Search results for "Pyramid"

showing 10 items of 410 documents

Molecular basis of the interaction of novel tributyltin(IV) 2/4-[(E)-2-(aryl)-1-diazenyl] benzoates endowed with an improved cytotoxic profile: Synth…

2010

A series of tributyltin(IV) complexes based on 2/4-[(E)-2-(aryl)-1-diazenyl]benzoate ligands was synthesized, wherein the position of the carboxylate and aryl substituents (methyl, tert-butyl and hydroxyl) varies. The complexes, Bu(3)SnL(1-4)H (1-4), have been structurally characterized by elemental analysis and IR, NMR ((1)H, (13)C, and (119)Sn) and (119)Sn Mossbauer spectroscopy. All have a tetrahedral geometry in solution and a trigonal bipyramidal geometry in the solid-state, except for Bu(3)SnL(4)H (4) that was ascertained to have tetrahedral coordination by X-ray crystallography. Cytotoxicity studies were carried out on human tumor cell lines A498 (renal cancer), EVSA-T (mammary cance…

Models MolecularQuantitative structure–activity relationshipMagnetic Resonance SpectroscopyStereochemistryCell SurvivalANTITUMOR-ACTIVITYHydrophobicityQuantitative Structure-Activity RelationshipAntineoplastic AgentsCrystallography X-RayBiochemistryBenzoatesVALIDATIONInorganic Chemistrychemistry.chemical_compoundAnti-cancer drugCell Line TumorOrganotin CompoundsTRIORGANOTIN(IV) COMPLEXESHumansCRYSTAL-STRUCTURESCarboxylateOPTIMIZATIONArylazobenzoateSpectroscopyX-ray crystallographyMolecular StructureQSARArylTetrahedral molecular geometryNuclear magnetic resonance spectroscopyBenzoatesTributyltin(IV) compoundTrigonal bipyramidal molecular geometryMOSQUITO LARVAEchemistryCELL-DEATHDocking (molecular)Settore CHIM/03 - Chimica Generale E InorganicaDocking studies RIBONUCLEOTIDE REDUCTASE INHIBITORSEMIEMPIRICAL METHODSTrialkyltin CompoundsCell lineAEDES-AEGYPTI
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Use of a reduced Schiff-Base ligand to prepare novel chloro-bridged chains of rare Cu(II) trinuclear complexes with mixed azido/oxo and chloro/oxo br…

2010

Two mixed bridged one-dimensional (1D) polynuclear complexes, [Cu(3)L(2)(mu(1,1)-N(3))(2)(mu-Cl)Cl](n) (1) and {[Cu(3)L(2)(mu-Cl)(3)Cl].0.46CH(3)OH}(n) (2), have been synthesized using the tridentate reduced Schiff-base ligand HL (2-[(2-dimethylamino-ethylamino)-methyl]-phenol). The complexes have been characterized by X-ray structural analyses and variable-temperature magnetic susceptibility measurements. In both complexes the basic trinuclear angular units are joined together by weak chloro bridges to form a 1D chain. The trinuclear structure of 1 is composed of two terminal square planar [Cu(L)(mu(1,1)-N(3))] units connected by a central Cu(II) atom through bridging nitrogen atoms of end…

Models MolecularSchiff baseLigandStereochemistrychemistry.chemical_elementCrystallography X-RayLigandsChlorideMagnetic susceptibilityCopperInorganic Chemistrychemistry.chemical_compoundTrigonal bipyramidal molecular geometryCrystallographyMagneticschemistryAtommedicineHydrocarbons ChlorinatedOrganometallic CompoundsPhysical and Theoretical ChemistryCopperSchiff Basesmedicine.drugGroup 2 organometallic chemistryInorganic chemistry
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Synthesis of and structural studies on lead(II) cysteamin complexes.

2004

The novel compounds PbCl(2).(SCH(2)CH(2)NH(3)) (1), Pb(SCH(2)CH(2)NH(2))(2).2PbCl(SCH(2)CH(2)NH(2)) (2), and Pb(SCH(2)CH(2)NH(2))(2) (3) were synthesized by reaction of PbO or PbCl(2) with [HSCH(2)CH(2)NH(3)]Cl and NaOH, and were characterized by elemental analysis, IR-, and UV/vis-spectroscopy. Single-crystal X-ray diffraction revealed different coordination modes for the two Pb atoms in 2. The Pb atom in the Pb(SCH(2)CH(2)NH(2))(2) unit forms two covalent Pb-S and two intramolecular dative Pb...N bonds, leading to a pseudo trigonal bipyramidal configuration with a stereochemically active lone pair. The Pb atom in the PbCl(SCH(2)CH(2)NH(2)) unit, the first moiety structurally characterized…

Molecular StructureStereochemistryChemistryCysteamineIntermolecular forceInorganic ChemistryTrigonal bipyramidal molecular geometryCrystallographyOctahedronLeadModels ChemicalCovalent bondIntramolecular forceAtomMoietyPhysical and Theoretical ChemistryLone pairInorganic chemistry
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Identification of Synaptic Integration Mode in CA3 Pyramidal Neuron Model

2019

International audience; A morphologically realistic and anisotropic model of CA3 pyramidal neuron was developed to determine the synaptic integration modes the neuron is able to perform. Linearity and nonlinearity were identified in different synaptic locations with varying active mechanisms such as the presence of ionic channels in the dendritic arbor and the types of receptors in the synapse. Quantification of synaptic integration was performed using paired-pulse stimulation protocol and subthreshold input/output (sI/O) transformation. Results show that the mode of synaptic integration is location-dependent while the linearity or nonlinearity in the integration is mainly influenced by the…

MorphologyShaftsionic channelsResistancereceptorstwo-layer networksynaptic integration modesimple CA3 pyramidal neuronSynapselinear integrationdendritic arbormedicinesynaptic locationsCA3 pyramidal neuron model[SDV.IB] Life Sciences [q-bio]/BioengineeringNeuronsbiomembrane transportcomputational powerPhysicssubthreshold input-output transformationSynaptic integrationSubthreshold conductionmorphologically realistic modelMode (statistics)Linearitypaired-pulse stimulation protocolactive channelsanisotropic modelNonlinear systemmedicine.anatomical_structurenervous systemsublinear integrationCa3 pyramidal neuronbioelectric phenomena[SDV.IB]Life Sciences [q-bio]/BioengineeringAction potentialsNeuronneurophysiologysupralinear integrationNeuroscienceNeckProtocols2019 9th International IEEE/EMBS Conference on Neural Engineering (NER)
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The frontal agranular cortex and the organization of purposeful movements

1985

A critical review of the traditional concepts of cortical association and motor areas is followed by a description of the functional organization and intrinsic and extrinsic cortical connectivity of the arcuate premotor area (APA). It is concluded that the frontal cortical organization of externally triggered purposeful movements is made possible by the associative character of Brodmann's area 6 and by its peculiar pattern of intra-areal connectivity.

MovementPyramidal TractsSensationDermatologyEfferent Pathwaysbehavioral disciplines and activitiesAssociationCortex (anatomy)medicineAnimalsHumansCerebral CortexNeuronsAfferent PathwaysBrain MappingNeocortexMotor areaGeneral NeuroscienceMotor CortexHaplorhiniGeneral MedicineFrontal LobePsychiatry and Mental healthmedicine.anatomical_structureCatsRabbitsNeurology (clinical)Functional organizationPsychologyNeurosciencepsychological phenomena and processesThe Italian Journal of Neurological Sciences
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Multi-focus image fusion using local variability

2018

In this thesis, we are interested in the multi-focus image fusion method. This technique consists of fusing several captured images with different focal lengths of the same scene to obtain an image with better quality than the two source images. We propose an image fusion method based on Laplacian pyramid technique using Discrete Wavelet Transform (DWT) as a selection rule. We then develop two multi-focus image fusion methods based on the local variability of each pixel. It takes into account the information in the surrounding pixel area. The first method is to use local variability as an information in the Dempster-Shafer theory. The second method uses a metric based on local variability. …

Multi-Focus image fusionLa variabilité locale[INFO.INFO-TI] Computer Science [cs]/Image Processing [eess.IV][INFO.INFO-TI]Computer Science [cs]/Image Processing [eess.IV]La transformée en ondelettes discrèteLes pyramidales LaplaciennesLa fusion d'images multi focalesLa théorie de Dempster-ShaferLocal variabilityLaplacian pyramidDempster-Shafer theoryDiscrete Wavelet Transform
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Dendritic Ih selectively blocks temporal summation of unsynchronized distal inputs in CA1 pyramidal neurons.

2004

The active dendritic conductances shape the input-output properties of many principal neurons in different brain regions, and the various ways in which they regulate neuronal excitability need to be investigated to better understand their functional consequences. Using a realistic model of a hippocampal CA1 pyramidal neuron, we show a major role for the hyperpolarization-activated current, I-h, in regulating the spike probability of a neuron when independent synaptic inputs are activated with different degrees of synchronization and at different distances from the soma. The results allowed us to make the experimentally testable prediction that the I-h in these neurons is needed to reduce ne…

N-MethylaspartateTime FactorsComputer scienceCognitive NeuroscienceModels NeurologicalNeural ConductionHippocampal formationSummationHippocampusSynaptic TransmissionCA1Cellular and Molecular NeurosciencemedicineExcitatory Amino Acid AgonistsAnimalsComputer Simulationalpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic AcidI-hProbabilityCa1 pyramidal neuronPyramidal CellsExcitatory Postsynaptic PotentialsReproducibility of ResultsmodelingDendritesSensory Systemsdendritic integrationmedicine.anatomical_structurenervous systemSomaNeuronNeuroscience
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Action of anticonvulsants on hippocampal slices in Mg-free medium

1989

The effects of six prototype anticonvulsant drugs were investigated on epileptiform field potential discharges evoked in hippocampal slices of rats by removing magnesium ions from the perfusion fluid in order to reveal a possible interaction with N-methyl-D-aspartate (NMDA) receptor activation. All drugs reduced the multiple discharges with the following order of potency: midazolam greater than carbamazepine = phenytoin = phenobarbital greater than ethosuximide = valproate. They had a stronger depressant effect on the later population spikes but none of them abolished the epileptiform discharge. These effects can be explained by known mechanisms of action of the anticonvulsants tested and l…

N-Methylaspartatemedicine.medical_treatmentPopulationPyramidal TractsIn Vitro TechniquesPharmacologyHippocampusReceptors N-Methyl-D-AspartatemedicineAnimalsMagnesiumeducationMagnesium ionPharmacologyAspartic Acideducation.field_of_studyEpilepsyDose-Response Relationship DrugChemistryElectroencephalographyRats Inbred StrainsGeneral MedicineCarbamazepineElectric StimulationRatsReceptors NeurotransmitterPerfusionEthosuximideAnticonvulsantnervous systemMechanism of actionNMDA receptorAnticonvulsantsPhenobarbitalmedicine.symptommedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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Cell expression of GDAP1 in the nervous system and pathogenesis of Charcot-Marie-Tooth type 4A disease

2007

Abstract Mutations in the mitochondrial protein GDAP1 are the cause of Charcot-Marie-Tooth type 4A disease (CMT4A), a severe form of peripheral neuropathy associated with either demyelinating, axonal or intermediate pheno-types. GDAP1 is located in the outer mitochondrial membrane and it seems that may be related with the mitochondrial network dynamics. We are interested to define cell expression in the nervous system and the effect of mutations in mitochondrial morphology and pathogenesis of the disease. We investigated GDAP1 expression in the nervous system and dorsal root ganglia (DRG) neuron cultures. GDAP1 is expressed in motor and sensory neurons of the spinal cord and other large neu…

Nervous systemCMT4A mutations and pathogenesisPathologymedicine.medical_specialtyperipheral neuropathyCharcot-Marie-Tooth type 4A diseaseMutation MissenseGene ExpressionImages in Cellular / Molecular MedicineNerve Tissue ProteinsGDAP1MitochondrionBiologymedicine.disease_causeNervous SystemPathogenesisMicePurkinje CellsCharcot-Marie-Tooth DiseaseInterneuronsGanglia SpinalChlorocebus aethiopsmedicineAnimalsHumansNeurons AfferentCells CulturedMotor NeuronsMutationfusion and fission pathwayPyramidal CellsCell Biologymedicine.diseaseSpinal cordImmunohistochemistrymitochondrial dynamicsCell biologyOlfactory bulbRatsmedicine.anatomical_structurePeripheral neuropathynervous systemAnimals NewbornSpinal CordCOS CellsMolecular MedicineNeuronHeLa CellsJournal of Cellular and Molecular Medicine
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Monoclonal antibodies SMI 311 and SMI 312 as tools to investigate the maturation of nerve cells and axonal patterns in human fetal brain

1998

Neurofilaments, which are exclusively found in nerve cells, are one of the earliest recognizable features of the maturing nervous system. The differential distribution of neurofilament proteins in varying degrees of phosphorylation within a neuron provides the possibility of selectively demonstrating either somata and dendrites or axons. Non-phosphorylated neurofilaments typical of somata and dendrites can be visualized with the aid of monoclonal antibody SMI 311, whereas antibody SMI 312 is directed against highly phosphorylated axonal epitopes of neurofilaments. The maturation of neuronal types, the development of area-specific axonal networks, and the gradients of maturation can thus be …

Nervous systemHistologyNeurofilamentmedicine.drug_classeducationImmunocytochemistryGolgi ApparatusGestational AgeBiologyMonoclonal antibodyPathology and Forensic MedicineEpitopeschemistry.chemical_compoundNeurofilament ProteinsmedicineHumansParaformaldehydeNeuronsPyramidal CellsfungiInfant NewbornAntibodies MonoclonalBrainAbortion InducedDendritesCell BiologyImmunohistochemistryAxonsmedicine.anatomical_structurenervous systemchemistryImmunohistochemistryNeuronNeuroscienceImmunostainingCell and Tissue Research
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