Search results for "Stimulation"

showing 10 items of 2192 documents

U-46619-induced potentiation of noradrenergic constriction in the human saphenous vein: antagonism by thromboxane receptor blockade.

2001

Objective: We investigated the potentiating effect of U-46619, a synthetic analogue of thromboxane A2 (TXA2), on the adrenergic responses in human saphenous vein. Methods: Saphenous vein rings were obtained from 35 patients undergoing coronary artery bypass surgery. The rings were suspended in organ bath chambers for isometric recording of tension. Results: U-46619 (10−10–3×10−7 mol/l) produced concentration-dependent and endothelium-independent contractile responses. U-46619 (10−10 mol/l) potentiated the contractions elicited by electrical stimulation and potassium chloride, and produced leftward shifts of the concentration–response curve for noradrenaline. The TXA2 receptor antagonist SQ-…

Malemedicine.medical_specialtyDihydropyridinesNifedipinePhysiologymedicine.drug_classThromboxaneReceptors ThromboxaneAdrenergicIn Vitro TechniquesPotassium ChlorideThromboxane receptorThromboxane A2chemistry.chemical_compoundNorepinephrineThromboxane A2Physiology (medical)Internal medicinemedicineHumansVasoconstrictor AgentsSaphenous VeinAgedVoltage-dependent calcium channelDose-Response Relationship DrugChemistryCalcium channelDihydropyridineDrug SynergismMiddle AgedReceptor antagonistCalcium Channel BlockersElectric StimulationStimulation ChemicalEndocrinology15-Hydroxy-11 alpha9 alpha-(epoxymethano)prosta-513-dienoic AcidFemaleEndothelium VascularCardiology and Cardiovascular Medicinemedicine.drugCardiovascular research
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On the peptidergic hypothesis for non-adrenergic non-cholinergic innervation in the rat duodenum

1992

1. The nature of the non-adrenergic, non-cholinergic (NANC) transmitter was studied in vitro in the rat duodenum, by use of an isometric-isovolumic preparation. 2. Electrical field stimulation (EFS) induced a tetrodotoxin (TTX)-sensitive fall both in luminal pressure and in isometric tension. 3. Neurotensin (NT) induced TTX-insensitive inhibitory responses similar to those induced by EFS. Vasoactive intestinal peptide (VIP) caused a delayed, slow, concentration-dependent, TTX-insensitive inhibitory effect, detected only by a change in luminal pressure. 4. alpha-chymotrypsin prevented the NT- and VIP-induced inhibitory effects and antagonized the response to EFS. 5. Apamin antagonized the EF…

Malemedicine.medical_specialtyDuodenumMuscle RelaxationVasoactive intestinal peptideIn Vitro TechniquesBiologyAutonomic Nervous SystemApaminInhibitory postsynaptic potentialchemistry.chemical_compoundDesensitization (telecommunications)Isometric ContractionInternal medicinemedicineAnimalsChymotrypsinReceptorNeurotensinPharmacologymusculoskeletal neural and ocular physiologyGeneral NeuroscienceNeuropeptidesMuscle SmoothRats Inbred StrainsElectric StimulationRatsmedicine.anatomical_structureEndocrinologyApaminchemistryTetrodotoxinDuodenumhormones hormone substitutes and hormone antagonistsVasoactive Intestinal PeptideNeurotensinJournal of Autonomic Pharmacology
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Effects of Substantia Nigra Stimulation on Electrical and Mechanical Activities of the Duodeno-Jejunal Loop, in the Cat

1985

The effect of substantia nigra stimulation on duodeno-jejunal intraluminal pressure and electrical activity was analysed in the cat. An inhibitory influence was noted to occur on both the intestinal pressure and the electrical response activity (ERA): the effect seemed to be in correlation with the stimulus parameters employed. After bilateral vagotomy, the inhibition remained substantially unchanged. The possibility of the existence of a sympathetic pathway mediating the effect is emphasized.

Malemedicine.medical_specialtyDuodenumPhysiologymedicine.medical_treatmentStimulationSubstantia nigraInhibitory postsynaptic potentialBiochemistryFunctional LateralityMidbrainIleumInternal medicinemedicineCarnivoraAnimalsbiologyFissipediaElectric Conductivitybiology.organism_classificationVagotomyElectric StimulationSubstantia NigraEndocrinologyCatsFemalemedicine.symptomMuscle contractionArchives Internationales de Physiologie et de Biochimie
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Modulation of adrenergic contraction of dog pulmonary arteries by nitric oxide and prostacyclin.

1999

Abstract The aim of this work was to investigate the influence of endothelium-derived nitric oxide and prostaglandins on the contractile responses of isolated dog pulmonary arteries to electrical field stimulation and noradrenaline. Electrical field stimulation (1–8 Hz, 20 v, 0.25 ms duration, for 30 s) produced frequency-dependent contractions that were abolished by tetrodotoxin, guanethidine and, prazosin (all at 10−6 M). Noradrenaline induced concentration-dependent contractions with an EC50 of 1.85 × 10−6 M. The increases in tension induced by electrical stimulation and noradrenaline were of greater magnitude in arteries denuded of endothelium. In segments with endothelium, NG-nitro- l …

Malemedicine.medical_specialtyEndotheliumArginineIndomethacinAdrenergicProstacyclinStimulationIn Vitro TechniquesPulmonary ArteryNitric OxideNitric oxidechemistry.chemical_compoundNorepinephrineDogsInternal medicinePrazosinmedicineAnimalsCyclooxygenase InhibitorsDrug InteractionsEnzyme InhibitorsGuanethidineAntihypertensive AgentsPharmacologyEpoprostenolElectric Stimulationmedicine.anatomical_structureEndocrinologyNG-Nitroarginine Methyl EsterchemistryVasoconstrictionProstaglandinsFemalemedicine.drugGeneral pharmacology
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β-Adrenoceptors differentially regulate vascular tone and angiogenesis of rat aorta via ERK1/2 and p38

2014

β-Adrenoceptors (β-ARs) modulate ERK1/2 and p38 in different cells, but little is known about the contribution of these signaling pathways to the function of β-ARs in vascular tissue. Immunoblotting analysis of rat aortic rings, primary endothelial (ECs) and smooth muscle cells (SMCs) isolated from aorta showed that β-AR stimulation with isoprenaline activated p38 in aortic rings and in both cultured cell types, whereas it had a dual effect on ERK1/2 phosphorylation, decreasing it in ECs while increasing it in SMCs. These effects were reversed by propranolol, which by itself increased p-ERK1/2 in ECs. Isoprenaline β-AR mediated vasodilation of aortic rings was potentiated by the ERK1/2 inhi…

Malemedicine.medical_specialtyEndotheliumPhysiologyAngiogenesisVasodilator AgentsAdrenergic beta-AntagonistsMyocytes Smooth MuscleNeovascularization PhysiologicAorta ThoracicStimulationVasodilationFibroblast growth factorp38 Mitogen-Activated Protein KinasesMuscle Smooth VascularInternal medicineIsoprenalinemedicine.arteryReceptors Adrenergic betamedicineAnimalsHumansRats WistarMitogen-Activated Protein Kinase 1PharmacologyMatrigelAortaMitogen-Activated Protein Kinase 3business.industryAdrenergic beta-AgonistsPropranololRatsVasodilationHEK293 Cellsmedicine.anatomical_structureEndocrinologycardiovascular systemMolecular MedicineEndothelium Vascularbusinessmedicine.drugVascular Pharmacology
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Contribution of both ?- and ?-adrenoceptors to the inotropic effects of catecholamines in the rabbit heart

1992

The functional role of alpha-adrenoceptors was investigated in different parts of the rabbit heart. Phenylephrine (PE) caused a marked increase in force of contraction (Fc) and a prolongation of the action potential (AP) in preparations from the left atrium and the right ventricle. The response was less pronounced in the right atrium and in the left ventricle, whereas APs of spontaneously beating sinoatrial preparations remained completely unchanged. Phentolamine as well as the diesters phorbol 12,13 dibutyrate (PDBu) or 12-O-tetradecanoyl-phorbol-13-acetate (TPA) eliminated the effects of PE. The contribution of alpha-adrenoceptors to the effects of adrenaline (Adr) and noradrenaline (NA) …

Malemedicine.medical_specialtyEpinephrineAction PotentialsStimulationPropranololNorepinephrinechemistry.chemical_compoundPhentolamineInternal medicineIsoprenalinePhorbol EstersReceptors Adrenergic betamedicineAnimalsDrug InteractionsPhentolaminePhenylephrinePharmacologyChemistryMyocardiumHeartGeneral MedicineReceptors Adrenergic alphaMyocardial ContractionPropranololEndocrinologymedicine.anatomical_structureVentricleCirculatory systemPhorbolFemaleRabbitsmedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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Fixation-related potentials in naming speed: A combined EEG and eye-tracking study on children with dyslexia.

2021

Abstract Objective We combined electroencephalography (EEG) and eye-tracking recordings to examine the underlying factors elicited during the serial Rapid-Automatized Naming (RAN) task that may differentiate between children with dyslexia (DYS) and chronological age controls (CAC). Methods Thirty children with DYS and 30 CAC (Mage = 9.79 years; age range 7.6 through 12.1 years) performed a set of serial RAN tasks. We extracted fixation-related potentials (FRPs) under phonologically similar (rime-confound) or visually similar (resembling lowercase letters) and dissimilar (non-confounding and discrete uppercase letters, respectively) control tasks. Results Results revealed significant differe…

Malemedicine.medical_specialtyEye MovementsElectroencephalographyAudiologyDyslexiaPhysiology (medical)medicineReaction TimedysleksiaHumansEEGSet (psychology)ChildEye-Tracking Technologyeye-trackingmedicine.diagnostic_testDyslexiaFixation-Related PotentialsElectroencephalographyNeurophysiologymedicine.diseaseSensory SystemsRANNeurologyReadingpsykologiset testitFixation (visual)RankatseenseurantaEye trackingFemaleNeurology (clinical)PsychologyNeurocognitivePhotic StimulationClinical neurophysiology : official journal of the International Federation of Clinical Neurophysiology
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Modulation of cytosolic free calcium concentration by ?1-adrenoceptors in rat atrial cells

1992

The effects of α1-adrenoceptor stimulation by phenylephrine (PE) and β-adrenoceptor stimulation by isoprenaline (ISO) on Ca2+ current (ICa) and free intracellular Ca2+ concentration ([Ca2+]i) were studied in isolated atrial myocytes from rat hearts. PE did not significantly affect the magnitude of ICa, whereas large increases of peak ICa were observed in response to ISO. In electrically driven cells, PE evoked a concentration-dependent, gradual increase in diastolic [Ca2+]i and, initially, an increase in the height of peak [Ca2+]i transients. When the diastolic [Ca2+]i was increased to a greater extent, the amplitude of [Ca2+]i transients was decreased. Simultaneous measurements of [Ca2+]i …

Malemedicine.medical_specialtyFura-2chemistry.chemical_elementStimulationIn Vitro TechniquesCalciumPhenylephrinechemistry.chemical_compoundInternal medicineIsoprenalinemedicineAnimalsHeart AtriaPhenylephrinePharmacologyMembrane potentialIsoproterenolRats Inbred StrainsDepolarizationGeneral MedicineReceptors Adrenergic alphaRatsElectrophysiologyElectrophysiologyEndocrinologychemistryCalciumAdrenergic alpha-Agonistsmedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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Increase by ?-adrenolytic drugs of acetylcholine release evoked by field stimulation of the guinea-pig ileum

1979

The release of acetylcholine evoked by field stimulation of the guinea-pig ileum (3 Hz) is increased by yohimbine and tolazoline but not affected by phentolamine. It is proposed that yohimbine and tolazoline by blocking alpha-adrenoceptors of the cholinergic nerves abolish the inhibition caused by endogenous noradrenaline, and thus facilitate the output of acetylcholine.

Malemedicine.medical_specialtyGuinea PigsAlpha (ethology)IleumEndogenyIn Vitro TechniquesPhentolamineIleumInternal medicinemedicineAnimalsTolazolineAdrenergic alpha-AntagonistsMyenteric plexusPharmacologyChemistryMuscle SmoothGeneral MedicineAcetylcholineElectric StimulationYohimbinemedicine.anatomical_structureEndocrinologyFemaleAcetylcholinemedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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Differential effects of nitric oxide donors on basal and electrically evoked release of acetylcholine from guinea-pig myenteric neurones

1996

1. The effects of the nitric oxide (NO) donors, 3-morpholino-sydnonimine (SIN-1), S-nitroso-N-acetylpenicillamine (SNAP) and sodium nitroprusside on basal and electrically evoked release of [3H]-acetylcholine were studied in myenteric plexus longitudinal muscle preparations of the guinea-pig small intestine preincubated with [3H]-choline. 2. The NO donors concentration-dependently increased basal release of [3H]-acetylcholine. The increase in release was calcium-dependent and was prevented in the presence of tetrodotoxin. Superoxide dismutase (150 u ml-1) potentiated the effect of SIN-1. The selective inhibitor of soluble guanylyl cyclase, 1H-[1,2,4]oxadiazolo[4,3-alpha]quinoxalin-1-one (OD…

Malemedicine.medical_specialtyGuinea PigsMyenteric PlexusNitric Oxidechemistry.chemical_compoundInternal medicinemedicineAnimalsEnzyme InhibitorsPhosphodiesterase inhibitorMyenteric plexusPharmacologyDose-Response Relationship DrugEndothelium-derived relaxing factorAcetylcholineElectric StimulationEndocrinologychemistryMolsidomineFemaleSodium nitroprussideS-Nitroso-N-acetylpenicillamineSoluble guanylyl cyclaseZaprinastAcetylcholineResearch Articlemedicine.drugBritish Journal of Pharmacology
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