Search results for "Benzene"

showing 10 items of 1701 documents

Inhibition of Delayed-Type Hypersensitivity by Cucurbitacin R through the Curbing of Lymphocyte Proliferation and Cytokine Expression by Means of Nuc…

2009

Cucurbitacin R is known to exhibit an anti-inflammatory effect in different experimental models of inflammation. In this article, we outline the effect of cucurbitacin R on T lymphocyte proliferation, cytokine production, and nuclear factor activation, as well as its influence on various experimental models of delayed-type hypersensitivity (DTH) in mice. Cucurbitacin R reduced the proliferation of phytohemagglutinin A-stimulated human T lymphocytes (IC(50), 18 microM), modifying the cell cycle, as well as the production of cytokines [interleukin (IL)-2, IL-4, IL-10, and especially interferon-gamma] and the induction of the principal cyclins implicated in the cell cycle (A(1), B(1), D(2), an…

Interleukin 2medicine.medical_specialtyT-Lymphocytesmedicine.medical_treatmentAnti-Inflammatory AgentsLymphocyte proliferationBiologyPharmacologyJurkat cellsDrug HypersensitivityJurkat CellsMiceCyclinsInternal medicinemedicineAnimalsHumansHypersensitivity DelayedInterleukin 4Cell ProliferationPharmacologyNFATC Transcription FactorsFootCell CycleIntracellular Signaling Peptides and ProteinsOxazoloneEarNFATCell cycleTriterpenesInterleukin 10EndocrinologyCytokineCytokinesMolecular MedicineDinitrofluorobenzeneFemalemedicine.drugJournal of Pharmacology and Experimental Therapeutics
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Effect of sodium dodecyl sulphate and Brij-35 on the analysis of sulphonamides in physiological samples using direct injection and acetonitrile gradi…

2016

Micellar liquid chromatography (MLC) is a reversed-phase (RP) mode, which often does not require gradient elution, since the peaks of mixtures of compounds within a large range of polarities appear more evenly distributed in the chromatograms of isocratic elution, giving rise to a “gradient effect”. However, the use of a gradient of organic solvent may still be convenient to shorten the total analysis time. This work compares the separation of 15 sulphonamides using conventional hydro-organic RPLC and MLC with the surfactants sodium dodecyl sulphate (SDS) and Brij-35, and both isocratic and gradient elution with acetonitrile. The observed behaviour is rationalized attending to the interacti…

Isocratic elutionChromatographyChemistryElutionGeneral Chemical EngineeringSodium010401 analytical chemistryGeneral EngineeringAnalytical chemistrychemistry.chemical_element010402 general chemistry01 natural sciences0104 chemical sciencesAnalytical Chemistrychemistry.chemical_compoundStationary phaseMicellar liquid chromatographyPhase (matter)AlkylbenzenesAcetonitrileAnalytical Methods
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Preparation, separation and identification of some para-substituted ONN and NNO trans-azoxybenzenes

2001

A series of para-substituted azoxybenzenes was obtained as model compounds for the investigation on the mechanism of Wallach rearrangement. Oxidation of azobenzenes with hydrogen peroxide in acetic acid solution, provided mixtures of α and β isomers. Some couples of the products were separated, using chromatography and crystallization techniques, and identified on the basis of their carbon NMR and mass spectra. The SCSD algorithm can be applied to the interpretation of the 13C-NMR spectra. Recognition of the ipso and para carbons suffice to the identification of an isomer, hence there are no strong interactions between the azoxy group and another substituent across the aromatic ring. Fragme…

IsomerismMass spectrometryAzoxybenzenesNMRPolish Journal of Chemistry
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Thermodynamics of transfer of polar additives from the aqueous to the dodecylsurfactant micellar phases

1990

The enthalpies of transfer from water to aqueous surfactant solutions, ΔH(W→W+S), of polar additives have been determined as a function of the surfactant concentration at fixed additive concentration. The surfactants used are sodium dodecylsulfate (NaDS), dodecyltrimethylammonium bromide and dodecyldimethylamine oxide (DDAO). The additives used are iso-butanol t-butanol, butoxyethanol, phenol, benzene, tributylphosphine oxide (TBPO), octyldimethylphosphine oxide (ODPO), octydimethylamine oxide (ODAO), DDAO and NaDS. A maximum was observed in the plots of ΔH(W→W+S) vs. fsms curves for ODPO and ODAO in NaDS while a small minimum was observed for TBPO. The experimental data are rationalized on…

Isothermal microcalorimetryAqueous solutionChemistryThermodynamics of micellizationInorganic chemistryEnthalpyBiophysicsOxideThermodynamicsFlory–Huggins solution theoryBiochemistryMicellechemistry.chemical_compoundlipids (amino acids peptides and proteins)Physical and Theoretical ChemistryBenzeneMolecular BiologyJournal of Solution Chemistry
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Hydrophobic effects in the stabilisation of copper(I) by the macrocyclic ligands 16,17,19,20-tetramethyl-2,6,9,13-tetraaza[14]paracyclophane and 14,1…

1996

Abstract The interaction of Cu 2+ with the para -azacychlophanes 16,17,19,20-tetramethyl-2,6,9,13-tetraazal[14]paracyclophane (L1) and 14,15,17,18-tetramethyl-2,5,8,11-tetraaza[12]paracyclophane (L2) has been studied by potentiometry, and direct microcalorimetry at 298.1±0.1 K in 0.15 mol dm −3 NaClO 4 . The stability constants (log K CuLi = 13.35(3), log K CuL2 = 9.32(4)) and the thermodynamic parameters ( ΔH ° CuL1 = −47.3(8) kJ mol −1 , ΔH ° CuL2 = 20.9(8) kJ mol −1 ) evidence that not all four nitrogen atoms in the ligands are involved in the coordination to the metal centre. These results, particulary in the case of L1, are similar to those reported for the analogous cyclophanes contai…

Isothermal microcalorimetryStereochemistrychemistry.chemical_elementNitrogenCopperMedicinal chemistryInorganic ChemistryMetalchemistry.chemical_compoundchemistryvisual_artMaterials Chemistryvisual_art.visual_art_mediumPhysical and Theoretical ChemistryBenzeneInorganica Chimica Acta
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Synthesis of azobenzene substituted tripod-shaped bi(p-phenylene)s. Adsorption on gold and CdS quantum-dots surfaces

2013

We report here the synthesis of several tripod-shaped oligo(p-phenylene)s with legs composed of two phenylene units. Each leg is end-capped with a thioacetate group for adhesion to metallic surfaces. An azobenzene chromophore group is present on the functional arm of the tripod. The key step in the synthesis is the Pd-catalyzed Suzuki cross-coupling reaction of the silicon derivative core molecule with substituted phenyl moieties and azobenzene derivatives. Gold surfaces prepared by thermal evaporation and CdS quantum-dots surfaces were covered by the tripod-shaped molecules. Modified surfaces were characterized by atomic force microscopy (AFM), fluorescence, and Kelvin Probe analyses.

Kelvin probe force microscopeNanostructureOrganic ChemistryTripod (photography)ChromophoreBiochemistrychemistry.chemical_compoundCrystallographyAzobenzenechemistryQuantum dotPhenyleneDrug DiscoveryOrganic chemistryMoleculeTetrahedron
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Enhanced expression of IL-8 in normal human keratinocytes and human keratinocyte cell line HaCaT in vitro after stimulation with contact sensitizers,…

1994

Abstract To investigate the interleukin-8 production of keratinocytes after stimulation in vitro we have used various agents: (i) contact sensi-tizer (2,4-dinitrofiuorobenzene, 3-n-penladecylcatechol); (ii) tolerogen (5-methyl-3-n-pentadecylcatechol); (iii) irritant (sodium lauryl sulfate). Interleukin-8 gene expression was assessed by northern blot hybridization of the total cytoplasmic RNA extracted from subconfluent normal human keratinocyte cultures and the keratinocyte cell line HaCaT using a radiolabeled DNA probe specific for human interleukin-8. Intcrleukin-8 gene expression was markedly increased upon in vitro stimulation after 1-6 h with contact sensitizers, tolerogen and the irri…

KeratinocytesCatecholsStimulationDermatologyDermatitis ContactBiochemistryGene expressionmedicineImmune ToleranceHumansInterleukin 8Northern blotRNA MessengerMolecular BiologyCells CulturedCell Line TransformedChemistryInterleukin-8Sodium Dodecyl SulfateMolecular biologyIn vitroHaCaTmedicine.anatomical_structureGene Expression RegulationCell cultureImmunologyIrritantsDinitrofluorobenzeneKeratinocyteExperimental dermatology
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Cannabinoid 1 Receptors in Keratinocytes Modulate Proinflammatory Chemokine Secretion and Attenuate Contact Allergic Inflammation

2013

Abstract Epidermal keratinocytes (KCs) and cannabinoid (CB) receptors both participate in the regulation of inflammatory responses in a mouse model for allergic contact dermatitis, the contact hypersensitivity (CHS) response to the obligate sensitizer 2,4-dinitrofluorobenzene. In this study, we investigated the cellular and molecular mechanisms how CB1 receptors attenuate CHS responses to 2,4-dinitrofluorobenzene. We used a conditional gene-targeting approach to identify the relative contribution of CB1 receptors on epidermal KCs for the control of CHS responses. To determine the underlying cellular and molecular mechanisms that regulate inflammatory responses in the effector phase of CHS, …

KeratinocytesChemokineImmunologyInflammationStimulationBiologyProinflammatory cytokineAllergic inflammationInterferon-gammaMiceReceptor Cannabinoid CB1medicineAnimalsChemokine CCL8Immunology and AllergyCXCL10ReceptorCells CulturedCell ProliferationInflammationMice Knockoutintegumentary systemEarAdoptive TransferChemokine CXCL10Mice Inbred C57BLDermatitis Allergic ContactImmunologyChemokine secretionbiology.proteinDinitrofluorobenzenemedicine.symptomThe Journal of Immunology
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Cellular and molecular mechanisms in the induction phase of contact sensitivity.

1995

During the induction phase of contact sensitivity, hapten-specific Th1 cells are primed by epidermal Langerhans cells. These Langerhans cells present hapten on MHC class II molecules and provide costimulatory signals. This presentation discusses the induction of cytokines in Langerhans cells and keratinocytes by haptens and their regulatory effects on contact sensitivity. Haptens were painted on the skin of normal BALB/c mice and epidermal cells were prepared at various times thereafter. Langerhans cell-derived interleukin (IL)-1 beta mRNA was observed as early as 15 min after hapten paining. In keratinocytes, tumor necrosis factor-alpha, IL-1 alpha, IP-10, MIP-2 and IL-10 were found to be …

KeratinocytesImmunologyAntigen presentationCD1chemical and pharmacologic phenomenaInduction PhasePicryl ChlorideBiologyMiceCytokines metabolismCricetinaeDinitrochlorobenzeneImmune ToleranceImmunology and AllergyAnimalsNitrobenzenesMHC class IIAntigen PresentationMice Inbred BALB Cintegumentary systemHistocompatibility Antigens Class IIAntibodies MonoclonalGeneral MedicineContact sensitivityCell biologyDinitrobenzenesLangerhans CellsImmunologyDermatitis Allergic Contactbiology.proteinCytokinesDinitrofluorobenzeneAntibodyHaptenHaptensInternational archives of allergy and immunology
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On the Nucleophilic Reactivity of 4,6-Dichloro-5-nitrobenzofuroxan with Some Aliphatic and Aromatic Amines: Selective nucleophilic substitution

2020

The reaction rates for the nucleophilic aromatic substitution of 4,6-dichloro-5-nitrobenzofuroxan 1 with eight aliphatic amines (characterized by very different basicities/ nucleophilicities) and three anilines have been measured in both methanol and toluene. The obtained rates have been related to the basicity (pKaH in water and Kb in benzene) or nucleophilicity (N Mayr constants) of the tested amines. The whole of the obtained kinetic data has furnished useful information on the high nucleophilic reactivity of benzofuroxan derivatives, which has been related essentially to two factors: the high electron-drawing ability/power of the condensed furoxan ring and the low aromatic character of …

KineticOrganic ChemistryFuroxanBenzofuroxanTolueneMedicinal chemistrySNArchemistry.chemical_compoundchemistryNucleophileNucleophilic aromatic substitutionAromaticity IndexNucleophilic substitutionMayr constantReactivity (chemistry)MethanolBenzene
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