Search results for "Antibacterial Activity"

showing 10 items of 169 documents

Activity against Microorganisms Affecting Cellulosic Objects of the Volatile Constituents of Leonotis nepetaefolia from Nicaragua

2014

The chemical composition of the essential oil from aerial parts of L. nepetaefolia (L.) R. Br. collected in Nicaragua was evaluated by GC and GC-MS. The main components were ( Z)-phytol (22.8%), caryophyllene oxide (18.9%) and hexahydrofarnesylacetone (9.0%). The antibacterial activity against several Gram + and Gram - bacteria, including Bacillus cereus and B. subtilis, both infesting historical cellulosic material, was also determined. B. cereus, B. subtilis and Staphylococcus epidermis were the most affected by the action of the oil.

MicroorganismBacillus cereusNicaraguaMicrobial Sensitivity TestsPlant ScienceGram-Positive Bacterialaw.inventionBacillus cereusPhytollawVolatile componentGram-Negative BacteriaDrug DiscoveryOils VolatileFood scienceEssential oilPolycyclic SesquiterpenesPharmacologyLamiaceaebiologyTerpenesChemistryfungiLeonotis nepetaefoliadisinfestation of museum objects.General MedicineHexahydrofarnesylacetonebiology.organism_classification(Z)-PhytolAnti-Bacterial AgentsComplementary and alternative medicineCereusCaryophyllene oxideLamiaceaeAntibacterial activitySesquiterpenesBacteriaBacillus subtilisLeonotis
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The Effect of Pesticides on the Tomato Bacterial Speck Disease Pathogen Pseudomonas Syringae pv. Tomato

2020

A significant part of the used pesticides does not reach the target organisms and, while remaining in the agrophytocenosis, influences all living organisms in it. Having a toxic and often mutagenic effect, pesticides induce morphological and physiological changes in the cells of microorganisms and are the cause of phenotypic heterogeneity of their populations. However, the effect of pesticides on phytopathogenic bacteria as non-target microorganisms remains out of the field of view for most researchers. However, the use of pesticides can lead to expansion of the diversity of existing phytopathogens and, as a consequence, complications of identification of the pathogens, loss of resistance b…

MicroorganismMutant010501 environmental sciencesBiology01 natural scienceslcsh:TechnologyMicrobiologylcsh:Chemistry03 medical and health scienceschemistry.chemical_compoundmorphological dissociation<i>Pseudomonas syringae</i> pv. <i>tomato</i>antibacterial activityPseudomonas syringaeGeneral Materials ScienceInstrumentationPathogenlcsh:QH301-705.5030304 developmental biology0105 earth and related environmental sciencesFluid Flow and Transfer Processes0303 health sciencesaluminium phosethyllcsh:TProcess Chemistry and TechnologyfungiGeneral Engineeringfood and beveragesPseudomonas syringae pv. tomatopesticidesdeltamethrinPesticidebiology.organism_classificationlcsh:QC1-999Computer Science ApplicationsFungicideDeltamethrinchemistrylcsh:Biology (General)lcsh:QD1-999lcsh:TA1-2040mutagenic actionlcsh:Engineering (General). Civil engineering (General)Bacterialcsh:PhysicsApplied Sciences
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Antimicrobial activity of essential oil ofArtemisia judaicaL. from Algeria against multi-drug resistant bacteria from clinical origin

2015

Artemisia judaica L. essential oil was studied for antibacterial activity against various clinical isolates of bacteria resistant to a number of antibiotics. The antibacterial activity was evaluated against 20 multidrug resistant (MDR) of clinical origin compared to standard ATCC strains. The strains that showed resistance against the maximum number of antibiotics tested were selected for an antibacterial assay by three methods: Disc diffusion method, microatmosphere and dilution method. The obtained results demonstrated that the A. judaica essential oil possessed an excellent inhibitory effect against all of the tested strains. The most potent results were obtained against MRSA (Methicilli…

Minimum bactericidal concentration010405 organic chemistryMulti drug resistant bacteriaChemistryGeneral ChemistryAntimicrobial01 natural sciences0104 chemical scienceslaw.inventionMicrobiologyArtemisia judaicaMultiple drug resistance010404 medicinal & biomolecular chemistryMinimum inhibitory concentrationlawBotanyAntibacterial activityEssential oilFood ScienceFlavour and Fragrance Journal
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Evaluation of the antibacterial activity of a new ozonized olive oil against oral and periodontal pathogens.

2018

Background In the present study, the antimicrobial properties of a new ozonized olive oil (O-zone gel) against oral and periodontal pathogens will be evaluated and compared with that of common CHX-based agents. Material and methods O-zone gel was compared with two agents based on chlorhexidine digluconate (CHX): Corsodyl Dental Gel and Plak Gel. A. actinomycetemcomitans, P. intermedia and S. mutans, were selected and the antibacterial capability of the compounds was tested by using direct contact agar diffusion test (DCT) and minimum inhibitory concentration (MIC) and minimum bactericidal concentration (MBC) evaluations. Differences between specific means were analyzed by a one-way analysis…

Minimum bactericidal concentrationbiologymedicine.drug_classChemistryResearch030206 dentistry02 engineering and technologyBacterial growth021001 nanoscience & nanotechnologyAntimicrobialbiology.organism_classification:CIENCIAS MÉDICAS [UNESCO]03 medical and health sciencesMinimum inhibitory concentration0302 clinical medicineAntisepticUNESCO::CIENCIAS MÉDICASmedicinePeriodontologyFood scienceAgar diffusion test0210 nano-technologyAntibacterial activityGeneral DentistryBacteriaJournal of clinical and experimental dentistry
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A peptide from human β thymosin as a platform for the development of new anti-biofilm agents for Staphylococcus spp. and Pseudomonas aeruginosa

2016

Conventional antibiotics might fail in the treatment of biofilm-associated infections causing infection recurrence and chronicity. The search for antimicrobial peptides has been performed with the aim to discover novel anti-infective agents active on pathogens in both planktonic and biofilm associated forms. The fragment 9-19 of human thymosin β4 was studied through 1 μs MD simulation. Two main conformations of the peptide were detected, both constituted by a central hydrophobic core and by the presence of peripheral charged residues suggesting a possible mechanism of interaction with two models of biological membranes, related to eukaryotic or bacterial membrane respectively. In addition, …

Models Molecular0301 basic medicineStaphylococcus aureusPhysiology030106 microbiologyAntimicrobial peptidesSettore BIO/05 - ZoologiaPeptideMicrobial Sensitivity TestsMolecular Dynamics SimulationBiologymedicine.disease_causeSettore BIO/19 - Microbiologia GeneraleApplied Microbiology and BiotechnologyMicrobiologyStructure-Activity Relationship03 medical and health sciencesAnti-Infective AgentsmedicineHumansAmino Acid SequencePeptide sequencechemistry.chemical_classificationPseudomonas aeruginosaAntimicrobial peptides Molecular dynamics Staphylococcal biofilms ThymosinBiofilmThymosinGeneral MedicineAntimicrobialSettore CHIM/08 - Chimica FarmaceuticaThymosin030104 developmental biologychemistryBiochemistrySettore CHIM/03 - Chimica Generale E InorganicaBiofilmsPseudomonas aeruginosaPeptidesAntibacterial activityBiotechnology
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Polyketide Derivatives from Mangrove Derived Endophytic Fungus Pseudopestalotiopsis theae

2020

Chemical investigation of secondary metabolites from the endophytic fungus Pseudopestalotiopsis theae led to the isolation of eighteen new polyketide derivatives, pestalotheols I&ndash

Models MolecularMagnetic Resonance SpectroscopyStereochemistryPharmaceutical Science010402 general chemistry01 natural sciencesArticlePolyketidepolyketideDrug DiscoverymedicineEndophytesCytotoxicityPharmacology Toxicology and Pharmaceutics (miscellaneous)IC50lcsh:QH301-705.5endophytic fungusbiologyMolecular Structure010405 organic chemistryChemistryAbsolute configurationFungibiology.organism_classification0104 chemical sciencesAcinetobacter baumanniiPseudopestalotiopsis theaelcsh:Biology (General)<i>Pseudopestalotiopsis theae</i>PolyketidesFermentationColistincytotoxicityRhizophoraceaeAntibacterial activityTwo-dimensional nuclear magnetic resonance spectroscopymedicine.drugMarine Drugs
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Discrimination and selection of new potential antibacterial compounds using simple topological descriptors.

2003

Abstract The aim of the work was to discriminate between antibacterial and non-antibacterial drugs by topological methods and to select new potential antibacterial agents from among new structures. The method used for antibacterial activity selection was a linear discriminant analysis (LDA). It is possible to obtain a QSAR interpretation of the information contained in the discriminant function. We make use of the pharmacological distribution diagrams (PDDs) as a visualizing technique for the identification and selection of new antibacterial agents.

Models MolecularQuantitative structure–activity relationshipMolecular StructureComputer sciencebusiness.industryDiscriminant AnalysisQuantitative Structure-Activity RelationshipPattern recognitionLinear discriminant analysisTopologyComputer Graphics and Computer-Aided DesignDiscriminant function analysisAnti-Infective AgentsSimple (abstract algebra)Drug DesignMaterials ChemistryComputer SimulationArtificial intelligencePhysical and Theoretical ChemistryAntibacterial activitybusinessSpectroscopySelection (genetic algorithm)SoftwareJournal of molecular graphicsmodelling
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Comparing the antibacterial activity of gaseous ozone and chlorhexidine solution on a tooth cavity model

2013

Objective: To evaluate the antibacterial activity of gaseous ozone andchlorhexidine solution on a tooth cavity model. Study Design: Twenty-one human molars were divided into 3 groups. Cavities were then cut into the teeth (4 per tooth, 28 cavities per group). After sterilization, the teeth wereleft in broth cultures of 106 colony-forming units (CFU) ml-1 of Streptococcus mutans (S. mutans) at 36°C for 48 h. The appropriate treatment followed (group A, control; group B, 2% chlorhexidine solution; and group C, 80s of treatment with ozone, and the cavities were thenfilled with compositeresin. After 72h, the restorations were removed, dentin chips were collected with an excavator, and the total…

MolarOzoneDentistryOdontologíaStreptococcus mutanschemistry.chemical_compoundOzonestomatognathic systemClinical and Experimental DentistrymedicineDentinGeneral Dentistrybiologybusiness.industryResearchChlorhexidineChlorhexidineSterilization (microbiology)biology.organism_classification:CIENCIAS MÉDICAS [UNESCO]Streptococcus mutansCiencias de la saludTooth cavitymedicine.anatomical_structurechemistryUNESCO::CIENCIAS MÉDICASTooth cavityAntibacterial activitybusinessAntibacterial activitymedicine.drug
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Search compounds with antimicrobial activity by applying molecular topology to selected quinolones.

2003

Molecular topology was used to obtain substances with antimicrobial activity. Selected quinolones were employed to develop the corresponding connectivity functions and discriminant equation. Limiting functions were selected that allowed the discriminant function to more efficiently distinguish substances with and without antibacterial activity. Antibacterial tests were run to confirm the theoretically established activity.

Molecular modelStereochemistryClinical BiochemistryPharmaceutical ScienceQuantitative Structure-Activity RelationshipMicrobial Sensitivity TestsQuinolonesBiochemistryDiscriminant function analysisDrug DiscoveryAnimalsMolecular BiologyTopology (chemistry)Antibacterial agentBacteriaChemistryOrganic ChemistryDiscriminant AnalysisAntimicrobialAnti-Bacterial AgentsDiscriminantDrug DesignMolecular MedicineMolecular topologyBiological systemAntibacterial activityBioorganicmedicinal chemistry letters
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New potent antibacterials against Gram-positive multiresistant pathogens: effects of side chain modification and chirality in linezolid-like 1,2,4-ox…

2014

The effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles have been studied to design new potent antibacterials against Gram-positive multidrug-resistant pathogens. The adopted strategy involved a molecular modelling approach, the synthesis and biological evaluation of new designed compounds, enantiomers separation and absolute configuration assignment. Experimental determination of the antibacterial activity of the designed (S)-1-((3-(4-(3-methyl-1,2,4-oxadiazol-5- yl)phenyl)-oxazolidin-2-one-5-yl)methyl)-3-methylthiourea and (S)-1-((3-(3-fluoro-4-(3-methyl-1,2,4- oxadiazol-5-yl)phenyl)-oxazolidin-2-one-5-yl)methyl)-3-methylthiourea against multidrug resistan…

Multidrug-resistant bacteriaClinical BiochemistryAntibioticsDrug ResistanceMolecular ConformationPharmaceutical ScienceBiochemistrychemistry.chemical_compoundAntibioticsDrug Resistance Multiple BacterialDrug DiscoveryAcetamidesSide chainOxadiazolesAbsolute configurationBacterialStereoisomerismHep G2 CellsBIO/10 - BIOCHIMICA23SAnti-Bacterial AgentsMolecular Docking SimulationRNA Ribosomal 23SDrug design Linezolid Antibiotics Multidrug-resistant bacteria EnantiomersMolecular MedicineAntibacterial activityMultipleMethicillin-Resistant Staphylococcus aureusStaphylococcus aureusmedicine.drug_classStereochemistryCell SurvivalMicrobial Sensitivity TestsGram-Positive BacteriaDrug designmedicineHumansMolecular BiologyOxazolidinonesRibosomalBinding SitesOrganic ChemistryAntibioticLinezolidSettore CHIM/06 - Chimica OrganicaSettore CHIM/08 - Chimica FarmaceuticaMultiple drug resistancechemistryEnantiomersMED/07 - MICROBIOLOGIA E MICROBIOLOGIA CLINICALinezolidRNANucleic Acid ConformationEnantiomerChirality (chemistry)Bioorganicmedicinal chemistry
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