Search results for "FUNCTIONAL"

showing 10 items of 4822 documents

New Reactions of Amino-Functionalized 3-Vinyl-1H-indoles and Tetrahydropyridin-4-yl Analogues with Dienophiles

1991

Reactions of 3-[2-(morpholin-4-yl)vinyl]-1H-indole (1), the 1,2-dihydro-9H-carbazole 2, as well as the 3-(tetrahydropyridin-4-yl)-1H-indoles 3a and 3b with some carbo- and heterodienophiles are described. The scope and limitations of the synthetic utility of these amino- (or homoamino)-functionalized 3-vinyl-1H-indoles are reported and some MO calculations for the qualitative prediction of their reactivities are presented. The reactions gave rise to substitution products, redox products, Diels-Alder adducts, ene adducts, and Michael-type adducts (Schemes 2 and 3).

Bicyclic moleculeChemistryOrganic ChemistryBiochemistryRedoxCatalysisQualitative predictionAmino functionalizedAdductEnamineInorganic Chemistrychemistry.chemical_compoundDrug DiscoveryOrganic chemistryPhysical and Theoretical ChemistryEne reactionHelvetica Chimica Acta
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Carbon nanotube supported aluminum porphyrin-imidazolium bromide crosslinked copolymer

2022

The increased awareness of the catastrophic consequences caused by the accumulation of greenhouse gases into the atmosphere has generated a large mobilization aimed at CO2 mitigation. Herein, in the spirit of the transformation of a waste as CO2 into value added products, we propose an efficient preparation of two different hybrid systems based on aluminum chloride tetrastyrylporphyrin (TSP-Al-Cl) and 1,4-butanediyl-3,3′-bis-1-vinylimidazolium dibromide copolymerized in the presence (MWCNT-TSP-AlCl-imi) and in absence (TSP-AlCl-imi) of multi-walled carbon nanotubes (MWCNTs) for the CO2 utilization in the synthesis of cyclic carbonates. The so-prepared materials have been thoroughly characte…

Bifunctional catalystCarbon dioxide fixationProcess Chemistry and TechnologyCarbon nanotubesCyclic carbonatesChemical Engineering (miscellaneous)Al-porphyrinWaste Management and DisposalJournal of CO2 Utilization
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Estimation of total electricity consumption curves of small areas by sampling in a finite population

2016

International audience; Many studies carried out in the French electricity company EDF are based on the analysis of the total electricity consumption curves of groups of customers. These aggregated electricity consumption curves are estimated by using samples of thousands of curves measured at a small time step and collected according to a sampling design. Small area estimation is very usual in survey sampling. It is often addressed by using implicit or explicit domain models between the interest variable and the auxiliary variables. The goal here is to estimate totals of electricity consumption curves over domains or areas. Three approaches are compared: the rst one consists in modeling th…

Big dataEnergyMSC: 62H25Functional principal component analysis[MATH.MATH-ST]Mathematics [math]/Statistics [math.ST]Regression trees[ MATH.MATH-ST ] Mathematics [math]/Statistics [math.ST]Mixed modelsFunctional data[MATH.MATH-ST] Mathematics [math]/Statistics [math.ST]
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Diorganotin(IV) N-acetyl-L-cysteinate complexes: synthesis, solid state, solution phase, DFT and biological investigations.

2009

Diorganotin(IV) complexes of N-acetyl-L-cysteine (H(2)NAC; (R)-2-acetamido-3-sulfanylpropanoic acid) have been synthesized and their solid and solution-phase structural configurations investigated by FTIR, Mössbauer, (1)H, (13)C and (119)Sn NMR spectroscopy. FTIR results suggested that in R(2)Sn(IV)NAC (R = Me, Bu, Ph) complexes NAC(2-) behaves as dianionic tridentate ligand coordinating the tin(IV) atom, through ester-type carboxylate, acetate carbonyl oxygen atom and the deprotonated thiolate group. From (119)Sn Mössbauer spectroscopy it could be inferred that the tin atom is pentacoordinated, with equatorial R(2)Sn(IV) trigonal bipyramidal configuration. In DMSO-d(6) solution, NMR spectr…

Binding SitesMolecular StructureLigandStereochemistryCell SurvivalSpectrum Analysischemistry.chemical_elementAntineoplastic AgentsNuclear magnetic resonance spectroscopyBiochemistryMedicinal chemistryAcetylcysteineCell LineInorganic Chemistrychemistry.chemical_compoundTrigonal bipyramidal molecular geometryDeprotonationchemistryMössbauer spectroscopyOrganotin CompoundsOrganotin(IV) FTIR Mössbauer NMR DFT Antitumor activityHumansDensity functional theoryCarboxylateTinJournal of inorganic biochemistry
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Interaction of Au16 Nanocluster with Defects in Supporting Graphite: A Density-Functional Study

2011

Soft-landed adsorption of Au-16 on bilayered graphene is investigated using density functional theory. The orientation of the Au-16 cluster and number of neighboring surface vacancies affect the overall structural and electronic properties of the cluster. The results of the PBE, vdW-DF, and vdW-DF2 exchange-correlation functionals are compared for the cluster-substrate interaction for systems with and without defects. In the presence of defects size two and greater, an Au atom adsorbs into the topmost graphene layer; this strongly influences the binding energy (>3 eV), while inducing substantial bending in the carbon plane and altering electronic properties of the system. Though the T-d-sym…

Binding energyNanotechnology02 engineering and technology010402 general chemistry01 natural scienceslaw.inventionDelocalized electronlawAtomCluster (physics)GraphitePhysical and Theoretical Chemistryta114ChemistryGraphene021001 nanoscience & nanotechnologyElectron localization function0104 chemical sciencesSurfaces Coatings and FilmsElectronic Optical and Magnetic MaterialsJGeneral EnergyChemical physicsddc:540Density functional theory0210 nano-technologyJournal of Physical Chemistry C
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Pyrene derived functionalized low molecular weight organic gelators and gels

2008

Pyrene derived binary functionalized low molecular weight organic gelators (FLMOGs) and gels thereof in selected organic solvents were synthesized and characterized. The functionality refers to a functional group that does not take part in formation of the supramolecular gel network, but remains free and available for other purposes, such as to bind nanoparticles or other molecules into the gel structure. Functional groups were observed to disturb gel formation strongly, if they interact with each other within the same supramolecule due to the formation of competitive structures. Preventing such interactions restored the original gel properties. A gel with weaker supramolecular bonding than…

Binding energySupramolecular chemistryGeneral ChemistryCatalysisFluorescence spectroscopySolventchemistry.chemical_compoundsymbols.namesakechemistryFunctional groupPolymer chemistryMaterials ChemistrysymbolsMoleculePyrenevan der Waals forceNew Journal of Chemistry
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Exponential Relaxation out of Nonequilibrium

1989

Simulation results are presented for a quench from a disordered state to a state below the coexistence curve. The model which we consider is the Ising model but with the dynamics governed by the Swendsen-Wang transition probabilities. We show that the resulting domain growth has an exponential instead of a power law behaviour and that the system is non-self-averaging while in nonequilibrium. The simulations were carried out on a parallel computer with up to 128 processors.

BinodalPhysicsCondensed Matter::Statistical MechanicsGeneral Physics and AstronomyRelaxation (physics)Non-equilibrium thermodynamicsIsing modelStatistical physicsState (functional analysis)Power lawDomain (mathematical analysis)Exponential functionEurophysics Letters (EPL)
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MANOTA: a promising bifunctional chelating agent for copper-64 immunoPET

2017

International audience; Improved bifunctional chelating agents (BFC) are required for copper-64 radiolabelling of monoclonal antibodies (mAbs) under mild conditions to yield stable, target-specific imaging agents. Four different bifunctional chelating agents (BFC) were evaluated for Fab (Fragment antigen binding) conjugation and radiolabelling with copper-64. Two DOTA- (1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid) and two NOTA- (1,4,7-triazacyclononane-1,4,7-triacetic acid) derivatives bearing a p-benzyl-isothiocyanate group were conjugated to Fab-trastuzumab - which targets the HER2/neu receptor - and the average number of chelators attached ranged from 2.4 to 4.3 macrocycles …

BiodistributionImmunoconjugatesmedicine.drug_class[SDV.CAN]Life Sciences [q-bio]/CancerMonoclonal antibody030218 nuclear medicine & medical imaging[ SDV.CAN ] Life Sciences [q-bio]/CancerInorganic ChemistryHeterocyclic Compounds 1-RingImmunoglobulin Fab FragmentsMice03 medical and health scienceschemistry.chemical_compound0302 clinical medicineCell Line TumormedicineAnimalsHumansDOTA[ SDV.IMM ] Life Sciences [q-bio]/ImmunologyTissue DistributionChelationBifunctionalChelating AgentsRadiochemistryMammary Neoplasms ExperimentalTrastuzumabIn vitroImmunoconjugateCopper RadioisotopesBiochemistrychemistryPositron-Emission Tomography030220 oncology & carcinogenesis[SDV.IMM]Life Sciences [q-bio]/ImmunologyCopper-64
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Evaluation of proton MR spectroscopy at 3 Tesla without endorectal coil in patients with a localized prostate cancer treated with exclusive radiother…

2011

Prostate cancer is the most frequent tumour affecting the male population. When the prostate is not removed and is treated with radiation therapy, PSA slowly decreases over time to reach its nadir, even sometimes 18 to 24 months after the completion of radiation therapy without combined androgen suppression therapy. When combined with hormones, PSA falls abruptely with no possibility to perceive the impact of either hormones or radiation effects on PSA.The optimal value of PSA that should be reached after radiation therapy (nadir) and time to this nadir are still unclear.Even when a satisfactory value of the PSA nadir is reached, on-going variations of the PSA and its “bounce” effects, whic…

BiomarqueursRéponse thérapeutique[SDV.MHEP] Life Sciences [q-bio]/Human health and pathologyProstate cancerTherapeutic responseRadiotherapySpectroscopieCancer de la prostateIRM fonctionnelle[ SDV.MHEP ] Life Sciences [q-bio]/Human health and pathologyBiomarkersSpectroscopy[SDV.MHEP]Life Sciences [q-bio]/Human health and pathologyFunctional MRIRadiothérapie
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An ab initio potential energy surface for the C2H2-N2 system

2012

International audience; An ab initio potential energy surface determined at the CCSD(T) level of theory is presented for the van der Waals complex C2H2-N2. Additional calculations performed with the HF- and DFT-SAPT methods compare well with the CCSD(T) results and allow a better understanding of the main features of this interaction potential surface. An expansion of this surface over spherical harmonics has also been performed. The global energy minimum of the complex is obtained for the linear conformation. The T conformations are the least attractive. Such characteristics mainly arise because of the variation, in sign and in absolute value of the electrostatic energy between all these c…

BiophysicsAb initioAbsolute valueINFRARED-SPECTRUM010402 general chemistry01 natural sciences[ CHIM ] Chemical SciencesCROSS-SECTIONSDENSITY-FUNCTIONAL THEORYsymbols.namesakeMOLECULES0103 physical sciencesPhysics::Atomic and Molecular Clusters[CHIM]Chemical SciencesPhysical and Theoretical ChemistryMolecular BiologyACETYLENEPERTURBATION-THEORY APPROACHDIMERSPECTROSCOPY010304 chemical physicsChemistryElectric potential energyDER-WAALS COMPLEXESSpherical harmonicsCondensed Matter Physics0104 chemical sciencesEnergy profileKOHN-SHAM ORBITALSPotential energy surfacesymbolsDensity functional theoryvan der Waals forceAtomic physics
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