Search results for "ALTER"

showing 10 items of 2368 documents

Vascular Activity of (-)-Anonaine, (-)-Roemerine and (-)-Pukateine, Three Natural 6a(R)-1,2-Methylenedioxyaporphines with Different Affinities for α1…

2004

We have studied the mechanism of action of three 6a( R)-1,2-methylenedioxyaporphines as vasorelaxant compounds. The alkaloids assayed showed different affinities for the three human cloned alpha (1)-adrenoceptor (AR) subtypes stably expressed in rat-1 fibroblasts, showing lower affinity for alpha(1B)-AR with regard to the alpha(1A)- or alpha(1D)-subtypes. These three natural compounds are more potent inhibitors of [ (3)H]-prazosin binding than of [ (3)H]-diltiazem binding to rat cerebral cortical membranes. As all these alkaloids inhibited noradrenaline (NA)-induced [ (3)H]-inositol phosphate formation in cerebral cortex and rat tail artery, they may be safely viewed as alpha (1)-AR antagon…

AporphinesPhosphodiesterase InhibitorsStereochemistryPharmaceutical ScienceAorta ThoracicDioxolesBiologyMuscle Smooth VascularAnalytical ChemistryHydroxylationchemistry.chemical_compoundAlkaloidsDrug DiscoverymedicineAnonaineAnimalsHumansAporphineRats WistarBinding sitePukateineCerebral CortexPharmacologyPlants MedicinalVoltage-dependent calcium channelAlkaloidOrganic ChemistryArteriesReceptors Adrenergic alphaIsoquinolinesRatsComplementary and alternative medicineMechanism of actionchemistryMolecular MedicineFemaleCalcium Channelsmedicine.symptomDrugs Chinese HerbalPhytotherapyPlanta Medica
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Educar

2015

El presente artículo describe una experiencia de formación en alternancia en un contexto de educación superior; en concreto, a partir de la iniciativa desarrollada por Florida Universitaria, centro adscrito a la Universidad de Valencia. La formación en alternancia implica alternar el aprendizaje entre períodos desarrollados en el centro educativo y momentos desarrollados en el contexto laboral. El objetivo del presente trabajo es identificar una iniciativa que, de forma empírica, muestre cómo estos periodos impactan en el aprendizaje de competencias de los estudiantes. La metodología que se ha aplicado en la experiencia de formación en alternancia se basa en el aprendizaje basado en problem…

Aprendizaje basado en problemassolución de problemasProblem-based learningUniversity-industry relationsCompetenciasaprendizaje basado en problemasformación alternadaCompetenciesEducationTransferencia del aprendizajeTransfer of learningAlternance trainingProfessional trainingAprenentatgeAprenentatge basat en problemesL7-991Col·laboració empresa-universitatFormació en alternançaCommunicationRelación universidad-empresaaprendizaje profesionalrelación universidad-empresaEducation (General)competenciasHuman-Computer InteractionRelació universitat-empresatransferencia del aprendizajeAprenentatge professional-- FormacióCompetènciesTransferència de l'aprenentatgeAprendizaje profesionalFormación alternada
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Aproximaciones al apócrifo en la órbita de Max Aub : del modelo francés a las últimas manifestaciones peninsulares

2009

En este trabajo se realiza una lectura del mapa de manifestaciones apócrifas alrededor de la figura de Max Aub, escritor que construye un universo de superchería literaria desde sus obras iniciales, abarcando y fusionando diferentes géneros. A partir del contraste con algunos de los textos franceses que leyó, y que supusieron una herencia cultural de gran valor, se esbozará un panorama que incluya tanto a los maestros y predecesores en la práctica apócrifa aubiana, André Gide y Valéry Larbaud fundamentalmente, como a sus sucesores más representativos: los narradores leoneses creadores de Sabino Ordás. Entre unos y otros, se rastrearán los casos peninsulares de mayor trascendencia, con el fi…

ApócrifoLiterature and Literary Theorymax aubFrench literature - Italian literature - Spanish literature - Portuguese literatureApocryphea.o. barnaboothapócrifoMax AubSupercheríaFakeCultural inheritanceAndré WaltersupercheríaSabino Ordásfalso literarioA.O. BarnaboothSubversionOrder (virtue)LiteratureFalso literariolcsh:French literature - Italian literature - Spanish literature - Portuguese literatureA. O. Barnaboothbusiness.industryPhilosophyBiographysabino ordás:CIENCIAS DE LAS ARTES Y LAS LETRAS::Teoría análisis y crítica literarias::Análisis literario [UNESCO]Apocryphe ; Max Aub ; Fake ; Sabino Ordás ; André Walter ; A. O. Barnaboothlcsh:PQ1-3999UNESCO::CIENCIAS DE LAS ARTES Y LAS LETRAS::Teoría análisis y crítica literarias::Análisis literarioPQ1-3999businessHumanitiesApócrifo ; Max Aub ; Superchería ; Sabino Ordás ; André Walter ; A.O. Barnabooth ; Falso literarioandré walter
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A laboratory cave for the study of wall degradation in rock art caves : an implementation in the Vézère area

2013

The aim of this proposal is to present an original approach to the study and preservation of rock art caves. A multidisciplinary study of cave wall alteration will be performed to understand the impact of environmental context on the evolution of wall surfaces. The approach involves the choice of a cave with characteristics similar to painted caves in the studied area (Vézère Valley in Dordogne, France): e.g., cave wall alteration, lithology, morphology, etc. This selected cave is intended to become a laboratory cave, monitored for the acquisition of chemical, physical and biological environmental data on bedrock, air and fluids along with their characteristics. A cave without art or archae…

Archeology[SHS.ARCHEO]Humanities and Social Sciences/Archaeology and PrehistoryLithology[SDV]Life Sciences [q-bio]STAPHYLOCOCCUS-EQUORUMContext (language use)010501 environmental sciences01 natural sciencesArchaeological scienceDatabaseRock art caves03 medical and health sciencesLASCAUX CAVECavepréhistoireComputingMilieux_MISCELLANEOUSLaboratory cave0105 earth and related environmental sciencesCave survey0303 health sciencesgeographygeography.geographical_feature_categoryIDENTIFICATION030306 microbiologyBedrockCave wall alterationsIn situ measurementsArchaeologyPreservationIn situ analysis[SDE]Environmental SciencesRock artSimulationGeology
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A transcription of MS Vatican, Borgh. 129: Gualterus Burlaeus Expositio super libros Politicorum, lib. 1, tract. 1, cap. 1

2021

This is a transcription of the beginning of Walter Burley’s (c. 1275–after 1344) commentary on Aristotle’s Politics (book one, tractate one, chapter one). The transcription reproduces the text of Vatican, MS Borgh. 129, fol. 1r–148v (here fol. 2rb–6va), which has been accessed in a high quality digital reproduction in colour. The commentary has been dated between 1338/39 and 1342. The transcription includes two apparatuses. The first of them is dedicated to references, mainly to Aristotle’s Politics. The other apparatus is for critical notes, and its main function is to reproduce marginalia. The manuscript contains several corrections by another hand (marked here as V1), and since these cor…

Aristotelian traditionPractical philosophykeskiajan filosofiamanuscriptsMedieval manuscriptWalter BurleykäsikirjoituksetAristotelianismkeskiajan latinaMedieval LatinMedieval philosophypaleografiaTranscriptionaristotelismiCommentary on Politicspaleography
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Isolation and characterization of a complement-activating lipid extracted from human atherosclerotic lesions.

1990

The major characteristics of human atherosclerotic lesions are similar to those of a chronic inflammatory reaction, namely fibrosis, mesenchymal cell proliferation, the presence of resident macrophages, and cell necrosis. Atherosclerosis exhibits in addition the feature of lipid (mainly cholesterol) accumulation. The results of the present report demonstrate that a specific cholesterol-containing lipid particle present in human atherosclerotic lesions activates the complement system to completion. Thus, lipid could represent a stimulatory factor for the inflammatory reaction, whose underlying mechanistic basis may be, at least in part, complement activation. The complement-activating lipid …

ArteriosclerosisComplement Pathway AlternativeImmunologyInflammationMuscle Smooth VascularC5-convertasechemistry.chemical_compoundMesenchymal cell proliferationmedicineHumansImmunology and AllergyComplement ActivationImmunoelectrophoresisAortaTriglyceridesCholesterolFatty AcidsComplement System ProteinsArticlesLipidsComplement systemCarotid ArteriesCholesterolchemistryBiochemistryLow-density lipoproteinChromatography GelAlternative complement pathwaylipids (amino acids peptides and proteins)Lipid particlemedicine.symptomJournal of Experimental Medicine
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A Methanol Extract ofBrugmansia arboreaAffects the Reinforcing and Motor Effects of Morphine and Cocaine in Mice

2013

Previous reports have shown that several of the effects of morphine, including the development of tolerance and physical withdrawal symptoms, are reduced by extracts ofBrugmansia arborea(L.) Lagerheim (Solanaceae) (B. arborea). In the present study we evaluate the action of the methanol extract ofB. arborea(7.5–60 mg/kg) on the motor and reinforcing effects of morphine (20 and 40 mg/kg) and cocaine (25 mg/kg) using the conditioned place preference (CPP) procedure. At the doses employed,B. arboreadid not affect motor activity or induce any effect on CPP. The extract partially counteracted morphine-induced motor activity and completely blocked the CPP induced by 20 mg/kg morphine. On the othe…

Article Subjectbiologybusiness.industryDopaminergiclcsh:Other systems of medicinePharmacologylcsh:RZ201-999biology.organism_classificationConditioned place preferenceComplementary and alternative medicineMechanism of actionBrugmansiaMorphinemedicineCholinergicMotor activitymedicine.symptombusinessCocaine abuseResearch Articlemedicine.drugEvidence-Based Complementary and Alternative Medicine
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Safer chemicals using less animals: kick-off of the European ONTOX project

2021

The 3Rs concept, calling for replacement, reduction and refinement of animal experimentation, is receiving increasing attention around the world, and has found its way to legislation, in particular in the European Union. This is aligned by continuing high-level efforts of the European Commission to support development and implementation of 3Rs methods. In this respect, the European project called "ONTOX: ontology-driven and artificial intelligence-based repeated dose toxicity testing of chemicals for next generation risk assessment" was recently initiated with the goal to provide a functional and sustainable solution for advancing human risk assessment of chemicals without the use of animal…

Artificial intelligenceComputer science010501 environmental sciencesOntology (information science)In Vitro TechniquesAnimal Testing AlternativesToxicology01 natural sciencesRisk Assessment3Rs03 medical and health sciencesIn vitroSAFERAdverse Outcome PathwayToxicity TestsEuropean projectmedia_common.cataloged_instanceAnimalsHumansComputer SimulationEuropean UnionAnimal testingEuropean union0105 earth and related environmental sciencesExposure assessmentmedia_common0303 health sciencesOntologyIn silico030311 toxicology3. Good healthVariety (cybernetics)Gene OntologyRisk analysis (engineering)Systemic toxicityONTOXRisk assessment
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All-sky search for continuous gravitational waves from isolated neutron stars using Advanced LIGO O2 data

2019

We present results of an all-sky search for continuous gravitational waves (CWs), which can be produced by fast-spinning neutron stars with an asymmetry around their rotation axis, using data from the second observing run of the Advanced LIGO detectors. We employ three different semi-coherent methods ($\textit{FrequencyHough}$, $\textit{SkyHough}$, and $\textit{Time-Domain $\mathcal{F}$-statistic}$) to search in a gravitational-wave frequency band from 20 to 1922 Hz and a first frequency derivative from $-1\times10^{-8}$ to $2\times10^{-9}$ Hz/s. None of these searches has found clear evidence for a CW signal, so we present upper limits on the gravitational-wave strain amplitude $h_0$ (the …

AstronomyAstrophysicsRotation01 natural sciencesrotationGravitation Cosmology & AstrophysicsGeneral Relativity and Quantum CosmologyPhysics Particles & Fieldscontinuous gravitational waveLIGOneutron starGeneralLiterature_REFERENCE(e.g.dictionariesencyclopediasglossaries)media_commonHigh Energy Astrophysical Phenomena (astro-ph.HE)Settore FIS/01Physicsastro-ph.HEPhysicsPhysical SystemsAmplitudeGeneral relativitygravitational wavesPhysical Sciences[PHYS.GRQC]Physics [physics]/General Relativity and Quantum Cosmology [gr-qc]Gravitational wave detectionAstrophysics - High Energy Astrophysical Phenomenacontinuous gravitational waves; Advanced LIGOcontinuous gravitational wavesasymmetryGravitationNeutron stars & pulsarsGeneral relativityFrequency bandmedia_common.quotation_subjectgr-qcFOS: Physical sciencesalternative theories of gravityGeneral Relativity and Quantum Cosmology (gr-qc)Astronomy & AstrophysicsGravitational waves0103 physical sciencesAdvanced LIGOddc:530Gravitation Cosmology & Astrophysics010306 general physicsgravitational radiation: frequencySTFCgravitational wavesneutron starsGravitational wave sourcesScience & TechnologyGravitational wave sources Gravitational waves Physical Systems Neutron stars and pulsars Gravitational wave detection010308 nuclear & particles physicsGravitational waveRCUKGravitational Wave PhysicsLIGONeutron stars & pulsarsNeutron starSkyNeutron stars and pulsarsDewey Decimal Classification::500 | Naturwissenschaften::530 | Physik[PHYS.ASTR]Physics [physics]/Astrophysics [astro-ph]
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All-sky search for short gravitational-wave bursts in the second Advanced LIGO and Advanced Virgo run

2019

We present the results of a search for short-duration gravitational-wave transients in the data from the second observing run of Advanced LIGO and Advanced Virgo. We search for gravitational-wave transients with a duration of milliseconds to approximately one second in the 32-4096 Hz frequency band with minimal assumptions about the signal properties, thus targeting a wide variety of sources. We also perform a matched-filter search for gravitational-wave transients from cosmic string cusps for which the waveform is well-modeled. The unmodeled search detected gravitational waves from several binary black hole mergers which have been identified by previous analyses. No other significant event…

AstronomyGravitational waves detectionAstrophysicsdetector: network01 natural sciencesSignalGeneral Relativity and Quantum CosmologyPhysics Particles & FieldsGravitational waves detection Stochastic gravitational-wavebinary [black hole]LIGOgravitational waveQCQBmedia_commonastro-ph.HEPhysicsHigh Energy Astrophysical Phenomena (astro-ph.HE)Settore FIS/01Physicsgravitational waves neutron starsgravitational wavesGeneral relativityburst [gravitational radiation]network [detector]Physical Sciences[PHYS.GRQC]Physics [physics]/General Relativity and Quantum Cosmology [gr-qc]direct detection [gravitational radiation]Advanced VirgoAstrophysics - High Energy Astrophysical PhenomenaFrequency bandsensitivity [detector]gr-qcmedia_common.quotation_subjectAstrophysics::High Energy Astrophysical PhenomenaFOS: Physical sciencesalternative theories of gravityGeneral Relativity and Quantum Cosmology (gr-qc)Astronomy & Astrophysicsgravitational radiation: direct detectionemission [gravitational radiation]Binary black holeSettore FIS/05 - Astronomia e Astrofisicabinary: coalescence0103 physical sciencesgravitational radiation: burstAdvanced LIGOWaveformddc:530010306 general physicscosmic stringSTFCScience & Technology010308 nuclear & particles physicsGravitational waveRCUKStochastic gravitational-waveGravitational Wave PhysicsLIGOgravitational radiation detectorgravitational waves; Advanced LIGO; Advanced VirgoCosmic stringdetector: sensitivityVIRGOPhysics and Astronomyblack hole: binarySkygravitational radiation: emissionDewey Decimal Classification::500 | Naturwissenschaften::530 | Physikcoalescence [binary][PHYS.ASTR]Physics [physics]/Astrophysics [astro-ph]
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