Search results for "Pyoluteorin"

showing 2 items of 2 documents

Synthesis and antimicrobial activity of new bromine-rich pyrrole derivatives related to monodeoxypyoluteorin

2006

The synthesis and antimicrobial activity of new pyrrole derivatives structurally related to monodeoxypyoluteorin are described. The insertion of a keto or methylene spacer between the phenol group and the pyrroloyl moiety of brominated 2-(2'-hydroxybenzoyl)pyrroles leads to a decrease of the antibacterial activity.

Antifungal AgentsMagnetic Resonance SpectroscopyKetoneMicrobial Sensitivity Testspyoluteorin analogsChemical synthesischemistry.chemical_compoundPhenolsSpectroscopy Fourier Transform InfraredDrug DiscoveryMoietyPhenolOrganic chemistryPyrrolesPhenolsMethyleneantimicrobicbromopyrrolePharmacologychemistry.chemical_classificationOrganic ChemistryGeneral MedicineBromineAntimicrobialAnti-Bacterial AgentschemistryAntibacterial activity
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Pharmaceutical potential of synthetic and natural pyrrolomycins

2015

The emergence of antibiotic resistance is currently considered one of the most important global health problem. The continuous onset of multidrug-resistant Gram-positive and Gram-negative bacterial strains limits the clinical efficacy of most of the marketed antibiotics. Therefore, there is an urgent need for new antibiotics. Pyrrolomycins are a class of biologically active compounds that exhibit a broad spectrum of biological activities, including antibacterial, antifungal, anthelmintic, antiproliferative, insecticidal, and acaricidal activities. In this review we focus on the antibacterial activity and antibiofilm activity of pyrrolomycins against Gram-positive and Gram-negative pathogens…

Pyoluteorinantibiotic resistancemedicine.drug_classAntibioticsPharmaceutical ScienceMicrobial Sensitivity TestsReviewPharmacologyAntibiofilm agentpyrrolomycinSettore BIO/19 - Microbiologia GeneraleAnalytical Chemistrylcsh:QD241-441Antibiotic resistancelcsh:Organic chemistryDrug DiscoveryDrug Resistance BacterialMedicineAnimalsHumansPyrrolesClinical efficacyPhysical and Theoretical ChemistrypyrrolomycinspentabromopseudilinLow toxicityBacteriabusiness.industryOrganic ChemistryBiological activityBacterial Infectionsantibiofilm agentsAntimicrobialSettore CHIM/08 - Chimica FarmaceuticaAnti-Bacterial AgentsChemistry (miscellaneous)BiofilmsPentabromopseudilinMolecular MedicinebusinessAntibacterial activity
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