Search results for "Osmolar Concentration"

showing 10 items of 106 documents

Response of yeast cells to high glucose involves molecular and physiological differences when compared to other osmostress conditions.

2015

Yeast cells can be affected by several causes of osmotic stress, such as high salt, sorbitol or glucose concentrations. The last condition is particularly interesting during natural processes where this microorganism participates. Response to osmostress requires the HOG (High Osmolarity Glycerol) pathway and several transcription factors, including Hot1, which plays a key role in high glucose concentrations. In this work, we describe how the yeast response to osmotic stress shows differences in accordance with the stress agent responsible for it. Compared with other conditions, under high glucose stress, delocalization of MAPK (Mitogen-Activated Protein Kinase) Hog1 is slower, induction of …

Snf3Saccharomyces cerevisiae ProteinsOsmotic shockTranscription GeneticSaccharomyces cerevisiaeChitinSaccharomyces cerevisiaeOsmosisApplied Microbiology and BiotechnologyMicrobiologychemistry.chemical_compoundOsmotic PressureGene Expression Regulation FungalSorbitolProtein kinase AbiologyGlycogenEthanolBenzenesulfonatesOsmolar ConcentrationGeneral Medicinebiology.organism_classificationYeastDNA-Binding ProteinsRepressor ProteinsBasic-Leucine Zipper Transcription FactorsGlucosechemistryBiochemistrySorbitolMitogen-Activated Protein KinasesTranscription FactorsFEMS yeast research
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Ion-exchange fibers and drugs: an equilibrium study

2001

The purpose of this study was to investigate the mechanisms of drug binding into and drug release from cation-exchange fibers in vitro under equilibrium conditions. Ion-exchange groups of the fibers were weakly drug binding carboxylic acid groups (-COOH), strongly drug binding sulphonic acid groups (-SO(3)H), or combinations thereof. Parameters determining the drug absorption and drug release properties of the fibers were: (i) the lipophilicity of the drug (tacrine and propranolol are lipophilic compounds, nadolol is a relatively hydrophilic molecule), (ii) the ion-exchange capacity of the fibers, which was increased by activating the cation-exchange groups with NaOH, (iii) the ionic streng…

SodiumCarboxylic acidPharmaceutical Sciencechemistry.chemical_element02 engineering and technology030226 pharmacology & pharmacyDivalent03 medical and health sciencesDrug Delivery Systems0302 clinical medicineFiberchemistry.chemical_classificationChromatographyOsmolar Concentration021001 nanoscience & nanotechnologyPropranololIon ExchangeNadololSolubilitychemistryIonic strengthLipophilicityTacrineCalcium0210 nano-technologyDrug carrierDrug metabolismNuclear chemistry
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Dispersive solid-phase extraction based on oleic acid-coated magnetic nanoparticles followed by gas chromatography-mass spectrometry for UV-filter de…

2011

Abstract A sensitive analytical method to concentrate and determine extensively used UV filters in cosmetic products at (ultra)trace levels in water samples is presented. The method is based on a sample treatment using dispersive solid-phase extraction (dSPE) with laboratory-made chemisorbed oleic acid-coated cobalt ferrite (CoFe 2 O 4 @oleic acid) magnetic nanoparticles (MNPs) as optimized sorbent for the target analytes. The variables involved in dSPE were studied and optimized in terms of sensitivity, and the optimum conditions were: mass of sorbent, 100 mg; donor phase volume, 75 mL; pH, 3; and sodium chloride concentration, 30% (w/v). After dSPE, the MNPs were eluted twice with 1.5 mL …

SorbentBiochemistrySensitivity and SpecificityGas Chromatography-Mass SpectrometryAnalytical ChemistryTap waterRiversSample preparationSolid phase extractionMagnetite NanoparticlesDetection limitChromatographyElutionChemistryOrganic ChemistryExtraction (chemistry)Osmolar ConcentrationSolid Phase ExtractionReproducibility of ResultsWaterGeneral MedicineHydrogen-Ion ConcentrationGas chromatography–mass spectrometrySunscreening AgentsWater Pollutants ChemicalOleic AcidJournal of chromatography. A
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Different Dissolution Media Lead to Different Crystal Structures of Talinolol with Impact on Its Dissolution and Solubility

2003

During the performance of dissolution tests with immediate and controlled-release talinolol tablets it was detected that the type of the buffer used as dissolution medium had a strong influence on the solubility and the dissolution behavior of the drug. It was proven that talinolol appeared in different crystal structures with strongly differing solubilities when pure water, acetate, or phosphate buffers were employed as dissolution media. The resulting crystal structures were characterized by means of light microscopy, differential scanning calorimetry, and X-ray powder diffraction. All methods were adjuvant to detect changes in talinolol crystal structures. The different solubility and di…

Surface PropertiesSodiumAdrenergic beta-AntagonistsPharmaceutical Sciencechemistry.chemical_elementSodium ChlorideDosage formlaw.inventionPropanolamineschemistry.chemical_compoundX-Ray DiffractionPulmonary surfactantlawDrug DiscoverySolubilityCrystallizationDissolutionPharmacologyChromatographyCalorimetry Differential ScanningChemistryOsmolar ConcentrationOrganic ChemistryHydrogen-Ion ConcentrationSolubilityIonic strengthDelayed-Action PreparationsSolventsCrystallizationTalinololNuclear chemistryDrug Development and Industrial Pharmacy
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Analysis of intrapulmonary O2concentration by MR imaging of inhaled hyperpolarized helium-3

1999

Inhalation of hyperpolarized 3He allows magnetic resonance imaging (MRI) of ventilated airspaces.3He hyperpolarization decays more rapidly when interacting with paramagnetic O2. We describe a method for in vivo determination of intrapulmonary O2 concentrations ([O2]) based on MRI analysis of the fate of measured amounts of inhaled hyperpolarized3He in imaged regions of the lung. Anesthetized pigs underwent controlled normoventilation in a 1.5-T MRI unit. The inspired O2 fraction was varied to achieve different end-tidal [O2] fractions ([Formula: see text]). With the use of a specifically designed applicator,3He (100 ml, 35–45% polarized) was administered at a predefined time within single …

SwinePhysiologychemistry.chemical_elementHyperpolarized Helium 3HeliumOxygenIsotopesPhysiology (medical)Administration InhalationTidal VolumemedicineAnimalsHyperpolarization (physics)Respiratory systemLungTidal volumeLungmedicine.diagnostic_testInhalationbusiness.industryRespirationOsmolar ConcentrationMagnetic resonance imagingMagnetic Resonance ImagingOxygenmedicine.anatomical_structurechemistryFeasibility StudiesNuclear medicinebusinessJournal of Applied Physiology
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Use of the Transglutaminase Reaction To Study the Dissociation of Histone N-Terminal Tails from DNA in Nucleosome Core Particles

1997

We have recently shown that core histones are glutaminyl substrates for transglutaminase (TGase) and that when native nucleosome cores are incubated with monodansylcadaverine (DNC) as donor amine, this fluorescent probe is incorporated into Gln5 and Gln19 of H3 and in Gln22 of H2B [Ballestar et al. (1996) J. Biol. Chem. 271, 18817-18825]. In the present paper, we report that the cause by which Gln22 of H2B is modified in nucleosomes but not in the free histone is the interaction of the region containing that glutamine with DNA. We have used the specificity of the TGase reaction to study the changes induced by increasing ionic strength in the interaction between the histone N-terminal tails …

TransglutaminasesbiologyMovementOsmolar ConcentrationFluorescence PolarizationDNABiochemistryLinker DNAMolecular biologyNucleosomesHistoneschemistry.chemical_compoundHistoneModels ChemicalchemistryIonic strengthCadaverineChromatosomeBiophysicsbiology.proteinNucleosomeHistone octamerFluorescence anisotropyDNABiochemistry
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Fractionated precipitation of acid macropolyanions by dialysis, a simple method for the estimation of DNA in complex biological samples.

1976

Abstract After efficient extraction by para-aminosalicylate, (hopping, grinding and eventual sonication, the macropolyanions are transformed into their cetyltrimethylammonium salts. These have differing solubilities, strongly depending on ionic strength. The cationic detergent-macropolyanionic salts are solubilized by high salt concentration. Salt is then dialysed out, rendering the polyanions highly insoluble in a sequential fashion. The insolubilized components are determined quantitatively by monitoring turbidity, which in case of DNA is strictly proportionate to its concentration. This relation is not affected by other components. This makes DNA determination possible even in crude aque…

chemistry.chemical_classificationAnionsChromatographyAqueous solutionPrecipitation (chemistry)TroutSonicationExtraction (chemistry)Osmolar ConcentrationSalt (chemistry)DNASaccharomyces cerevisiaeBiologyGeneral Biochemistry Genetics and Molecular BiologySoilActivated sludgechemistryIonic strengthCetrimonium CompoundsMethodsAnimalsChemical PrecipitationTurbidityDialysisZeitschrift fur Naturforschung. Section C, Biosciences
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Sequence-specific and DNA structure-dependent interactions of Escherichia coli MutS and human p53 with DNA

2013

Many proteins involved in DNA repair systems interact with DNA that has structure altered from the typical B-form helix. Using magnetic beads to immobilize DNAs containing various types of structures, we evaluated the in vitro binding activities of two well-characterized DNA repair proteins, Escherichia coli MutS and human p53. E. coli MutS bound to double-stranded DNAs, with higher affinity for a G/T mismatch compared to a G/A mismatch and highest affinity for larger non-B-DNA structures. E. coli MutS bound best to DNA between pH 6 and 9. Experiments discriminated between modes of p53-DNA binding, and increasing ionic strength reduced p53 binding to nonspecific double-stranded DNA, but had…

chemistry.chemical_classificationDNA ligaseDNA clampHMG-boxBase pairEscherichia coli ProteinsOsmolar ConcentrationBiophysicsDNACell BiologyBiologyBiochemistryMutS DNA Mismatch-Binding ProteinDNA binding siteBiochemistrychemistryMutS-1Escherichia coliHumansNucleic Acid ConformationProtein–DNA interactionAmino Acid SequenceTumor Suppressor Protein p53Molecular BiologyReplication protein AAnalytical Biochemistry
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Competing salt effects on phase behavior of protein solutions: tailoring of protein interaction by the binding of multivalent ions and charge screeni…

2014

The phase behavior of protein solutions is affected by additives such as crowder molecules or salts. In particular, upon addition of multivalent counterions, a reentrant condensation can occur; i.e., protein solutions are stable for low and high multivalent ion concentrations but aggregating at intermediate salt concentrations. The addition of monovalent ions shifts the phase boundaries to higher multivalent ion concentrations. This effect is found to be reflected in the protein interactions, as accessed via small-angle X-ray scattering. Two simulation schemes (a Monte Carlo sampling of the counterion binding configurations using the detailed protein structure and an analytical coarse-grain…

chemistry.chemical_classificationIonsCondensationOsmolar ConcentrationSurfaces Coatings and FilmsIonProtein–protein interactionProtein structurechemistryX-Ray DiffractionIonic strengthComputational chemistryPhase (matter)Scattering Small AngleMaterials ChemistryMoleculeHumansSaltsPhysical and Theoretical ChemistryCounterionSerum AlbuminThe journal of physical chemistry. B
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A minireview on NHE1 inhibitors. A rediscovered hope in oncohematology.

2015

Background: Na+/H+ exchanger-1 (NHE-1) is involved in pH regulation and is up-regulated in different malignancies. Activation of NHE-1 is one way for allowing cells to avoid intracellular acidification and protect them against apoptosis. Inhibitors of NHE-1 are able to decrease intracellular pH and induce apoptosis. Some statins can also act by partial inhibition of NHE-1. This review presents progress in understanding the mechanisms of action of these inhibitors, connections with certain genetic mutations and acquired treatment resistance, as well as new patents on them. Methods: A MEDLINE search for original and review articles using key terms, Na+/H+ exchanger, leukemia, cariporide, and …

lovastatinlcsh:MedicineApoptosisPharmacologyGuanidinesAmiloridep-glycoproteinhemic and lymphatic diseasesDrug InteractionsSulfonesCation Transport ProteinsSodium-Hydrogen Exchanger 1leukemiaMyeloid leukemiaHydrogen-Ion ConcentrationSorafenibUp-RegulationLeukemiaLeukemia Myeloid AcuteImatinib MesylateSignal transductionTyrosine kinasemedicine.drugSignal TransductionSorafenibNiacinamideisoprenylationSodium-Hydrogen Exchangersbcr/ablAntineoplastic AgentsGenes ablGeneral Biochemistry Genetics and Molecular BiologystatinsPatents as TopicCell Line TumorLeukemia Myelogenous Chronic BCR-ABL PositivemedicineHumansProtein Kinase Inhibitorscariporidena+/h+ exchangerTumor hypoxiabusiness.industryPhenylurea Compoundslcsh:ROsmolar Concentrationintracellular phmedicine.diseaseImatinib mesylatefms-Like Tyrosine Kinase 3Fms-Like Tyrosine Kinase 3MutationCancer researchTumor Hypoxiaflt3/itdHydroxymethylglutaryl-CoA Reductase InhibitorsbusinessHeme Oxygenase-1DNA DamageBiomedical papers of the Medical Faculty of the University Palacky, Olomouc, Czechoslovakia
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