Search results for "Pines"

showing 10 items of 421 documents

Synthesis and biological evaluation of papain-family cathepsin L-like cysteine protease inhibitors containing a 1,4-benzodiazepine scaffold as antipr…

2014

Novel papain-family cathepsin L-like cysteine protease inhibitors endowed with antitrypanosomal and antimalarial activity were developed, through an optimization study of previously developed inhibitors. In the present work, we studied the structure-activity relationships of these derivatives, with the aim to develop new analogues with a simplified and more synthetically accessible structure and with improved antiparasitic activity. The structure of the model compounds was significantly simplified by modifying or even eliminating the side chain appended at the C3 atom of the benzodiazepine scaffold. In addition, a simple methylene spacer of appropriate length was inserted between the benzod…

Trypanosomamedicine.drug_classPeptidomimeticStereochemistryAntiparasiticCell SurvivalCathepsin LAntiprotozoal AgentsCysteine Proteinase InhibitorsBiochemistryCathepsin BCell LineCathepsin Lchemistry.chemical_compoundBenzodiazepinesMiceStructure-Activity RelationshipDrug DiscoverymedicineMoietyAnimalsGeneral Pharmacology Toxicology and PharmaceuticsPharmacologyCathepsinbiologyOrganic ChemistryCombinatorial chemistryCysteine proteasePapainantiprotozoal agents; inhibitors; Malaria; Peptidomimetics; structure-activity relationshipsCysteine EndopeptidaseschemistryAntiprotozoalbiology.proteinMolecular MedicineProtein BindingChemMedChem
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Bene vivere politice

2022

Abstract This chapter approaches the question of biopolitics in ancient political thought looking not at specific political techniques but at notions of the final aim of the political community. It argues that the “happiness” (eudaimonia, beatitudo) that constitutes the greatest human good in the tradition from Aristotle to Thomas Aquinas is not a “biopolitical” ideal, but rather a metabiopolitical one, consisting in a contemplative activity situated above and beyond the biological and the political. It is only with Thomas Hobbes that civic happiness becomes “biopolitically” identified with simple survival; for modernity, as Hannah Arendt puts it, mere being alive becomes the greatest human…

Tuomas Akvinolainensupreme goodAristotelespoliittinen osallistuminenkeskiajan filosofiaelämänlaatupoliittinen filosofiahyväArendt HannahbiopoliticsHobbes ThomasAristotleThomas AquinasFoucault Michelhappinessmetabiopolitiikkaantiikin filosofiabiopolitiikkaonnellisuushyvä elämäOjakangas Mikametabiopolitics
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Liderazgo transformacional, capacidad de aprendizaje organizativo y felicidad en el trabajo

2013

En los últimos veinte años se ha producido un incremento de los artículos que buscan cómo mejorar el resultado económico en las empresas. No hay duda de la importancia que tiene esta variable como fin último de cualquier investigación, sin embargo, en este estudio queremos proponer una variable que consideramos de especial relevancia para la investigación en el área de organización de empresas como es la felicidad en el trabajo. La felicidad en general está directamente conectada con beneficios tan importantes como la salud física o mental, y las medidas que hasta ahora se han aproximado a la felicidad en el trabajo se han relacionado con variables tan importantes como la mejora de la motiv…

UNESCO::CIENCIAS ECONÓMICAS::Organización y dirección de empresas ::Organización de recursos humanosliderazgocapacidad de aprendizaje organizativoUNESCO::CIENCIAS ECONÓMICASsatisfacción laboral:CIENCIAS ECONÓMICAS [UNESCO]UNESCO::CIENCIAS ECONÓMICAS::Organización y dirección de empresasorganizational learning capability:CIENCIAS ECONÓMICAS::Organización y dirección de empresas ::Organización de recursos humanos [UNESCO]transformational leadershipaprendizaje organizativohappinessliderazgo transformacionalfelicidad:CIENCIAS ECONÓMICAS::Organización y dirección de empresas [UNESCO]job satisfaction
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Development of the Happiness Index in a country

2016

[EN] In this paper, a Happiness Index is built through the Human Dignity Respect Index which is explained by Author (2014). The index is created using three main values: development, freedom and equality. But the equality is explained by solidarity, justice and peace. Then, the Happiness Index is developed with this five concepts. The aim of this paper is to obtain the minimum quantitative variables to explain these values as well as to obtain a generic formula, which allows measuring the happiness of a country/region. The term “generic” is introduced because this formula could be extrapolated to any country. The variables to obtain the Development Index are health (Life Expectancy at birth…

Value (ethics)Index (economics)media_common.quotation_subjectOverall Life Satisfaction IndexEconomic JusticeSolidarityHappiness indexSocial groupDignityUNDPHappinessmedia_common.cataloged_instanceSociologyClassical economicsEuropean unionSocial psychologymedia_commonLibro de Actas - Systems & Design: Beyond Processes and Thinking (IFDP - SD2016)
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Operationalization of un-captured GDP - Innovation stream under new global mega-trends

2016

With the understanding that current ICT-driven global development depends on a trend shifting from traditional co-evolution of computer-initiated ICT, captured GDP, and economic functionality to new co-evolution of the Internet, un-captured GDP, and supra-functionality beyond economic value, the following hypothetical view was postulated: The disparity between the world's ICT leader countries with respect to happiness/welfare amidst great stagnation (Finland) or conspicuous economic growth (Singapore) can be attributed to the difference of the state in the above shifting trends. The foregoing hypothetical view was demonstrated on the basis of an empirical analysis measuring dependency on un…

Value (ethics)Sociology and Political Science020209 energymedia_common.quotation_subjectHuman Factors and ErgonomicsContext (language use)02 engineering and technologyEducationinteractive return gain structure0502 economics and business0202 electrical engineering electronic engineering information engineeringEconomicsBusiness and International Managementmedia_commonta113GovernmentOperationalizationmuscular economic environment05 social sciencesVirtuous circle and vicious circleco-evolution of 3 mega-trendsEconomyHappinessun-captured GDPEconomic systemInternational developmentWelfare050203 business & managementTechnology in Society
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Co-Creation of Value for IT-Enabled Services : A Case of Geocaching

2013

This study explores how value is co-created in one particular IT-enabled service, geocaching. Consumer Information Systems (CIS) framework is used as a sensitizing framework to study experienced geocachers' (n=14) perceptions of what they value in geocaching. The following core values emerged that motivate people to co-create value in geocaching: challenging oneself and others, joy of success, learning, and social relations. The results reveal that geocaching is distinctively hedonic in nature, as people pursue happiness and utility via geocaching. Even support for the geocaching community was motivated by such values. In addition, the results reveal that the environment of geocaching and s…

Value (ethics)media_common.quotation_subjectInternet privacyContext (language use)information systemskäyttäjälähtöisyysConsumer informationGlobal Positioning SystemCo-creationInformation systemSociologymedia_commontietojärjestelmätService (business)ta113geographic information systemsbusiness.industryyhteisöllisyysgeokätköilyPublic relationsSocial relationvalue co-creationHappinessbusinessIT enabled servicesmotivointi
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Sense-Making, Meaningfulness, and Instrumental Music Education

2020

The purpose of this paper is to re-examine the nature of "meaning" and "meaningfulness" in the context of instrumental music education. By doing so, I propose to expand the ways in which instrumental music educators conceive their mission and the ways in which we may instill meaning in people's lives. Traditionally, pursuits of philosophical deliberation have claimed that meaningfulness comes from either personal happiness (e.g., Jeremy Bentham and John Stuart Mill) or an impersonal sense of duty (e.g., St. Augustine, St. Thomas Aquinas, and Immanuel Kant). However, philosopher Wolf (2010) criticizes these positions in favor of a broader perspective, one that arises from understanding that …

Value (ethics)media_common.quotation_subjectinstrumental music teaching and learninglcsh:BF1-990Context (language use)DeliberationMusic educationsense-makingeudaimonia (well being)EudaimoniaEpistemologylcsh:PsychologyHypothesis and Theoryenaction and embodied cognitionmeaningfulness and motivationHappinessPsychologyMeaning (existential)PsychologyDutyGeneral Psychologymedia_commonFrontiers in Psychology
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Staphylococcus aureus alpha toxin mediates polymorphonuclear leukocyte-induced vasocontraction and endothelial dysfunction.

2002

The effect of Staphylococcus aureus alpha toxin (alpha-toxin) on selectin-mediated neutrophil adhesion was investigated in polymorphonuclear leukocyte- (PMN) induced vasocontraction and endothelial dysfunction. Adherence of human PMNs to rat aortic endothelium increased significantly following stimulation of the endothelium with alpha-toxin (0.1, 0.5, and 1 microg/mL). This effect could be significantly attenuated by monoclonal antibodies directed against P-selectin or fucoidin, a carbohydrate known to block selectins. Unstimulated human PMNs (10(6)cells/mL) were added to organ chambers containing rat aortic rings stimulated with alpha-toxin (0.5 microg/mL). PMNs elicited a significant vaso…

Vascular smooth muscleEndotheliumNeutrophilsBacterial ToxinsPharmacologyBiologyIn Vitro TechniquesCritical Care and Intensive Care MedicineMicrocirculationHemolysin ProteinsFibrinolytic AgentsmedicineCell AdhesionAnimalsHumansEndothelial dysfunctionStaphylococcus aureus alpha toxinAortaThrombinAzepinesTriazolesmedicine.diseaseRatsmedicine.anatomical_structureVasoconstrictionImmunologyEmergency MedicineEndothelium Vascularmedicine.symptomVasoconstrictionSelectinBlood vesselShock (Augusta, Ga.)
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Fatigue, sleep, and nocturnal complaints in patients with amyotrophic lateral sclerosis

2012

Background and purpose: Fatigue is a common symptom in amyotrophic lateral sclerosis (ALS). Although sleep disturbances are a candidate factor that may interfere with fatigue in patients with ALS, the role of sleep-related abnormalities in determining fatigue in ALS is unknown. Objective: To evaluate the frequency and determinants of fatigue in a group of 91 consecutive patients with ALS, with special attention to the relationship between fatigue and sleep problems. Methods: Measures included the Fatigue Severity Scale (FSS), Pittsburgh Sleep Quality Index (PSQI), Epworth Sleepiness Scale (ESS), ALS Functional Rating ScaleRevised (ALSFRS-R), and Beck Depression Inventory (BDI). Results: The…

Vital capacitymedicine.medical_specialtybusiness.industryEpworth Sleepiness ScaleBeck Depression Inventorymedicine.diseasePittsburgh Sleep Quality IndexPhysical medicine and rehabilitationNeurologySeverity of illnessmedicinePhysical therapyNocturiaNeurology (clinical)medicine.symptomAmyotrophic lateral sclerosisbusinessMuscle crampEuropean Journal of Neurology
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The Conceptions of Quality of Life, Wellness and Well-Being: A Literature Review

2022

In the last few years, a growing body of research has been interested in wellness, quality of life, and well-being issues. Furthermore, institutions, governments, and policymakers start to introduce numerous physical and mental well-being programs, whereas scholars interested in well-being research use different indicators to evaluate them. Although these terms are popular in the scientific debate, they are variously interpreted and at the conceptual level do not have a standard definition. This disagreement is particularly relevant when considering the questions related to their measurement and application in empirical research. This review explores the main theoretical conceptions of qual…

WellneQuality of lifeSubjective well-beingSettore SPS/08 - Sociologia Dei Processi Culturali E ComunicativiHappinessLife satisfactionSettore SPS/07 - Sociologia Generale
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