Search results for "OBIA"

showing 10 items of 2471 documents

SKRINING FITOKIMIA, UJI AKTIVITAS ANTIMIKROBA DAN ANTITUMOR TUMBUHAN OBAT KABUPATEN MANOKWARI

2008

<p><em>Pythochemistry screening and testing of antimicrobial and antitumor activities was carried out on 31 species of medicinal plants distributed around Manokwari Regency.  All parts of the plants were collected and screened for the presence of alkaloids, saponins, and tannins; antimicrobial and antitumor activity. The number of positive tests obtained are 17 (55, 3%) for alkaloids, 6 (19, 4%) for saponins, and 26 (84, 7%) for tannins. Eleven species shown inhibition activities (antimicrobial) to Candida albicans, Staphyloccocus aureus, and Echericia colii while only seven species have antitumor activity, especially against tumor cell P-388. </em></p>

Antitumor activitychemistry.chemical_classificationchemistryTraditional medicineSaponinTanninStaphyloccocus aureusTumor cellsBiologyMedicinal plantsAntimicrobialCandida albicansbiology.organism_classificationJurnal Natural
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A new method for creating sparse design velocity fields

2006

We present a novel method for the computation of mesh node sensitivities with respect to the boundary node movement. The sensitivity field is sparse in a sense that movement of each boundary node affects only given amount of inner mesh nodes, which can result in considerable savings in the storage space. The method needs minimal control from the user, and it does not place any restrictions (such as block structure) on the mesh. Use of the method is demonstrated with a shape optimization problem using CAD-free parametrization. A solution to the classical die-swell free boundary problem by coupling the boundary node locations with the state variables is also presented. In that case, sparsity …

Mathematical optimizationMechanical EngineeringComputationComputational MechanicsGeneral Physics and AstronomyBoundary (topology)ResidualComputer Science Applicationssymbols.namesakeMechanics of MaterialsMesh generationJacobian matrix and determinantsymbolsFree boundary problemNode (circuits)Sensitivity (control systems)AlgorithmMathematicsComputer Methods in Applied Mechanics and Engineering
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The Application of the Essential Oils of Thymus vulgaris L. and Crithmum maritimum L. as Biocidal on Two Tholu Bommalu Indian Leather Puppets

2021

The chemical profile of the Thymus vulgaris (Lamiaceae) essential oil (EO) was investigated in order to evaluate its biological properties against microorganisms affecting two Tholu Bommalu, typical Indian leather puppets stored at the International Puppets Museum “Antonio Pasqualino” of Palermo, Italy. A GC–MS analysis, using both polar and apolar columns, was used to determine the chemical composition of the essential oil. The aim of this study was to evaluate the antimicrobial effectiveness of the Thymus vulgaris and Crithmum maritimum essential oils in vapor phase to disinfect heritage leather puppets. Pieces of leather artifacts that were affected by different bacterial colonies were e…

BiocideMicroorganismThymus vulgarisPlant ScienceThymus vulgari01 natural sciencesArticleessential oillaw.inventionThymus vulgarisanti-bacterial activitylawCrithmum<i>Thymus vulgaris</i>Food scienceleather artifactsessential oilsEcology Evolution Behavior and SystematicsEssential oil<i>Crithmum maritimum</i>ApiaceaeEcologybiology010405 organic chemistryChemistrytechnology industry and agricultureBotanyCrithmum maritimumbiology.organism_classificationAntimicrobial0104 chemical sciences010404 medicinal & biomolecular chemistryleather artifactQK1-989LamiaceaePlants
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Real-Time Polymerase Chain Reaction for Detection of Schistosoma DNA in Small-Volume Urine Samples Reflects Focal Distribution of Urogenital Schistos…

2014

Schistosoma haematobium eggs and Schistosoma DNA levels were measured in urine samples from 708 girls recruited from 18 randomly sampled primary schools in South Africa. Microscopic analysis of two 10-mL urine subsamples collected on three consecutive days confirmed high day-to-day variation; 103 (14.5%) girls had positive results at all six examinations, and at least one positive sample was seen in 225 (31.8%) girls. Schistosoma-specific DNA, which was measured in a 200-μL urine subsample by using real-time polymerase chain reaction, was detected in 180 (25.4%) cases, and levels of DNA corresponded significantly with average urine egg excretion. In concordance with microscopic results, pol…

Pathologymedicine.medical_specialtyConcordancePhysiologyUrineBiologyReal-Time Polymerase Chain ReactionSensitivity and Specificitylaw.inventionExcretionSchistosomiasis haematobiaSouth AfricalawVirologyParasite Egg CountmedicineAnimalsHumansChildParasite Egg CountPolymerase chain reactionSchistosomaSchistosoma haematobiumArticlesDNA Helminthbiology.organism_classificationInfectious DiseasesReal-time polymerase chain reactionSchistosoma haematobiumParasitologyFemale
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Bioactive pyrrole-based compounds with target selectivity

2020

The discovery of novel synthetic compounds with drug-like properties is an ongoing challenge in medicinal chemistry. Natural products have inspired the synthesis of compounds for pharmaceutical application, most of which are based on N-heterocyclic motifs. Among these, the pyrrole ring is one of the most explored heterocycles in drug discovery programs for several therapeutic areas, confirmed by the high number of pyrrole-based drugs reaching the market. In the present review, we focused on pyrrole and its hetero-fused derivatives with anticancer, antimicrobial, and antiviral activities, reported in the literature between 2015 and 2019, for which a specific target was identified, being resp…

Coronavirus disease 2019 (COVID-19)Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2)Antineoplastic AgentsReview ArticlePyrroleAntiviral Agentschemistry.chemical_compoundAnti-Infective AgentsDrug DiscoveryHumansPyrrolesMolecular Targeted TherapyAntiviralTargeted compoundsPyrrolePharmacologyDrug discoveryChemistryOrganic ChemistryCOVID-19Biological activityGeneral MedicineAntimicrobialSettore CHIM/08 - Chimica FarmaceuticaCombinatorial chemistryAnticancerDrug DesignAntimicrobialPharmacophoreSelectivityEuropean Journal of Medicinal Chemistry
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Development of a real-time PCR assay for detection and quantification of enterotoxigenic members of Bacillus cereus group in food samples

2009

A highly sensitive real-time PCR (qPCR) procedure, targeting the phosphatidylcholine-specific phospholipase C gene (pc-plc), was developed for specific detection and quantification of strains belonging to Bacillus cereus group. The target region was selected based on the enterotoxigenic profiles of 75 Bacillus strains. The inclusivity and exclusivity of the RTi-PCR assay were assessed with 59 isolates of the B. cereus group, 16 other Bacillus spp., and 4 non-Bacillus strains. The assay was also used to construct calibration curves for different food matrices, and it had a wide quantification range of 6 log units using both serial dilutions of purified DNA and calibrated cell suspensions of …

DNA BacterialSerial dilutionEggsMolecular Sequence DataColony Count MicrobialBacillus cereusFood ContaminationPolymerase Chain ReactionSensitivity and SpecificityMicrobiologyMicrobiologyEnterotoxinsBacillus cereusSpecies SpecificityHumansFood microbiologyDetection limitBacillus (shape)ChromatographybiologyfungiInfant NewbornInfantReproducibility of ResultsSequence Analysis DNAGeneral Medicinebiology.organism_classificationBacillalesInfant FormulaCereusCalibrationFood MicrobiologyFood ScienceFood contaminantInternational Journal of Food Microbiology
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Monoclonal anti-fosB antibody specific for predetermined, nonstructural region of the fosB protein.

1997

Comparison of the primary structures and theoretical prediction of the potential antigenic determinant of the deduced Fos proteins reveals the presence of a nonstructural and hydrophilic region juxtaposed to the leucine zipper and nonconserved among the Fos protein family. To develop monoclonal anti-peptide antibodies capable of distinguishing all Fos-proteins, synthetic peptides specific for the mentioned predicted region were synthesized manually by the "tea-bag" method. Immunization of Balb/c mice with fosB-related synthetic peptide BSA gave rise to mouse hybridoma cell line K21 (IgG1, kappa) secreting highly specific antibodies against corresponding human fosB protein. Fine mapping of t…

Leucine zippermedicine.drug_classImmunologyMolecular Sequence DataEnzyme-Linked Immunosorbent AssayMonoclonal antibodyEpitopeMiceAntibody SpecificityGeneticsmedicineAnimalsHumansAmino Acid SequencePeptide sequencebiologyProtein primary structureDrug Resistance MicrobialMolecular biologyPeptide FragmentsEpitope mappingbiology.proteinAntibodyProto-Oncogene Proteins c-fosEpitope MappingFOSBHybridoma
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Peptide Processing Is Critical for T-Cell Memory Inflation and May Be Optimized to Improve Immune Protection by CMV-Based Vaccine Vectors.

2016

Cytomegalovirus (CMV) elicits long-term T-cell immunity of unparalleled strength, which has allowed the development of highly protective CMV-based vaccine vectors. Counterintuitively, experimental vaccines encoding a single MHC-I restricted epitope offered better immune protection than those expressing entire proteins, including the same epitope. To clarify this conundrum, we generated recombinant murine CMVs (MCMVs) encoding well-characterized MHC-I epitopes at different positions within viral genes and observed strong immune responses and protection against viruses and tumor growth when the epitopes were expressed at the protein C-terminus. We used the M45-encoded conventional epitope HGI…

0301 basic medicineMuromegalovirusEpitopes T-LymphocyteCD8-Positive T-LymphocytesLymphocyte ActivationPathology and Laboratory MedicineBiochemistryEpitopeMass SpectrometryMiceWhite Blood Cells0302 clinical medicineAnimal CellsMedicine and Health SciencesCytotoxic T celllcsh:QH301-705.5Antigens ViralImmune ResponseStainingVaccines SyntheticbiologyT CellsCell StainingHerpesviridae InfectionsFlow CytometryRecombinant Proteins3. Good healthmedicine.anatomical_structureMedical MicrobiologyViral PathogensVirusesHuman CytomegalovirusCellular TypesPathogensResearch Articlelcsh:Immunologic diseases. AllergyHerpesvirusesT cellImmune CellsAntigen presentationImmunologyCytotoxic T cellsMajor histocompatibility complexResearch and Analysis MethodsMicrobiology03 medical and health sciencesViral ProteinsImmune systemAntigenVirologyGeneticsmedicineAnimalsAntigen-presenting cellMolecular Biology TechniquesMolecular BiologyMicrobial PathogensBlood CellsImmunodominant EpitopesOrganismsBiology and Life SciencesProteinsViral VaccinesCell BiologyVirology030104 developmental biologylcsh:Biology (General)Specimen Preparation and Treatmentbiology.proteinMutagenesis Site-DirectedParasitologylcsh:RC581-607PeptidesDNA virusesImmunologic Memory030215 immunologyChromatography LiquidCloningPLoS pathogens
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Gene expression specificity of the mussel antifungal mytimycin (MytM)

2011

Abstract We previously reported the nucleotide sequences and diversity of mytimycin (MytM) from the Mediterranean mussel, Mytilus galloprovincialis. Using real-time PCR (q-PCR), we observed that the MytM gene was mainly expressed in circulating hemocytes and to a less extent in the mantle. In vivo challenge with bacteria or with the yeast, Candida albicans, did not increase the expression as measured by q-PCR in hemocytes. By contrast, injection of the filamentous fungus, Fusarium oxysporum, induced a sudden and strong increase of expression at 9h p.i. (stimulation index of 25.7 ± 2.1). Optimum stimulating dose was 104 spores of F. oxysporum per mussel. In the same samples, AMP mytilin and …

Hemocytesbeta-GlucansspecificityStimulationAquatic ScienceMicrobiologyMicrococcusAntifungal peptidechemistry.chemical_compoundAdjuvants ImmunologicFusariumGene expressionEnvironmental ChemistryAnimalsCandida albicansVibrioMytilusInnate immunitybiologyQ-PCRMytilinGene Expression ProfilingGeneral MedicineMyticinbiology.organism_classificationYeastGene expression profilingchemistryGene Expression RegulationchallengeBacteriaAntimicrobial Cationic Peptides
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Inhibitory effect of sweet whey fermented by Lactobacillus plantarum strains against fungal growth: A potential application as an antifungal agent

2020

Abstract: The presence of mycotoxigenic fungi such as Aspergillus, Penicillium, and Fusarium genera represents a problem in food preservation and consequently, its spoilage. During the fermentation process with lactic acid bacteria, a range of secondary metabolites associated with beneficial health effects were released. In the present study, goat whey fermented by Lactobacillus plantarum (CECT 220, 221, 223, and 748) species has shown a satisfactory inhibitory effect against 28 fungi, showing for certain species of Fusarium genus and also, for Aspergillus steynii, a value of minimum inhibitory concentration until 1.95 g/L. In addition, phenyllactic acid was identified in each sample of fer…

FusariumPreservativeAntifungal Agentsfermentation proceFood spoilageMicrobial Sensitivity TestsShelf lifeFusariumWheymycotoxigenic fungiAnimalsFood sciencephenyllactic acidbiologyChemistryGoatsantifungal activitydigestive oral and skin physiologyPenicilliumFood preservationfood and beveragesbiology.organism_classificationAspergillusWhey ProteinsFermentationPenicilliumFermentationLactobacillus plantarumLactobacillus plantarumFood ScienceJournal of Food Science
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