Search results for "Opioides"

showing 3 items of 3 documents

Search for potential Angiotensin Converting Enzyme (ACE)-inhibitors from plants

2001

MeOH extracts, fractions and pure substances from Musanga cecropioides, Cecropia species and Crataegus oxyacantha /C. monogyna were screened by using an in vitro bio-assay based on the inhibition of Angiotensin Converting Enzyme (ACE), as measured from the enzymatic cleavage of the chromophore-fluorophore-labelled substrate dansyltriglycine into dansylglycine and diglycine. Phenolic acids showed no significant ACE-inhibition whereas flavonoids and proanthocyanidins demonstrated inhibitory activity at 0.33 mg/ml using this test system.

Musanga cecropioidesPharmaceutical ScienceAngiotensin-Converting Enzyme InhibitorsCrataegus oxyacanthaCleavage (embryo)AnthocyaninsDiglycineDrug DiscoveryHumansProanthocyanidinsFlavonoidsPharmacologychemistry.chemical_classificationPlants MedicinalbiologyPlant ExtractsChemistryAngiotensin-converting enzymebiology.organism_classificationIn vitroEnzymeComplementary and alternative medicineBiochemistryProanthocyanidinbiology.proteinMolecular MedicinePhytomedicine
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Recomendaciones prácticas para el manejo del paciente con dolor crónico durante la pandemia de COVID-19

2021

Resumen La infeccion por SARS-CoV-2 ha evolucionado hasta convertirse progresivamente en una pandemia y en una emergencia de salud publica de importancia internacional que ha obligado a las organizaciones de salud a nivel mundial, regional y local a adoptar una serie de medidas para hacer frente a la COVID-19 e intentar disminuir su impacto, no solo en el ambito social sino tambien en el ambito sanitario, modificandose las pautas de actuacion en los servicios de salud. Dentro de estas recomendaciones, que incluyen las unidades de tratamiento del dolor, los pacientes con sospecha o infeccion confirmada por SARS-CoV-2 pueden encontrase en situacion de espera para consulta medica o tecnicas in…

medicine.medical_specialtyCoronavirus disease 2019 (COVID-19)Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2)Critical Care and Intensive Care MedicineArticleHealth servicesHealth personnelSpecial Article03 medical and health sciences0302 clinical medicinePandemicHumansPain ManagementMedicine030212 general & internal medicineOpioidesPandemicsSARS-CoV-2business.industryRisk of infectionPublic healthChronic painManejo del dolorCOVID-19General Medicinemedicine.diseaseDolor crónicoOpioidsAnesthesiology and Pain MedicineEsteroidesSteroidsMedical emergencyChronic PainbusinessHumanities030217 neurology & neurosurgeryRevista Española de Anestesiología y Reanimación
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Prolonged-release buprenorphine formulations: Perspectives for clinical practice

2020

International audience; Buprenorphine and methadone are the two main opioid agonist treatments approved for opioid use disorder. Buprenorphine is a partial agonist of the mu opioid receptors, which has been merely available through sublingual form until now. In practice, the use of buprenorphine is smoother than that of methadone, and it induces reduced risks of overdose. However, sublingual buprenorphine also exposes to risks (e.g., withdrawal, misuse) and constraints (e.g., daily intake). Three new galenic formulations of prolonged-release buprenorphine (PRB) are being commercialized and should allow some improvements in patients' comfort and safety. This narrative review aims to describe…

medicine.medical_specialtyDoseNarcotic Antagonists[SDV.MHEP.PSM] Life Sciences [q-bio]/Human health and pathology/Psychiatrics and mental healthReceptors Opioid mu030226 pharmacology & pharmacyPartial agonistOpioid dependenceDependance aux opioides03 medical and health sciencesSubcutaneous injection0302 clinical medicineProlonged releasemedicineHumansProlonged-releasePharmacology (medical)OpiacésAction prolongeebusiness.industryOpioid use disorderOpioid-Related Disordersmedicine.disease3. Good healthBuprenorphineAnalgesics OpioidOpiatesOpioid[SDV.MHEP.PSM]Life Sciences [q-bio]/Human health and pathology/Psychiatrics and mental healthEmergency medicinebusinessSubstitutionMethadoneBuprenorphinemedicine.drugMethadone
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