Search results for "TG"

showing 10 items of 2275 documents

Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor

2013

The Eph–ephrin system plays a critical role in tumor growth and vascular functions during carcinogenesis. We had previously identified cholanic acid as a competitive and reversible EphA2 antagonist able to disrupt EphA2-ephrinA1 interaction and to inhibit EphA2 activation in prostate cancer cells. Herein, we report the synthesis and biological evaluation of a set of cholanic acid derivatives obtained by conjugation of its carboxyl group with a panel of naturally occurring amino acids with the aim to improve EphA2 receptor inhibition. Structure-activity relationships indicate that conjugation of cholanic acid with linear amino acids of small size leads to effective EphA2 antagonists whereas …

EphA2 antagonistsStereochemistryStructure-activity relationship studiesPharmaceutical Sciencemedicine.disease_causeArticleProtein Structure SecondaryAnalytical Chemistrylcsh:QD241-441Inhibitory Concentration 50Structure-Activity Relationshipchemistry.chemical_compoundamino acid conjugateslcsh:Organic chemistryEphA2 anatgonistscholanic acid; amino acid conjugates; EphA2 antagonists; structure-activity relationshipsCell Line TumorDrug DiscoveryAromatic amino acidsmedicineHumansPhosphorylationPhysical and Theoretical ChemistryReceptorbile acids; EphA2 anatgonists; Structure-activity relationship studies; amino acid conjugatesbile acidschemistry.chemical_classificationBinding SitesReceptor EphA1Receptor EphA2structure-activity relationshipsOrganic ChemistryAntagonistCholic AcidsHydrogen BondingEPH receptor A2Amino acidMolecular Docking SimulationCholanic acidcholanic acidchemistryBiochemistryChemistry (miscellaneous)Molecular MedicineCarcinogenesisProtein Processing Post-TranslationalProtein BindingConjugateMolecules
researchProduct

Evaluating the citywide Edinburgh 20mph speed limit intervention effects on traffic speed and volume: A pre-post observational evaluation.

2021

Objectives Traffic speed is important to public health as it is a major contributory factor to collision risk and casualty severity. 20mph (32km/h) speed limit interventions are an increasingly common approach to address this transport and health challenge, but a more developed evidence base is needed to understand their effects. This study describes the changes in traffic speed and traffic volume in the City of Edinburgh, pre- and 12 months post-implementation of phased city-wide 20mph speed limits from 2016–2018. Methods The City of Edinburgh Council collected speed and volume data across one full week (24 hours a day) pre- and post-20mph speed limits for 66 streets. The pre- and post-sp…

EpidemiologyGeography Planning and DevelopmentSocial SciencesTransportation/dk/atira/pure/core/keywords/exercise_nutrition_and_health_sciences20mph speed limitsCognitionAccident PreventionRA0421RA0421 Public health. Hygiene. Preventive Medicine/dk/atira/pure/subjectarea/asjc/3300/3313Medicine and Health SciencesPsychologyPublic and Occupational Health/dk/atira/pure/sustainabledevelopmentgoals/industry_innovation_and_infrastructureEvaluationGeographic AreasMultidisciplinaryGeographyHealth PolicyTraumatic Injury Risk FactorsQFOS: Social sciencesRAccidents Traffic/dk/atira/pure/subjectarea/asjc/2700/27393rd-DASSPEED LIMITSResearch AssessmentTransportation InfrastructureSDG 11 - Sustainable Cities and CommunitiesTreatment Outcome/dk/atira/pure/subjectarea/asjc/3300/3322Evaluation Studies as TopicRoad Traffic Collisions/dk/atira/pure/sustainabledevelopmentgoals/good_health_and_well_beingEngineering and TechnologyMedicinePublic HealthSafetyResearch ArticleUrban AreasAutomobile DrivingScienceDecision MakingHuman GeographyResearch and Analysis MethodsCivil EngineeringUrban Geography/dk/atira/pure/sustainabledevelopmentgoals/sustainable_cities_and_communitiesSDG 3 - Good Health and Well-beingHumansUrban InfrastructureCitiespre-post observational evaluationPublic Health Environmental and Occupational HealthCognitive PsychologyBiology and Life Sciences/dk/atira/pure/subjectarea/asjc/3300/3305FOS: Engineering and technologyRoadsUrban StudiesLogistic ModelsScotlandMedical Risk FactorstransportEarth SciencesCognitive Science20mphSDG 9 - Industry Innovation and InfrastructureSPS Exercise Nutrition and Health SciencesNeuroscience
researchProduct

“Living in Contaminated Areas”—Consideration of Different Perspectives

2020

Following large-scale nuclear power plant accidents such as those that occurred at Chernobyl (Ukraine) in 1986 and Fukushima Daiichi (Japan) in 2011, large populations are living in areas containing residual amounts of radioactivity. As a key session of the ConRad conference, experts were invited from different disciplines to provide state-of-the-art information on the topic of "living in contaminated areas." These experts provided their different perspectives on a range of topics including radiation protection principles and dose criteria, environmental measurements and dose estimation, maintaining decent living and working conditions, evidence of health risks, and social impact and risk c…

EpidemiologyHealth Toxicology and MutagenesisSocial impact030218 nuclear medicine & medical imaginglaw.invention03 medical and health sciences0302 clinical medicineGeographyFukushima daiichiSDG 3 - Good Health and Well-beinglaw030220 oncology & carcinogenesisDose estimationNuclear power plant/dk/atira/pure/sustainabledevelopmentgoals/good_health_and_well_beingRisk communicationRadiology Nuclear Medicine and imagingEnvironmental planningHealth Physics
researchProduct

Differential Effect on the Determinants of the Late Payments According to the Economic Cycle

2018

From 2004 to 2007, the Spanish financial system grew at a very rapid rate. However, from 2008 to 2012 impairment losses amounted equivalent to 25% of Spanish GDP.The objective of this paper is investigate how have affected the main problems that have suffered the Spanish economy on the late payments on Spanish credit institutions. And to check whether the effect of these problems is different on stages of growth with respect to the stages of crisis.The main results, according the test Chow, confirmed that there is a structural break in the model in 2007. Also the increase in unemployment increases the late payments   and this increase is greater in the stages of growth compared to the stage…

Equity (economics)Rapid ratemedia_common.quotation_subjectStructural breakBancs hipotecarisAturDifferential (mechanical device)PaymentRecessionHabitatge FinançamentUnemploymentPréstecs hipotecaris d'alt riscEconomicsBusiness cycleDemographic economicshealth care economics and organizationsmedia_common
researchProduct

Odwrócony kredyt hipoteczny jako źródło uposażenia emerytalnego (Reverse mortgage as a source of pension equipment)

2016

Equity releaseReverse mortgageEconomicsEconomic historyPrace Naukowe Uniwersytetu Ekonomicznego we Wrocławiu
researchProduct

Jutekliskās uztveres tematizācija Pētera Handkes stāstā „Senviktuāras kalna mācība”

2015

Bakalaura darbs ir veltīts tēmai „Jutekliskās uztveres tematizācija Pētera Handkes stāstā Senviktuāra kalna mācība”. Darba mērķis ir izmeklēt un aplūkot Pētera Handkes jutekliskās uztveres atspoguļojumu stāstā Senviktuāra kalna mācība. Darba uzdevums ir izpētīt rakstnieka Pētera Handkes personību un viņa slaveno tetraloģiju, it īpaši tetraloģijas otro daļu. Darbs ir sadalīts trijās nodaļās. Pirmajā nodaļā tiek apskatīts un visparēji raksturots jēdziens „mūsdienu literatūra”, kā arī tiek apskatīta tā laika politiskā un sabiedriskā situācija Vācijā un Austrijā. Papildus tiek apskatīta mūsdienu rakstnieku paaudze un Pēters Handke tiek prezentēts kā mūsdienu vācu rakstnieku paaudzes populārs pā…

Erläuterung des Begriffs Gegenwartsliteratur. Charakterisierung der zeitgenössischen Literatur und des Epochenhitergrundes.ValodniecībaBekannte Tetralogie Peter Handkes mit dem Titel Langsame Heimkehr (1979 - 1981); Darstellung der Handlung der drei Erzählungen Langsame Heimkehr Die Lehre der Sainte-Victoire und Kindergeschichte und dem dramatischen Gedicht Über die Dörfer.Thema der Bakkalaureusarbeit lautet „Thematisierung der sinnlichen Wahrnehmung in Peter Handkes Erzählung Die Lehre der Sainte-Victoire“.Übersicht über die Schriftstellergeneration der Gegenwart. Peter Handke als einer der bekanntesten zeitgenössischen deutschsprachigen Autoren; seine Biographie und literariche Entwicklung.Untersuchungsobjekt für diese Arbeit – das 1980 mit einem Vorwort von Karl Krolow herausgegebene Buch von Peter Handke „Die Lehre der Sainte-Victoire“.
researchProduct

Programa experimental per al foment de l'ús de llibres de text en dispositius electrònics : estudi d'un cas

2015

L'aparició al mercat de les tauletes digitals ha marcat un abans i un després en l'ensenyament. Aquesta eina tecnològica es perfila com un recurs innovador de cara a la seua utilització educativa. I, com tots sabem, l'escola no pot quedar-se al marge d'aquesta revolució tecnològica. Analitzar l'impacte sobre l'alumnat de l'ús de les tauletes digitals, extraure els seus avantatges i inconvenients i generar idees sobre el seu ús ens pot portar a una educació de qualitat. En aquest article s’analitza la posada en pràctica d’aquest nou projecte anomenat Programa experimental per al foment de l'ús de llibres de text en dispositius electrònics anomenats tauletes digitals en un centre de titularit…

EscolaAlumnatLibros electrónicosMestresSchool teacherVentajasLlibres electrònicsAvantatgesAlumnadoTauletes digitalsEscuelaMaestrasAdvantagesTabletStudentsElectronic booksDIM: Didáctica, Innovación y Multimedia
researchProduct

Poesias con que han adornado la fachada de su templo los PP. de la Escuela Pia con el plausible motivo de la venida de SS. MM. y AA. a Valencia.

Sign.: [ ]2, A-M2, N3

Escolapis (València) 1802Poesia llatina S.XIXVisites oficials Comunitat valenciana València 1802Poesia castellana S.XIXCarles IV rei d'Espanya 1748-1819 Viatges València (Comunitat Valenciana) 1802
researchProduct

Ioan. Bapt. Cardonae ... De regia S. Laurentii bibliotheca ; De Pontificia Vaticana ; De expungendis haereticor. propiis nominib. ; De dyptichis.

1587

Orn.

Escorial El (Monestir : Comunitat de Madrid). Biblioteca Obres anteriors a 1800Escorial (Monestir). Biblioteca Obres anteriors al 1800Heretges cristiansBiblioteca apostolica vaticana Obres anteriors al 1800Biblioteca Apostolica Vaticana Obres anteriors a 1800DIG-BH
researchProduct

Poblacion general de España : Sus trofeos, blasones y conquistas heroycas : Descripciones agradables, grandezas notables, excelencias gloriosas y su…

1675

Esc. real xil. a la f. 259 [i. e. 257 Port. a dues tintes Text a dues col. Sign.: ^8, A8, B-Z6, Aa-Vu6, Xx4 Errates tip. a la fol.: de la 258 passa a la 261

Espanya Història CronologiaEspanya Descripció i viatges Obres anteriors a 1800
researchProduct