Search results for "Plant extracts"

showing 10 items of 510 documents

Antiproliferative Effects of St. John’s Wort, Its Derivatives, and Other Hypericum Species in Hematologic Malignancies

2021

Hypericumis a widely present plant, and extracts of its leaves, flowers, and aerial elements have been employed for many years as therapeutic cures for depression, skin wounds, and respiratory and inflammatory disorders. Hypericum also displays an ample variety of other biological actions, such as hypotensive, analgesic, anti-infective, anti-oxidant, and spasmolytic abilities. However, recent investigations highlighted that this species could be advantageous for the cure of other pathological situations, such as trigeminal neuralgia, as well as in the treatment of cancer. This review focuses on the in vitro and in vivo antitumor effects of St. John’s Wort (Hypericum perforatum), its derivat…

MyeloidAngiogenesisDrug Evaluation PreclinicalReviewPharmacologylcsh:Chemistrychemistry.chemical_compoundhyperforinDrug InteractionsMyeloid CellsLymphocyteslcsh:QH301-705.5SpectroscopybiologyapoptosisleukemiaHypericum perforatumGeneral MedicineComputer Science ApplicationsHypericinLeukemiamedicine.anatomical_structurephotodynamic therapyHematologic NeoplasmsHypericumHypericumSt. John’s wortlymphomaCatalysisInorganic ChemistryStructure-Activity Relationshipmultidrug resistanceIn vivoCell Line TumormedicineAnimalsHumansPhysical and Theoretical ChemistryMolecular BiologyCell ProliferationPlant Extractsbusiness.industryOrganic Chemistry<i>Hypericum</i>biology.organism_classificationmedicine.diseaseAntineoplastic Agents PhytogenicApoptosis; Hyperforin; Hypericin; Hypericum; Leukemia; Lymphoma; Mul-tidrug resistance; Photodynamic therapy; St. John’s wort; Animals; Antineoplastic Agents Phytogenic; Apoptosis; Cell Line Tumor; Cell Proliferation; Drug Evaluation Preclinical; Drug Interactions; Drug Resistance Neoplasm; Hematologic Neoplasms; Humans; Hypericum; Lymphocytes; Myeloid Cells; Plant Extracts; Structure-Activity RelationshipHyperforinchemistrylcsh:Biology (General)lcsh:QD1-999Drug Resistance NeoplasmhypericinbusinessInternational Journal of Molecular Sciences
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A Two-Year Bio-Agronomic and Chemotaxonomic Evaluation of Wild Sicilian Myrtle (Myrtus communis L.) Berries and Leaves.

2019

A collection of nine Myrtus communis samples from different localities of Sicily was evaluated. Morphological traits and production characteristics have been chosen as parameters to arrange the samples into homogeneous groups and to identify the best biotypes for possible future agro-industrial exploitation. The plant material has been subjected to taxonomic characterization from biometric and phytochemical perspectives. Myrtle berries and leaves have been analyzed for their content in metabolites, applying a cascade extraction protocol for M. communis leaves and a single hydroalcoholic extraction for berries, whereas hydrodistillation procedures have been applied to obtain the essential oi…

Myrtus communis L.FlavonolsCyanidinPhytochemicalsBioengineeringLinalyl acetate01 natural sciencesBiochemistryMediterranean areaessential oillaw.inventionAnthocyaninschemistry.chemical_compoundFlavonolsLinaloollawPetunidinOils VolatileMolecular BiologySicilyEssential oilbiodiversitychemistry.chemical_classificationMyrtus communisMolecular Structure010405 organic chemistryPlant ExtractsMyrtus communis L. essential oil polyphenol biodiversity Mediterranean area phytochemistry.General ChemistryGeneral MedicineMyrtus0104 chemical sciencesPlant Leaves010404 medicinal & biomolecular chemistryHorticulturepolyphenolchemistryPhytochemicalFruitMolecular MedicinephytochemistryChemistrybiodiversity
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Screening of some rare endemic Italian plants for inhibitory activity on 5-lipoxygenase

2003

Abstract The extracts of four rare plants found on the islands of Sicily, Vulcano and Marettimo, Southern Italy, were screened for their inhibitory effect on the production of leukotriene B 4 by 5-lipoxygenase in intact cells. The methanol extracts of pods of Cytisus aeolicus and aerial parts of Thymus richardii were the most active extracts, inhibiting almost completely the leukotriene B 4 production at 200 and 50 μg/ml, respectively.

NeutrophilsLeukotriene B4PharmacognosyInhibitory postsynaptic potentialLeukotriene B4MicrobiologyThymus PlantLipoxygenasechemistry.chemical_compoundPlumbaginaceaeDrug DiscoveryBotanyAnimalsLipoxygenase InhibitorsGenistaRats WistarCytotoxicitySicilyCytisusPharmacologychemistry.chemical_classificationbiologyPlant ExtractsCytisusGeneral MedicinePlant Components Aerialbiology.organism_classificationRatsEnzymechemistryArachidonate 5-lipoxygenasebiology.proteinFitoterapia
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An Aqueous Extract of Ilex paraguariensis Reduces Carrageenan-Induced Edema and Inhibits the Expression of Cyclooxygenase-2 and Inducible Nitric Oxid…

2014

Mate (Ilex paraguariensis) is a highly popular herbal beverage in South America due to its high content of caffeine. Its hypolipidemic and antioxidant properties are of increasing interest in the treatment of cardiovascular disorders and for weight control. In the present study, we show for the first time both the local and systemic anti-inflammatory effects of an aqueous extract of mate in three classic in vivo models, namely acute and chronic 12-O-tetradecanoylphorbol 13-acetate-induced mouse ear edema and acute carrageenan-induced mouse paw edema. Caffeine, rutin, chlorogenic acid, 3,5-dicafeoyl quinic acid, and 4,5-dicafeoyl quinic acid, accompanied by a complex mixture of other simple …

Nitric Oxide Synthase Type IIPharmaceutical ScienceMice Inbred StrainsPharmacologyCarrageenanAnalytical Chemistrychemistry.chemical_compoundPhenolsDermisChlorogenic acidIlex paraguariensisIn vivoEdemaDrug DiscoveryAnimalsEdemaMedicineSkinInflammationPharmacologyCyclooxygenase 2 InhibitorsbiologyPlant Extractsbusiness.industryOrganic ChemistryQuinic acidNitric oxide synthaseDisease Models Animalmedicine.anatomical_structureComplementary and alternative medicinechemistryCyclooxygenase 2biology.proteinTetradecanoylphorbol AcetateMolecular MedicineFemaleCyclooxygenasemedicine.symptomCaffeinebusinessPhytotherapyPlanta Medica
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Ursolic acid from the Chinese herb Danshen (Salvia miltiorrhiza L.) upregulates eNOS and downregulates Nox4 expression in human endothelial cells

2007

Danshen, the dried root of Salvia miltiorrhiza Bunge (Lamiaceae), is one of the most commonly used traditional Chinese medicines for cardiovascular indications. In EA.hy 926 cells, a cell line derived from human umbilical vein endothelial cells (HUVEC), an aqueous extract of danshen, and also a methanol extract of the plant, increased eNOS promoter activity, eNOS mRNA and protein expression, as well as endothelial NO production. A dichloromethane extract, in contrast, did not change eNOS gene expression. Thus, the active danshen constituent(s) responsible for eNOS upregulation is (are) hydrophilic and/or alcohol-soluble. One such compound is ursolic acid that significantly increased eNOS ex…

Nitric Oxide Synthase Type IIIEndotheliumSalvia miltiorrhizaBiologyPharmacologySalvia miltiorrhizaGene Expression Regulation Enzymologicchemistry.chemical_compoundRibonucleasesUrsolic acidDownregulation and upregulationGenes ReporterEnosmedicineHumansRNA MessengerCells CulturedNADPH oxidasePlant ExtractsMethanolNADPH OxidasesNOX4biology.organism_classificationTriterpenesNitric oxide synthaseOxidative Stressmedicine.anatomical_structureBiochemistrychemistryNADPH Oxidase 4Alcoholsbiology.proteinEndothelium VascularCardiology and Cardiovascular MedicineAtherosclerosis
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In vitro blood brain barrier exposure to mycotoxins and carotenoids pumpkin extract alters mitochondrial gene expression and oxidative stress.

2021

Abstract Food and feed are daily exposed to mycotoxin contamination which effects may be counteracted by antioxidants like carotenoids. Some mycotoxins as well as carotenoids penetrate the blood brain barrier (BBB) inducing alterations related to redox balance in the mitochondria. Therefore, the in vitro BBB model ECV304 was subcultured for 7 days and exposed to beauvericine, enniatins, ochratoxin A, zearalenone (100 nM each), individually and combined, and pumpkin extract (500 nM). Reactive oxygen species were measured by fluorescence using the dichlorofluorescein diacetate probe at 0 h, 2 h and 4 h. Intracellular ROS generation reported was condition dependent. RNA extraction was performe…

Ochratoxin ADown-RegulationGene ExpressionMitochondrionToxicologymedicine.disease_causeCell LineElectron Transport Complex IV03 medical and health scienceschemistry.chemical_compound0404 agricultural biotechnologyCucurbitaDichlorofluoresceinDepsipeptidesGene expressionmedicineHumansOxidoreductases Acting on Sulfur Group DonorsUncoupling Protein 2MycotoxinCarotenoid030304 developmental biologychemistry.chemical_classification0303 health sciencesReactive oxygen speciesChemistryPlant Extractsfood and beverages04 agricultural and veterinary sciencesGeneral MedicineMycotoxins040401 food scienceCarotenoidsMitochondriaUp-RegulationOxidative StressGenes MitochondrialBiochemistryBlood-Brain BarrierCarrier ProteinsReactive Oxygen SpeciesOxidative stressFood ScienceFood and chemical toxicology : an international journal published for the British Industrial Biological Research Association
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The role of pumpkin pulp extract carotenoids against mycotoxin damage in the blood brain barrier

2021

Some mycotoxins such as beauvericin (BEA), ochratoxin A (OTA), and zearalenone (ZEA) can cross the blood brain barrier, which is why we tested the anti-inflammatory action of a pumpkin carotenoid extract (from the pulp) against these mycotoxins and their combinations (OTA+ZEA and OTA+ZEA+BEA) on a blood brain barrier model with co-cultured ECV304 and C6 cells using an untargeted metabolomic approach. The cells were added with mycotoxins at a concentration of 100 nmol/L per mycotoxin and pumpkin carotenoid extract at 500 nmol/L. For control we used only vehicle solvent (cell control) or vehicle solvent with pumpkin extract (extract control). After two hours of exposure, samples were analysed…

Ochratoxin AMetaboliteProstaglandinToxicologychemistry.chemical_compoundCucurbitametabolomikaFood scienceMycotoxinZearalenoneCarotenoidchemistry.chemical_classificationzearalenonPlant ExtractsECV304fungibeauvericinzearalenonePublic Health Environmental and Occupational Healthfood and beveragesMycotoxinsCarotenoidsOchratoxinsmetabolomicsBeauvericinchemistryBlood-Brain Barrierbovericinokratoksin AArachidonic acidOriginal Articleochratoxin AArhiv za higijenu rada i toksikologiju
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Nopal Cactus (Opuntia ficus-indica) as a Source of Bioactive Compounds for Nutrition, Health and Disease

2014

Opuntia ficus-indica, commonly referred to as prickly pear or nopal cactus, is a dicotyledonous angiosperm plant. It belongs to the Cactaceae family and is characterized by its remarkable adaptation to arid and semi-arid climates in tropical and subtropical regions of the globe. In the last decade, compelling evidence for the nutritional and health benefit potential of this cactus has been provided by academic scientists and private companies. Notably, its rich composition in polyphenols, vitamins, polyunsaturated fatty acids and amino acids has been highlighted through the use of a large panel of extraction methods. The identified natural cactus compounds and derivatives were shown to be e…

Opuntia ficus-indicaOpuntia ficusAnti-Inflammatory AgentsPharmaceutical ScienceDiseaseReviewHealth benefitsBiologyAntioxidantsAnalytical Chemistrylcsh:QD241-441lcsh:Organic chemistryDrug DiscoveryBotanycell signalingAnimalsHumansPhysical and Theoretical Chemistryanti-inflammatorychemistry.chemical_classificationPEARPlant ExtractsOrganic ChemistryOpuntiaPolyphenolschemistryChemistry (miscellaneous)CactusMolecular MedicineExtraction methodsDrug Screening Assays AntitumorPolyunsaturated fatty acidMolecules
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A Review of the Phytochemistry, Traditional Uses, and Biological Activities of the Genus Ballota and Otostegia

2019

AbstractThe 2 genera Ballota and Otostegia, belonging to the Lamiaceae family, are closely related taxonomically and found mainly in the Mediterranean area, Middle East, and North Africa. Since ancient times, they have been largely employed in traditional medicine for their biological properties such as antimicrobial, anti-inflammatory, antispasmodic, insecticidal, anti-malaria, etc. Phytochemical investigations of Ballota and Otostegia species have revealed that diterpenoids are the main constituents of the genera. A large number of flavonoids and other metabolites were also identified. This review, covering literature from 1911 up to 2018, includes traditional uses, chemical profiles (bot…

OtostegiaantioxidantPhytochemistryfood.ingredientPharmaceutical Sciencesecondary metabolite01 natural sciencesAnalytical ChemistryfoodGenusBiological propertyDrug DiscoveryAnimalsHumansSettore BIO/15 - Biologia FarmaceuticaPharmacologyLamiaceaebiologyTraditional medicinePlant Extracts010405 organic chemistryOrganic ChemistrySettore CHIM/06 - Chimica OrganicaBallotabiology.organism_classification0104 chemical sciencesantibacterial010404 medicinal & biomolecular chemistryTaxonComplementary and alternative medicinePhytochemicalMolecular MedicineLamiaceaeMedicine TraditionalOtostegiaBallotaantifungalPhytotherapyPlanta Medica
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Kavapyrone enriched extract fromPiper methysticum as modulator of the GABA binding site in different regions of rat brain

1994

Regional differences in the modulation of [3H] muscimol binding to GABAA receptor complexes by kavapyrones, compounds of the rhizome of the plant Piper methysticum which possess sedative activity, were demonstrated using membrane fractions obtained from target brain centers of kavapyrone action: hippocampus (HIP), amygdala (AMY) and medulla oblongata (MED), and from brain centers outside the main kavapyrone effects as frontal cortex (FC) and cerebellum (CER). The kava extract enhanced the binding of [3H] muscimol in a concentration-dependent manner with maximal potentiation of 358% over control in HIP followed by AMY and MED (main target brain centers). Minimal stimulation was observed in C…

OvariectomyStimulationIn Vitro TechniquesPharmacologyBiologyBinding CompetitiveRats Sprague-Dawleychemistry.chemical_compoundReceptors GABAmedicineAnimalsBinding siteKavainReceptorPentobarbitalBrain ChemistryPharmacologyDiazepamPlants MedicinalMuscimolPlant ExtractsGABAA receptorLong-term potentiationRatsnervous systemMechanism of actionMuscimolchemistryPyronesFemaleSteroidsmedicine.symptomNeurosciencePsychopharmacology
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