Search results for "RED"

showing 10 items of 23890 documents

Case-specific performance of MM-PBSA, MM-GBSA, and SIE in virtual screening.

2015

In drug discovery the reliable prediction of binding free energies is of crucial importance. Methods that combine molecular mechanics force fields with continuum solvent models have become popular because of their high accuracy and relatively good computational efficiency. In this research we studied the performance of molecular mechanics generalized Born surface area (MM-GBSA), molecular mechanics Poisson-Boltzmann surface area (MM-PBSA), and solvated interaction energy (SIE) both in their virtual screening efficiency and their ability to predict experimentally determined binding affinities for five different protein targets. The protein-ligand complexes were derived with two different app…

molecular mechanics generalized Born surface areaPhosphodiesterase InhibitorsMolecular Dynamics Simulationta3111Molecular mechanicsMolecular Docking Simulationbeta-LactamasesMolecular dynamicssolvated interaction energyBacterial ProteinsComputational chemistryAldehyde ReductaseDrug DiscoveryMaterials ChemistryHumansHSP90 Heat-Shock ProteinsPhysical and Theoretical ChemistryBeta-Lactamase InhibitorsSpectroscopymolecular mechanics Poisson-Boltzmann surface areaMM-GBSAVirtual screeningBinding SitesChemistryPhosphoric Diester Hydrolasesta1182Hydrogen BondingInteraction energyvirtual screeningComputer Graphics and Computer-Aided DesignMolecular Docking SimulationMM-PBSAModels ChemicalROC CurveSolvent modelsDocking (molecular)Area Under CurveBiological systemReceptors Progesteronebeta-Lactamase InhibitorsHydrophobic and Hydrophilic InteractionsProtein BindingJournal of molecular graphicsmodelling
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A magnetic look into the protecting layer of Au25 clusters

2016

The field of molecular metal clusters protected by organothiolates is experiencing a very rapid growth. So far, however, a clear understanding of the fine interactions between the cluster core and the capping monolayer has remained elusive, despite the importance of the latter in interfacing the former to the surrounding medium. Here, we describe a very sensitive methodology that enables comprehensive assessment of these interactions. Pulse electron nuclear double resonance (ENDOR) was employed to study the interaction of the unpaired electron with the protons of the alkanethiolate ligands in four structurally related paramagnetic Au25(SR)0 18 clusters (R ¼ ethyl, propyl, butyl, 2-methylpro…

molecular metal clusterselectronic distributionkemiaIcosahedral symmetryAnalytical chemistry02 engineering and technologychemistry010402 general chemistrygold clusters01 natural sciencesSpectral lineAu25ParamagnetismMolecular dynamicsNMR spectroscopyMonolayerthiolate-cappedCluster (physics)ta116Electron nuclear double resonanceChemistryChemistry (all)paramagnetic gols nanoclustersGeneral ChemistryENDOR spectroscopy021001 nanoscience & nanotechnology0104 chemical sciencesUnpaired electronChemical physics0210 nano-technology
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CHANGES IN THE EUROPEAN CENTRAL BANK (ECB) APPROACHES IN MATTERS OF MONETARY POLICY AFTER THE OUTBREAK OF THE INTERNATIONAL FINANCIAL CRISIS

2012

The problem of monetary policy is a current one, given the fact that now, through this component of the economic policy, the monetary authority of each state tries to solve the problems considered essential for each economy separately. Through this article I have tried to capture the major changes regarding the implementation of the ECB's monetary policy before and after the outbreak of the international financial crisis. Following the analysis I have shown that the monetary policy of the ECB is not a constant one in its actions and instruments used but it is adapted to a conjuncture context through which the European economy is passing through. Therefore, in this paper I have broadly shown…

monetary policy monetary policy interest rate credit financial crisisStudies in Business and Economics
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Quelques observations récentes sur des sites de l'Antiquité tardive à Autun (2001-2008)

2011

This article describes the result of ten or so fairly limited preventive archaeology operations (surveillance of works, diagnostics not followed up with excavations) carried out over the last ten years that have nonetheless finalised knowledge of several deposits from Late Antiquity in Autun located intra muros but also outside the walls. The works have enabled us to renew our knowledge of the reduced enclosure and of three Late Antiquity necropolises, to discover the remains of a lime kiln from the end of the 4th century at the centre of a public zone (perhaps the forum), and lastly to point up the difficulties of interpretation of an occupation of two zones from the end of the 4th century…

monumental zonelime kiln[SHS.ARCHEO] Humanities and Social Sciences/Archaeology and Prehistory[SHS.ARCHEO]Humanities and Social Sciences/Archaeology and PrehistoryReduced enclosuredomusîlot monumental[ SHS.ARCHEO ] Humanities and Social Sciences/Archaeology and PrehistoryEnceinte réduiteforumatelier de chaufourniernécropolenecropolis
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Mašīntulkotu nosaukto entitāšu gramatisko locījumu noteikšana automātiskajā pēcrediģēšanā

2020

Dziļās mašīnmācīšanās sasniegumi ir veicinājuši ievērojamu attīstību mašīntulkošanas jomā. Tomēr joprojām bieži tiek novērots, ka retas nosauktās entitātes neironu mašīntulkošanas sistēmas iztulko nepareizi. Kļūdaini tulkotu nosaukto entitāšu labošanu var veikt, izmantojot automātisko pēcrediģēšanu. Pēcrediģēšana kā vienu no soļiem ietver teikuma kontekstā iederīgas morfoloģiskās formas noteikšanu. Šī darba mērķis bija izstrādāt un apmācīt klasifikatoru nosauktās entitātes teikumā iederīgo morfoloģisko kategoriju formu paredzēšanai. Darba ietvaros tika izpētīts, kā risinātas līdzīgas ar vārdu kontekstuālu morfoloģisko analīzi saistītas problēmas, sagatavoti klasifikatoram piemēroti apmācība…

morfoloģiskā formveidošanaperceptronsDatorzinātneautomātiskā pēcrediģēšanamašīnmācīšanāsdabisko valodu apstrāde
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Modelo predictivo de mortalidad a largo plazo en el trasplante hepático del adulto

2015

El trasplante hepático es el tratamiento de elección de muchas hepatopatías terminales y un procedimiento que ha ido evolucionando desde sus inicios, mejorando sus resultados con el paso del tiempo. A pesar de que nuestro país es uno de los que presentan las tasas de donación más altas del mundo, debido al incremento en el número de indicaciones para la realización de un trasplante hepático, porcentaje de pacientes que fallecen en lista de espera se cifra en torno al 5 %. Por ello se continúa investigando y buscando modelos predictivos y de asignación de injertos a fin de mejorar la eficiencia global del procedimiento. En nuestro trabajo planteamos como objetivo el desarrollo de un modelo p…

mortalidad receptortrasplante hepáticoUNESCO::CIENCIAS MÉDICASmodelo predictivo:CIENCIAS MÉDICAS [UNESCO]
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Laulunopetuksen psyykkisistä vaikutuksista : opetuksen kriittisiä tekijöitä ja terapeuttisia piirteitä

2015

Tutkimuksessa tarkasteltiin laulunopetuksen tuntitapahtumia psyykkisten ilmiöiden näkökulmasta ja pyrittiin selvittämään millaisia kriittisiä ja terapeuttisia tekijöitä laulunopetus sisältää. Tätä tutkittiin laulunopiskelijoille lähetetyllä sähköisellä kyselyllä, joka sisälsi sekä monivalintakysymyksiä että avoimia kysymyksiä. Kysymyksillä pyrittiin selvittämään mitä opiskelijat mielsivät sisältyvän hyvään laulutuntiin ja laulunopettajaan. Myös opettajien näkökulma tuotiin esiin kolmessa haastattelussa, joissa kysyttiin opettajien mielipiteitä hyvän laulutunnin edellytyksistä, onnistuneen opettaja-oppilassuhteen edellytyksistä, opetuksen tyypillisimmistä kipupisteistä sekä opettavimmista ja…

motivaatiooppiminenlaulaminenlaulunopettajatBion Wilfred Rpsykodynamiikkaopetus
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MOTIVACIÓN Y ESTILO ATRIBUCIONAL SOBRE EL RENDIMIENTO ACADÉMICO EN EDUCACIÓN INFANTIL

2016

El presente trabajo tiene como objetivo examinar el poder predictivo de variables del sistema motivacional sobre las habilidades iniciales de lectura y matemáticas en una muestra de niños de Educación Infantil. Participaron 209 preescolares (5-6 años) y sus maestros. Se evaluaron las  habilidades matemáticas de conteo, conocimiento de los números, cálculo y resolución de problemas. Para determinar el rendimiento en lectura se administraron tareas de identificación de letras y de lectura de palabras. Respecto al sistema motivacional, se analizaron las variables de competencia-motivación, atención-persistencia y actitud hacia el aprendizaje, así como las dimensiones de internalidad, globalida…

motivación hacia el aprendizajeMathematical problemmedia_common.quotation_subjectestilo atribucionallcsh:BF1-99005 social scienceslecturaStability (learning theory)050301 educationGlobalitymatemáticaseducación infantillcsh:PsychologyMath skillsReading (process)Predictive powerMathematics educationMathematical ability0501 psychology and cognitive sciences0503 education050104 developmental & child psychologymedia_commonVariable (mathematics)
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Neural Correlates of Age-Related Changes in Precise Grip Force Regulation: A Combined EEG-fNIRS Study

2020

Motor control is associated with suppression of oscillatory activity in alpha (8–12 Hz) and beta (12–30 Hz) ranges and elevation of oxygenated hemoglobin levels in motor-cortical areas. Aging leads to changes in oscillatory and hemodynamic brain activity and impairments in motor control. However, the relationship between age-related changes in motor control and brain activity is not yet fully understood. Therefore, this study aimed to investigate age-related and task-complexity-related changes in grip force control and the underlying oscillatory and hemodynamic activity. Sixteen younger [age (mean ± SD) = 25.4 ± 1.9, 20–30 years] and 16 older (age = 56.7 ± 4.7, 50–70 years) healthy men were…

motor recoveryagingneuroplasticitymotor controlfunctional near-infrared spectroscopylcsh:Neurosciences. Biological psychiatry. Neuropsychiatryelectroencephalographylcsh:RC321-571Frontiers in Aging Neuroscience
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Commentary: Concurrent Imitative Movement During Action Observation Facilitates Accuracy of Outcome Prediction in Less-Skilled Performers

2018

motor scenarioMovement (music)tacticslcsh:BF1-99005 social sciences030229 sport sciences050105 experimental psychology03 medical and health scienceslcsh:Psychology0302 clinical medicinemodalities' ladderAction observationBernstein's theory0501 psychology and cognitive sciencesmotor habitOutcome predictionPsychologyGeneral PsychologyCognitive psychologyFrontiers in Psychology
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