Search results for "Platinum"

showing 10 items of 629 documents

Characterization of Hydrophilic Gold(I) N-Heterocyclic Carbene (NHC) Complexes as Potent TrxR Inhibitors Using Biochemical and Mass Spectrometric App…

2017

We report here on the synthesis of a series of mono-and dinuclear gold(I) complexes exhibiting sulfonated bis(NHC) ligands and novel hydroxylated mono(NHC) Au(I) compounds, which were also examined for their 'biological activities. Initial cell viability assays show strong antiproliferative activities of the hydroxylated mono(NHC) gold compounds (8 > 9 > 10) against 2008 human ovarian cancer cells even after 1 h incubation. In order to gain insight into the mechanism of biological action of the gold compounds, their effect on the pivotal cellular target seleno-enzyme thioredoxin reductase (TrxR), involved in the maintenance of intracellular redox balance, was investigated in depth. Th…

Thioredoxin Reductase 1AuranofinSilverStereochemistryThioredoxin reductaseThioredoxin Reductase 2WATER-SOLUBLE RUTHENIUM(II)Antineoplastic Agents010402 general chemistryG-quadruplexLigandsIN-VITRO CYTOTOXICITYLIGANDS SYNTHESIS01 natural sciencesInorganic Chemistrychemistry.chemical_compoundDrug StabilityThioredoxin Reductase 1Coordination ComplexesTHIOREDOXIN REDUCTASE INHIBITIONCell Line TumormedicineOrganogold CompoundsAnimalsHumansCRYSTAL-STRUCTURESPhysical and Theoretical ChemistryCANCER CELLSBIOLOGICAL-PROPERTIES010405 organic chemistryChemistryMOLECULAR-MECHANISMSDNA0104 chemical sciencesRatsG-QuadruplexesGlutathione ReductaseSolubilityBiological targetCancer cellPLATINUM ANTICANCER DRUGSMETAL-COMPLEXESGoldReactive Oxygen SpeciesCarbeneHydrophobic and Hydrophilic InteractionsOrganogold Compoundsmedicine.drugInorganic Chemistry
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Divergent route to the preparation of hybrid Pt–Fe 2,4,6-Tris(4-ethynyl)phenyl-1,3,5-triazine metallodendrimers for nonlinear optics

2013

Abstract: The synthesis strategy for the preparation of novel platinum acetylide homometallic and heterobimetallic dendrimers (containing Fe as the other metal fragment) based on a 2,4,6-tris(4-ethynyl)phenyl-1,3,5-triazine core (3) is reported. All the dendrimer generations (G0G2) were synthesized under copper-free conditions following a divergent route. The G0-Pt dendrimer (4) was synthesized using the 1,3,5-triazine core (3) and cis-[Pt(PEt3)2Cl2] with a molar ratio of 1/4. The advantage of the current method is that different dendrimers can be prepared by following the same procedure with only changes in the molar ratios of the reactants involved. For instance, when 3 reacts with 4 in a…

TrisMolarPreparation of hybrid Pt−Fe 246-Tris(4ethynyl)phenyl-135-triazinePhysicsAcetylideOrganic Chemistrychemistry.chemical_element.Inorganic ChemistryMetalChemistrychemistry.chemical_compoundMetallodendrimers for nonlinear opticsFaculdade de Ciências Exatas e da Engenhariachemistry135-Triazinevisual_artDendrimerPolymer chemistryvisual_art.visual_art_mediumMoietyPhysical and Theoretical ChemistryPlatinumta116
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New light on an old debate: does the RCN–PtCl2 bond include any back-donation? RCN←PtCl2 backbonding vs. the IR νCN blue-shift dichotomy in organoni…

2019

For a series of organonitrile [RCN (R = Me, CF3, Ph, CH3Ph, CF3Ph)] ligands, the nature of the N–Pt bond in the related cis-/trans-(RCN)2PtCl2 complexes has been computationally investigated by Density Functional Theory. A fragment based bond analysis has been performed in the canonical Kohn–Sham molecular orbitals framework, and it has been ultimately assessed that this bond is characterized both by N→Pt σ and by N←Pt π contributions. Voronoi Deformation Density charges further confirms the occurrence of N←Pt π interactions. Moreover, the Energy Decomposition Analysis-Natural Orbital for Chemical Valence (EDA-NOCV) method shows that the strength of the N←Pt π interaction is not negligible …

Valence (chemistry)010405 organic chemistrychemistry.chemical_element010402 general chemistryTriple bond01 natural sciences0104 chemical sciencesInorganic ChemistryCrystallographychemistryMolecular orbitalDensity functional theoryLewis acids and basesVoronoi deformation densityPlatinumPi backbondingDalton Transactions
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An Open-Label Phase II Study Evaluating the Safety and Efficacy of Ramucirumab Combined With mFOLFOX-6 as First-Line Therapy for Metastatic Colorecta…

2014

Abstract Author Summary Background. Vascular endothelial growth factor (VEGF) and VEGF receptor 2 (VEGFR-2) are believed to mediate angiogenesis in colorectal cancer (CRC). Ramucirumab (RAM; IMC-1121B) is a human IgG1 monoclonal antibody that inhibits VEGF ligand binding to VEGFR-2, inhibiting VEGFR-2 activation and signaling. Methods. Patients with metastatic CRC, Eastern Cooperative Oncology Group performance status 0–1, and adequate organ function who had not received chemotherapy for metastatic disease received RAM and the modified FOLFOX-6 regimen every 2 weeks. Endpoints included progression-free survival (PFS), objective response rate, overall survival, and safety. The sample size wa…

Vascular Endothelial Growth Factor ACancer ResearchPathologymedicine.medical_specialtyOrganoplatinum CompoundsAngiogenesisColorectal cancerLeucovorinAntibodies Monoclonal HumanizedDisease-Free SurvivalDrug Administration ScheduleRamucirumabchemistry.chemical_compoundAntineoplastic Combined Chemotherapy ProtocolsmedicineHumansNeoplasm Metastasisbusiness.industryClinical Trial ResultsAntibodies MonoclonalKinase insert domain receptormedicine.diseaseVascular Endothelial Growth Factor Receptor-2Vascular endothelial growth factorVascular endothelial growth factor ATreatment OutcomeOncologychemistryFluorouracilMonoclonalCancer researchFluorouracilbusinessColorectal Neoplasmsmedicine.drugProtein Binding
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Voltammetric determinations of platinum and rhodium in particulate of Palermo (Italy) area

2012

Traffic has an important impact on the air quality which affects both the environmental and human health. Since the introduction of PGE-containing catalytic converters, a number studies have been undertaken to determine the effects of PGE emissions on human and to environment. This requires the development of good analytic methods to measure Pt and Rh concentrations in environmental matrices, as well to estimate background concentrations. In this paper are presented the results concerning Pt and Rh concentrations in PM10 samples collected at five stations within the urban area of Palermo. The highest mean values (Pt= 13 pg/m3, Rh=9.8 pg/m3) were recorded at an urban station, and the lowest …

Voltammetric platinumrhodiumSettore CHIM/12 - Chimica Dell'Ambiente E Dei Beni Culturali
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One- and Two-Dimensional Diffusion of Metal Atoms in Graphene

2008

In the present work, individual Au or Pt atoms in layersconsisting of one or twographene planes have been monitoredin real time at high temperature by high-resolution TEM. Weobtain information about the location of metal atoms ingrapheneandthediffusionmechanisms.Activationenergiesfordiffusion are obtained in a temperature range close to thetemperature of the technically important metal-assisted CVDprocess.Thematerialwassynthesizedinanarcdischarge

Work (thermodynamics)Materials scienceMacromolecular SubstancesSurface PropertiesDiffusionMolecular Conformationchemistry.chemical_elementMolecular physicslaw.inventionDiffusionBiomaterialsMetallawMaterials TestingNanotechnologyGeneral Materials ScienceParticle SizePlatinumNanotubes CarbonGrapheneCarbon chemistryGeneral ChemistryAtmospheric temperature rangechemistryvisual_artvisual_art.visual_art_mediumGraphiteGoldParticle sizeAtomic physicsCrystallizationCarbonBiotechnologySmall
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CCDC 1970145: Experimental Crystal Structure Determination

2020

Related Article: Ariadna Lázaro, Carla Cunha, Ramon Bosque, João Pina, Jas S. Ward, Khai-Nghi Truong, Kari Rissanen, João Carlos Lima, Margarita Crespo, J. Sérgio Seixas de Melo, Laura Rodríguez|2020|Inorg.Chem.|59|8220|doi:10.1021/acs.inorgchem.0c00577

[2-({[2-(dimethylamino)ethyl]imino}methyl)-5-fluorophenyl]-[(4-fluorophenyl)ethynyl]-platinumSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Experimental and theoretical studies on electropolymerization of polar amino acids on platinum electrode

2017

International audience; The anodic oxidation of polar amino acids (L-serine, L-threonine, L-asparagine, and L-glutamine) in aqueous electrolyte on smooth platinum electrode was carried out by cyclic voltammetry coupled to electrochemical quartz crystal microbalance (EQCM). pH (zwitterion, acidic and alkaline) effects on their electrochemical behavior were examined. The maximum current values are measured for zwitterion species. In addition, the current increases with increasing of concentration and scan rate, and decreases with increasing pH. The resulting passivation was studied by spectroscopic analysis such as attenuated total reflection FT infrared spectroscopy (ATR-FTIR), X-ray photoel…

[SPI.OTHER]Engineering Sciences [physics]/Otherab-initiopotentiometric phInorganic chemistryAnalytical chemistryl-alaninechemistry.chemical_elementInfrared spectroscopy02 engineering and technology010402 general chemistry01 natural sciencesDFTpolyanilinechemistry.chemical_compoundX-ray photoelectron spectroscopyGeneral Materials ScienceSpectroscopyl-serinepH sensingElectropolymerizationQuartz crystal microbalance[CHIM.MATE]Chemical Sciences/Material chemistry021001 nanoscience & nanotechnologyCondensed Matter Physics0104 chemical sciencesthin-filmchemistryadsorptionZwitterionAttenuated total reflection[ CHIM.MATE ] Chemical Sciences/Material chemistryThin polymer filmElectrodel-lysinepeptidesgold electrodeCyclic voltammetryPolar amino acid0210 nano-technologyPlatinum
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CCDC 2031113: Experimental Crystal Structure Determination

2021

Related Article: Margarita Bulatova, Daniil M. Ivanov, Matti Haukka|2021|Cryst.Growth Des.|21|974|doi:10.1021/acs.cgd.0c01314

[cycloocta-15-diene]-di-iodo-platinum(ii) triiodomethaneSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Racemization of Secondary-Amine-Containing Natural Products Using Heterogeneous Metal Catalysts

2018

amineschemistry.chemical_element010402 general chemistry01 natural sciencescatalystsCatalysisInorganic ChemistrykatalyytitOrganic chemistryIridiumMetal catalystPhysical and Theoretical Chemistryta116Racemizationamiinit010405 organic chemistryChemistryOrganic Chemistryluonnonaineetseoksetnaturally occurring substances0104 chemical sciencesmixturesracemizationAmine gas treatingPlatinumChemCatChem
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