Search results for "Diene"

showing 10 items of 623 documents

Pharmacogenomic and molecular docking studies on the cytotoxicity of the natural steroid wortmannin against multidrug-resistant tumor cells

2014

Wortmannin is a cytotoxic compound derived from the endophytic fungi Fusarium oxysporum, Penicillium wortmannii and Penicillium funiculosum that occurs in many plants, including medicinal herbs. The rationale to develop novel anticancer drugs is the frequent development of tumor resistance to the existing antineoplasic agents. Therefore, it is mandatory to analyze resistance mechanisms of novel drug candidates such as wortmannin as well to bring effective drugs into the clinic that have the potential to bypass or overcome resistance to established drugs and to substantially increase life span of cancer patients. In the present project, we found that P-glycoprotein-overexpressing tumor cells…

DrugATP Binding Cassette Transporter Subfamily BClass I Phosphatidylinositol 3-Kinasesmedia_common.quotation_subjectPharmaceutical ScienceAntineoplastic AgentsATP-binding cassette transporterDrug resistancePharmacologyBiologyWortmanninPhosphatidylinositol 3-Kinaseschemistry.chemical_compoundCell Line TumorDrug DiscoveryCluster AnalysisHumansCytotoxicityProtein kinase BPI3K/AKT/mTOR pathwayOligonucleotide Array Sequence Analysismedia_commonPharmacologyDrug Resistance MultipleAndrostadienesMolecular Docking SimulationMultiple drug resistanceComplementary and alternative medicinechemistryDrug Resistance NeoplasmPharmacogeneticsMolecular MedicineWortmanninSignal TransductionPhytomedicine
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Design and characterization of the SiPM tracking system of NEXT-DEMO, a demonstrator prototype of the NEXT-100 experiment

2013

NEXT-100 experiment aims at searching the neutrinoless double-beta decay of the Xe-136 isotope using a TPC filled with a 100 kg of high-pressure gaseous xenon, with 90% isotopic enrichment. The experiment will take place at the Laboratorio Subterraneo de Canfranc (LSC), Spain. NEXT-100 uses electroluminescence (EL) technology for energy measurement with a resolution better than 1% FWHM. The gaseous xenon in the TPC additionally allows the tracks of the two beta particles to be recorded, which are expected to have a length of up to 30 cm at 10 bar pressure. The ability to record the topological signature of the beta beta 0 nu events provides a powerful background rejection factor for the bet…

Enginyeria -- InstrumentsMECANICA DE LOS MEDIOS CONTINUOS Y TEORIA DE ESTRUCTURASBar (music)Tracking (particle physics)7. Clean energy01 natural sciencesEngineering instrumentsTECNOLOGIA ELECTRONICAchemistry.chemical_compoundData acquisitionSilicon photomultiplierOptics0103 physical sciencesPhysical instrumentsVisible and IR photons (solid-state)010306 general physicsInstrumentationPhoton detectors for UVMathematical PhysicsDetectors de radiacióPhysics010308 nuclear & particles physicsDynamic rangebusiness.industryTime projection Chambers (TPC)Electrical engineeringTetraphenyl butadieneFísicaTracking systemDetectorsGaseous imaging and tracking detectorschemistryNuclear countersParticle tracking detectors (Solid-state detectors)Física -- InstrumentsbusinessDark current
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Polar organic marker compounds in PM2.5 aerosol from a mixed forest site in western Germany

2008

The molecular composition of PM2.5 (particulate matter with an aerodynamic diameter2.5 microm) aerosol samples collected during a very warm and dry 2003 summer period at a mixed forest site in Jülich, Germany, was determined by gas chromatography/mass spectrometry in an effort to evaluate photooxidation products of biogenic volatile organic compounds (BVOCs) and other markers for aerosol source characterization. Six major classes of compounds represented by twenty-four individual organic species were identified and measured, comprising tracers for biomass combustion, short-chain acids, fatty acids, sugars/sugar alcohols, and tracers for the photooxidation of isoprene and alpha-/beta-pinene.…

Environmental EngineeringHealth Toxicology and MutagenesisCarbohydratescomplex mixturesGas Chromatography-Mass SpectrometryTreesBridged Bicyclo Compoundschemistry.chemical_compoundHemiterpenesGermanyPentanesButadienesEnvironmental ChemistryVolatile organic compoundBiomassOrganic ChemicalsChemical compositionBicyclic MonoterpenesAerosolschemistry.chemical_classificationPhotolysisChemistryPharmacology. TherapyLevoglucosanFatty AcidsPublic Health Environmental and Occupational HealthGeneral MedicineGeneral ChemistryParticulatesPollutionAerosolChemistryHydrocarbonPyrogallolEnvironmental chemistryMonoterpenesParticulate MatterAcids AcyclicMalic acidVolatilizationOxidation-ReductionChemosphere
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Towards an accurate molecular orbital theory for excited states : Ethene, butadiene, and hexatriene

1993

A newly proposed quantum chemical approach for ab initio calculations of electronic spectra of molecular systems is applied to the molecules ethene, trans‐1,3‐butadiene, and trans‐trans‐1,3,5‐hexatriene. The method has the aim of being accurate to better than 0.5 eV for excitation energies and is expected to provide structural and physical data for the excited states with good reliability. The approach is based on the complete active space (CAS) SCF method, which gives a proper description of the major features in the electronic structure of the excited state, independent of its complexity, accounts for all near degeneracy effects, and includes full orbital relaxation. Remaining dynamic ele…

ErrorsGeneral Physics and AstronomyPolyenesElectronic structuresymbols.namesakeRydberg StatesAb initio quantum chemistry methodsComputational chemistrySinglet statePhysical and Theoretical ChemistryTriplet state:FÍSICA::Química física [UNESCO]AccuracyExcitationCalculation MethodsButadieneTripletsChemistryMolecular orbital theoryScf CalculationsExcited StatesCalculation Methods ; Quantum Chemistry ; Ab Initio Calculations ; Electron Spectra ; Butadiene ; Accuracy ; Scf Calculations ; Triplets ; Rydberg States ; Excitation ; Errors ; Polyenes ; Excited StatesQuantum ChemistryUNESCO::FÍSICA::Química físicaElectron SpectraExcited stateRydberg formulasymbolsRydberg stateAtomic physicsAb Initio Calculations
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Linked cyclopentadienyl-amido titanium catalysts supported on pyridylethylsilane-modified silica for heterogeneous ethylene homo- and copolymerization

2003

Abstract Linked cyclopentadienyl-amido titanium dimethyl and dichloro complexes, Ti(η 5 :η 1 -C 5 Me 4 SiMe 2 N t Bu)X 2 (X=Me, Cl), were reacted with trityl tetrakis(pentafluorophenyl)borate (TB), Ph 3 C + [B(C 6 F 5 ) 4 ] − , and methylaluminoxane (MAO), followed by treatment with toluene suspension of pyridylethylsilane-modified silica, to give two new supported-type titanium catalysts, PySTiTB and PySTiMAO. PySTiTB polymerized ethylene in the presence of triisobutylaluminum (TIBA) in hexane at 60 °C and 5 bar with slightly higher activity than the corresponding homogeneous system under the same conditions. PySTiMAO showed relatively high activity even without any use of alkylaluminum co…

EthyleneCyclopentadieneProcess Chemistry and TechnologyMethylaluminoxanechemistry.chemical_elementPolyethyleneCatalysisCatalysischemistry.chemical_compoundCyclopentadienyl complexchemistryPolymer chemistryCopolymerPhysical and Theoretical ChemistryTitaniumJournal of Molecular Catalysis A: Chemical
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Interaction of half-sandwich alkylmolybdenum(III) complexes with B(C6F5)3. The X-ray structure of [CpMo(η4-C4H6)(μ-Cl)(μ-CH2)(O)MoCp][CH3B(C6F5)3]

2001

Abstract The reactions of the half-sandwich molybdenum(III) complexes CpMo(η 4 -C 4 H 4 R 2 )(CH 3 ) 2 , where Cpη 5 -C 5 H 5 and RH or CH 3 , with equimolar amounts of B(C 6 F 5 ) 3 have been investigated in toluene. EPR monitoring shows the formation of an addition product which does not readily react with Lewis bases such as ethylene, pyridine, or PMe 3 . The analysis of the EPR properties and the X-ray structure of a decomposition product obtained from dichloromethane, [CpMo(η 4 -C 4 H 6 )(μ-Cl)(μ-CH 2 )(O)MoCp][CH 3 B(C 6 F 5 ) 3 ], indicate that the borane attack has occurred at the methyl position.

EthyleneStereochemistrychemistry.chemical_elementBorane010402 general chemistry01 natural sciencesBiochemistryMedicinal chemistrylaw.inventionInorganic Chemistrychemistry.chemical_compoundlawPyridineMaterials Chemistry[CHIM.CRIS]Chemical Sciences/Cristallography[CHIM.COOR]Chemical Sciences/Coordination chemistryLewis acids and basesPhysical and Theoretical ChemistryElectron paramagnetic resonanceDichloromethaneMolybdenumEPR properties010405 organic chemistryOrganic ChemistryTolueneButadiene ligand0104 chemical sciences3. Good healthchemistryHalf-sandwichMolybdenumX-ray structure
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Synthèse et caractérisation de phosphine, borane, amine sur plateforme ferrocène polyfonctionnelle

2016

Ferrocene platforms are useful in coordination chemistry and catalysis thanks to their robustness and versatile functionalization. Ferrocene backbone allows the implantation of several key functional groups in a restricted space, inducing close proximity and potential polyfunctional cooperation (see for instance ferrocenyl polyphosphine chemistry). Ansa ferrocene and ferrocene bearing conformational control inducing groups maximizing the proximity of key groups have been widely reported.The first part of this thesis focuses on the synthesis of new borylated cyclopentadienyl, and their use in formation of borylated metallocenes bearing conformational constraints. NMR analysis and DFT calcula…

Frustrated Lewis pairAmbiphilic ligandCouplage de spinPhosphorusPaire frustrée de Lewis[CHIM.COOR] Chemical Sciences/Coordination chemistryCyclopentadiénureCyclopentadienideBorePhosphore[CHIM.COOR]Chemical Sciences/Coordination chemistryFerroceneNon-bonded spin couplingLigand ambiphileAmineCyclopentadieneBoronMetallocene
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On the enhancement of stereoselection by cooperation between chiral auxiliaries. Asymmetric diels-alder reactions with fumaric acid bis ((S)-proline …

1989

Abstract Fumaric acid bis ((S)-proline benzyl ester) amide reacts with cyclopentadiene in thermal and Lewis acid catalyzed Diels-Alder reactions to give the cycloadducts with high yields and diastereomeric ratios up to 100:1.

Fumaric acidCyclopentadieneOrganic ChemistryDiastereomerBiochemistryCatalysischemistry.chemical_compoundchemistryAmideDrug DiscoveryDiels alderOrganic chemistryLewis acids and basesProline benzyl esterTetrahedron Letters
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Ab initio SCF and CI calculations on the barrier to internal rotation of 1,3-butadiene

1972

Ab initio SCF and CI calculations employing a set of gaussian lobe functions have been carried out for the ground and excited states of five geometrical C4H6-structures occurring in the course of rotation from cis-butadiene to the trans-isomer. The rotational potential curves are discussed for the ground and excited states. Particularly the potential curve of the lowest triplet state is considered in this connection thereby substantiating quantitatively the proposed mechanism for induced dimerisation of C4H6. Possible assignments of the lowest singlet excited states in trans-butadiene are discussed.

GaussianInternal rotationAb initio13-ButadieneRotationchemistry.chemical_compoundsymbols.namesakechemistryExcited statesymbolsChiropracticsSinglet statePhysics::Chemical PhysicsPhysical and Theoretical ChemistryAtomic physicsTriplet stateTheoretica Chimica Acta
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The Program of Health Volunteer Promoters for OlderAdults: The Well-Being of the Volunteers at Leisure Time

2018

The study of ageing processes has gained increased attention in recent years, partly due to the growth of this population group (United Nations, World population prospects: The 2015 revision. New York: United Nations Department of Economic and Social Affairs. https://esa.un.org/unpd/wpp/publications/files/key_findings_wpp_2015.pdf. Accessed 25 Sep 2016, 2015). Research into this area has focused on older adult well-being (Au et al, Clinical Gerontologist 38:203–210, 2015) and the identification of factors having an influence on well-being at this stage of the life cycle (Carstensen, Current Directions in Psychological Science 4:151–156, 1995). These lines of research have emphasized the con…

Gerontologyeducation.field_of_studybiologySocializationGarciaPopulationWorld populationbiology.organism_classificationSolidarityActive ageingDienerWell-beingeducationPsychology
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