Search results for "ACEA"

showing 10 items of 2814 documents

New sesquiterpene lactones and acetylenes from chrysanthemum lavandulifolium

1990

Abstract The aerial parts of Chrysanthemum lavandulifolium Mak. (Asteraceae) yielded three new acetylenes of the spiroacetal type 1-3, as well as two new germacranolides 4-5 and several known lactones.

chemistry.chemical_classificationbiologyStereochemistryOrganic ChemistryAsteraceaeSesquiterpenebiology.organism_classificationBiochemistryTerpenechemistry.chemical_compoundchemistryDrug DiscoveryOrganic chemistryLactoneTetrahedron
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Rollimembrin, a novel acetogenin inhibitor of mammalian mitochondrial complex I

1997

Abstract Rollimembrin (3), is a new adjacent bis-tetrahydrofuranic acetogenin with a scarce relative configuration, threo/cis/threo/cis/erythro, isolated from Rollinia membranacea seeds. The mechanism of cytotoxic activity, determined by NADH-oxidase experiments, establish that rollimembrin (3) is the most potent inhibitor of mammalian mitochondrial complex I.

chemistry.chemical_classificationbiologyStereochemistryOrganic ChemistryClinical BiochemistryAbsolute configurationPharmaceutical ScienceBiological activitybiology.organism_classificationBiochemistryIn vitrochemistry.chemical_compoundEnzymechemistryAnnonaceaeEnzyme inhibitorDrug DiscoveryAcetogeninbiology.proteinMolecular MedicineMolecular BiologyLactoneBioorganic & Medicinal Chemistry Letters
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Triterpene Saponins from Four Species of the Polygalaceae Family

2005

Twelve triterpene saponins were isolated by successive MPLC over silica gel from four species of Polygalaceae: From Polygala ruwenzoriensis, five new saponins 1–5 of which 1–4 as two pairs of (E)/(Z)-isomers, together with the four known compounds tenuifoline, (E)- and (Z)-senegasaponin b, (E)- and (Z)-senegin II, and polygalasaponin XXVIII, from the genus Carpolobia, one new saponin 6 from C. alba and the known arilloside (11) from C. lutea, and another new triterpene glycoside 7 from Polygala arenaria. Their structures were established mainly by 600-MHz 2D-NMR techniques (1H,1H-COSY, TOCSY, NOESY, HSQC, HMBC) as 3-O-(β-D-glucopyranosyl)presenegenin 28-{O-α-L-arabinopyranosyl-(1  4)-O-β-D-…

chemistry.chemical_classificationbiologyStereochemistryOrganic ChemistrySaponinGlycosidePolygalasaponin XXVIIIbiology.organism_classificationBiochemistryPresenegeninCatalysisPolygalaInorganic ChemistryCarpolobiaTriterpenechemistryDrug DiscoveryPolygalaceaePhysical and Theoretical ChemistryHelvetica Chimica Acta
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LC-NMR applied to the characterisation of cardiac glycosides from three micropropagatedIsoplexisspecies

2002

Species of the genus Isoplexis are of particular interest with respect to the biochemical pathway leading to the cardenolides. It is important to determine whether or not 5β-configured compounds, typically produced by Digitalis species and used in medicine, are present together with their respective α-isomers in Isoplexis spp. Structure elucidation by LC-NMR of the products isolated from in vitro regenerated Isoplexis canariensis, I. chalcantha and I. isabelliana was carried out, and similarities were observed among the products of the three species, including the presence of digitoxigenin-type cardenolides in I. canariensis and xysmalogenin and canarigenin derivatives in I. chalcantha neve…

chemistry.chemical_classificationbiologyStereochemistryScrophulariaceaePregnaneGlycosideDigitalisPlant ScienceGeneral Medicinebiology.organism_classificationBiochemistryAnalytical ChemistryIsoplexis canariensisCanarigeninchemistry.chemical_compoundComplementary and alternative medicinechemistryGenusDrug DiscoveryIsoplexisBotanyMolecular MedicineFood SciencePhytochemical Analysis
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Metabolic cross-talk between pathways of terpenoid backbone biosynthesis in spike lavender

2015

Abstract The metabolic cross-talk between the mevalonate (MVA) and the methylerythritol phosphate (MEP) pathways in developing spike lavender ( Lavandula latifolia Med) was analyzed using specific inhibitors and on the basis of 13 C-labeling experiments. The presence of mevinolin (MEV), an inhibitor of the MVA pathway, at concentrations higher than 0.5 μM significantly reduced plant development, but not the synthesis of chlorophylls and carotenoids. On the other hand, fosmidomycin (FSM), an inhibitor of the MEP pathway, at concentrations higher than 20 μM blocked the synthesis of chlorophyll, carotenoids and essential oils, and significantly reduced stem development. Notably, 1.2 mM MVA cou…

chemistry.chemical_classificationbiologyTerpenesPhysiologyLavandula latifoliaPlant ScienceReductasebiology.organism_classificationFosmidomycinchemistry.chemical_compoundCytosolLavandulaEnzymeBiosynthesischemistryBiochemistryHydroxymethylglutaryl-CoA-Reductases NADP-dependentGeneticsmedicineLamiaceaeCarotenoidPlant ShootsPlant Proteinsmedicine.drugPlant Physiology and Biochemistry
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Exopolysaccharides favor the survival of Erwinia amylovora under copper stress through different strategies.

2010

Erwinia amylovora causes fire blight, a destructive disease of rosaceous plants very difficult to control. We demonstrated that copper, employed to control plant diseases, induces the "viable-but-nonculturable" (VBNC) state in E. amylovora. Moreover, it was previously reported that copper increases production of its main exopolysaccharide (EPS), amylovoran. In this work, the copper-complexing ability of amylovoran and levan, other major EPS of E. amylovora, was demonstrated. Following this, EPS-deficient mutants were used to determine the role of these EPSs in survival of this bacterium in AB mineral medium with copper, compared to their wild type strain and AB without copper. Tot…

chemistry.chemical_classificationbiologyVirulenceMutantPolysaccharides BacterialVirulenceGeneral MedicineErwiniaPolysaccharidebiology.organism_classificationMicrobiologyEnterobacteriaceaeMicrobiologyAnti-Bacterial AgentsFructansFructanchemistryGenes BacterialFire blightMutationErwinia amylovoraMolecular BiologyBacteriaCopperPlant DiseasesResearch in microbiology
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Molecular characterization of the phenolic acid metabolism in the lactic acid bacteria Lactobacillus plantarum

2001

The lactic acid bacteria Lactobacillus plantarumdisplays substrate-inducible decar- boxylase activities on p-coumaric, caffeic and ferulic acids. Purification of the p-coumaric acid decarboxylase (PDC) was performed. Sequence of the N-terminal part of the PDC led to the cloning of the corresponding pdc gene. Expression of this gene in Escherichia colirevealed that PDC displayed a weak activity on ferulic acid, detectable in vitro in the presence of ammonium sulfate. Transcrip- tional studies of this gene in L. plantarum demonstrated that the pdc transcription is phenolic acid- dependent. A mutant deficient in the PDC activity, designated LPD1, was constructed to study phe- nolic acid altern…

chemistry.chemical_classificationbiologyhemic and immune systemsmacromolecular substancesLactobacillaceaePhenolic acidbiology.organism_classificationLactic acidFerulic acidchemistry.chemical_compoundEnzymechemistryBiochemistryLactobacillusLactobacillus plantarumBacteriaFood ScienceLe Lait
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Steroidal saponins and flavan-3-ol glycosides from Dioscorea villosa

2006

chemistry.chemical_classificationchemistrybiologyDioscorea villosaDioscoreaceaeBotanyGlycosideFlavan-3-olbiology.organism_classificationBiochemistryEcology Evolution Behavior and SystematicsBiochemical Systematics and Ecology
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A New Flavonol Glycoside from Tristemma hirtum (Melastomataceae)

2018

chemistry.chemical_classificationchemistrybiologyTraditional medicineMelastomataceaeOrganic ChemistryDrug DiscoveryGlycosidebiology.organism_classificationNatural Product Sciences
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Triterpene saponins from Schefflera abyssinica

2006

chemistry.chemical_classificationchemistry.chemical_compoundHederageninbiologyTriterpenechemistryTraditional medicineAraliaceaebiology.organism_classificationBiochemistryOleanolic acidEcology Evolution Behavior and SystematicsScheffleraBiochemical Systematics and Ecology
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