Search results for "Rauvolfia serpentina"

showing 10 items of 29 documents

Ligand structures of synthetic deoxa-pyranosylamines with raucaffricine and strictosidine glucosidases provide structural insights into their binding…

2014

Insight into the structure and inhibition mechanism of O-β-d-glucosidases by deoxa-pyranosylamine type inhibitors is provided by X-ray analysis of complexes between raucaffricine and strictosidine glucosidases and N-(cyclohexylmethyl)-, N-(cyclohexyl)- and N-(bromobenzyl)-β-d-gluco-1,5-deoxa-pyranosylamine. All inhibitors anchored exclusively in the catalytic active site by competition with appropriate enzyme substrates. Thus facilitated prospective elucidation of the binding networks with residues located at <3.9 A distance will enable the development of potent inhibitors suitable for the production of valuable alkaloid glucosides, raucaffricine and strictosidine, by means of synthesis in …

Models MolecularStereochemistryCyclopentanesLigandsRauwolfiaStructure-Activity RelationshipSugar AlcoholsRauvolfia serpentinaDrug DiscoveryHydrolasePharmacologychemistry.chemical_classificationBinding SitesDose-Response Relationship DrugMolecular StructurebiologyAlkaloidActive siteGeneral Medicinebiology.organism_classificationLigand (biochemistry)EnzymeBiochemistrychemistryStrictosidinebiology.proteinGlucosidasesGlucosidasesJournal of Enzyme Inhibition and Medicinal Chemistry
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The Structure of Rauvolfia serpentina Strictosidine Synthase Is a Novel Six-Bladed β-Propeller Fold in Plant Proteins

2006

Abstract The enzyme strictosidine synthase (STR1) from the Indian medicinal plant Rauvolfia serpentina is of primary importance for the biosynthetic pathway of the indole alkaloid ajmaline. Moreover, STR1 initiates all biosynthetic pathways leading to the entire monoterpenoid indole alkaloid family representing an enormous structural variety of ∼2000 compounds in higher plants. The crystal structures of STR1 in complex with its natural substrates tryptamine and secologanin provide structural understanding of the observed substrate preference and identify residues lining the active site surface that contact the substrates. STR1 catalyzes a Pictet-Spengler–type reaction and represents a novel…

Models MolecularTryptamineProtein FoldingStrictosidine synthaseProtein ConformationMolecular Sequence DataSequence alignmentPlant ScienceCatalysisRauwolfiaSubstrate Specificitychemistry.chemical_compoundRauvolfia serpentinaCarbon-Nitrogen LyasesAmino Acid SequenceResearch ArticlesConserved SequencePlant ProteinsBinding SitesSequence Homology Amino AcidbiologyIndole alkaloidActive siteCell BiologyLyasebiology.organism_classificationTryptamineschemistryBiochemistrybiology.proteinSecologaninSequence AlignmentThe Plant Cell
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New Alkaloids of the Sarpagine Group from Rauvolfia serpentina Hairy Root Culture

2002

Three new monoterpenoid indole alkaloids, 19(S),20(R)-dihydroperaksine (1), 19(S),20(R)-dihydroperaksine-17-al (2), and 10-hydroxy-19(S),20(R)-dihydroperaksine (3), along with 16 known alkaloids 4-19 were isolated from hairy root culture of Rauvolfia serpentina, and their structures were elucidated by 1D and 2D NMR analyses. Taking into account the stereochemistry of the new alkaloids and results of preliminary enzymatical studies, the putative biosynthetical relationships between the novel alkaloids are discussed.

Monoterpenoid Indole AlkaloidsStereochemistryPharmaceutical SciencePharmacognosyPlant RootsRauwolfiaIndole AlkaloidsAnalytical ChemistryRauvolfia serpentinaDrug DiscoveryNuclear Magnetic Resonance BiomolecularPharmacologyFolk medicinePlants MedicinalMolecular StructurebiologyApocynaceaeChemistryAlkaloidOrganic ChemistryStereoisomerismbiology.organism_classificationSecologanin Tryptamine AlkaloidsTerpenoidComplementary and alternative medicineHairy root cultureMolecular MedicineChromatography Thin LayerRhizobiumJournal of Natural Products
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Molecular cloning and functional bacterial expression of a plant glucosidase specifically involved in alkaloid biosynthesis.

2000

Monoterpenoid indole alkaloids are a vast and structurally complex group of plant secondary compounds. In contrast to other groups of plant products which produce many glycosides, indole alkaloids rarely occur as glucosides. Plants of Rauvolfia serpentina accumulate ajmaline as a major alkaloid, whereas cell suspension cultures of Rauvolfia mainly accumulate the glucoalkaloid raucaffricine at levels of 1.6 g/l. Cell cultures do contain a specific glucosidase. known as raucaffricine-O-beta-D-glucosidase (RG), which catalyzes the in vitro formation of vomilenine, a direct intermediate in ajmaline biosynthesis. Here, we describe the molecular cloning and functional expression of this enzyme in…

RauvolfiaDNA ComplementaryStereochemistryMolecular Sequence DataPlant ScienceHorticultureMolecular cloningBiochemistryIndole AlkaloidsSubstrate SpecificityMagnoliopsidaAlkaloidsRauvolfia serpentinamedicineAmino Acid SequenceCloning MolecularMolecular BiologybiologyBase SequenceGeneral Medicinebiology.organism_classificationSecologanin Tryptamine AlkaloidsAjmalineBlotting SouthernBiochemistryVomilenineStrictosidinebiology.proteinHeterologous expressionGlucosidasesGlucosidasesmedicine.drugPhytochemistry
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Vinorine synthase from Rauvolfia: the first example of crystallization and preliminary X-ray diffraction analysis of an enzyme of the BAHD superfamily

2004

Abstract Crystals of vinorine synthase (VS) from medicinal plant Rauvolfia serpentina expressed in Escherichia coli have been obtained by the hanging-drop technique at 305 K with ammonium sulfate and PEG 400 as precipitants. The enzyme is involved in the biosynthesis of the antiarrhythmic drug ajmaline and is a member of the BAHD superfamily of acyltransferases. So far, no three-dimensional structure of a member of this enzyme family is known. The crystals belong to the space group P 2 1 2 1 2 1 with cell dimensions of a =82.3 A, b =89.6 A and c =136.2 A. Under cryoconditions (120 K), a complete data set up to 2.8 A was collected at a synchrotron source.

RauvolfiaIndolesStereochemistryBiophysicsCrystallography X-RayBiochemistryRauwolfiaAnalytical Chemistrychemistry.chemical_compoundAlkaloidsBiosynthesisRauvolfia serpentinamedicineMolecular Biologychemistry.chemical_classificationATP synthasebiologybiology.organism_classificationEnzymesAjmalineEnzymechemistryBiochemistryAcyltransferasesAcetyltransferasebiology.proteinCrystallizationmedicine.drugBiochimica et Biophysica Acta (BBA) - Proteins and Proteomics
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Heterologous expression, purification, crystallization and preliminary X-ray analysis of raucaffricine glucosidase, a plant enzyme specifically invol…

2006

Raucaffricine glucosidase (RG) is an enzyme that is specifically involved in the biosynthesis of indole alkaloids from the plant Rauvolfia serpentina. After heterologous expression in Escherichia coli cells, crystals of RG were obtained by the hanging-drop vapour-diffusion technique at 293 K with 0.3 M ammonium sulfate, 0.1 M sodium acetate pH 4.6 buffer and 11% PEG 4000 as precipitant. Crystals belong to space group I222 and diffract to 2.30 A, with unit-cell parameters a = 102.8, b = 127.3, c = 215.8 A.

RauvolfiaStereochemistryBiophysicsmedicine.disease_causeCrystallography X-RayBiochemistryRauwolfiachemistry.chemical_compoundBiosynthesisStructural BiologyRauvolfia serpentinaGeneticsmedicineEscherichia coliCloning MolecularEscherichia colichemistry.chemical_classificationIndole testbiologyCondensed Matter Physicsbiology.organism_classificationEnzymechemistryBiochemistryCrystallization Communicationsbiology.proteinHeterologous expressionCrystallizationGlucosidasesGlucosidases
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Hydroquinone: O-glucosyltransferase from cultivated Rauvolfia cells: enrichment and partial amino acid sequences.

2000

Plant cell suspension cultures of Rauvolfia are able to produce a high amount of arbutin by glucosylation of exogenously added hydroquinone. A four step purification procedure using anion exchange, hydrophobic interaction, hydroxyapatite-chromatography and chromatofocusing delivered in a yield of 0.5%, an approximately 390 fold enrichment of the involved glucosyltransferase. SDS-PAGE showed a M(r) for the enzyme of 52 kDa. Proteolysis of the pure enzyme with endoproteinase LysC revealed six peptide fragments with 9-23 amino acids which were sequenced. Sequence alignment of the six peptides showed high homologies to glycosyltransferases from other higher plants.

RauvolfiaStereochemistryMolecular Sequence DataPeptidePlant ScienceHorticultureBiochemistryRauwolfiachemistry.chemical_compoundRauvolfia serpentinaAmino Acid SequenceMolecular BiologyCells Culturedchemistry.chemical_classificationChromatographyPlants MedicinalbiologyChromatofocusingArbutinGeneral Medicinebiology.organism_classificationChromatography Ion ExchangePeptide FragmentsAmino acidMolecular WeightKineticsEnzymeDurapatitechemistryBiochemistryGlucosyltransferasesbiology.proteinGlucosyltransferaseElectrophoresis Polyacrylamide GelPhytochemistry
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Crystallization and preliminary X-ray crystallographic analysis of strictosidine synthase from Rauvolfia: the first member of a novel enzyme family.

2004

Strictosidine synthase is a central enzyme involved in the biosynthesis of almost all plant monoterpenoid indole alkaloids. Strictosidine synthase from Rauvolfia serpentina was heterologously expressed in Escherichia coli. Crystals of the purified recombinant enzyme have been obtained by the hanging-drop technique at 303 K with potassium sodium tartrate tetrahydrate as precipitant. The crystals belong to the space group R3 with cell dimensions of a=b=150.3 A and c=122.4 A. Under cryoconditions (120 K), the crystals diffract to about 2.95 A.

RauvolfiaStrictosidine synthaseDNA PlantStereochemistryBiophysicsmedicine.disease_causeCrystallography X-RayBiochemistryRauwolfiaAnalytical Chemistrylaw.inventionchemistry.chemical_compoundBiosynthesislawRauvolfia serpentinaCarbon-Nitrogen LyasesmedicineEscherichia coliCrystallizationMolecular BiologyEscherichia colichemistry.chemical_classificationTetrahydratebiologyBase Sequencebiology.organism_classificationRecombinant ProteinsEnzymechemistryBiochemistrybiology.proteinBiochimica et biophysica acta
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Purification and partial amino acid sequences of the enzyme vinorine synthase involved in a crucial step of ajmaline biosynthesis.

2004

The acetyl-CoA-dependent enzyme vinorine synthase was isolated from hybrid cell suspension cultures of Rauvolfia serpentina and Rhazya stricta. The sarpagan-type alkaloid gardneral was used as a substrate of the enzyme leading to the ajmalan-type 10-methoxyvinorine. An HPLC-based assay was developed to monitor vinorine synthase activity, which allowed establishing a five step purification procedure combining anion exchange, hydrophobic interaction, hydroxyapatite and gel filtration. Purification resulted in a yield of 0.2% and an approximately 991-fold enrichment of the acetyltransfer activity. SDS-PAGE analysis showed a Mr for the enzyme of approximately 50 kDa. The four peptide fragments …

Sequence analysisStereochemistryClinical BiochemistryMolecular Sequence DataPharmaceutical ScienceHybrid CellsBiochemistryRauwolfiaIndole Alkaloidschemistry.chemical_compoundVinorine synthase activityBiosynthesisRauvolfia serpentinaSequence Analysis ProteinDrug DiscoveryAmino Acid SequenceAcetyl-CoA C-AcetyltransferaseMolecular BiologyPeptide sequencechemistry.chemical_classificationAjmalinebiologyATP synthaseMolecular StructureOrganic ChemistrySubstrate (chemistry)biology.organism_classificationApocynaceaeEnzymeBiochemistrychemistrybiology.proteinMolecular MedicineBioorganicmedicinal chemistry
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Crystallization and preliminary X-ray analysis of native and selenomethionyl vinorine synthase from Rauvolfia serpentina.

2005

Vinorine synthase (VS) is a central enzyme of the biosynthesis of the antiarrhythmic drug ajmaline and is a member of the BAHD superfamily of acyltransferases. So far, no three-dimensional structure with significant sequence homology with VS is known. Crystals of VS and selenomethionyl-labelled VS from the medicinal plant Rauvolfia serpentina have been obtained by the hanging-drop technique at 305 K with ammonium sulfate and PEG 400 as precipitants. VS crystals diffract to 2.8 Å and belong to space group P212121, with unit-cell parameters a = 82.3, b = 89.6, c = 136.2 Å. The selenomethionyl VS crystal was nearly isomorphous with the VS crystal.

StereochemistryCrystallography X-RayRauwolfialaw.inventionIndole AlkaloidsLigaseschemistry.chemical_compoundBiosynthesisStructural BiologylawRauvolfia serpentinamedicineCrystallizationSelenomethioninePlant ProteinsPEG 400chemistry.chemical_classificationATP synthasebiologyGeneral Medicinebiology.organism_classificationAjmalineEnzymechemistryAcyltransferasesbiology.proteinCrystallizationmedicine.drugActa crystallographica. Section D, Biological crystallography
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