Search results for "Benzene Derivative"

showing 10 items of 44 documents

Free radical scavenging abilities of flavonoids as mechanism of protection against mutagenicity induced by tert-butyl hydroperoxide or cumene hydrope…

2003

Mutagenicity induced by tert-butyl hydroperoxide (BHP) or cumene hydroperoxide (CHP) in Salmonella typhimurium TA102 was effectively reduced by flavonols with 3',4'-hydroxyl groups such as fisetin, quercetin, rutin, isoquercitrin, hyperoxide, myricetin, myricitrin, robinetin, and to a lesser extent also by morin and kaempferol (ID50=0.25-1.05 micromol per plate). With the exception of isorhamnetin, rhamnetin, morin, and kaempferol, closely similar results were obtained with both peroxides. Hydrogenation of the double bond between carbons 2 and 3 (dihydroquercetin, dihydrorobinetin) as well as the additional elimination of the carbonyl function at carbon 4 (catechins) resulted in a loss of a…

Salmonella typhimuriumFree RadicalsHealth Toxicology and MutagenesisMedicinal chemistrychemistry.chemical_compoundFlavonolstert-ButylhydroperoxideBenzene DerivativesGeneticsButylated hydroxytolueneIsorhamnetinFlavonoidschemistry.chemical_classificationDose-Response Relationship DrugDeferoxamine mesylateHydroxyl RadicalMutagenicity TestsAntimutagenic AgentsFree Radical ScavengersHydrogen PeroxideOxidantsBiochemistrychemistryCumene hydroperoxidetert-Butyl hydroperoxideMyricetinQuercetinMutation Research/Genetic Toxicology and Environmental Mutagenesis
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Three 2,5-dialkoxy-1,4-diethynylbenzene derivatives

2008

2,5-Dieth­oxy-1,4-bis­[(trimethyl­silyl)ethyn­yl]benzene, C20H30O2Si2, (I), constitutes one of the first structurally characterized examples of a family of compounds, viz. the 2,5-dialk­oxy-1,4-bis­[(trimethyl­silyl)ethyn­yl]benzene derivatives, used in the preparation of oligo(phenyl­ene­ethynylene)s via Pd/Cu-catalysed cross-coupling. 2,5-Dieth­oxy-1,4-diethynylbenzene, C14H14O2, (II), results from protodesilylation of (I). 1,4-Diethynyl-2,5-bis­(hept­yloxy)benzene, C24H34O2, (III), is a long alk­yloxy chain analogue of (II). The molecules of compounds (I)–(III) are located on sites with crystallographic inversion symmetry. The large substituents either in the alkynyl group or in the benz…

SilylationStereochemistryThree 25-dialkoxy-14-diethynylbenzene derivativesEtherGeneral MedicineCrystal structure.Ring (chemistry)Medicinal chemistryGeneral Biochemistry Genetics and Molecular BiologyFaculdade de Ciências Exatas e da Engenhariachemistry.chemical_compoundsymbols.namesakechemistryAtomsymbolsMoleculeVan der Waals radiusBenzeneActa Crystallographica Section C Crystal Structure Communications
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Nitramino, NRNO2 (R = H, CH3), as a substituent.13C and15N NMR spectroscopic study of nitraminobenzenes and -pyridines

1993

In order to clarify the special properties of the aryl-bound nitramino substituent NRNO 2 (R=H, CH 3 ), 13 C and 15 N NMR spectra of six nitraminobenzenes and nine nitraminopyridines were measured in DMSO-d 6 and their chemical shifts assigned. 1 H NMr chemical shifts and spin-spin coupling constants of all the compounds were also determined. In contrast to the behaviour of nitropyridines or -benzenes studied previously, most of the present compounds gave very broad 17 O NMR lines even at elevated temperatures and their 17 O NMR data were not useful for any reliable conclusions

StereochemistryChemical shiftSubstituentGeneral ChemistryNuclear magnetic resonance spectroscopyNmr dataMedicinal chemistryNMR spectra databasechemistry.chemical_compoundchemistryBenzene derivativesProton NMRNitroamineGeneral Materials ScienceMagnetic Resonance in Chemistry
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Development of a versatile, easy and rapid atmospheric monitor for benzene, toluene, ethylbenzene and xylenes determination in air

2009

Abstract A new procedure for the passive sampling in air of benzene, toluene, ethylbenzene and xylene isomers (BTEX) is proposed. A low-density polyethylene layflat tube filled with a mixture of solid phases provided a high versatility tool for the sampling of volatile compounds from air. Several solid phases were assayed in order to increase the BTEX absorption in the sampler and a mixture of florisil and activated carbon provided the best results. Direct head-space-gas chromatography–mass spectrometry (HS-GC–MS) measurement of the whole deployed sampler was employed for a fast determination of BTEX. Absorption isotherms were used to develop simple mathematical models for the estimation of…

Time FactorsBTEXXylenesBiochemistryEthylbenzenePermeabilityAnalytical Chemistrychemistry.chemical_compoundBenzene DerivativesBenzeneAir quality indexChromatographyAirOrganic ChemistryXyleneTemperatureBenzeneMembranes ArtificialGeneral MedicineToluenechemistryAdsorptionGas chromatographyGas chromatography–mass spectrometryEnvironmental MonitoringTolueneJournal of Chromatography A
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Effects of cyclooxygenase-1/cyclooxygenase-2 inhibition on leukocyte/endothelial cell interactions in the rat mesentery.

2002

Nonsteroidal anti-inflammatory drugs (NSAID) inhibit cyclooxygenase activity and cause gastrointestinal damage in part by promoting leukocyte accumulation in the mucosa. Our aim was to evaluate the effects of selective blockade of the isoenzymes cyclooxygenase-1 and cyclooxygenase-2 on leukocyte adhesion in vivo. Leukocyte/endothelial cell interactions were examined in rat mesenteric venules before and after treatment with indomethacin, SC-560 (5-(4-chlorophenyl)-1-(4-methoxyphenyl)-3-trifluoromethylpyrazole, cyclooxygenase-1 inhibitor), DFP (5,5-dimethyl-3-(2-propoxy)-4-(4-methanesulfonyl)-2(5H)-furanone, cyclooxygenase-2 inhibitor), or SC-560 plus DFP (20 mg/kg, i.v. each). Indomethacin i…

Time FactorsEndotheliumIndomethacinCell CommunicationPharmacologyRats Sprague-DawleyIn vivomedicineBenzene DerivativesCell AdhesionLeukocytesTumor Cells CulturedAnimalsHumansCyclooxygenase InhibitorsMesenteryFuransPharmacologybiologyCyclooxygenase 2 InhibitorsChemistryAnti-Inflammatory Agents Non-SteroidalMembrane ProteinsBiological activityDrug SynergismRatsEndothelial stem cellIsoenzymesmedicine.anatomical_structureMechanism of actionEnzyme inhibitorCyclooxygenase 2Prostaglandin-Endoperoxide SynthasesImmunologybiology.proteinCyclooxygenase 1PyrazolesCyclooxygenaseEndothelium Vascularmedicine.symptomBlood vesselEuropean journal of pharmacology
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Oxidative stress induces distinct physiological responses in the two Trebouxia phycobionts of the lichen Ramalina farinacea

2010

† Background and Aims Most lichens form associations with Trebouxia phycobionts and some of them simultaneously include genetically different algal lineages. In other symbiotic systems involving algae (e.g. reef corals), the relative abundances of different endosymbiotic algal clades may change over time. This process seems to provide a mechanism allowing the organism to respond to environmental stress. A similar mechanism may operate in lichens with more than one algal lineage, likewise protecting them against environmental stresses. Here, the physiological responses to oxidative stress of two distinct Trebouxia phycobionts (provisionally named TR1 and TR9) that coexist within the lichen R…

TrebouxiaAntioxidantLichensmedicine.medical_treatmentGlutathione reductasePlant ScienceGenes PlantPhotosynthesismedicine.disease_causeRamalina farinaceaSuperoxide dismutaseChlorophytaBotanyBenzene DerivativesmedicineHSP70 Heat-Shock ProteinsPhotosynthesisChlorophyll fluorescencebiologySuperoxide DismutaseGenetic VariationOriginal Articlesbiology.organism_classificationOxidative StressGlutathione ReductaseBiochemistrybiology.proteinOxidative stressAnnals of Botany
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The organic air pollutant cumene hydroperoxide interferes with NOantioxidant role in rehydrating lichen

2013

Organic pollutants effects on lichens have not been addressed. Rehydration is critical for lichens, a burst of free radicals involving NO occurs. Repeated dehydrations with organic pollutants could increase oxidative damage. Our aim is to learn the effects of cumene hydroperoxide (CP) during lichen rehydration using Ramalina farinacea (L.) Ach., its photobiont Trebouxia spp. and Asterochloris erici. Confocal imaging shows intracellular ROS and NO production within myco and phycobionts, being the chloroplast the main source of free radicals. CP increases ROS, NO and lipid peroxidation and reduces chlorophyll autofluorescence, although photosynthesis remains unaffected. Concomitant NO inhibit…

TrebouxiaChlorophyllAntioxidantLichensHealth Toxicology and Mutagenesismedicine.medical_treatmentBOTANICAToxicologymedicine.disease_causePhotosynthesisRamalina farinaceaLipid peroxidationchemistry.chemical_compoundBotanymedicineBenzene DerivativesDesiccationPhotosynthesisVolatile organic pollutantsBIOLOGIA VEGETALAir PollutantsbiologyDehydrationROSNitric oxideGeneral Medicinebiology.organism_classificationPollutionOxidative StressBiochemistrychemistryCumene hydroperoxideChlorophyllTrebouxiaNitrogen OxidesOxidation-ReductionOxidative stress
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Determination of optical purity of phosphonic acid analogues of aromatic amino acids by capillary electrophoresis with alpha-cyclodextrin.

2000

A simple and efficient method for the determination of enantiomeric purity of structurally diverse phosphonic and phosphinic acid analogues of phenylalanine and phenylglycine using capillary electrophoresis is presented. These preliminary studies indicated that the enantiomer separation is strongly dependent on the structure of the aminophosphonic acid.

chemistry.chemical_classificationCyclodextrinsalpha-CyclodextrinsChromatographyCyclodextrinOrganic ChemistryOrganophosphonatesElectrophoresis CapillaryPhenylalanineGeneral MedicineBiochemistryAnalytical ChemistryAmino acidchemistry.chemical_compoundCapillary electrophoresischemistryBenzene derivativesAromatic amino acidsphosphonic acidsEnantiomerenantiomer separationAmino AcidsEnantiomeric excessJournal of chromatography. A
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Biofiltration of ethylbenzene vapours: influence of the packing material.

2006

In order to investigate suitable packing materials, a soil amendment composed of granular high mineralized peat (35% organic content) locally available has been evaluated as carrier material for biofiltration of volatile organic compounds in air by comparison with a fibrous peat (95% organic content). Both supports were tested to eliminate ethylbenzene from air streams in laboratory-scale reactors inoculated with a two-month conditioned culture. In pseudo-steady state operation, experiments at various ethylbenzene inlet loads (ILs) were carried out. Maximum elimination capacity of about 120 g m(-3) h(-1) for an IL of 135 g m(-3) h(-1) was obtained for the fibrous peat. The soil amendment re…

chemistry.chemical_classificationEnvironmental EngineeringPeatSoil testRenewable Energy Sustainability and the EnvironmentChemistryEnvironmental engineeringAmendmentBioengineeringGeneral MedicineBiodegradationModels Theoreticalmedicine.diseasePulp and paper industryEthylbenzenechemistry.chemical_compoundSoilSpainBiofiltermedicineBenzene DerivativesVolatile organic compoundWaste Management and DisposalVapoursFiltrationBioresource technology
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ChemInform Abstract: Multi-Arm 1,2,3-Thiadiazole Systems.

2010

Benzene derivatives 2a–c with 6, 4, and 3 side chains bearing terminal 1,2,3-thiadiazole rings, respectively, have been prepared. Alkaline cleavage of 2a–c led to the corresponding alkynethiolates 6a–c, which were trapped by electrophiles such as benzyl bromide or iodomethane. The method provides an alternative to the thermal or photochemical cleavage of 1,2,3-thiadiazoles to thioketenes, which react further with nucleophiles.

chemistry.chemical_compoundBenzyl bromideNucleophileChemistryElectrophileBenzene derivativesSide chainNanotechnologyGeneral MedicineCleavage (embryo)Medicinal chemistryChemInform
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