Search results for "44"

showing 10 items of 1507 documents

New Tripentone Analogs with Antiproliferative Activity

2017

Tripentones represent an interesting class of compounds due to their significant cytotoxicity against different human tumor cells in the submicro-nanomolar range. New tripentone analogs, in which a pyridine moiety replaces the thiophene ring originating the fused azaindole system endowed with anticancer activity viz 8H-thieno[2,3-b]pyrrolizinones, were efficiently synthesized in four steps with fair overall yields (34–57%). All tripentone derivatives were tested in the range of 0.1–100 μM for cytotoxicity against two human tumor cell lines, HCT-116 (human colorectal carcinoma) and MCF-7 (human breast cancer). The most active derivative, with GI50 values of 4.25 µM and 20.73 µM for HCT-116 a…

8H-thieno[23-b]pyrrolizinonePyridinesPharmaceutical SciencetripentonesApoptosis01 natural sciencesAnalytical Chemistrychemistry.chemical_compoundDrug DiscoveryThiopheneCytotoxic T cellCytotoxicityMolecular StructureCell Cycletripentoneproapoptotic agentsCell cycleBiochemistryChemistry (miscellaneous)MCF-7 CellsMolecular Medicineaza-indolesAntineoplastic Agents010402 general chemistryArticlelcsh:QD241-441Structure-Activity Relationshiplcsh:Organic chemistryCell Line TumormedicineHumansantitumor activityPhysical and Theoretical ChemistryMode of actionCell ProliferationDose-Response Relationship Drug010405 organic chemistryOrganic ChemistryCancermedicine.diseaseHCT116 CellsSettore CHIM/08 - Chimica Farmaceutica0104 chemical sciences8H-thieno[23-b]pyrrolizinoneschemistryApoptosisCell cultureaza-indoletripentones; aza-indoles; 8<i>H</i>-thieno[23-<i>b</i>]pyrrolizinones; antitumor activity; proapoptotic agentsCaco-2 CellsMolecules; Volume 22; Issue 11; Pages: 2005
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Reflexiones a propósito de la protección de datos en el escenario global digital: El derecho de daños en la litigiosidad internacional

2021

La circulación internacional de datos personales constituye un sector pujante en la esfera socio-económica. En tales condiciones, ante la existencia de un tratamiento ilícito de aquellos, el agraviado está legitimado para exigir una indemnización por los daños y perjuicios que se hubieran podido originar en el marco transfronterizo. Tal situación plantea dos cuestiones fundamentales: por un lado, determinar el órgano jurisdiccional competente para conocer de un eventual litigio, y, por otro, precisar la Ley aplicable para resolver la controversia suscitada. En la presente investigación cabe destacar las significativas novedades que introduce el Reglamento (UE) 2016/679, de 27 de abril de 20…

:CIENCIAS JURÍDICAS [UNESCO]Derecho aplicablenon-contractual obligations 442 475David La circulación internacional de datos personales constituye un sector pujante en la esfera socio-económica. En tales condicionesresponsabilidad civil extracontractual.2070-8157 22082 Revista Boliviana de Derecho 565487 2021 31 7730065 Reflexiones a propósito de la protección de datos en el escenario global digital El derecho de daños en la litigiosidad internacional Carrizo Aguadodeterminar el órgano jurisdiccional competente para conocer de un eventual litigionormas de competencia judicial internacionalpor otropor un lado [el agraviado está legitimado para exigir una indemnización por los daños y perjuicios que se hubieran podido originar en el marco transfronterizo. Tal situación plantea dos cuestiones fundamentales]el agraviado está legitimado para exigir una indemnización por los daños y perjuicios que se hubieran podido originar en el marco transfronterizo. Tal situación plantea dos cuestiones fundamentales: por un ladoUNESCO::CIENCIAS JURÍDICASde 27 de abril de 2016en lo relativo a su dimensión transnacional y cómo deben ser comprendidas en conjunción con las normas preexistentes de Derecho internacional privado en sede de obligaciones extracontractuales Protección de datos de carácter personaljurisdiction rulesLaw applicableante la existencia de un tratamiento ilícito de aquellosprecisar la Ley aplicable para resolver la controversia suscitada. En la presente investigación cabe destacar las significativas novedades que introduce el Reglamento (UE) 2016/679yData protection
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Análisis jurisprudencial de la legitimación pasiva de las entidades financieras en las reclamaciones realizadas por consumidores derivadas de una com…

2021

Consumers, who acquired real estate through a deed of sale with a mortgage subrogation, have made numerous claims against the financial entities. They request the nullity of the clause that imposes upon them all the expenses cause by the notarial deed. Financial entities have alleged that they do not have the capacity to be sued. Courts decisions have been diverse.

:CIENCIAS JURÍDICAS [UNESCO]Roberto Consumersmortgage subrogationcapacity to be sued 966 979who acquired real estate through a deed of sale with a mortgage subrogationunfair termshave made numerous claims against the financial entities. They request the nullity of the clause that imposes upon them all the expenses cause by the notarial deed. Financial entities have alleged that they do not have the capacity to be sued. Courts decisions have been diverse. ConsumidoresUNESCO::CIENCIAS JURÍDICASlegitimación pasiva2070-8157 22082 Revista Boliviana de Derecho 584568 2021 32 8055244 Análisis jurisprudencial de la legitimación pasiva de las entidades financieras en las reclamaciones realizadas por consumidores derivadas de una compraventa con subrogación hipotecaria especial referencia a la de nulidad de la cláusula de gastos. Martín LópezConsumerssubrogación hipotecariacláusulas abusivas
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Gestación subrogada y dignidad de la mujer

2018

The situation of the surrogate pregnancy in Spain demands action by our legislators and / or our public authorities. The reason is that the current legal system in which there is a ban of the surrogacy contract is not being attended. In this issue an analysis of the situation in Spain and in other countries is made, to conclude from the right to the dignity of women, that possible actions could be taken to adapt the reality to the legal system.

:CIENCIAS JURÍDICAS [UNESCO]the right to the dignity of womenfiliation. 10 44dignidad de la mujerUNESCO::CIENCIAS JURÍDICASthat possible actions could be taken to adapt the reality to the legal system. Gestación por sustituciónSurrogate pregnancyMaría Dolores The situation of the surrogate pregnancy in Spain demands action by our legislators and / or our public authorities. The reason is that the current legal system in which there is a ban of the surrogacy contract is not being attended. In this issue an analysis of the situation in Spain and in other countries is madeto conclude from the right to the dignity of women2386-4567 22661 Actualidad jurídica iberoamericana 502169 2018 9 6653319 Gestación subrogada y dignidad de la mujer Cervilla Garzónfiliación
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Un cuento de robots : La hija cibernética de descartes

2021

French philosopher René Descartes is today valued as a forerunner of the studies of human mind, artificial intelligence and robotic systems. Throughout his work there are large references to automata and the possibility of artificial life, as well as an assessment of the differences between rational behavior of human beings and the purely mechanical of animals and automata. In addition to these references, there is a fable about the creation by the philosopher of an automaton that replicated his deceased daughter Francine, a story that is well known among the French and Anglo-Saxon specialists, but not so much in the Spanish ones, which is what settles this short work

:CIENCIAS JURÍDICAS [UNESCO]which is what settles this short work René DescartesFrancine Descartesinteligencia artificialautómatasautomataas well as an assessment of the differences between rational behavior of human beings and the purely mechanical of animals and automata. In addition to these referencesthere is a fable about the creation by the philosopher of an automaton that replicated his deceased daughter Francinebut not so much in the Spanish onesartificial intelligence2070-8157 22082 Revista Boliviana de Derecho 565487 2021 31 7730064 Un cuento de robots La hija cibernética de descartes Lacruz MantecónMiguel L. French philosopher René Descartes is today valued as a forerunner of the studies of human mindartificial intelligence and robotic systems. Throughout his work there are large references to automata and the possibility of artificial lifea story that is well known among the French and Anglo-Saxon specialistsRené DescartesUNESCO::CIENCIAS JURÍDICASrobots. 422 441robots
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Characterizing the initial conditions of heavy-ion collisions at the LHC with mean transverse momentum and anisotropic flow correlations

2022

Physics letters / B 834, 137393 (2022). doi:10.1016/j.physletb.2022.137393

:Kjerne- og elementærpartikkelfysikk: 431 [VDP]heavy ion: scatteringNuclear Experiment; Nuclear Experiment; High Energy Physics - Experimenthiukkasfysiikkanucl-exElliptic-flowHigh Energy Physics - ExperimentHigh Energy Physics - Experiment (hep-ex)ALICE5020: 5440 GeV-cms/nucleon[PHYS.HEXP]Physics [physics]/High Energy Physics - Experiment [hep-ex]Quark-gluon plasma elliptic flow Pb collisionsNuclear Experiment (nucl-ex)Nuclear ExperimentViscosityelliptic flowQuark-gluon plasmaheavy ion: scattering ; flow: anisotropy ; gluon: saturation ; correlation: higher-order ; initial state ; transverse momentum ; ALICE ; boundary condition ; CERN LHC Coll ; hydrodynamics ; color glass condensate ; numerical calculations ; experimental results ; 5020: 5440 GeV-cms/nucleonflow: anisotropyHigh Energy Heavy Ion Collisions:Nuclear and elementary particle physics: 431 [VDP]CERN LHC CollPerspectiveydinfysiikkahigher-order [correlation]Particle Physics - Experimentanisotropy [flow]Nuclear and High Energy PhysicsEvolutionFOS: Physical sciencesPb collisionstransverse momentum[PHYS.NEXP]Physics [physics]/Nuclear Experiment [nucl-ex]114 Physical sciences530scattering [heavy ion]Nuclear Physics - Experimentddc:530saturation [gluon]numerical calculationsinitial statehep-exkvarkki-gluoniplasmaheavy-ion collisions nuclear physics correlations LHCcorrelation: higher-orderboundary condition5440 GeV-cms/nucleon [5020]hydrodynamicsgluon: saturationcolor glass condensateexperimental results
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Análisis coste-utilidad de la triple terapia con telaprevir en pacientes con hepatitis C no tratados previamente

2014

Introducción: En España, con una prevalencia del 2,5%, la hepatitis C (VHC) se asocia a una elevada morbi-mortalidad. El tratamiento combinado de telaprevir y peginterferon/ribavirina ([T/PR]) es eficaz en pacientes con VHC-G1. El objetivo primario de este estudio fue evaluar la relación coste-utilidad (RCUI) de [T/PR] versus peginterferon alfa 2a/ribavirina ([PR]) en pacientes naïve VHC-G1, según el grado de fibrosis y bajo la perspectiva del sistema sanitario español. Metodología: La eficacia y la incidencia de efectos adversos (EAs) se obtuvieron de los estudios ADVANCE y OPTIMIZE. La estimación de los costes de monitorización, de manejo de EAs y de la enfermedad por estados de salud (€,…

; Genotype 1lcsh:RRibavirinalcsh:Medicinelcsh:RS1-441Genotype 1Hepatitis CTelaprevirGenotipo 1lcsh:Pharmacy and materia medicaCoste-utilidadCost-effectivenessPeginterferon alfa 2aRibavirinehealth care economics and organizationsFarmacia Hospitalaria
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Chemical Composition and antimicrobial activity of the essential oils from two species of Thimus growing wild in southern Italy

2009

The volatile constituents of the aerial parts of two samples of Thymus longicaulis C. Presl, collected in Campania and in Sicily, and two samples of Thymus pulegioides L. from the same regions, were extracted by hydrodistillation and analyzed. Considering the four oils together, seventy-eight different compounds were identified: 57 for Thymus longicaulis from Sicily (91.1% of the total oil), 40 for Thymus longicaulis from Campania (91.5% of the oil), 39 for Thymus pulegioides from Sicily (92.5% of the oil) and 29 for Thymus pulegioides from Campania (90.1% of the oil). The composition of the oils is different, although the most abundant components are identical in T. pulegioides. The essent…

<em>Thymus longicaulis</em> C. Presl; <em>Thymus pulegioides </em>L.; essential oil composition; thymol; geraniol; antibacterial activityThymus pulegioidesPharmaceutical ScienceMicrobial Sensitivity TestsArticleAnalytical Chemistrylcsh:QD241-441Thymus Plantchemistry.chemical_compoundlcsh:Organic chemistryantibacterial activitythymolDrug DiscoveryBotanyOils VolatilePlant OilsThymus PlantSettore BIO/15 - Biologia FarmaceuticaPhysical and Theoretical ChemistrygeraniolThymolChemical compositionessential oil compositionThymus longicaulisbiologyBacteriaThymus pulegioides L.Organic ChemistrySettore CHIM/06 - Chimica Organicabiology.organism_classificationAntimicrobialAnti-Bacterial AgentschemistryItalyantimicrobial activity essential oils Thimus longicaulis Thimus pulegioidesChemistry (miscellaneous)Molecular MedicineComposition (visual arts)Thymus longicaulis C. PreslGeraniol
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Antitumor Mechanism of the Essential Oils from Two Succulent Plants in Multidrug Resistance Leukemia Cell

2019

Drug resistance remains a major challenge in the treatment of cancer. The multiplicity of the drug resistance determinants raises the question about the optimal strategies to deal with them. Essential oils showed to inhibit the growth of different tumor cell types. Essential oils contain several chemical classes of compounds whose heterogeneity of active moieties can help prevent the development of drug resistance. In the present paper, we analyzed, by gas chromatography-mass spectrometry the chemical composition of the essential oil of the leaves of Kalanchoe beharensis obtained by hydrodistillation and compared the chemical composition of its essential oil with that of Cyphostemma juttae.…

<i>Kalanchoe beharensis</i>Celllcsh:Medicinelcsh:RS1-441Pharmaceutical ScienceKalanchoe beharensiDrug resistanceArticleessential oilNF-κBlaw.inventionlcsh:Pharmacy and materia medica03 medical and health sciences0302 clinical medicineKalanchoe beharensislawmultidrug resistanceCyphostemma juttaeDrug DiscoverymedicineNF-kappaBSettore BIO/15 - Biologia FarmaceuticaEssential oilacute myeloid leukemia cell030304 developmental biology0303 health sciences<i>Cyphostemma juttae</i>biologylcsh:RMyeloid leukemiaCyphostemma juttaebiology.organism_classificationmedicine.diseaseMultiple drug resistanceLeukemiamedicine.anatomical_structureBiochemistry030220 oncology & carcinogenesisSettore BIO/03 - Botanica Ambientale E ApplicataSettore BIO/14 - FarmacologiaMolecular MedicineKalanchoe beharensisPharmaceuticals
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Feasibility of a Responsibility-Based Leadership Training Program for Novice Physical Activity Instructors

2021

Most coaches and instructors would like to teach more than just sport skills to their athletes and children. However, to promote athletes' or children's holistic development and teach them to take responsibility and lead, requires the coaches and instructors to first master the skills themselves. Therefore, feasible, high quality leadership training programs where coaches and physical activity instructors are taught to teach and share leadership are needed. The aim of the current study was to evaluate the feasibility of a leadership training program to optimize it and to determine whether to proceed with its evaluation. In the leadership training program, eight Finnish novice physical activ…

AFTER-SCHOOL PROGRAMliikunnanohjaajat515 PsychologySOCIAL-RESPONSIBILITYvastuullisuusIMPLEMENTATION FIDELITYphysical activitykoulutusohjelmatBasic Behavioral and Social ScienceSPORTshared leadershipClinical ResearchBehavioral and Social ScienceADOLESCENTSPsychologyEDUCATION TEACHERSteaching personal and social responsibility modeljohtajuusOriginal Researchpositive youth developmentleadership trainingRANDOMIZATIONSHARED LEADERSHIPMODEL5144 Social psychologyammatillinen kehitys5141 Sociology516 Educational sciencesCognitive Sciencesnovice instructorPOSITIVE YOUTH DEVELOPMENTfeasibility
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