Search results for "AGENTS"

showing 10 items of 7330 documents

Targeting the vascular endothelial growth factor system to prevent ovarian hyperstimulation syndrome

2008

BACKGROUND: Ovarian hyperstimulation syndrome (OHSS) typically occurs when ovaries are primed with FSH/ LH and subsequently exposed to hCG. The ultimate pathophysiological step underlying this clinical picture is increased vascular permeability (VP). METHODS: A search of the literature was carried out using PubMed and the authors’ files. RESULTS: In rodents and humans, the expression of vascular endothelial growth factor (VEGF) and VEGF receptor 2 (VEGFR-2) mRNA increases during ovarian stimulation. With the administration of hCG, the expression of each rises to a maximum. Expression of VEGF/VEGFR-2 mRNAs correlates with enhanced VP, with both peaking 48 h following an injection of hCG. Imm…

endocrine systemmedicine.medical_specialtyCabergolineIndolesOvarian hyperstimulation syndromeVascular permeabilityBiologyChorionic GonadotropinDopamine agonistCapillary PermeabilityOvarian Hyperstimulation Syndromechemistry.chemical_compoundInternal medicineCabergolinemedicineAnimalsHumansPyrrolesErgolinesPhosphorylationCells CulturedClinical Trials as TopicEstradiolVascular Endothelial Growth FactorsObstetrics and GynecologyEstrogensKinase insert domain receptormedicine.diseaseRatsVascular endothelial growth factorActin CytoskeletonVascular endothelial growth factor Amedicine.anatomical_structureEndocrinologyReproductive MedicinechemistryDopamine AgonistsReproductive Control AgentsFemaleCorpus luteumSignal Transductionmedicine.drugHuman Reproduction Update
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Expression and regulation of mPer1 in immortalized GnRH neurons.

2003

Hypothalamic GnRH (gonadotropin-releasing hormone) neurons play a critical role in the initiation and maintenance of reproduction competence. Using the mouse GnRH neuronal cell line, GT1-7, we have characterized the expression of the gene mPer1, a recognized key element of the mammalian circadian clockwork. Both mPer1 transcripts and the 136 kDa mPER1 gene product could be detected in these cells. Immunocytochemical analysis also confirmed expression of mPER1 both in vitro and in vivo in GnRH neurons. Activation of cyclic AMP signalling pathways in vitro elevated GnRH secretion as well as mPer1 expression and nuclear mPER1 immunoreactivity. As mPER1 is known to feedback on transcriptional a…

endocrine systemmedicine.medical_specialtyCellImmunoblottingCell Cycle ProteinsBiologyGene productGonadotropin-Releasing HormoneMiceInternal medicineGene expressionmedicineAnimalsGeneCells CulturedRegulation of gene expressionNeuronsReverse Transcriptase Polymerase Chain ReactionGeneral NeuroscienceColforsinNuclear ProteinsPeriod Circadian ProteinsImmunohistochemistryPreoptic AreaIn vitromedicine.anatomical_structureEndocrinologyNeuroprotective AgentsGene Expression RegulationCell cultureHypothalamushormones hormone substitutes and hormone antagonistsVasoactive Intestinal PeptideNeuroreport
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Effects of sulphonylureas on spontaneous motility and induced contractions in rat isolated uterus

1986

Abstract To clarify the action of sulphonylureas on calcium, the effect of tolbutamide and ghbenclamide has been investigated on a Ca-dependent process, the contractile activity of uterine smooth muscle. Both sulphonylureas antagonized the contractions evoked by CaCl2 in a non-competitive manner when the uterus was maintained in depolarizing solution and did not affect the spontaneous contractions of rat uterus. The capacity of tolbutamide and ghbenclamide to relax vanadate-induced contraction of rat uterus in Ca-free medium suggests that sulphonylureas may have an intracellular site of action related to cytosolic free Ca levels, or effect a reduction in Ca action.

endocrine systemmedicine.medical_specialtyContraction (grammar)TolbutamideUterusPharmaceutical ScienceMotilitychemistry.chemical_elementIn Vitro TechniquesBiologyCalciumGlibenclamideContractilityUterine ContractionTolbutamideInternal medicineGlyburidemedicineAnimalsHypoglycemic AgentsPharmacologyRats Inbred StrainsVanadiumRatsSulfonylurea CompoundsEndocrinologymedicine.anatomical_structureMechanism of actionchemistryCalciumFemaleVanadatesmedicine.symptommedicine.drugJournal of Pharmacy and Pharmacology
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Memory for time intervals is impaired in left hemi-Parkinson patients.

2004

The basal ganglia have been proposed as one of the neural correlates of timekeeping functions. Both encoding and memory retrieval components for time perception are impaired in Parkinson's disease (PD). The aim of our study was to investigate in hemi-Parkinsonian patients the existence of a specific alteration in memory for time depending on the affected side, to better understand the contribution of the left or right basal ganglia circuits in different components of time perception. Right and left hemi-PD patients performed a time reproduction task in which they were required to reproduce in the same session short (5 s) and long (15 s) time intervals, in off- and on-therapy condition. Whil…

endocrine systemmedicine.medical_specialtyParkinson's diseaseTime FactorsParkinson's diseaseCognitive NeuroscienceHemi-Parkinsonian patientsTime perceptionTime perception Parkinson's disease Memory Migration effect Cognitive functions Hemi-Parkinsonian patients Basal gangliaExperimental and Cognitive PsychologyAudiologyFunctional LateralityNOAntiparkinson AgentsLevodopaBehavioral NeuroscienceMemoryBasal gangliaTask Performance and AnalysismedicineHumansLevodopa; Analysis of Variance; Parkinson Disease; Humans; Task Performance and Analysis; Antiparkinson Agents; Aged; Middle Aged; Time Factors; Memory Disorders; Functional Laterality; FemaleMemory disorderAgedNeural correlates of consciousnessAnalysis of VarianceMemory DisordersSettore M-PSI/02 - Psicobiologia E Psicologia FisiologicaMemoriaCognitive disorderCognitionParkinson DiseaseBasal ganglia; Cognitive functions; Hemi-Parkinsonian patients; Memory; Migration effect; Parkinson's disease; Time perception;Time perceptionMiddle Agedmedicine.diseaseCognitive functionsBasal gangliaSettore MED/26 - NeurologiaMigration effectFemalePsychologyNeuroscienceNeuropsychologia
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Energy harvesting for mobile agents supporting wireless sensor networks

2022

Abstract Wireless sensor networks (WSNs) have been deployed widely in many different application including in civil and military fields. The sensing data from the networks is very diverse and may cost huge energy consumption for transmission. Hence, mobile sensors with high capacity are deployed to support the static sensors dealing with longer range communicating distances and also supplying power wirelessly the sensors if possible. This paper focuses on an energy harvesting (EH) design for either mobile agents or sensor nodes in WSNs. A hybrid EH system can harvest energy from ambient environment around to power the mobile sensors and static sensors. In addition, these mobile sensors and …

energy harvestingRenewable Energy Sustainability and the EnvironmentElectrochemistryEnergy Engineering and Power Technologysensor nodeshybrid RF-solar energyElectrical and Electronic Engineeringmobile agentswireless sensor networks
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Les épouses comme agents de rupture dans l’entreprise familiale ?

2014

International audience

entreprise familiale[SHS.SOCIO]Humanities and Social Sciences/Sociology[SHS.SOCIO] Humanities and Social Sciences/Sociologyépousesrupture[ SHS.SOCIO ] Humanities and Social Sciences/SociologyComputingMilieux_MISCELLANEOUSagents
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Peripheral Alterations in Cytokine and Chemokine Levels After Antidepressant Drug Treatment for Major Depressive Disorder: Systematic Review and Meta…

2017

Mounting evidence suggests that aberrations in immune-inflammatory pathways contribute to the pathophysiology of major depressive disorder (MDD), and individuals with MDD may have elevated levels of predominantly pro-inflammatory cytokines and C-reactive protein. In addition, previous meta-analyses suggest that antidepressant drug treatment may decrease peripheral levels of interleukin-1 beta (IL-1β) and IL-6. Recently, several new studies examining the effect of antidepressants on these cytokines have been published, and so we performed an updated meta-analysis of studies that measured peripheral levels of cytokines and chemokines during antidepressant treatment in patients with MDD. The P…

epressionChemokinemedicine.drug_classmedicine.medical_treatmentNeuroscience (miscellaneous)InflammationAntidepressantPharmacology03 medical and health sciencesCellular and Molecular Neuroscience0302 clinical medicinemedicineHumansMeta-analysiCytokineInflammationDepressive Disorder MajorbiologyDepressionbusiness.industrymedicine.diseaseReceptor antagonistAntidepressive Agents030227 psychiatryMeta-analysisCytokineTreatment OutcomeAntidepressant; Chemokines; Cytokines; Depression; Inflammation; Meta-analysis; Cellular and Molecular NeuroscienceNeurologyChemokineMeta-analysisbiology.proteinCytokinesMajor depressive disorderAntidepressantTumor necrosis factor alphamedicine.symptomChemokinesbusiness030217 neurology & neurosurgeryMolecular neurobiology
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Synthesis and Antiproliferative Activity of 2,5-bis(3′-Indolyl)pyrroles, Analogues of the Marine Alkaloid Nortopsentin

2013

2,5-bis(3′-Indolyl)pyrroles, analogues of the marine alkaloid nortopsentin, were conveniently prepared through a three step procedure in good overall yields. Derivatives 1a and 1b exhibited concentration-dependent antitumor activity towards a panel of 42 human tumor cell lines with mean IC50 values of 1.54 μM and 0.67 μM, respectively. Investigating human tumor xenografts in an ex-vivo clonogenic assay revealed selective antitumor activity, whereas sensitive tumor models were scattered among various tumor histotypes.

ex-vivo xenograftsIndolesStereochemistryPharmaceutical ScienceMice NudeAntineoplastic AgentsArticleInhibitory Concentration 50MiceCell Line TumorNeoplasmsDrug Discoverybis-indolyl-pyrroles; nortopsentin analogues; marine alkaloids; antitumor; <i>ex-vivo </i>xenograftsIc50 valuesAnimalsHumansnortopsentin analoguePyrrolesClonogenic assayPharmacology Toxicology and Pharmaceutics (miscellaneous)lcsh:QH301-705.5Tumor Stem Cell AssayMice nudeantitumorAntitumor activityDose-Response Relationship DrugChemistryAlkaloidbis-indolyl-pyrroles; nortopsentin analogues; marine alkaloids; antitumor; ex-vivo xenograftsImidazolesTumor Stem Cell AssaySettore CHIM/08 - Chimica FarmaceuticaXenograft Model Antitumor Assaysbis-indolyl-pyrrolemarine alkaloidHuman tumornortopsentin analogueslcsh:Biology (General)Cell culturebis-indolyl-pyrrolesmarine alkaloidsMarine Drugs
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Cytotoxicity of 91 Kenyan indigenous medicinal plants towards human CCRF-CEM leukemia cells.

2015

Abstract Ethnopharmacological relevance Plants from Kenyan flora are traditionally used against many ailments, including cancer and related diseases. Cancer is characterized as a condition with complex signs and symptoms. Recently there are recommendations that ethnopharmacological usages such as immune and skin disorders, inflammatory, infectious, parasitic and viral diseases should be taken into account when selecting plants that treat cancer. Aim The present study was aimed at investigating the cytotoxicity of a plethora of 145 plant parts from 91 medicinal plants, most of which are used in the management of cancer and related diseases by different communities in Kenya, against CCRF-CEM …

food.ingredientCell Survival01 natural sciences03 medical and health sciences0302 clinical medicinefoodCell Line TumorDrug DiscoveryHumansMedicinal plantsCytotoxicityPharmacologyLeukemiaPlants MedicinalbiologyTraditional medicinePlant ExtractsZanthoxylum gilletiiSolanum aculeastrumBridelia micranthabiology.organism_classificationAntineoplastic Agents PhytogenicKenyaGrowth Inhibitors0104 chemical sciences010404 medicinal & biomolecular chemistry030220 oncology & carcinogenesisHerbvisual_artvisual_art.visual_art_mediumBarkErythrina sacleuxiiJournal of ethnopharmacology
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Fruits and vegetables protect against the genotoxicity of heterocyclic aromatic amines activated by human xenobiotic-metabolizing enzymes expressed i…

2010

Heterocyclic aromatic amines (HAAs) can be formed during the cooking of meat and fish at elevated temperatures and are associated with an increased risk for cancer. On the other hand, epidemiological findings suggest that foods rich in fruits and vegetables can protect against cancer. In the present study three teas, two wines, and the juices of 15 fruits and 11 vegetables were investigated for their protective effect against the genotoxic effects of 2-amino-3-methylimidazo[4,5-f]quinoline (IQ) and 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (PhIP). To closely mimic the enzymatic activation of these HAAs in humans, genetically engineered V79 Chinese hamster fibroblasts were employed tha…

food.ingredientCytochrome P-450 CYP1A2 InhibitorsHealth Toxicology and Mutagenesismedicine.disease_causeGrapefruit juiceCell LineBeveragesCricetulusfoodCherry juiceHeterocyclic CompoundsCricetinaeVegetablesBotanyGeneticsmedicineAnimalsFood scienceAminescomic_books.seriesOrange juicebiologyChemistryCucumber juicefood and beveragesAntimutagenic Agentsbiology.organism_classificationfood.foodEnzyme assayEnzyme ActivationComet assayFruitRed currantcomic_booksbiology.proteinGenotoxicityMutagensMutation Research/Genetic Toxicology and Environmental Mutagenesis
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