Search results for "Phenanthrene"
showing 10 items of 101 documents
CCDC 783766: Experimental Crystal Structure Determination
2011
Related Article: V.Blanco, M.D.Garcia, A.Terenzi, E.Pia, A.Fernandez-Mato, C.Peinador, J.M.Quintela|2010|Chem.-Eur.J.|16|12373|doi:10.1002/chem.201002051
CCDC 2074636: Experimental Crystal Structure Determination
2021
Related Article: Jaroslav Jacko, Monika Staś, Lubomír Rulíšek, Ivana Císařová, Martin Kotora|2022|J.Org.Chem.|87|744|doi:10.1021/acs.joc.1c01118
CCDC 766950: Experimental Crystal Structure Determination
2010
Related Article: S.Ikonen, Nonappa, A.Valkonen, R.Juvonen, H.Salo, E.Kolehmainen|2010|Org.Biomol.Chem.|8|2784|doi:10.1039/c003228j
CCDC 910388: Experimental Crystal Structure Determination
2013
Related Article: Y.Inokuma,S.Yoshioka,J.Ariyoshi,T.Arai,Y.Hitora,K.Takada,S.Matsunaga,K.Rissanen,M.Fujita|2013|Nature (London)|495|461|doi:10.1038/nature11990
CCDC 2074635: Experimental Crystal Structure Determination
2021
Related Article: Jaroslav Jacko, Monika Staś, Lubomír Rulíšek, Ivana Císařová, Martin Kotora|2022|J.Org.Chem.|87|744|doi:10.1021/acs.joc.1c01118
CCDC 804367: Experimental Crystal Structure Determination
2015
Related Article: Kathrin Wehming, Moritz Schubert, Gregor Schnakenburg, Siegfried R. Waldvogel|2014|Chem.-Eur.J.|20|12463|doi:10.1002/chem.201403442
3,4-Dihydroxy- and 3,4-methylenedioxy- phenanthrene-type alkaloids with high selectivity for D2 dopamine receptor.
2013
Abstract Dopamine-mediated neurotransmission plays an important role in relevant psychiatric and neurological disorders. Nowadays, there is an enormous interest in the development of new drugs acting at the dopamine receptors (DR) as potential new targets for the treatment of schizophrenia or Parkinson’s disease. Previous studies have revealed that isoquinoline compounds such as tetrahydroisoquinolines (THIQs) can behave as selective D 2 dopaminergic alkaloids. In the present study we have synthesized five aporphine compounds and five phenanthrene alkaloids and evaluated their potential dopaminergic activity. Binding studies on rat striatal membranes were used to evaluate their affinity and…
Synthesis of Polyfused Heterocycle Derivatives Containing the Dipyridoimidazole Core by Friedländer’s Reaction: Access to Analogs of Ellipticine
2005
Reaction of 3-amino-2-formylimidazo[l,2-a]pyridine with various aldehydes and ketones by Friedlander's methodology afforded an entry to dipyridoimidazole, tri(tetra)azacyclopenta[b]fluorene, tri(tetra)azabenzo[b]-fluorene and triazaindeno[2,1-b]phenanthrene derivatives. Intercalation with a synthetic oligodeoxynucleotide was examined.
Differential Enantioselectivity of Murine GlutathioneS-Transferase Isoenzymes in the Glutathione Conjugation ofTrans-3,4-dihydroxy-1,2-oxy- 1,2,3,4-t…
1998
Abstract The kinetics of the glutathione (GSH) conjugation of (+)- and (−)-enantiomers ofanti- as well assyn-3,4-dihydroxy-1,2-oxy-1,2,3,4-tetrahydrobenzo[c]phenanthrene (B[c]PDE) catalyzed by murine GSHS-transferase (GST) isoenzymes has been investigated. Murine GSTs exhibited significant differences in their enantioselectivity toward B[c]PDE stereoisomers. For example, while pi class isoenzyme mGSTP1-1 was virtually inactive toward stereoisomers with 1Sconfiguration [(−)-syn-and (+)-anti-B[c]PDE], these stereoisomers were good substrates for alpha class isoenzyme mGSTA1-2. When GST activity was measured as a function of varying B[c]PDE concentration (10–320 μM) at a fixed saturating conce…
DFT studies of COOH tip-functionalized zigzag and armchair single wall carbon nanotubes
2011
Structure and energy calculations of pristine and COOH-modified model single wall carbon nanotubes (SWCNTs) of different length were performed at B3LYP/6-31G* level of theory. From 1 to 9 COOH groups were added at the end of the nanotube. The differences in structure and energetics of partially and fully functionalized SWCNTs at one end of the nanotube are observed. Up to nine COOH groups could be added at one end of (9,0) zigzag SWCNT in case of full functionalization. However, for (5,5) armchair SWCNT, the full functionalization was impossible due to steric crowding and rim deformation. The dependence of substituent attachment energy on the number of substituents at the carbon nanotube ri…