Search results for "TF"

showing 10 items of 1652 documents

Synchronizing the release rates of salicylate and indomethacin from degradable chitosan hydrogel and its optimization by definitive screening design.

2018

Abstract Three types of ionically crosslinked (with citric acid) chitosan discs were loaded with the highly water- soluble drug, sodium salicylate (SS) and the poorly water-soluble drug, indomethacin (Ind). In separate experiments the hydrated discs were immersed in a de-crosslinking solution comprising of different concentrations of calcium chloride, which induced a controlled erosion of the discs, a process which was optimized to synchronize the release rates of the two drugs over a predetermined period of time. The optimization was accomplished by manipulating six factors: chitosan MW, its amount in the formulation, the concentration of the crosslinker agent, the concentration of the de-…

3003DrugSynchronized release ratemedia_common.quotation_subjectIndomethacinPharmaceutical Sciencechemistry.chemical_elementmacromolecular substances02 engineering and technologyCalciumTriggered erosionCitric AcidChitosan03 medical and health scienceschemistry.chemical_compoundCrosslinked chitosan0302 clinical medicineDrug Delivery SystemsScreening designMultifactorial definitive screening designDissolutionSodium salicylatemedia_commonChitosanChromatographytechnology industry and agricultureHydrogelsCrosslinked chitosanDual drug platform021001 nanoscience & nanotechnologyDrug LiberationCross-Linking Reagentschemistry030220 oncology & carcinogenesisDrug Design0210 nano-technologyCitric acidSalicylic AcidEuropean journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
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Antidiabetic Drugs in NAFLD: The Accomplishment of Two Goals at Once?

2018

Non-Alcoholic Fatty Liver Disease (NAFLD) is the most common cause of chronic liver disease in Western countries, accounting for 20–30% of general population and reaching a prevalence of 55% in patients with type 2 diabetes mellitus (T2DM). Insulin resistance plays a key role in pathogenic mechanisms of NAFLD. Many drugs have been tested but no medications have yet been approved. Antidiabetic drugs could have a role in the progression reduction of the disease. The aim of this review is to summarize evidence on efficacy and safety of antidiabetic drugs in patients with NAFLD. Metformin, a biguanide, is the most frequently used drug in the treatment of T2DM. To date 15 randomized controlled t…

3003medicine.medical_specialtymedicine.drug_classmedicine.medical_treatmentlcsh:Medicinelcsh:RS1-441Pharmaceutical Sciencehepatic cirrhosis030209 endocrinology & metabolismReviewChronic liver diseaseGastroenterologylcsh:Pharmacy and materia medica03 medical and health sciences0302 clinical medicineInsulin resistanceInternal medicineDiabetes mellitusDrug DiscoverymedicineBiguanidebusiness.industryLiraglutideInsulinlcsh:RFatty liverThiazolidinedionenutritional and metabolic diseasesnon-alcoholic fatty liver diseaseLiraglutidemedicine.diseaseMetforminMetforminHepatic cirrhosiMolecular Medicine030211 gastroenterology & hepatologyThiazolidinedionesnon-alcoholic steatohepatitisbusinessNon-alcoholic steatohepatitimedicine.drugPharmaceuticals (Basel, Switzerland)
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Wind accretion in the massive X-ray binary 4U 2206+54: abnormally slow wind and a moderately eccentric orbit

2006

Massive X-ray binaries are usually classified depending on the properties of the donor star in classical, supergiant and Be X-ray binaries. The massive X-ray binary 4U 2206+54 does not fit in any of these groups, and deserves a detailed study to understand how the transfer of matter and the accretion on to the compact object take place. To this end we study an IUE spectrum of the donor and obtain a wind terminal velocity (v_inf) of ~350 km/s, which is abnormally slow for its spectral type. We also analyse here more than 9 years of available RXTE/ASM data. We study the long-term X-ray variability of the source and find it to be similar to that observed in the wind-fed supergiant system Vela …

4U 2206+54X-ray binaryBinary numberFOS: Physical sciencesOutflows Emission-lineOrbital eccentricityAstrophysicsWindsCompact starUNESCO::ASTRONOMÍA Y ASTROFÍSICAVelaAstrophysicsIndividual starsPhysicsAstrophysics (astro-ph)BD +53◦2790BeAstronomy and AstrophysicsOrbital period:ASTRONOMÍA Y ASTROFÍSICA::Cosmología y cosmogonia [UNESCO]Accretion (astrophysics)X-rays binariesX-rays individualsX-rays binaries ; X-rays individuals ; 4U 2206+54 ; Individual stars ; BD +53◦2790 ; Winds ; Outflows Emission-line ; BeSpace and Planetary ScienceUNESCO::ASTRONOMÍA Y ASTROFÍSICA::Cosmología y cosmogoniaSupergiant:ASTRONOMÍA Y ASTROFÍSICA [UNESCO]
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A flexible and reconfigurable 5G networking architecture based on context and content information

2017

The need for massive content delivery is a consolidated trend in mobile communications, and will even increase for next years. Moreover, while 4G maturity and evolution is driven by video contents, next generation (5G) networks will be dominated by heterogeneous data and additional massive diffusion of Internet of Things (IoT). The current network architecture is not sufficient to cope with such traffic, which is heterogeneous in terms of latency and QoS requirements, and variable in space and time. This paper proposes architectural advances to endow the network with the necessary flexibility helping to adapt to these varying traffic needs by providing content and communication services whe…

5G networkingComputer scienceflexible HW/SW platforms 5G networking context-awareness content-centric networks reconfigurability050801 communication & media studies02 engineering and technologyflexible HW/SW platforms 5G networking context-awareness; content-centric networks; reconfigurability.0508 media and communications0202 electrical engineering electronic engineering information engineeringReference architectureArchitectureNetwork architecturebusiness.industrySettore ING-INF/03 - TelecomunicazioniQuality of service05 social sciencesflexible HW/SW platformscontent-centric networkscontext-awarenessReconfigurability020206 networking & telecommunicationsApplications architectureMobile telephonybusinessreconfigurability5GComputer network
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Designing the 5G network infrastructure: a flexible and reconfigurable architecture based on context and content information

2018

5G networks will have to offer extremely high volumes of content, compared to those of today’s. Moreover, they will have to support heterogeneous traffics, including machine-to-machine, generated by a massive volume of Internet-of-Things devices. Traffic demands will be variable in time and space. In this work, we argue that all this can be achieved in a cost-effective way if the network is flexible and reconfigurable. We present the Flex5Gware network architecture, designed to meet the above requirements. Moreover, we discuss the links between flexibility and reconfigurability, on the one side, and context awareness and content awareness, on the other; we show how two of the building…

5G networkingStandardizationFlexible HW/SW platformComputer Networks and CommunicationsComputer scienceContext-awareneDistributed computinglcsh:TK7800-8360050801 communication & media studies02 engineering and technologylcsh:Telecommunication0508 media and communicationslcsh:TK5101-6720flexible HW/SW platforms 5G networking context-awareness; content-awareness; reconfigurability0202 electrical engineering electronic engineering information engineeringContext awarenessArchitecturecontent-awarenessNetwork architectureAccess networklcsh:Electronicsflexible HW/SW platforms05 social sciencescontext-awarenessReconfigurabilityControl reconfigurationComputer Science Applications1707 Computer Vision and Pattern Recognition020206 networking & telecommunicationsComputer Science ApplicationsContent-awareneSignal Processingreconfigurability5GEURASIP Journal on Wireless Communications and Networking
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Tactics of invisibility : How people in vulnerable positions make datafied everyday life livable

2022

Various data platforms force the individual into constant presence and visibility. However, the ways in which datafied environments relate to experienced vulnerabilities in our everyday lives remain unclear. Through diaries produced by and interviews with participants from three groups who occupy presumably vulnerable positions and who currently live in Finland, we explore the ways in which people challenge expectations and prior assumptions related to forced visibility. Using the concept of tactics developed by de Certeau, we aim to understand how individuals make everyday surveillance culture livable through what we call tactics of invisibility. Based on our analysis, we identify three k…

6131 Theatre dance music other performing artsvulnerabilitiesSociology and Political ScienceCommunicationtacticssurveillancenäkymättömyysinvisibilitytarkkailudata platformshaavoittuvuustaktiikka
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Servicios de intermediación en línea en Europa : diseño de un sistema específico de solución de controversias

2021

Este trabajo analiza el sistema de solución de controversias específicamente diseñado, con la introducción de alternativas a la jurisdicción, en el Reglamento (UE) 2019/1150 sobre el fomento de la equidad y la transparencia para los usuarios profesionales de servicios de intermediación en línea, que ha entrado recientemente en vigor.

:CIENCIAS JURÍDICAS [UNESCO]online intermediate servicesOnline platformsque ha entrado recientemente en vigor. This paper analyses the specific designed dispute resolution systemthe right to take judicial action 560 585dispute resolution methodsinternal complainthandling systemwith the introduction of alternatives to jurisdictioncon la introducción de alternativas a la jurisdicciónin the Regulation (EU) 2019/1150 on promoting fairness and transparency for business users of online intermediation services2070-8157 22082 Revista Boliviana de Derecho 584568 2021 32 8055231 Servicios de intermediación en línea en Europa diseño de un sistema específico de solución de controversias Fernández MasiáUNESCO::CIENCIAS JURÍDICASen el Reglamento (UE) 2019/1150 sobre el fomento de la equidad y la transparencia para los usuarios profesionales de servicios de intermediación en líneaEnrique Este trabajo analiza el sistema de solución de controversias específicamente diseñadomediationhas recently entered into force
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Polyoxypregnanes as safe, potent, and specific ABCB1-inhibitory pro-drugs to overcome multidrug resistance in cancer chemotherapy in vitro and in vivo

2021

Multidrug resistance (MDR) mediated by ATP binding cassette subfamily B member 1 (ABCB1) is significantly hindering effective cancer chemotherapy. However, currently, no ABCB1-inhibitory drugs have been approved to treat MDR cancer clinically, mainly due to the inhibitor specificity, toxicity, and drug interactions. Here, we reported that three polyoxypregnanes (POPs) as the most abundant constituents of Marsdenia tenacissima (M. tenacissima) were novel ABCB1-modulatory pro-drugs, which underwent intestinal microbiota-mediated biotransformation in vivo to generate active metabolites. The metabolites at non-toxic concentrations restored chemosensitivity in ABCB1-overexpressing cancer cells v…

ABCC1 ATP binding cassette subfamily C member 1IC50 half maximal inhibitory concentrationMultidrug resistancePharmacologyNADPH reduced nicotinamide adenine dinucleotide phosphateF bioavailabilitychemistry.chemical_compoundPCR polymerase chain reaction0302 clinical medicineMDR multidrug resistanceECL electrochemiluminescencet1/2 elimination half-lifeLC–MS liquid chromatography coupled with mass spectrometryN.D. not detectedGeneral Pharmacology Toxicology and PharmaceuticsBBB blood–brain barriermedia_commonATF3 activating transcription factor 30303 health sciencesChemistryABC ATP-binding cassetteNMPA National Medical Products AdministrationPXR pregnane X receptorSDS-PAGE sodium dodecyl sulfate-polyacrylamide gel electrophoresisHBSS Hankʹs balanced salt solutionABCB1Combination chemotherapyProdrugMarsdenia tenacissimaCmax peak concentrationPaclitaxelGAPDH glyceraldehyde-3-phosphate dehydrogenase030220 oncology & carcinogenesisBHI brain heart infusionOriginal ArticleAUC0–∞ area under plasma concentration vs. time curveMRT mean residence timeDrugmedia_common.quotation_subjectRM1-950Vd volume of distributionABCB1 ATP binding cassette subfamily B member 1UIC-2 mouse monoclonal ABCB1 antibodyABCG2 ATP binding cassette subfamily G member 2Combination chemotherapyCYP cytochrome P450 isozymePI propidium iodideTEER transepithelial electrical resistance03 medical and health sciencesPBS phosphate buffer salineFBS fetal bovine serumDox doxorubicinIn vivoPOP polyoxypregnanemedicine030304 developmental biologyEVOM epithelial tissue voltohmmeterTmax time for peak concentrationCancerLBE lowest binding energyPE phycoerythrinmedicine.diseaseMultiple drug resistancePolyoxypregnanePapp apparent permeabilityN.A. not applicableCancer cellH&E hematoxylin and eosinMDR1a multidrug resistance protein 1aTherapeutics. PharmacologyqPCR quantitative PCRM. tenacissima Marsdenia tenacissimaCL clearanceSD standard derivationActa Pharmaceutica Sinica B
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Accretion in strong field gravity with eXTP

2019

In this paper we describe the potential of the enhanced X-ray Timing and Polarimetry (eXTP) mission for studies related to accretion flows in the strong field gravity regime around both stellar-mass and supermassive black-holes. eXTP has the unique capability of using advanced 'spectral-timing-polarimetry' techniques to analyze the rapid variations with three orthogonal diagnostics of the flow and its geometry, yielding unprecedented insight into the inner accreting regions, the effects of strong field gravity on the material within them and the powerful outflows which are driven by the accretion process.

ACTIVE GALACTIC NUCLEIAccretionaccretion; black holes physics; X-ray; Physics and Astronomy (all)black holes physicAstronomyAstrophysics::High Energy Astrophysical PhenomenaBlack holes physicsPolarimetryFOS: Physical sciencesBLACK-HOLE SPINGeneral Physics and AstronomyStrong fieldAstrophysicsAstrophysics::Cosmology and Extragalactic Astrophysics01 natural sciencesX-rayPhysics and Astronomy (all)ELECTROMAGNETIC EMISSIONSettore FIS/05 - Astronomia e Astrofisicablack holes physicsaccretion0103 physical sciencesAstrophysics::Solar and Stellar Astrophysics010306 general physics010303 astronomy & astrophysicsAstrophysics::Galaxy AstrophysicsHigh Energy Astrophysical Phenomena (astro-ph.HE)XMM-NEWTONPhysicsLENS-THIRRING PRECESSION[SDU.ASTR]Sciences of the Universe [physics]/Astrophysics [astro-ph]QUASI-PERIODIC OSCILLATIONS[SDU.ASTR.HE]Sciences of the Universe [physics]/Astrophysics [astro-ph]/High Energy Astrophysical Phenomena [astro-ph.HE]IRON KAccretion (astrophysics)X ray[SDU]Sciences of the Universe [physics]ULTRA-FAST OUTFLOWSAstrophysics::Earth and Planetary AstrophysicsSPECTRAL FEATURESAstrophysics - High Energy Astrophysical Phenomena[PHYS.ASTR]Physics [physics]/Astrophysics [astro-ph]X-RAY BINARIESScience China Physics, Mechanics & Astronomy
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Ethical Requirements Stack : A framework for implementing ethical requirements of AI in software engineering practices

2023

AI ethicsAIAI ethics principlesEthical requirementsEthical requirements stackAgile portfolio managementetiikkatekoäly
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