Search results for "CONTRACT"

showing 10 items of 1719 documents

Selective chiral inhibition of Ca2+ entry promoted by bisbenzyltetrahydroisoquinolines in rat uterus.

1992

Abstract The effects of diltiazem and six bisbenzyltetrahydroisoquinoline alkaloids (antioquine, 7-O-methylantioquine, dimethylantioquine, monterine, granjine and cordobimine) were studied in rat isolated uterus in order to clarify the mechanisms of their relaxant actions. All the compounds tested completely relaxed KCl-induced contractions and totally or partially inhibited oxytocin-induced rhythmic contractions. Only alkaloids with absolute configurations (1R,1′S or 1R,1′R) acted intracellularly, promoting relaxation of contractile responses induced by oxytocin in a Ca2+-free medium, as does papaverine. Alkaloids of the antioquine series (1S,1′R) selectively inhibited Ca2+ entry. The grea…

endocrine systemStereochemistryMuscle RelaxationUterusBiologyOxytocinBenzylisoquinolinesPotassium ChlorideDiltiazemUterine ContractionAlkaloidsmedicineAnimalsheterocyclic compoundsDiltiazemRats WistarPharmacologyPapaverineAlkaloidUterusCalcium Channel BlockersIn vitroRatsmedicine.anatomical_structureOxytocinStereoselectivityFemalemedicine.symptommedicine.drugMuscle contractionEuropean journal of pharmacology
researchProduct

Effects of sulphonylureas on spontaneous motility and induced contractions in rat isolated uterus

1986

Abstract To clarify the action of sulphonylureas on calcium, the effect of tolbutamide and ghbenclamide has been investigated on a Ca-dependent process, the contractile activity of uterine smooth muscle. Both sulphonylureas antagonized the contractions evoked by CaCl2 in a non-competitive manner when the uterus was maintained in depolarizing solution and did not affect the spontaneous contractions of rat uterus. The capacity of tolbutamide and ghbenclamide to relax vanadate-induced contraction of rat uterus in Ca-free medium suggests that sulphonylureas may have an intracellular site of action related to cytosolic free Ca levels, or effect a reduction in Ca action.

endocrine systemmedicine.medical_specialtyContraction (grammar)TolbutamideUterusPharmaceutical ScienceMotilitychemistry.chemical_elementIn Vitro TechniquesBiologyCalciumGlibenclamideContractilityUterine ContractionTolbutamideInternal medicineGlyburidemedicineAnimalsHypoglycemic AgentsPharmacologyRats Inbred StrainsVanadiumRatsSulfonylurea CompoundsEndocrinologymedicine.anatomical_structureMechanism of actionchemistryCalciumFemaleVanadatesmedicine.symptommedicine.drugJournal of Pharmacy and Pharmacology
researchProduct

Relaxation induced by N-terminal fragments of chromogranin A in mouse gastric preparations.

2007

Abstract A definitive role for chromogranin A (CGA)-derived fragments in the control of the gastrointestinal smooth muscle contractility has not been yet established. The purpose of the present study was to evaluate, in vitro , the effects of the recombinant vasostatin 1–78 (VS-1), CGA 7–57 and CGA 47–66 on the mouse gastric mechanical activity, recording the changes of intraluminal pressure. VS-1, CGA 7–57 and CGA 47–66 produced concentration-dependent relaxations. Mouse anti-vasostatin-1 monoclonal antibody 5A8, recognising the region 53–57, abolished the relaxation induced by VS-1, indicating the specificity of the effect. The relaxation was significantly reduced by tetrodotoxin (TTX), b…

endocrine systemmedicine.medical_specialtyPhysiologyMuscle RelaxationClinical BiochemistryBiologyIn Vitro TechniquesApaminInhibitory postsynaptic potentialBiochemistrySettore BIO/09 - FisiologiaNitric oxideContractilityGastric relaxationCellular and Molecular Neurosciencechemistry.chemical_compoundMiceEndocrinologyInternal medicinemedicineAnimalsGastrointestinal tractCGA-derived peptideDose-Response Relationship DrugStomachChromogranin ANitric oxideMuscle SmoothMolecular biologyIn vitroPeptide FragmentsRecombinant ProteinsMice Inbred C57BLEndocrinologychemistryTetrodotoxinbiology.proteinVasostatinChromogranin ACalreticulinRegulatory peptides
researchProduct

Muscle function in monozygotic female twin pairs discordant for hormone replacement therapy

2011

Introduction: Postmenopausal monozygotic twin pairs discordant for hormone replacement therapy (HRT) provide an advantageous study design controlling for genetic background for elucidating the relationships between aging, sex hormone levels, muscle strength, contractile capacity, and fatigability. Methods: Thirteen postmenopausal monozygotic twin pairs discordant for HRT were measured for maximal voluntary torque (MVC) and twitch characteristics using electrical stimulation before and after intermittent dynamic plantarflexor exercise until exhaustion. Results: Peak twitch torque was 32% higher in HRT users than in their non-HRT, genetically identical sisters (P = 0.002), but MVC did not dif…

estradiolimedicine.medical_specialtygenetic structuresPhysiology030310 physiologyMonozygotic twinStimulationplantarflexor03 medical and health sciencesCellular and Molecular NeuroscienceMuscle nerveSex hormone-binding globulinPhysiology (medical)Internal medicinemedicineHumansvoimaMuscle StrengthtwitchMuscle Skeletalväsyminen030304 developmental biology0303 health sciencesPostmenopausal womenbiologyEstradiolbusiness.industryElectromyographyEstrogen Replacement TherapySkeletal muscleTwins MonozygoticMiddle AgedestrogeeniEndocrinologymedicine.anatomical_structureTransgender hormone therapyMuscle Fatiguebiology.proteinTime to peakfatigueFemalesense organsNeurology (clinical)strengthbusinesshuman activitiesMuscle ContractionMuscle & Nerve
researchProduct

Union representation and prevention of occupational risks during the crisis: impact and limits

2019

La investigación que presentamos estudia el impacto de la intervención sindical en materia de salud laboral, en lo que se refiere tanto a la gestión preventiva y creación de una cultura participativa como en los procesos de vigilancia y control de las condiciones de trabajo. A tal efecto, se han consultado las principales encuestas nacionales e internacionales sobre gestión de riesgos laborales en las empresas, analizando los datos más relevantes en base a modelos de regresión logística y lineal, lo que ha permitido constatar que la representación sindical de los trabajadores en la empresa (generalista y especializada) correlaciona positivamente con el desarrollo de las principales dimensio…

externalización preventivaSociología del Trabajocontractual precariousnessSociology of WorkOccupational riskmedia_common.quotation_subjectLabor. Work. Working classparticipative management.RecessionOccupational safety and healthHM401-1281OutsourcingDeregulationrepresentación sindical0502 economics and businessTrade unionSociology (General)precariedad contractualmedia_commonpreventive outsourcingOccupational healthbusiness.industryWelfare economicsunion representation05 social sciencesNegociación Colectivagestión participativa.050209 industrial relationsSalud laboralHD4801-8943Intervention (law)Participatory culturebusiness050203 business & managementSociología del Trabajo
researchProduct

Attività extralavorativa durante l'infortunio, obblighi contrattuali e doveri di correttezza e buona fede

2021

Il contributo, a partire da una pronuncia del Tribunale di Roma, affronta la questione della legittimità del licenziamento per giusta causa di un lavoratore, che svolga attività lavorativa presso terzi o extra lavorativa, quando sia infortunato e perciò assente dal lavoro. The essay deals with the legitimacy of dismissal for cause, starting from a decision of the Court of Rome. It’s about an employee who carries out other work or does some extracurriculars, when he is out sick.

extracurricularobblighi contrattualiLicenziamento per giusta causalegittimitàSettore IUS/07 - Diritto Del Lavorogood faith and fair dealinglegitimacyinfortunioattività extralavorativabuona fede e correttezzacontractual obligationsDismissal for cause
researchProduct

Sécurité juridique et relations commerciales internationales

2006

Colloque des 26 et 27 octobre 2006; National audience

favor contractus[SHS.DROIT]Humanities and Social Sciences/Law[SHS.DROIT] Humanities and Social Sciences/Lawprévisibilité du droit applicableDroit du commerce internationalprévisibilité du for compétentintangibilité du contratprévisibilité de l'efficacité internationale des jugements et des sentences arbitralesprévisibilité des lois de police applicablessolidarisme contractuel[ SHS.DROIT ] Humanities and Social Sciences/Law
researchProduct

Los Derechos Humanos en la Filosofía Analítica: Ronald Dworkin

2013

Este artículo atiende la manera en que Ronald Dworkin –como H. L. A. Hart y John Rawls, a quienes él sigue– enuncia el fundamento de los derechos humanos. Cierta presencia de iusnaturalismo en ese fundamento es señalado por Dworkin, Hart y Rawls y ellos buscan cuáles serían los derechos naturales del hombre (uno de ellos dice que sería la libertad y los otros dos dicen que sería la igualdad), i.e., ellos son derechos que no pueden depender de un contrato social porque ellos son primeros para estos y son presupuestos; debido a esto, ellos no pueden depender de la sola positivación. Hay, entonces, un iusnaturalismo escondido o latente en el fundamento de los derechos humanos como derechos mor…

filosofía analíticaSocial contractHuman rightslcsh:Philosophy (General)Philosophymedia_common.quotation_subjectFoundation (evidence)Moral rightsPhilosophyH. L. A. Hartfundamento.John RawlsLawDerechos humanosNatural (music)Ronald Dworkinlcsh:B1-5802media_commonTópicos, Revista de Filosofía
researchProduct

Fixed point results for α-implicit contractions with application to integral equations

2016

Recently, Aydi et al. [On fixed point results for α-implicit contractions in quasi-metric spaces and consequences, Nonlinear Anal. Model. Control, 21(1):40–56, 2016] proved some fixed point results involving α-implicit contractive conditions in quasi-b-metric spaces. In this paper we extend and improve these results and derive some new fixed point theorems for implicit contractions in ordered quasi-b-metric spaces. Moreover, some examples and an application to integral equations are given here to illustrate the usability of the obtained results.

fixed pointsApplied Mathematics010102 general mathematicsMathematical analysisimplicit contractionslcsh:QA299.6-433Alpha (ethology)implicit contractionlcsh:AnalysisFixed point01 natural sciencesIntegral equation010101 applied mathematicsfixed pointSettore MAT/05 - Analisi Matematicaquasi-b-metric spacesSettore MAT/03 - Geometria0101 mathematicsAnalysisMathematicsNonlinear Analysis: Modelling and Control
researchProduct

Il contratto a termine nelle fondazioni liriche

2020

The discipline of the fixed term contracts in opera foundations has been repeatedly modified in the last years. The attempts of the legislator to avoid the application of ordinary rules to these subjects has been nullified by the European Court of Justice. It has been therefore introduced a new regulation, that applies to these contracts some of the limits provided for in EU Directive 1999/70, but not the sanction of the conversion of the fixed term contract into a contract of indeterminate duration, in case of violation of the above mentioned limits. The workers have rights only to a monetary compensation, that can be considered an effective protection to unlawful use of flexible contracts.

fixed term contract operaSettore IUS/07 - Diritto Del Lavoro
researchProduct