Search results for "Screen"

showing 10 items of 1374 documents

Cytotoxicity of some Cameroonian spices and selected medicinal plant extracts

2011

Abstract Ethnopharmacological relevance Several medicinal plants and spices are used traditionally to treat cancers in Cameroon. Aim Methanol extracts from thirty-four spices and plants, with related ethnobotanical use were investigated for their in vitro cytotoxicity on the human pancreatic cancer cell line MiaPaCa-2, leukemia CCRF-CEM cells and their multidrug resistant (MDR) subline CEM/ADR5000, and the normal human umbilical vein endothelial cells (HUVECs). In addition the anti-angiogenic properties of the most active extracts were investigated. Material and methods The MTS [3-(4,5-dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4-sulfophenyl)-2H-tetrazolium] assay was used for cyto…

PharmacologyXylopia aethiopicaEchinopsPlants MedicinalbiologyTraditional medicinePlant ExtractsAngiogenesis Inhibitorsbiology.organism_classificationAntineoplastic Agents PhytogenicPancreatic NeoplasmsMultiple drug resistanceDorsteniaCell Line TumorDrug DiscoveryCancer cellOfficinalisHumansCameroonDrug Screening Assays AntitumorSpicesCytotoxicityMedicinal plantsCells CulturedJournal of Ethnopharmacology
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Optimization of anti-proliferative activity using a screening approach with a series of bis-heterocyclic G-quadruplex ligands

2013

Abstract Using a phenotypic screening and SAR optimization approach, a phenyl-bis-oxazole derivative has been identified with anti-proliferative activity, optimized with the use of a panel of cancer cell lines. The lead compound was synthesized by means of a short and effective two-step synthesis using Pd-catalyzed direct arylation. The compound stabilizes several quadruplex DNA sequences including a human telomeric DNA and one from the promoter of the HSP90 gene, although the structure–activity relationships of the series are not obviously related to the quadruplex binding.

Phenotypic screeningClinical BiochemistryPharmaceutical ScienceG-quadruplexLigandsBiochemistrychemistry.chemical_compoundInhibitory Concentration 50Structure-Activity RelationshipHeterocyclic CompoundsCell Line TumorDrug DiscoveryHumansMolecular BiologyGeneCell ProliferationOrganic ChemistryCombinatorial chemistrySmall moleculeSettore CHIM/08 - Chimica FarmaceuticaG-QuadruplexeschemistryMolecular MedicineHuman genomeQuadruplex Anti-proliferative Phenotypic screening Telomerase OxazolesDrug Screening Assays AntitumorLead compoundDerivative (chemistry)DNA
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Maternal phenylketonuria in two Sicilian families identified by maternal blood phenylalanine level screening and identification of a new phenylalanin…

1999

not available

Phenylketonuria MaternalPhenylalanine hydroxylasephenylalanine 4 monooxygenasePhenylalanineGene mutationMaternal bloodNeonatal ScreeningPregnancyPhenylketonuriasMedicineHumansMaternal phenylketonuriaGenetic TestingPhenylalanine levelGeneticsbiologybusiness.industryInfant NewbornPhenylalanine HydroxylasePedigreeItalyPediatrics Perinatology and Child HealthMutationbiology.proteinIdentification (biology)FemalebusinessEuropean journal of pediatrics
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Selective Excitation of Guided Waves into Bone Phantoms by a Time-Delayed Laser Diode Array

2012

We excite selectively the Ao and So plate mode into an acrylic bone phantom using a laser diode array. This is done by controlling the time delay between the signals driving the array elements. Selective mode generation is important because it can potentially increase the sensitivity of in vivo osteoporosis screening.

Photoacoustic effect0303 health sciencesMaterials scienceLaser diodebusiness.industry030209 endocrinology & metabolismSelective excitationImaging phantomlaw.inventionOsteoporosis screeningUltrasonic imaging03 medical and health sciences0302 clinical medicineTime delayedOptics030301 anatomy & morphologylawbusinessSensitivity (electronics)2012 Symposium on Photonics and Optoelectronics
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DNA-binding and in vitro cytotoxic activity of platinum(II) complexes of curcumin and caffeine

2019

Abstract Three Pt(II) complexes containing the natural ligands curcumin and caffeine, namely [Pt(curc)(PPh3)2]Cl (1), [PtCl(curc)(DMSO)] (2) (curc = deprotonated curcumin) and trans-[Pt(caffeine)Cl2(DMSO)] (3), were synthesized and fully characterized. The data obtained suggest that, for both 1 and 2, the anion of curcumin is coordinated to the platinum ion via the oxygen atoms of the β-diketonate moiety. Spectroscopic features reveal that in 2 and 3, a DMSO molecule is S-bonded to the metal centre. For 3, all data indicate a square-planar geometry formed by a 9-N bonded caffeine, two trans chloride anions and a DMSO. The three complexes undergo changes in solution upon incubation for 24 h;…

PhotoactivationCurcuminCytotoxicityIntercalation (chemistry)chemistry.chemical_elementCaffeine; Curcumin; Cytotoxicity; DNA interaction; Natural ligands; Photoactivation; Platinum(II) complexAntineoplastic Agents010402 general chemistryLigands01 natural sciencesBiochemistryMedicinal chemistryNucleobaseInorganic Chemistrychemistry.chemical_compoundDrug StabilityCoordination ComplexesCaffeineCell Line TumorMoietyMoleculeAnimalsHumansPlatinumMolecular Structure010405 organic chemistryDNA0104 chemical sciencesDNA interactionchemistryCurcuminPlatinum(II) complexCattleCaffeine Curcumin Cytotoxicity DNA interaction Natural ligands Photoactivation Platinum(II) complexCisplatinDrug Screening Assays AntitumorSelectivityPlatinumNatural ligandsCis–trans isomerism
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$^{222}$Rn emanation measurements for the XENON1T experiment

2021

The selection of low-radioactive construction materials is of utmost importance for the success of low-energy rare event search experiments. Besides radioactive contaminants in the bulk, the emanation of radioactive radon atoms from material surfaces attains increasing relevance in the effort to further reduce the background of such experiments. In this work, we present the $^{222}$Rn emanation measurements performed for the XENON1T dark matter experiment. Together with the bulk impurity screening campaign, the results enabled us to select the radio-purest construction materials, targeting a $^{222}$Rn activity concentration of 10 $\mu$Bq/kg in 3.2 t of xenon. The knowledge of the distribut…

Physics - Instrumentation and DetectorsPhysics and Astronomy (miscellaneous)Radon emanationFOS: Physical scienceschemistry.chemical_element01 natural sciencesNOHigh Energy Physics - Experimentradon: nuclideHigh Energy Physics - Experiment (hep-ex)XENONXenon222 RnPE2_2PE2_10103 physical sciencesActivity concentration[PHYS.HEXP]Physics [physics]/High Energy Physics - Experiment [hep-ex]Dark Matter[PHYS.PHYS.PHYS-INS-DET]Physics [physics]/Physics [physics]/Instrumentation and Detectors [physics.ins-det]010306 general physicsEngineering (miscellaneous)background: radioactivityPhysicsradon: admixture010308 nuclear & particles physicsdetector: surfacescreeningInstrumentation and Detectors (physics.ins-det)chemistryXenon Dark matter 222 Rn radioactivityDark Matter Radon emanation XENON Direct Dark MatterDirect Dark MatterradioactivityAtomic physics
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The analog Resistive Plate Chamber detector of the ARGO-YBJ experiment

2015

The ARGO-YBJ experiment has been in stable data taking from November 2007 till February 2013 at the YangBaJing Cosmic Ray Observatory (4300 m a.s.l.). The detector consists of a single layer of Resistive Plate Chambers (RPCs) (6700 m2) operated in streamer mode. The signal pick-up is obtained by means of strips facing one side of the gas volume. The digital readout of the signals, while allows a high space–time resolution in the shower front reconstruction, limits the measurable energy to a few hundred TeV. In order to fully investigate the 1–10 PeV region, an analog readout has been implemented by instrumenting each RPC with two large size electrodes facing the other side of the gas volume…

Physics - Instrumentation and DetectorsPhysics::Instrumentation and DetectorsAstrophysics::High Energy Astrophysical PhenomenaAir shower detectionFOS: Physical sciencesCosmic raySTRIPSCalorimetrySignallaw.inventionOpticsObservatorylawAir shower detection RPC detector CalorimetryCosmic-ray observatoryphysics.ins-detInstrumentation and Methods for Astrophysics (astro-ph.IM)PhysicsResistive touchscreenbusiness.industryDetectorSettore FIS/01 - Fisica SperimentaleAstrophysics::Instrumentation and Methods for AstrophysicsAstronomy and AstrophysicsInstrumentation and Detectors (physics.ins-det)Core (optical fiber)RPC detectorbusinessAstrophysics - Instrumentation and Methods for Astrophysicsastro-ph.IM
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Time structure of the extensive air shower front

1997

Abstract The GREX/COVER_PLASTEX experiment has measured the temporal and spatial fine structure of the EAS disc at sea level in a new and original way, using resistive plate counter detectors for direct measurements of the arrival time of each particle crossing the detector. Data were taken at EAS core distances up to 100 m for shower size N > 105 (PeV energy range). Arrival times of shower particles were measured with nanosecond accuracy. More than 450000 air shower events have been included in this analysis.

PhysicsCore (optical fiber)Nuclear physicsResistive touchscreenRange (particle radiation)ShowerAir showerDetectorParticleAstronomy and AstrophysicsNanosecondComputational physics
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The effect of dynamical screening on helium (e, 3e) differential cross-sections

2005

A simplified derivation of dynamic screening in the case of three Coulomb-interacting particles in the continuum is given and applied to describe the shapes of multi-differential cross-sections for the (e, 3e) process on the helium atom in which the incident fast electron is treated in first-order Born approximation. A very good agreement with experimental multi-differential cross-sections is obtained for two slow ejected electrons (specifically both electrons have 5 eV) but the strategy appears to be breaking down at intermediate emission energies.

PhysicsDynamic screeningHelium atomchemistry.chemical_elementElectronCondensed Matter PhysicsAtomic and Molecular Physics and Opticschemistry.chemical_compoundchemistryBasso continuoAtomic physicsBorn approximationElectron ionizationHeliumJournal of Physics B: Atomic, Molecular and Optical Physics
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Signal Characteristics of a Resistive-Strip Micromegas Detector with an Integrated Two-Dimensional Readout

2014

In recent years, micropattern gaseous detectors, which comprise a two-dimensional readout structure within one PCB layer, received significant attention in the development of precision and cost-effective tracking detectors in medium and high energy physics experiments. In this article, we present for the first time a systematic performance study of the signal characteristics of a resistive strip micromegas detector with a two-dimensional readout, based on test-beam and X-ray measurements. In particular, comparisons of the response of the two independent readout-layers regarding their signal shapes and signal reconstruction efficiencies are discussed.

PhysicsNuclear and High Energy PhysicsParticle physicsResistive touchscreenPhysics - Instrumentation and DetectorsSignal reconstructionbusiness.industryPhysics::Instrumentation and DetectorsDetectorFOS: Physical sciencesMicroMegas detectorInstrumentation and Detectors (physics.ins-det)Tracking (particle physics)SignalGaseous detectorsOpticsbusinessInstrumentation
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