Search results for "ATS"

showing 10 items of 6881 documents

Vascular Activity of (-)-Anonaine, (-)-Roemerine and (-)-Pukateine, Three Natural 6a(R)-1,2-Methylenedioxyaporphines with Different Affinities for α1…

2004

We have studied the mechanism of action of three 6a( R)-1,2-methylenedioxyaporphines as vasorelaxant compounds. The alkaloids assayed showed different affinities for the three human cloned alpha (1)-adrenoceptor (AR) subtypes stably expressed in rat-1 fibroblasts, showing lower affinity for alpha(1B)-AR with regard to the alpha(1A)- or alpha(1D)-subtypes. These three natural compounds are more potent inhibitors of [ (3)H]-prazosin binding than of [ (3)H]-diltiazem binding to rat cerebral cortical membranes. As all these alkaloids inhibited noradrenaline (NA)-induced [ (3)H]-inositol phosphate formation in cerebral cortex and rat tail artery, they may be safely viewed as alpha (1)-AR antagon…

AporphinesPhosphodiesterase InhibitorsStereochemistryPharmaceutical ScienceAorta ThoracicDioxolesBiologyMuscle Smooth VascularAnalytical ChemistryHydroxylationchemistry.chemical_compoundAlkaloidsDrug DiscoverymedicineAnonaineAnimalsHumansAporphineRats WistarBinding sitePukateineCerebral CortexPharmacologyPlants MedicinalVoltage-dependent calcium channelAlkaloidOrganic ChemistryArteriesReceptors Adrenergic alphaIsoquinolinesRatsComplementary and alternative medicineMechanism of actionchemistryMolecular MedicineFemaleCalcium Channelsmedicine.symptomDrugs Chinese HerbalPhytotherapyPlanta Medica
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A possible structural determinant of selectivity of boldine and derivatives for the alpha 1A-adrenoceptor subtype.

1996

1. The selectivity of action of boldine and the related aporphine alkaloids, predicentrine (9-O-methylboldine) and glaucine (2,9-O-dimethylboldine) and alpha 1-adrenoceptor subtypes was studied by examining [3H]-prazosin competition binding in rat cerebral cortex. WB 4101 and benoxathian were used as selective alpha 1A-adrenoceptor antagonists. 2. In the competition experiments [3H]-prazosin (0.2 nM) binding was inhibited by WB 4101 and benoxathian. The inhibition curves displayed shallow slopes which could be subdivided into high and low affinity components (pKi = 9.92 and 8.29 for WB 4101, 9.35 and 7.94 for benoxathian). The two antagonists recognized approximately 37% of the sites with h…

AporphinesStereochemistryAlpha (ethology)Binding CompetitiveAntioxidantsDioxanesOxathiinschemistry.chemical_compoundChloroethylclonidineBoldineAnimalsAporphineBinding siteRats WistarBenoxathianAdrenergic alpha-AntagonistsPharmacologyCerebral CortexAlkaloidPrazosinGlaucineRatschemistryAdrenergic alpha-1 Receptor AntagonistsFemaleResearch Article
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Simplification, not “tropicalization”, of temperate marine ecosystems under ocean warming and acidification

2021

Ocean warming is altering the biogeographical distribution of marine organisms. In the tropics, rising sea surface temperatures are restructuring coral reef communities with sensitive species being lost. At the biogeographical divide between temperate and tropical communities, warming is causing macroalgal forest loss and the spread of tropical corals, fishes and other species, termed “tropicalization”. A lack of field research into the combined effects of warming and ocean acidification means there is a gap in our ability to understand and plan for changes in coastal ecosystems. Here, we focus on the tropicalization trajectory of temperate marine ecosystems becoming coral-dominated systems…

Aquatic Organismsnatural analoguesEffects of global warming on oceanskelp forestswarm-temperateAnimalsEnvironmental ChemistrySeawaterMarine ecosystemEcosystembiogeographyEcosystemGeneral Environmental ScienceGlobal and Planetary Changegeographygeography.geographical_feature_categoryEcologyCoral ReefsEcologyfungitechnology industry and agricultureMarine habitatsOcean acidificationCoral reefHydrogen-Ion Concentrationbiochemical phenomena metabolism and nutritionrange shiftKelp forestclimate changeHabitat destructionEnvironmental sciencescleractinian coralsgeographic locationsGlobal Change Biology
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Gas-liquid chromatographic analyses

1983

Abstract The gas chromatography of mixtures of n -alkyl acetates (CH 3 COOR, R = C 1 —C 8 ) and methyl esters of aliphatic n -carboxylic acids (R′COOCH 3 , R′ = C 1 —C 8 ) and certain of their monochlorinated derivatives has been studied on Carbowax 20M and SE-30 glass capillary columns under the same operating conditions. The separation of the isomeric monochlorinated esters was complete on Carbowax 20M, whereas on SE-30 the peaks of 6- and 7-chlorooctyl acetates and methyl (ω − 1)- and (ω − 2)-chlorooctanoates and -nonanoates partly overlapped. The complete separation of the mixtures could not be achieved, however, on Carbowax 20M, in spite of the use of various operating conditions. The …

Aqueous normal-phase chromatographyValeric acidCapillary actionChlorine atomLiquid phasechemistry.chemical_elementAlcoholBiochemistryIsothermal processAnalytical ChemistryHomologous serieschemistry.chemical_compoundChain (algebraic topology)Capillary columnChlorineOrganic chemistryMethyleneChlorine substituentQuartzAlkylchemistry.chemical_classificationPrimary (chemistry)ChromatographyElutionChemistrySubstitution (logic)Organic ChemistryButanoic AcidsReversed-phase chromatographyGeneral MedicineCapillary gas chromatographyChromatographic separationAcyl chainembryonic structuresHalogenNitrocardiovascular systemPolarKovats retention indexGas chromatographyChromatography columnRetention timeGas liquid chromatographicJournal of Chromatography A
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Arbitrage international. Arbitrage multiparties, Groupe de contrats, Clauses compromissoires incompatibles, Consolidation (non)

1991

International audience; (Versailles, 7 mars 1990, Rev. arb. 1991. 326, note Loquin)

Arbitrage internationalUnité économique[SHS.DROIT]Humanities and Social Sciences/Law[SHS.DROIT] Humanities and Social Sciences/LawContrats multiplesARBITRAGECompétence
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Confirmation de l'application du principe de l'efficacité internationale de la clause compromissoire à la transmission de la convention d'arbitrage

2002

International audience; (Cass. 1re civ., 28 mai 2002, inédit, Sté Burkinabe des ciments et matériaux c/ Sté Des ciments d'Abidjan)

Arbitrage international[SHS.DROIT]Humanities and Social Sciences/LawChaîne de contrats[SHS.DROIT] Humanities and Social Sciences/LawARBITRAGEOpposabilitéClause compromissoire
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Clause compromissoire. Chaîne de contrats translatifs de propriété. Transmissibilité aux acquéreurs subséquents. Exception : preuve de l'ignorance ra…

2001

International audience; (Cass. 1re civ., 6 févr. 2001, Peavey Company c/ Organisme général des fourrages, D.2001.1135, obs. P. Delebecque)

Arbitrage international[SHS.DROIT]Humanities and Social Sciences/Law[SHS.DROIT] Humanities and Social Sciences/LawChaîne de contratsARBITRAGEOpposabilitéClause compromissoire
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De la transmission et de l'extension de la clause compromissoire : un « grand arrêt » de la première chambre civile de la Cour de cassation

2007

International audience; (Civ. 1re, 27 mars 2007, Sté Alcaltel Business Systems et autre c/ Sté Amkor Technology et autres, Rev. arb. 2007. 247 ; D. 2007. Jur. 2077, note S. Bollée)

Arbitrage international[SHS.DROIT]Humanities and Social Sciences/Law[SHS.DROIT] Humanities and Social Sciences/LawChaîne de contratsARBITRAGEOpposabilitéComputingMilieux_MISCELLANEOUS[ SHS.DROIT ] Humanities and Social Sciences/LawClause compromissoire
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Arbitrage international. Clause compromissoire - champs d'application, Chaîne non translative de contrats - Principe de l'effectivité de la clause co…

1996

International audience; (Paris, 22 mars 1995, Sté Aquaboulevard et autres c/ Sté Statinor et autres, inédit)

Arbitrage international[SHS.DROIT]Humanities and Social Sciences/Law[SHS.DROIT] Humanities and Social Sciences/LawChaîne non translative de contratsEffectivité de la clauseARBITRAGEClause compromissoire
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Société d'avocats. Cession d'action. Prix, Expertise, Article 1843-4 c. civ., Application en matière d'arbitrage

1997

International audience; (Paris, 21 mai 1996, CIP et autres c/ Soulier et autres, Rev. arb., 1996. 225, note Viandier)

ArbitrageCESSION DE DROITS SOCIAUX[SHS.DROIT]Humanities and Social Sciences/LawPrixSociété d'avocats[SHS.DROIT] Humanities and Social Sciences/LawExpert
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