlled by sucrose addition: The influence of the attractive forces on the sedimentation beha…

2022

In this work, we propose an easy strategy for the separation of halloysite/kaolinite mixtures in sucrose aqueous solution. Preliminarily, we investigated the influence of the sucrose addition on the colloidal stability of kaolinite nanoplates and halloysite nanotubes (HNTs) dispersed in water. Dynamic Light Scattering (DLS) measurements revealed that the HNTs aqueous mobility is dependent on the sucrose concentration, while the ζ-potential is negligibly affected by the addition of the carbohydrate in the aqueous solvent. On the other hand, any variations on the surface charge and dynamic behavior of kaolinite were detected in the presence of sucrose. The obtained ζ-potential and DLS results…

Aqueous colloidal stabilityTGAColloid and Surface ChemistryHalloysite nanotubesNanoclaysSeparationSettore CHIM/02 - Chimica FisicaColloids and Surfaces A: Physicochemical and Engineering Aspects
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Thermodynamic and kinetic aspects of the transport of small molecules in dispersed systems

1998

Abstract The knowledge of the behaviour of flavour compounds in complex multiphase systems with regard to their structure is of great importance in flavour perception of foods. The thermodynamic and kinetic behaviour of three selected flavour compounds belonging to a homologous series of esters, e.g. ethyl acetate, ethyl butanoate and ethyl hexanoate, were studied in simple and multiphase systems. The liquid system was composed of water (with or without sodium caseinate) and/or a lipid, Miglyol. First, the properties of the solutes were determined by means of their liquid–liquid partition at equilibrium and their diffusion in aqueous or lipid phases. This first step allowed to reveal the im…

Aqueous solutionChemistryDiffusionFlavourEthyl acetateAqueous two-phase systemEthyl hexanoateSurfaces and InterfacesGeneral MedicineSmall moleculechemistry.chemical_compoundHomologous seriesColloid and Surface ChemistryOrganic chemistryPhysical and Theoretical ChemistryBiotechnologyColloids and Surfaces B: Biointerfaces
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