Search results for "S1"

showing 10 items of 755 documents

STUDY ON NOISE LEVEL GENERATED BY HUMAN ACTIVITIES IN SIBIU CITY, ROMANIA

2014

In this paper I have proposed an analysis and monitoring of the noise sources in the open spaces of air traffic, rail and car in Sibiu. From centralizing data obtained from the analysis of the measurements performed with equipment noise levels, we concluded that the noise and vibration produced by means of Transportation (air, road, rail) can affect human health if they exceed limits. Noise is present and part of our lives and always a source of pollution as any of modern man is not conscious.

air trafficrail trafficcar trafficnoise levellcsh:Agriculture (General)lcsh:S1-972Scientific Papers Series : Management, Economic Engineering in Agriculture and Rural Development
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Phosphonic Acid Analogues of Phenylglycine as Inhibitors of Aminopeptidases: Comparison of Porcine Aminopeptidase N, Bovine Leucine Aminopeptidase, T…

2019

The inhibitory activity of 14 racemic phosphonic acid analogs of phenylglycine, substituted in aromatic rings, towards porcine aminopeptidase N (pAPN) and barley seed aminopeptidase was determined experimentally. The obtained patterns of the inhibitory activity against the two enzymes were similar. The obtained data served as a basis for studying the binding modes of these inhibitors by pAPN using molecular modeling. It was found that their aminophosphonate fragments were bound in a highly uniform manner and that the difference in their affinities most likely resulted from the mode of substitution of their phenyl rings. The obtained binding modes towards pAPN were compared, with these predi…

aminophosphonateMolecular modelStereochemistryPharmaceutical Sciencelcsh:Medicinelcsh:RS1-441AminopeptidaseArticlelcsh:Pharmacy and materia medica03 medical and health sciences0302 clinical medicineDrug Discoveryinhibitorsaminopeptidases030304 developmental biologychemistry.chemical_classification0303 health sciencesChemistrymolecular modelingAminopeptidase Nlcsh:RAromaticityAffinitiesEnzymefluorine substitutedAminophosphonate030220 oncology & carcinogenesisMolecular Medicinephenylglycine analoguesLeucinePharmaceuticals
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How Molecular Topology Can Help in Amyotrophic Lateral Sclerosis (ALS) Drug Development: A Revolutionary Paradigm for a Merciless Disease

2022

r Abstract: Even if amyotrophic lateral sclerosis is still considered an orphan disease to date, its prevalence among the population is growing fast. Despite the efforts made by researchers and pharmaceutical companies, the cryptic information related to the biological and physiological onset mechanisms, as well as the complexity in identifying specific pharmacological targets, make it almost impossible to find effective treatments. Furthermore, because of complex ethical and economic aspects, it is usually hard to find all the necessary resources when searching for drugs for new orphan diseases. In this context, computational methods, based either on receptors or ligands, share the capabil…

amyotrophic lateral sclerosisamyotrophic lateral sclerosis; orphan diseases; molecular topology; drug design; QSAR; drug repurposingdrug repurposingdrug designQSARRPharmaceutical ScienceArticlemolecular topologyRS1-441orphan diseasesPharmacy and materia medicaDrug DiscoveryMolecular MedicineMedicinePharmaceuticals; Volume 15; Issue 1; Pages: 94
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STUDY ON WASTE WATER TREATMENT PLANTS

2015

Biogas is more and more used as an alternative source of energy, considering the fact that it is obtained from waste materials and it can be easily used in cities and rural communities for many uses, between which, as a fuel for households. Biogas has many energy utilisations, depending on the nature of the biogas source and the local demand. Generally, biogas can be used for heat production by direct combustion, electricity production by fuel cells or micro-turbines, Combined Hest and Power generation or as vehicle fuel. In this paper we search for another uses of biogas and Anaerobe Digestion substrate, such as: waste water treatment plants and agricultural wastewater treatment, which are…

anaerobe digestionbi ogaswaste waterlcsh:Agriculture (General)lcsh:S1-972Scientific Papers Series : Management, Economic Engineering in Agriculture and Rural Development
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Sequence of vascular patterning and gene transcription in the chick chorioallantoic membrane (15.1)

2014

Introduction: The chick chorioallantoic membrane (CAM) is a well-established model of both vasculogenesis and angiogenesis; however, little is known about the genetic control of vascular patterning in the CAM. Methods: Using recent advances in chicken genomics, we investigated the relative expression of 84 angiogenesis genes during the growth and remodeling of the CAM microcirculatory network. Chick embryos, cultured ex ovo, were studied during embryonic development days (EDD) 8-14. UV laser microdissection was used to harvest capillary plexus and 1st, 2nd, and 3rd order conducting vessels for qRT-PCR analysis. Results: Two transcription peaks were observed between EDD 8 and 14. The first p…

animal structuresAngiogenesisChemistryEmbryogenesisEPAS1BiochemistryMolecular biologyChick chorioallantoic membraneVasculogenesisTranscription (biology)GeneticsMolecular BiologyGeneMicrodissectionBiotechnologyThe FASEB Journal
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Synthesis of curcumin derivatives and analysis of their antitumor effects in triple negative breast cancer (TNBC) cell lines

2019

We analyzed antitumor effects of a series of curcumin analogues. Some of them were obtained by reaction of substitution involving the two phenolic OH groups of curcumin while the analogues with a substituent at C-4 was prepared following an original procedure that regards the condensation of benzenesulfenic acid onto the nucleophilic central carbon of the curcumin skeleton. We analyzed cytotoxic effects of such derivatives on two TNBC (triple negative breast cancer) cell lines, SUM 149 and MDA-MB-231, but only three of them showed an IC50 in a lower micromolar range with respect to curcumin. We also focused on these three derivatives that in both cell lines exhibited a higher or at least eq…

antiproliferative activitySubstituentPharmaceutical Sciencelcsh:Medicinelcsh:RS1-441antioxidant activityprooxidant activitylcsh:Pharmacy and materia medicapro-apoptotic activity03 medical and health scienceschemistry.chemical_compound0302 clinical medicineDrug DiscoveryCytotoxic T cellNF-κB inhibitionAntioxidant activity Antiproliferative activity NF-κB inhibition Pro-apoptotic activity Prooxidant activity Sulfenic acidIC50Triple-negative breast cancer030304 developmental biology0303 health sciencesCommunicationlcsh:Rsulfenic acidchemistryCell culture030220 oncology & carcinogenesisCancer researchCurcuminSettore BIO/14 - FarmacologiaMolecular MedicineSulfenic acidLead compound
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Observation of Higgs boson production in association with a top quark pair at the LHC with the ATLAS detector

2018

Physics letters / B 784, 173 - 191 (2018). doi:10.1016/j.physletb.2018.07.035

associated production [Higgs particle]Yukawa [coupling]13000 GeV-cms01 natural sciencesStandard deviationSubatomär fysikscattering [p p]Z0: pair productionCollisionsmeasured [total cross section]протон-протонные столкновенияGeneralLiterature_REFERENCE(e.g.dictionariesencyclopediasglossaries)ComputingMilieux_MISCELLANEOUSLHC; Higgs; Top-QuarkLarge Hadron ColliderQ007THXlcsh:QC1-999Top-Quark:Mathematics and natural scienses: 400::Physics: 430::Nuclear and elementary particle physics: 431 [VDP]pair production [Z0]CERN LHC CollHiggs bosonХиггса бозонcolliding beams [p p]top: pair productionHiggs particle: decay modesp p: scatteringmass spectrum: (4lepton)Ciências Naturais::Ciências FísicasAstrophysics::High Energy Astrophysical PhenomenaSTANDARD MODELddc:500.2SEARCHddc:530High Energy Physics010306 general physicstop quarktwo-photon [mass spectrum]Science & TechnologyHiggs particle: coupling010308 nuclear & particles physics(4lepton) [mass spectrum]HIGGSExperimental High Energy PhysicsATLAS детекторp p: colliding beamslcsh:Physicscoupling: Yukawamass spectrum: two-photonHiggsTop quarkHiggs Top LHC observationБольшой адронный коллайдерAtlas detectorCiencias Físicasbranching ratio [Higgs particle]pair production [top]High Energy Physics - Experiment//purl.org/becyt/ford/1 [https]W: pair productionHigh Energy Physics - Experiment (hep-ex)Subatomic Physics[PHYS.HEXP]Physics [physics]/High Energy Physics - Experiment [hep-ex]Physicsscattering | p p: colliding beams | top: pair production | Higgs particle: associated production | Higgs particle: decay modes | bottom: pair production | W: pair production | Z0: pair production | tau: pair production | photon: pair production | Higgs particle: coupling | coupling: Yukawa | CERN LHC Coll | ATLAS | mass spectrum: two-photon | mass spectrum: (4lepton) | Higgs particle: branching ratio | total cross section: measured | experimental results | 13000 GeV-cms [p p]proton–proton collisionstau: pair productionSettore FIS/01 - Fisica SperimentaleTOPATLASpair production [bottom]pair production [tau]S126STHpair production [W]LHCphoton: pair productionCIENCIAS NATURALES Y EXACTASParticle Physics - Experimentpair production [photon]jetsParticle physicsNuclear and High Energy Physicscoupling [Higgs particle]Higgs boson530 Physics:Ciências Físicas [Ciências Naturais]decay modes [Higgs particle]FOS: Physical sciencesbottom: pair productionFísica de Partículas y Campos5300103 physical sciencesHigh Energy Physics::Phenomenology:Matematikk og naturvitenskap: 400::Fysikk: 430::Kjerne- og elementærpartikkelfysikk: 431 [VDP]//purl.org/becyt/ford/1.3 [https]Higgs particle: associated productionHiggs particle: branching ratiototal cross section: measuredHigh Energy Physics::ExperimentHadron-hadron collisionsexperimental results
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Atgriezeniskā dienas grāmata kā pedagoģiskais risinājums bērnu ar autisma spektra traucējumiem komunikatīvās kompetences veicināšanai

2018

Šajā Maģistra darbā tiek prezentēta inovatīva “atgriezeniskā dienas grāmata” kā pedagoģiskais risinājums (objekts) bērnu ar autisma spektra traucējumiem komunikatīvās kompetences attīstīšanai (priekšmets). Darbam ir 83 lpp., tā skaitā 2 tabulas, 9 attēli, 68 zinātniskās literatūras vienības un 3 pielikumi Ieraksti ko vecāki un skolotāji fiksē dienas grāmatā, atspoguļojot ikdienā veiktās aktivitātes un kritiskos notikumus, palīdz paredzēt attīstības grūtības un labāk izprast konkrētās situācijas. Tika pierādīts, ka šī metode veicina bērnu verbālās un neverbālās komunikācijas uzlabošanu, sekmējot viņu emocionāla uztraukuma samazināšanos, kā arī viņu iespējas sekmīgāk iekļauties darba tirgū un…

autistic spectrum disorders communication alternative systems of communication “round trip agenda” familyPedagoģijals16131
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Immunogenic hotspots in the spacer domain of ADAMTS13 in immune‐mediated thrombotic thrombocytopenic purpura

2021

International audience; Background Immune-mediated thrombotic thrombocytopenic purpura (iTTP) is caused by anti-ADAMTS13 autoantibodies inducing a severe deficiency of ADAMTS13. Epitope mapping studies on samples obtained during acute iTTP episodes have shown that the iTTP immune response is polyclonal, with almost all patients having autoantibodies targeting the spacer domain of ADAMTS13.Objectives To identify the immunogenic hotspots in the spacer domain of ADAMTS13.Patients/methods A library of 11 full-length ADAMTS13 spacer hybrids was created in which amino acid regions of the spacer domain of ADAMTS13 were exchanged by the corresponding region of the spacer domain of ADAMTS1. Next, th…

autoantibodiesADAMTS13 Protein030204 cardiovascular system & hematologyEpitope03 medical and health sciencesEpitopes0302 clinical medicineVon Willebrand factorimmunophenotypinghemic and lymphatic diseasesHumansthrombotic thrombocytopenic purpurachemistry.chemical_classificationbiologyPurpura Thrombotic ThrombocytopenicAutoantibodyHematologyMolecular biologyADAMTS13ADAMTS133. Good healthAmino acidepitope mappingEpitope mappingchemistryPolyclonal antibodiesImmunoglobulin Gbiology.proteinDNA IntergenicAntibody[SDV.MHEP]Life Sciences [q-bio]/Human health and pathology
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STUDY OF RASPBERRY EXTRACT APPLICATIONS AS TEXTILE COLORANT ON NATURAL FIBERS

2014

The present study deals with the biomordant assisted application of natural extracts obtained from red raspberry (Rubus idaeus L.) fruits onto two different cellulosic supports – flax and bamboo. The study relies on the improvement of multifunctionalities such as colour fastness, washing and rubbing fastness, due to the synergism provided by the co-assistance of both a biomordant, and the complex resulted by inclusion of the pigment molecule, in the cavity of MCT-β-CD; it is well known that natural dye molecule have a good selectivity binding to the hydrophobic monochloro-triazynil-cyclodextrin’s (MCT-β-CD) cavity to form inclusion complexes. An investigation system provided the characteriz…

bamboo knitted fabricfastness propertiesnatural extractlcsh:Manufacturesflax fabricscolour differencelcsh:TS1-2301Annals of the University of Oradea: Fascicle of Textiles, Leatherwork
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