Search results for "Polyp"

showing 10 items of 1415 documents

Stability of mycophenolate mofetil in polypropylene 5% dextrose infusion bags and chemical compatibility associated with the use of the Equashield ® …

2019

Stability studies are necessary in healthcare settings as they facilitate fast, cost-effective and efficient work related to batch manufacturing and availability of supplies. We studied the stability of 1-10 mg/mL mycophenolate mofetil (MMF) in polypropylene 5% dextrose infusion bags prepared from Cellcept® and with a generic brand name (Micofenolato de Mofetilo Accord) at different storage temperatures. To ensure chemical compatibility during preparation, we also tested MMF sorption to the Equashield® closed-system drug transfer device used in this step. For this, a validated stability-indicating high-performance liquid chromatography method was developed for the quantification and identif…

PharmacologyPolypropyleneDrug transferChromatography010401 analytical chemistryClinical BiochemistrySorptionGeneral MedicineMycophenolateBatch manufacturing030226 pharmacology & pharmacy01 natural sciencesBiochemistryWork related0104 chemical sciencesAnalytical ChemistryChemical compatibility03 medical and health scienceschemistry.chemical_compound0302 clinical medicinechemistryDrug Discovery5 dextroseMolecular BiologyBiomedical Chromatography
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Occurrence of resveratrol and pterostilbene in age-old darakchasava, an ayurvedic medicine from India

2000

'Darakchasava' is a well known Indian herbal preparation of which the main ingredient is Vitis vinifera L. This 'ayurvedic' medicine is prescribed as a cardiotonic and also given for other disorders. HPLC analysis of this age old formulation revealed the presence of polyphenols like resveratrol and pterostilbene. These phenolic compounds are now known as antioxidants, cancer chemopreventive agents, and also known to reduce mortality from coronary heart disease by increasing high density lipoproteins like cholesterol and inhibiting platelet aggregation (Soleas, J.S., Diamandis, E.P., Goldberg, D.M., 1997. Resveratrol: a molecule whose time has come? and gone? Clin. Biochem. 30 (2), 91-113). …

PharmacologyPterostilbeneTraditional medicinePlant ExtractsCholesterolIndiafood and beveragesPharmacognosyResveratrolAntineoplastic Agents PhytogenicAntioxidantsMedicine Ayurvedicchemistry.chemical_compoundIngredientPhenolschemistryResveratrolPolyphenolStilbenesDrug DiscoveryHypoglycemic AgentsPlatelet aggregation inhibitorVitis viniferaChromatography High Pressure LiquidPlatelet Aggregation InhibitorsJournal of Ethnopharmacology
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Multi or Single-Kinase Inhibitors to Counteract Drug Resistance in Cancer: What is New?

2023

The concept of protein kinase inhibition starts from the groundbreaking research on the role of these proteins in the regulation of fundamental processes, including proliferation, cell cycle, apoptosis, metabolism, and inflammation. Kinase genetic mutations, as well as overexpression and dysregulation, can contribute to the development of several diseases, including neoplasms, leading to relapses and resistance to standard drug chemotherapy [1-3].

PharmacologySmall molecules kinase inhibitorspolypharmacologycovalent kinase inhibitorsallosteric inhibitorsDrug DiscoveryOrganic ChemistryMolecular Medicineanticancer drug combinationsBiochemistrykinase genetic aberrationSettore CHIM/08 - Chimica Farmaceutica
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Bioactive Polyphenols from Grapes and Wine Emphasized with Resveratrol

2013

Grape polyphenols are abundant. They play essential roles in the plant's life, particularly in defence mechanisms. Moreover, the grape, fresh or dried, is a widely consumed fruit by humans, as are its by-products, grape juice and wine. They also contain vast and highly varied quantities of polyphenols. Like other phytophenols, grape and wine resveratrol is considered a protective micronutrient. Resveratrol is a well known antioxidant, for example, a protector of low-density lipoproteins against oxidation. Its applications are therefore highly varied. Research supports the idea that wine consumed regularly, without excess, is a natural biological product possesses preventive properties, and …

PharmacologyWineAntioxidantmedicine.medical_treatmentBiological Availabilityfood and beveragesWineContext (language use)Biological productBiologyResveratrolchemistry.chemical_compoundchemistryResveratrolPolyphenolStilbenesDrug DiscoverymedicineAnimalsHumansFrench paradoxVitisFood sciencePlants EdibleHuman speciesCurrent Pharmaceutical Design
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Inhibition of human P450 enzymes by natural extracts used in traditional medicine

2008

Different medicinal plants are widely used in Cuba and Mexico to treat several disorders. This paper reports in vitro inhibitory effects on the P450 system of herbal products commonly used by people in Cuba and Mexico in traditional medicine for decades. Experiments were conducted in human liver microsomes. The catalytic activities of CYP1A1/2, 2D6, and 3A4 were measured using specific probe substrates. The Heliopsis longipes extract exhibited a concentration-dependent inhibition of the three enzymes, and similar effects were produced by affinin (an alkamide isolated from the H. longipes extract) and two catalytically reduced alkamides. Mangifera indica L. and Thalassia testudinum extracts,…

Pharmacologychemistry.chemical_classificationbiologyTraditional medicineEnzyme assaylaw.inventionEnzymechemistrylawPolyphenolHeliopsis longipesbiology.proteinMangiferaPhytotherapyMedicinal plantsDrug metabolismPhytotherapy Research
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Pharmacological Properties of Polyphenols: Bioavailability, Mechanisms of Action, and Biological Effects in In Vitro Studies, Animal Models, and Huma…

2021

Este artículo se encuentra disponible en la siguiente URL: https://www.mdpi.com/2227-9059/9/8/1074 Este artículo de investigación pertenece al número especial "Oxidative Stress and Inflammation: From Mechanisms to Therapeutic Approaches 2.0". Drugs are bioactive compounds originally discovered from chemical structures present in both the plant and animal kingdoms. These have the ability to interact with molecules found in our body, blocking them, activating them, or increasing or decreasing their levels. Their actions have allowed us to cure diseases and improve our state of health, which has led us to increase the longevity of our species. Among the molecules with pharmacological activity …

Phenols - Physiological effect.Pharmacology.QH301-705.5Medicine (miscellaneous)Phenols - Properties.Farmacología.ReviewPharmacologyGeneral Biochemistry Genetics and Molecular BiologyDrugs - Bioavalability.drugsIn vivoconcomitanthumanBiology (General)Chemistrybiological effectsBiological activitypharmacologicalin vitroMedicamentos - Biodisponibilidad.In vitroBioavailabilityFenoles - Propiedades.mechanisms of actionpolyphenolin vivoPolyphenolFenoles - Efectos fisiológicos.bioavailabilityBiomedicines
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Do avian predators select for seasonal polyphenism in the European map butterfly Araschnia levana (Lepidoptera: Nymphalidae)?

2012

Seasonal polyphenism in animal colour patterns indicates that temporal variation in selection pressures maintains phenotypic plasticity. Spring generation of the polyphenic European map butterfly Araschnia levana has an orange–black fritillary-like pattern whilst individuals of the summer generation are black with white bands across the wings. What selects for the colour difference is unknown. Because predation is a major selection pressure for insect coloration, we first tested whether map butterfly coloration could have a warning function (i.e. whether the butterflies are unpalatable to birds). In a following field experiment with butterfly dummies we tested whether the spring form is bet…

Phenotypic plasticitybiologyPolyphenismEcologyCyanistesButterflyAposematismAdaptationbiology.organism_classificationNymphalidaeEcology Evolution Behavior and SystematicsPredationBiological Journal of the Linnean Society
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First record of Phlebia margaritae (Polyporales, Basidiomycota) in Italy

2017

A new record of Phlebia margaritae, a very rare corticoid fungus, is reported for the first time in Italy. Macro- and micro-morphological descriptions, supported by molecular analysis, are also provided and new information on the geographic distribution of this species has now been increased

Phlebia margaritaebiologySettore BIO/02 - Botanica SistematicaBotanydistributionPolyporalesBasidiomycotaPlant Sciencebiology.organism_classificationSicilyEcology Evolution Behavior and Systematicsrare corticoid speciesPistacia lentiscus
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Photo-oxidation of nano- and micro-filled polypropylene

2010

Photo-oxidation polypropylene BESED MICRO- NANO-COMPOSITES
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Influence of the electrodeposition conditions on the energetics of polypyrrole thin films

2008

The influence of the solvent used for the electrodeposition and that of the dopant anion on the energetics of electrochemically grown polypyrrole were studied by means of a non-destructive optical technique: Photocurrent Spectroscopy. Polypyrrole films doped with the same anion and grown in different solvents, both aqueous and non- aqueous, show the same HOMO-LUMO gap and the same Fermi level location in respect to HOMO. Polypyrrole films doped with different anions in aqueous solutions, present different values of indirect band gap and flat band potential, indicating that dopant anion influences both the defects band and the Fermi level locations.

Photocurrent Spectroscopy Band gap Flat Band Potential Fermi Level Polypyrrole.
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