Search results for "Plant Extract"

showing 10 items of 517 documents

Antiproliferative activity against leukemia cells of sesquiterpene lactones from the Turkish endemic plant Centaurea drabifolia subsp. detonsa

2017

The apolar organic extract obtained from aerial parts of Centaurea drabifolia Sibth. & Sm. subsp. detonsa (Bornm.) Wagenitz, growing wild in Turkey, was investigated for the first time for its secondary metabolite composition. Seven sesquiterpene lactones belonging to the guaiane class (1-7), including the new compound 4, along with a fatty acid lactone derivative (8), were isolated. The structures of these compounds were established by spectroscopic analysis, including 2D NMR spectroscopic techniques, with the stereostructure of the new guaiane 4 determined with the help of MTPA derivatization. Cytotoxic activities of compounds 1-7 were evaluated against two cancer cell lines, namely acute…

TurkeyCentaurea drabifoliaStereochemistryCynaropicrinCentaureaMultidrug-resistant cell lineSecondary metaboliteBiologySesquiterpene01 natural sciencesLactonesSesquiterpenes GuaianeStructure-Activity Relationshipchemistry.chemical_compoundCell Line TumorDrug DiscoverymedicineHumansDerivatizationPharmacologychemistry.chemical_classificationLeukemiaMolecular StructurePlant Extracts010405 organic chemistryFatty acidGeneral MedicinePlant Components AerialAntineoplastic Agents PhytogenicCynaropicrin0104 chemical sciences010404 medicinal & biomolecular chemistrychemistryDrug Resistance NeoplasmAntileukemic activityDrug Screening Assays AntitumorSesquiterpene lactonesSesquiterpenesTwo-dimensional nuclear magnetic resonance spectroscopyDerivative (chemistry)Lactonemedicine.drugFitoterapia
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Kinetic characterization of mitochondrial complex I inhibitors using annonaceous acetogenins

1999

The NADH:ubiquinone oxidoreductase (complex I) of the mitochondrial respiratory chain is by far the largest and most complicated of the proton-translocating enzymes involved in the oxidative phosphorylation. Many clues regarding the electron pathways from matrix NADH to membrane ubiquinone and the links of this process with the translocation of protons are highly controversial. Different types of inhibitors become valuable tools to dissect the electron and proton pathways of this complex enzyme. Therefore, further knowledge of the mode of action of complex I inhibitors is needed to understand the underlying mechanism of energy conservation. This study presents for the first time a detailed …

UbiquinoneSubmitochondrial ParticlesBiophysicsOxidative phosphorylationBiologyBiochemistryMitochondria HeartLactonesOxidoreductaseRotenoneNAD(P)H Dehydrogenase (Quinone)Mammalian enzymeAnimalsFuransMolecular Biologychemistry.chemical_classificationNADH-Ubiquinone OxidoreductasePlant ExtractsNADKineticsMitochondrial respiratory chainEnzymechemistryBiochemistryCattleAnnonaceous AcetogeninsMitochondrial Complex I
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Ultrasound-Assisted Extraction, Centrifugation and Ultrafiltration: Multistage Process for Polyphenol Recovery from Purple Sweet Potatoes

2016

This work provides an evaluation of an ultrasound-assisted, combined extraction, centrifugation and ultrafiltration process for the optimal recovery of polyphenols. A purple sweet potato (PSP) extract has been obtained using ultrasonic circulating extraction equipment at a power of 840 W, a frequency of 59 kHz and using water as solvent. Extract ultrafiltration, using polyethersulfone (PES), was carried out for the recovery of polyphenol, protein and anthocyanin. Pre-treatment, via the centrifugation of purple sweet potato extract at 2500 rpm over 6 min, led to better polyphenol recovery, with satisfactory protein removal (reused for future purposes), than PSP extract filtration without cen…

Ultrafiltrationpurple sweet potatoAgronomiaPharmaceutical Science01 natural sciencesArticleAnalytical Chemistrylaw.inventionAnthocyaninslcsh:QD241-441chemistry.chemical_compound0404 agricultural biotechnologylcsh:Organic chemistrylawDrug DiscoveryCentrifugation; Filtration; Polyphenols; Purple sweet potato; Ultrasound; Anthocyanins; Chromatography High Pressure Liquid; Ipomoea batatas; Plant Extracts; Polyphenols; Ultrasonics; Medicine (all); Organic ChemistryCentrifugationUltrasonicspurple sweet potato; ultrasound; polyphenols; filtration; centrifugationPhysical and Theoretical ChemistryIpomoea batatasFiltrationChromatography High Pressure LiquidpolyphenolsfiltrationcentrifugationQuímica agrícolaChromatographyChromatographyFoulingPlant ExtractsultrasoundMedicine (all)010401 analytical chemistryExtraction (chemistry)Organic Chemistry04 agricultural and veterinary sciences040401 food science0104 chemical sciencesSolventchemistryChemistry (miscellaneous)PolyphenolAnthocyaninHigh Pressure LiquidMolecular MedicineMolecules; Volume 21; Issue 11; Pages: 1584
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Antioxidant betalains from cactus pear (Opuntia ficus-indica) inhibit endothelial ICAM-1 expression.

2004

It has been suggested that some pigments would have antioxidant properties and that their presence in dietary constituents would contribute to reduce the risk of oxidative stress–correlated diseases. Among others, inflammatory response depends on redox status and may implicate oxidative stress. Vascular endothelial cells are a direct target of oxidative stress in inflammation. We have tested the impact of the free radical scavenger and antioxidant properties of betalains from the prickle pear in an in vitro model of endothelial cells. Here we show the capacity of betalains to protect endothelium from cytokine- induced redox state alteration, through ICAM-1 inhibition. KEYWORDS: endothelial …

Umbilical VeinsAntioxidantEndotheliumICAM-1Pyridinesmedicine.medical_treatmentAnti-Inflammatory AgentsBetalainsInflammationOxidative phosphorylationBiologymedicine.disease_causeModels BiologicalGeneral Biochemistry Genetics and Molecular BiologyAntioxidantschemistry.chemical_compoundHistory and Philosophy of ScienceSettore BIO/10 - BiochimicamedicineHumansCells CulturedInflammationICAM-1Dose-Response Relationship DrugPlant ExtractsGeneral NeurosciencebetalainOpuntiaFree radical scavengerFlow CytometryIntercellular Adhesion Molecule-1BetaxanthinsQuaternary Ammonium CompoundsOxidative Stressmedicine.anatomical_structurechemistryBiochemistryendothelial cellendothelial cells; ICAM-1; betalains; antiinflammatory drugsCytokinesEndothelium Vascularantiinflammatory drugsmedicine.symptomIndicaxanthinOxidation-ReductionOxidative stressAnnals of the New York Academy of Sciences
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Phytoestrogens increase the capacity of serum to stimulate prostacyclin release in human endothelial cells

2003

Both the estrogen receptor (ER) alpha and beta isoforms are expressed in the endothelium. The ER beta has been assigned a crucial role in normal vascular wall function. Prostacyclin has been ascribed a beneficial effect on vessel wall physiology. Isoflavones bind with higher affinity to ER beta. We investigated the hypothesis that their administration to postmenopausal women can promote endothelial prostacyclin production.Twenty-five healthy postmenopausal women with mild climacteric symptoms received capsules containing 55 mg/day isoflavones derived from soy and red clover for 6 months. Cultured human umbilical vein endothelial cells (HUVECs) were exposed for 24 h to serum collected before…

Umbilical Veinsmedicine.medical_specialtyTime FactorsEndotheliumAdministration OralAlpha (ethology)Estrogen receptorPhytoestrogensProstacyclinDrug Administration ScheduleUmbilical veinchemistry.chemical_compoundInternal medicinemedicineHumansEstrogens Non-SteroidalEstrogen receptor betaPlant Extractsbusiness.industryObstetrics and GynecologyGeneral MedicineMiddle AgedIsoflavonesBlood Physiological PhenomenaEpoprostenolIsoflavonesPostmenopauseEndocrinologymedicine.anatomical_structurechemistryFemaleTrifoliumPhytoestrogensEndothelium VascularPlant PreparationsSoybeansbusinessPlatelet Aggregation Inhibitorsmedicine.drugActa Obstetricia et Gynecologica Scandinavica
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Activity investigation of pinostrobin towards herpes simplex virus-1 as determined by atomic force microscopy

2009

In the present study, the antiviral activity of pinostrobin towards herpes simplex virus-1 (HSV-1) was investigated by MTT assay and atomic force microscopy. Pinostrobin can inhibit HSV-1 replication with 50% effective concentration (EC(50)) of 22.71 ± 1.72 μg/ml. MTT assay showed HSV-1 was significantly inhibited when pretreated with pinostrobin, with the inhibition of 85.69 ± 2.59%. Significant changes in morphology and size of HSV-1 were observed by atomic force microscopy (AFM) in response to pinostrobin treatment. AFM topography and phase images showed that with increasing time, the envelope was shedded and damaged, finally leading to virus inactivation. With increasing concentration, …

Virus inactivationPharmaceutical ScienceMice Inbred StrainsHerpesvirus 1 HumanMicrobial Sensitivity TestsMicroscopy Atomic Forcemedicine.disease_causePhase imageMiceIn vivoChlorocebus aethiopsDrug DiscoverymedicineAnimalsMTT assayTreatment effectVero CellsPharmacologyPlant ExtractsChemistryAtomic force microscopyHerpes SimplexVirologyHerpes simplex virusComplementary and alternative medicineFlavanonesBiophysicsVero cellMolecular MedicinePhytotherapyPhytomedicine
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Zizyphus lotus L. (Desf.) modulates antioxidant activity and human T-cell proliferation

2009

Abstract Background Zizyphus lotus L. (Desf.) also known as Jujube, is a deciduous shrub which belongs to Rhamnaceae family. This plant is used in Algerian traditional medicine for its anti-diabetic, sedative, analgesic, anti-inflammatory and hypoglycaemic activities. In the present study, we determined the concentrations of different vitamins (vitamin A, C and E) and fatty acids in root, stem, leaves, fruit pulp and seed of Zizyphus lotus L. (Desf.) and assessed the effects of their aqueous extracts on antioxidant status and human T-cell proliferation. Methods Aqueous filtrates from different parts, i.e, root, leaf, stem, fruit pulp and seed, of Zizyphus lotus L. (Desf.) were prepared. Vit…

VitaminAntioxidantLinolenic acidT-LymphocytesLinoleic acidmedicine.medical_treatmentGene ExpressionAscorbic AcidLymphocyte ActivationAntioxidantsCell LineLinoleic Acidchemistry.chemical_compoundBotanymedicineHumansVitamin EMicronutrientsFood scienceVitamin AbiologyVitamin CPlant ExtractsVitamin Efood and beveragesZiziphuslcsh:Other systems of medicineGeneral MedicineZiziphuslcsh:RZ201-999biology.organism_classificationAscorbic acidComplementary and alternative medicinechemistryFruitInterleukin-2Plant StructuresImmunosuppressive AgentsResearch Article
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Ultrasound as a Promising Tool for the Green Extraction of Specialized Metabolites from Some Culinary Spices

2021

Spices are a popular food of plant origin, rich in various phytochemicals and recognized for their numerous properties. The aim of the study was to evaluate the antioxidant and antimicrobial activity, as well as the content of specialized metabolites, of aqueous extracts of three spice species––garlic (Allium sativum L.), ginger (Zingiber officinalle L.) and turmeric (Curcuma longa L.)––prepared by green extraction methods. Ultrasound treatment increased the chromaticity parameter b value of turmeric and ginger extracts, thus indicating a higher yellow color predominantly due to curcuminoids characteristic of these species. Ultrasound-assisted extraction significantly increased the content …

VitaminAntioxidantmedicine.medical_treatmentPharmaceutical Scienceantioxidant capacityGinger01 natural sciencesArticleAnalytical Chemistrylcsh:QD241-441chemistry.chemical_compoundCurcuma0404 agricultural biotechnologylcsh:Organic chemistryDrug DiscoverymedicinePhenolsFood sciencePhysical and Theoretical ChemistryCurcumaGarlicCarotenoidComputingMilieux_MISCELLANEOUSspiceschemistry.chemical_classificationbioactive compoundsantimicrobial activityBacteriaVitamin CbiologyPlant Extracts010401 analytical chemistryOrganic ChemistryExtraction (chemistry)food and beverages04 agricultural and veterinary sciencesbiology.organism_classificationAllium sativum040401 food scienceAnti-Bacterial Agents0104 chemical scienceschemistryChemistry (miscellaneous)Bioactive compounds ; Antioxidant capacity ; Antimicrobial activity ; Ultrasonic extraction ; SpicesMolecular Medicineultrasonic extractionMolecules
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Inhibition of Folic Acid Uptake by Catechins and Tea Extracts in Caco-2 Cells

2006

In this present study it was aimed to determine whether the catechins contained in green tea and the whole extracts of Camellia sinensis (Theaceae) inhibit the uptake of folic acid by Caco-2 cell monolayers. Our results indicate that (-)-epigallocatechin 3-gallate (EGCG) and (-)-epicatechin 3-gallate (ECG) inhibit cellular folic acid uptake with IC50 values of 34.8 micromol/L and 30.8 micromol/L, respectively. Furthermore, green and black tea extracts were also found to inhibit folic acid uptake with IC50 values of approximately 7.5 and 3.6 mg/mL, respectively. According to these results, simultaneous intake of tea and folic acid may inhibit intestinal folic acid absorption. The consequence…

VitaminFlavonoidPharmaceutical SciencePharmacognosyAntioxidantsCamellia sinensisCatechinAnalytical Chemistrylaw.inventionInhibitory Concentration 50chemistry.chemical_compoundFolic AcidlawDrug DiscoveryHumansPhenolsTheaceaeFood sciencePharmacologychemistry.chemical_classificationbiologyPlant ExtractsOrganic Chemistryfood and beveragesCatechinbiology.organism_classificationIntestinal AbsorptionComplementary and alternative medicinechemistryBiochemistryPolyphenolMolecular MedicineCaco-2 CellsPhytotherapyPhytotherapyPlanta Medica
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Combined effect of natural antioxidants and antimicrobial compounds during refrigerated storage of nitrite-free frankfurter-type sausage.

2019

Abstract The effects of nisin (200 and 400 ppm), e-polylysine (0.1 and 0.2%) and chitosan (0.5 and 1%) in combination with a Mixed Extract (green tea, stinging nettle and olive leaves extracts) on the physicochemical, microbiological characteristics, fatty acid composition and sensory attributes of the nitrite-free frankfurter-type sausages were assessed during 45 days of storage. The results revealed no significant differences on moisture, fat, protein, ash, salt and water activity (aw) among treatments. 1% Chitosan + Mixed Extract sausages displayed the lowest thiobarbituric acid reactive substances (TBARS) and total volatile nitrogen (TVN) values compared to Control after 45 days of refr…

Water activity030309 nutrition & dieteticsThiobarbituric acidTotal Viable CountShelf lifeAntioxidants03 medical and health scienceschemistry.chemical_compound0404 agricultural biotechnologyFood PreservationOleaTBARSPolylysineFood scienceNitriteNisinNisinNitriteschemistry.chemical_classification0303 health sciencesChitosanTeaPlant Extracts04 agricultural and veterinary sciences040401 food scienceMeat ProductschemistryFood StorageFood MicrobiologyFood SciencePolyunsaturated fatty acidFood research international (Ottawa, Ont.)
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