Search results for "ANTIOXIDANTS"

showing 10 items of 827 documents

Targeting antioxidants to mitochondria: a potential new therapeutic strategy for cardiovascular diseases.

2007

Mitochondria produce large amounts of free radicals and play an important role in the life and death of a cell. Thus, mitochondrial oxidative damage and dysfunction contribute to a number of cell pathologies that manifest themselves through a range of conditions including ischemia-reperfusion injury, sepsis, diabetes, atherosclerosis and, consequently, cardiovascular diseases (CVD). In fact, endothelial dysfunction, characterized by a loss of nitric oxide (NO) bioactivity, occurs early on in the development of atherosclerosis, and determines future vascular complications. Although the molecular mechanisms responsible for mitochondria-mediated disease processes are not yet clear, oxidative s…

Oxidative phosphorylationPharmacologyMitochondrionBiologymedicine.disease_causeAntioxidantsNitric oxidechemistry.chemical_compoundDrug DiscoverymedicineAnimalsHumansEndothelial dysfunctionInner mitochondrial membranePharmacologychemistry.chemical_classificationReactive oxygen speciesMolecular Structuremedicine.diseaseMitochondriaOxidative StresschemistryCardiovascular DiseasesReactive Oxygen SpeciesReperfusion injuryOxidative stressCurrent pharmaceutical design
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Nutraceutical Value of Pantelleria Capers (Capparis spinosa L.)

2019

Abstract: Unopened flower buds of Capparis spinosa L. (capers), generally used in the Mediterranean area as food flavoring, are known to be a good source of bioactive compounds. The aim of this work was to evaluate the nutraceutical value of salt-fermented capers collected from different areas of Pantelleria Island (Italy), testing their methylglyoxal and glyoxal trapping capacity and antioxidant activity by 2,2-diphenyl-1-picryl hydrazyl (DPPH), [2,2-azinobis(3-ethylben- zothiazoline-6-sulfonic acid)] diammonium salt (ABTS), and oxygen radical absorbance capacity (ORAC) assays. Hydrophilic extracts were also characterized by high-performance liquid chromatography–electrospray ionization/ma…

Oxygen radical absorbance capacity030309 nutrition & dieteticsDPPHFlavonoidGlucosinolatesAntioxidantsCapparis spinosa03 medical and health scienceschemistry.chemical_compound0404 agricultural biotechnologyfoodFlavonolsPhenolsnutraceutical propertiesFood scienceKaempferolsChromatography High Pressure LiquidPantelleria Island caperschemistry.chemical_classificationFlavonoids0303 health sciencesABTSPlant ExtractsCapparis spinosa04 agricultural and veterinary sciencesnutraceutical propertie040401 food sciencefood.foodSettore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeCapparischemistryItalymethylglyoxal and glyoxal trapping capacityhydrophilic extract compositionDietary SupplementsSeedsQuercetinQuercetinKaempferolFood Science
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Multi-Functional Nanogels for Tumor Targeting and Redox-Sensitive Drug and siRNA Delivery

2016

(1) Background: A new family of nanosystems able to discern between normal and tumor cells and to release a therapeutic agent in controlled way were synthetized by e-beam irradiation. This technique permits to obtain biocompatible, sterile, carboxyl-functionalized polyvinylpyrrolidone (PVP-co-acrylic acid) nanogels (NGs); (2) Methods: Here, we performed a targeting strategy based on the recognition of over-expressed proteins on tumor cells, like the folate receptor. The selective targeting was demonstrated by co-culture studies and flow cytometry analysis, using folate conjugated NGs. Moreover, nanoparticles were conjugated to a chemotherapeutic drug or to a pro-apoptotic siRNA through a gl…

PVPPharmaceutical ScienceNanogels02 engineering and technologyPharmacology01 natural sciencesAntioxidantsAnalytical Chemistryfolate-targetingPolyethylene GlycolsNanogelchemistry.chemical_compoundMiceRNA interferenceNeoplasmsDrug DiscoveryFluorescence microscopePolyethyleneimineRNA Small InterferingCytotoxicitymedicine.diagnostic_testPovidone021001 nanoscience & nanotechnologyControlled releaseCell biologyChemistry (miscellaneous)Folate receptorMolecular Medicinee-beamGSH-responsive release0210 nano-technologyOxidation-Reduction010402 general chemistrydoxorubicinArticleFlow cytometryFolic AcidCell Line TumormedicineAnimalsHumansPhysical and Theoretical ChemistryParticle SizeOrganic ChemistryGlutathione0104 chemical scienceschemistryPVP; nanogels; e-beam; folate-targeting; doxorubicin; siRNA; GSH-responsive releasesiRNACancer cellNIH 3T3 CellsNanoparticlesSettore CHIM/07 - Fondamenti Chimici Delle TecnologieFolic Acid TransportersHeLa CellsMolecules
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Effects of pharmacological agents on the lifespan phenotype of Drosophila DJ-1beta mutants.

2010

Mutations in the DJ-1 gene cause autosomal recessive, early-onset Parkinsonism. The DJ-1 protein exerts a protective role against oxidative stress damage, working as a cellular oxidative stress sensor, and it seems to regulate gene expression at different levels. In Drosophila, two DJ-1 orthologs have been identified: DJ-1β and DJ-1β. Several studies have shown that loss of DJ-1β function causes Parkinson's disease (PD)-like phenotypes in flies such as age-dependent locomotor defects, reduced lifespan, and enhanced sensitivity to toxins that induce oxidative stress, like the herbicide paraquat. However, no dopaminergic neurodegeneration is observed. These results suggested that both locomot…

ParaquatDopamineMutantOxidative phosphorylationBiologymedicine.disease_causeAntioxidantsLipid peroxidationchemistry.chemical_compoundParkinsonian DisordersGeneticsmedicineAnimalsGeneticschemistry.chemical_classificationReactive oxygen speciesNeurodegenerationDopaminergicBrainParkinson DiseaseGeneral Medicinemedicine.diseasePhenotypeCell biologyOxidative StressPhenotypechemistryMutationDrosophilaReactive Oxygen SpeciesOxidative stressGene
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Protection of Flupirtine on β-Amyloid-Induced Apoptosis in Neuronal Cells In Vitro: Prevention of Amyloid-Induced Glutathione Depletion

2002

Effective drugs are not available to protect against beta-amyloid peptide (A beta)-induced neurotoxicity. Cortical neurons from rat embryos were treated with the toxic fragment A beta25-35 at 1 microM in the presence or absence of flupirtine, a triaminopyridine, successfully applied clinically as a nonopiate analgesic drug. Five days later 1 microM A beta25-35 caused reduction of cell viability to 31.1%. Preincubation of cells with flupirtine (1 or 5 microg/ml) resulted in a significant increase of the percentage of viable cells (74.6 and 65.4%, respectively). During incubation with A beta25-35 the neurons undergo apoptosis as determined by appearance of the characteristic stepladder-like D…

Pathologymedicine.medical_specialtyCell SurvivalAminopyridinesApoptosisPharmacologymedicine.disease_causeBiochemistryAntioxidantsCellular and Molecular NeurosciencemedicineAnimalsViability assaySenile plaquesRats WistarCerebral CortexNeuronsAmyloid beta-PeptidesChemistryNeurotoxicitymedicine.diseaseGlutathionePeptide FragmentsRatsOxidative StressNeuroprotective AgentsApoptosisCell cultureDNA fragmentationFlupirtineOxidative stressmedicine.drugJournal of Neurochemistry
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Effects of polyphenols and lipids from Pennisetum glaucum grains on T-cell activation: modulation of Ca2+ and ERK1/ERK2 signaling

2015

International audience; BACKGROUND: Pearl millet (PM), i.e., Pennisetum glaucum, is widely grown in Africa and known for its anti-oxidant and anti-hyperlipidemic properties.METHODS: The P. glaucum grains were obtained from the region of Ouled Aïssa (South of Algeria). We assessed the effects of phenolic compounds and lipids, extracted from seeds of P. glaucum, on rat lymphocyte proliferation, activated by phorbol 12-myristate 13-acetate and ionomycin. In order to explore signaling pathway, triggered by these compounds, we assessed interleukin-2 (IL-2) mRNA expression and extracellular signal-regulated kinase-1/2 (ERK1/ERK2) phosphorylation. Finally, we determined increases in free intracell…

PennisetumT-LymphocytesLymphocyte proliferationLymphocyte ActivationAntioxidantsPearl milletchemistry.chemical_compoundExtracellularAnimalsGallic acidExtracellular Signal-Regulated MAP KinasesCell ProliferationHypolipidemic AgentsMitogen-Activated Protein Kinase 1Mitogen-Activated Protein Kinase 3[SDV.MHEP] Life Sciences [q-bio]/Human health and pathologybiologyPlant ExtractsT-cellsPolyphenolsGeneral Medicinebiology.organism_classificationLipidsRatschemistryBiochemistryComplementary and alternative medicinePolyphenolIonomycinSeedsPhorbolPhosphorylationCalciumEdible GrainPennisetum[SDV.MHEP]Life Sciences [q-bio]/Human health and pathologySignal TransductionResearch Article
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Volatile constituents of Dianthus rupicola Biv. from Sicily: activity against microorganisms affecting cellulosic objects.

2014

Dianthus rupicola Biv. (cliffs carnation) is a camephytic, suffruticous, perennial plant growing up to 40 cm high. The plant is widespread in Sicily and neighbouring islands (Egadi, Lampedusa, Lipari) and in some areas of southern Italy. GC and GC-MS analyses of the essential oil distilled from the flowers showed the presence of 66 components. Its composition is characterised by the high content of thymol and carvacrol derivatives. A good antibacterial activity against Bacillus cereus and Bacillussubtilis, both infesting cellulosic historical material, was shown, whereas the antioxidant capacity was determined to be quite poor.

Perennial plantBacillus cereusCaryophyllaceaeBacillusPlant ScienceCarnationFlowersMicrobial Sensitivity TestsBiochemistryAntioxidantsAnalytical Chemistrylaw.inventionchemistry.chemical_compoundlawDianthusBotanyOils VolatilePlant OilsCarvacrolSettore BIO/15 - Biologia FarmaceuticaThymolSicilyEssential oilbiologyfungiOrganic ChemistryDianthus rupicola caryophyllaceae essential oils Thymol and carvacrol derivatives Bacillus ssp.Settore CHIM/06 - Chimica Organicabiology.organism_classificationThymolAnti-Bacterial AgentschemistryMonoterpenesCymenesAntibacterial activityNatural product research
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Comparative Chemical Compositions of Fresh and Stored Vesuvian PDO "Pomodorino Del Piennolo" Tomato and the Ciliegino Variety

2018

The Vesuvian Piennolo cherry tomato (Lycopersicon esculentum Miller) (PdP) is an old and typical variety grown in the Campania region (Italy). PdP is referred to as a long-storage tomato due to its thick and coriaceous skin that allows long post-harvest storage and it has been granted Protected Designation of Origin (PDO) status since 2009. In this study, the chemical composition, focusing in particular on organic acids, antioxidant molecules and volatile compounds, were investigated in PdP and compared to another typical variety in Campania, the Ciliegino tomato (CIL). Chemical characterization was evaluated for both the CIL and PdP varieties during storage in the same environmental condit…

Pharmaceutical Scienceantioxidants fractionsLycopersiconAntioxidantsArticleAnalytical ChemistryNOlcsh:QD241-441storagechemistry.chemical_compound0404 agricultural biotechnologyPomodorino del Piennolo del Vesuvio; antioxidants fractions; chemical composition; cherry tomato; organic acids; storage; volatile organic compoundsCherry tomatolcsh:Organic chemistrySolanum lycopersicumvolatile organic compoundsDrug Discoveryorganic acidschemical compositionPhysical and Theoretical ChemistryChemical compositionPomodorino del Piennolo del VesuviobiologyChemistryOrganic Chemistryfood and beverages04 agricultural and veterinary sciencesbiology.organism_classification040401 food scienceLycopeneHorticultureChemistry (miscellaneous)Geographic originFruitMolecular Medicinecherry tomato
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Extraction of Phenolic Compounds from Fresh Apple Pomace by Different Non-Conventional Techniques

2021

Red Delicious apple pomace was produced at laboratory scale with a domestic blender and different non-conventional extraction techniques were performed to isolate phenolic compounds, such as ultrasound-assisted extraction (UAE), ultraturrax extraction (UTE), accelerated solvent extraction (ASE) and pulsed electric field (PEF) extraction pre-treatment. Total phenolic content (TPC) was determined by Folin–Ciocalteu assay. Phloridzin, the main phenolic compound in apples, was determined by chromatographic analysis Q-TOF-LC/MS. The results obtained with these techniques were compared in order to identify the most efficient method to recover polyphenols. The highest value of TPC (1062.92 ± 59.80…

Pharmaceutical SciencephloridzinLaboratory scale01 natural sciencesArticleAntioxidantsMass SpectrometryASEQ-TOF-LC/MSAnalytical ChemistryQD241-4410404 agricultural biotechnologyNutraceuticalPhenolsFunctional foodDrug DiscoveryFood sciencenon-conventional extractionsPhysical and Theoretical ChemistryChromatography High Pressure LiquidpolyphenolsFlavonoidsEthanolPlant ExtractsChemistry010401 analytical chemistryOrganic ChemistryExtraction (chemistry)Pomace04 agricultural and veterinary sciencesPEF040401 food science0104 chemical sciencesAccelerated solvent extractionUAEChemistry (miscellaneous)PolyphenolMalusapple pomaceMolecular MedicineUTEMolecules
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Influence of fructose 1,6-diphosphate on the lung antioxidant defenses of mice with endotoxemia.

1990

PharmacologyLipopolysaccharidesAntioxidantLungFructose 1 6 diphosphateFree RadicalsChemistrymedicine.medical_treatmentMice Inbred StrainsShock SepticAntioxidantsMicemedicine.anatomical_structureBiochemistrySalmonella enteritidismedicineFructosediphosphatesAnimalsFemaleLungPharmacological research
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